首页 工具
登录
购物车

搜索结果

Search Results for " pseudomonas "

116

抑制剂 & 化合物

37

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T22269 Benzyldodecyldimethylammonium Chloride Dihydrate

Antibacterial Microbiology/Virology
Benzyldodecyldimethylammonium chloride dihydrate 可以用作杀虫试剂,可以靶向耐药性细菌,如耐甲氧西林金黄色葡萄球菌、耐多药铜绿假单胞菌等,且具有浓度依赖性。
T0396 Pipemidic acid

吡哌酸,Acido pipemidico

Antibacterial; Antibiotic Microbiology/Virology
Pipemidic acid (Acido pipemidico) 是一种新型抗菌剂,对革兰氏阴性菌和某些革兰氏阳性细菌具有活性,可研究肠道、泌尿和胆道感染。
T4201 Avibactam sodium

阿维巴坦,AVE-1330A,阿维巴坦钠,NXL-104

Antibacterial; Antibiotic Microbiology/Virology
Avibactam sodium (NXL-104) 是一种可逆的 β-内酰胺酶抑制剂,抑制 TEM-1,P99和KPC-2 β-内酰胺酶,IC50分别为8、80和38 nM。
T1293 Gatifloxacin

BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin (CG5501) 是一种具有广谱抗菌活性的氟喹诺酮类抗生素。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml) 和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml)。在动物模型中,它有抗细菌性结膜炎作用。
T38862 Nandrolone acetate

19-Nortestosterone 17β-acetate

Others Others
Nandrolone acetate (19-Nortestosterone 17β-acetate) 是一种甾体酮,是异构酶的竞争性抑制剂,对Δ5-3-酮甾体异构酶的 Ki 为 7 μM。
T6179 Moxalactam sodium salt

Latamoxef sodium,6059 S,拉氧头孢钠,Moxalactam Disodium,LY-127935,Antibiotic 6059S,Shiomarin,FestamoxinLy

Antibacterial; Antibiotic Microbiology/Virology
Moxalactam sodium salt (LY-127935) 是一种抗生素, 对大肠杆菌和绿脓杆菌有作用。
T40421 4,5-Dichlorocatechol

Others Others
4,5-Dichlorocatechol 是广谱的pseudomonas chlororaphisRW71 氯邻苯二酚 1,2-二加氧酶的底物。对于Pseudomonas putidaAC27 菌株双加氧酶和AcidovoraxPS14 菌株双加氧酶的Ki 都为 30 nM。
T20711 Hemipyocyanine

1-羟基吩嗪,528-71-2

Amylase Metabolism
Hemipyocyanine (528-71-2) 是一种 α-淀粉酶抑制剂。
T38137 3,5-Dimethylbenzaldehyde

Endogenous Metabolite; Antifungal Metabolism; Microbiology/Virology
3,5-Dimethylbenzaldehyde 具有广谱的抗菌活性,对枯草芽孢杆菌、白假丝酵母菌、大肠杆菌、铜绿假单胞菌、金黄色葡萄杆菌和肺炎链球菌具有抑制作用。
T18910 Acid Yellow 9 monosodium salt

Hydrogen 4-aminoazobenzene-3,4'-disulphonate (sodium salt)

Others Others
Acid Yellow 9 monosodium salt (Hydrogen 4-aminoazobenzene-3,4'-disulphonate (sodium salt)) 是一种可被Pseudomonas fluorescens 降解的含氮染料,是此类菌株碳、氮和能量的唯一来源。
T65309 S-Methyl methanesulfonothioate

Antibacterial Microbiology/Virology
S-Methyl methanesulfonothioate 是一种生物原料,具有细胞毒性和潜在的抗菌活性,可用于研究铜绿假单胞菌感染。
T38173 Propargylcholine

Propargylcholine (bromide)

Antibacterial Microbiology/Virology
Propargylcholine (Propargylcholine (bromide)) 是一种炔烃修饰的胆碱类似物,在铜绿假单胞菌中 Dgc 酶催化的二甲基甘氨酸去甲基化水平上抑制胆碱分解代谢。
T77686 1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone

Antifungal Microbiology/Virology
1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone 具有广谱的抗真菌活性,对白色念珠菌、黑曲霉、铜绿假单胞菌、金黄色葡萄球菌等具有抑制作用。
T67912 PA3552-IN-1

PA3552-IN-1 是一种抗生素佐剂, 可以降低 PA3552 的表达,恢复 MDR 铜绿假单胞菌 DK2 菌株对 Polymyxin B 的敏感性。
T1218 Cefoperazone sodium salt

CP 52640-2,头孢哌酮钠,Cefoperazone sodium

Antibacterial; Antibiotic Microbiology/Virology
Cefoperazone sodium salt (CP 52640-2) 是一种半合成的头孢菌素,具有广谱抗菌活性。
T7495 Hexa-D-arginine

Others Others
Hexa-D-arginine 是稳定的furin 抑制剂,能够作用于 furin (Ki:106 nM)、PACE4 (Ki:580 nM)、PC1 (Ki:13.2 nM)。它在体外和体内均可阻断假单胞菌外毒素 A 和炭疽毒素的毒性。
T9119 SU0268

Others Others
SU0268 是有效的 8-8-氧鸟嘌呤 DNA 糖基化酶1的选择性抑制剂,具有调控铜绿假单胞杆菌感染免疫反应的能力。
T8620 piperacillin

Pipril,Pipracil,哌拉西林,Pipercillin

Antibacterial Microbiology/Virology
Piperacillin (Pipercillin) 是半合成青霉素,可以作用于革兰氏阳性和革兰氏阴性需氧和厌氧菌。与其他青霉素相比,它对产生 β-内酰胺酶的菌类表现出更强的活性。
T37681 3-hydroxy Stearic Acid

3-hydroxystearic acid,3-hydroxyoctadecanoic acid

3-hydroxy Stearic Acid (3-hydroxystearic acid) 是从假单胞菌和菌丝桃属植物中发现的一种脂肪酸。
T77574 ROS inducer 1

ROS; Antibiotic Immunology/Inflammation; Microbiology/Virology
ROS inducer 1 是一种具有杀菌作用的小分子化合物,对 Xanthomonas axonopodis pv. citri (Xac)、Xanthomonas oryzae pv. oryzae (Xoo)和 Pseudomonas syringae pv. actinidiae (Psa) 具有抑制作用。ROS inducer 1 诱 Xanthomonas 细胞内 ROS 的产生可用于研究农作物细菌感染。
TP1050L Murepavadin acetate(944252-63-5 free base)

Antibacterial; Antibiotic Microbiology/Virology
Murepavadin acetate(944252-63-5 free base) 是一种有效且特异性的抗生素,用于治疗由铜绿假单胞菌引起的细菌感染。 Murepavadin acetate 靶向脂多糖转运蛋白 D。
T78226 Methyl 2-amino-5-bromobenzoate

Methyl 5-Bromoanthranilate

HCV Protease; Antifungal Microbiology/Virology; Proteases/Proteasome
Methyl 2-amino-5-bromobenzoate (Methyl 5-Bromoanthranilate) 是一种丙型肝炎病毒 NS5b RNA 聚合酶抑制剂,具有抗菌活性,可抑制铜绿假单胞菌感染,参与许多毒力因子的产生和生物膜的形成。
T4998L Cefpodoxime (free acid)

Others Others
Cefpodoxime (free acid) 是一种口服的第三代头孢菌素抗生素。除铜绿假单胞菌、肠球菌和脆弱拟杆菌外,它对大多数革兰氏阳性和革兰氏阴性微生物均有效。
T23858 WCK-5153

WCK 5153,WCK5153

Antibacterial Microbiology/Virology
WCK-5153 是 β-Lactamase 的增强剂和 PBP2 的抑制剂,对铜绿假单胞菌具有抗菌活性。 WCK-5153 可用于治疗由高度耐药的革兰氏阴性病原体引起的严重感染的研究。
T7858 Ceftezole sodium

Celoslin,Falomesin,头孢替唑钠,Alomen

Anti-infection; Antibacterial; Antibiotic; Glucosidase Metabolism; Microbiology/Virology
Ceftezole sodium (Falomesin) 是一种广谱 cephem 抗生素,具有抑制多种革兰氏阳性菌和革兰氏阴性菌活性。它是一种α-葡萄糖苷酶抑制剂,具有体内抗糖尿病活性。
T125115 Cyclo(L-Leu-L-Pro)

Antifungal Microbiology/Virology
Cyclo(L-Leu-L-Pro) 是一种来自芝麻假单胞菌BC42的化合物,具有抗真菌活性,抑制真菌病原体,抑制黄曲霉增殖。Cyclo(L-Leu-L-Pro) 抑制分生孢子的萌发和分生孢子的形成,可用于农业生物防治。
T124492 Imipenem

N-Formimidoyl thienamycin,MK0787

Antifungal Microbiology/Virology
Imipenem (MK0787) 是一种噻吩霉素衍生物,属于抗生素类,具有抗菌活性,对革兰氏阳性和革兰氏阴性菌具有部分的抑制作用。Imipenem 可用于研究碳青霉烯类非易感性感染和铜绿假单胞菌生物膜感染。
T60247 Diethylamine NONOate diethylammonium salt

NOC-18 Diethylamine,DEA NONOate diethylamine

Antibiotic Microbiology/Virology
Diethylamine NONOate diethylammonium salt (DEA NONOate diethylamine) 是一种一氧化氮供体,具有抗菌活性,是铜绿假单胞菌生物膜预形成生物膜的分散剂,可抑制大肠杆菌的生长。Diethylamine NONOate diethylammonium salt 可用于离体大鼠心脏的保存。
T77608 1H-Indole, 3,3'-(2-thienylmethylene)bis[2-methyl-

Antifungal Microbiology/Virology
1H-Indole, 3,3'-(2-thienylmethylene)bis[2-methyl- 可作为一种广谱抗菌剂,对黑曲霉枯草芽孢杆菌、白假丝酵母、大肠杆菌和金黄色葡萄球菌有抑制作用。1H-Indole, 3,3'-(2-thienylmethylene)bis[2-methyl- 在体外实验中显示出抗炎活性,可用于治疗细菌感染。
T13789 N-dodecanoyl-L-Homoserine lactone

C12-HSL,十二烷酰-L-高丝氨酸内酯

Others Others
N-dodecanoyl-L-Homoserine lactone (C12-HSL) 是群体感应 (QS) 信号分子的一种。它适配体可用于阻止群体感应,并能够阻碍铜绿假单胞菌 (Pseudomonas aeruginosa) 生物膜的形成。
T35449 α-(difluoromethyl)-DL-Arginine

DFMA,RMI 71897,α-(difluoromethyl)-DL-Arginine

Others Others
α-(difluoromethyl)-DL-Arginine (RMI 71897) 是一种酶激活的、不可逆的大肠杆菌(Ki = 800 μM)、铜绿假单胞菌和肺炎克雷伯菌精氨酸脱羧酶抑制剂。在0.01 mM 时,它已被证明可以防止渗透胁迫诱导的燕麦叶片细胞精氨酸脱羧酶活性和腐胺合成的增加。当α-(difluoromethyl)-DL-Arginine 与多种多胺类似物联用时,能在10 mM 的最低浓度下抑制克氏锥虫在哺乳动物宿主细胞中的生长,并在T 细胞受体α缺陷小鼠模型中阻止小锥虫的生长。
T37739 N-decanoyl-L-Homoserine lactone

C10-HSL,N-decanoyl-L-Homoserine lactone

Reactive Oxygen Species; Antibacterial Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
N-decanoyl-L-Homoserine lactone (C10-HSL) 是一种由克雷莫里色假单胞菌菌株 ND07产生的 N-acyl-homoserine lactone (AHL)。N-decanoyl-L-homoserine lactone 可抑制拟南芥的主根生长。N-decanoyl-L-homoserine lactone 处理可引起拟南芥根胞质游离 Ca2+ 和活性氧 (ROS) 浓度短暂和和立即升高,增加丝裂原激活蛋白激酶 6 (MPK6) 的活性,并促使一氧化氮 (NO) 的产生。
T33857 PA Autoinducer

3O-C12 autoinducer,PA-Autoinducer

PA Autoinducer is a Pseudomonas aeruginosa autoinducer.
T14923 Cefpiramide sodium

头孢匹胺钠,SM-1652,Wy-44635

Others Others
Cefpiramide sodium (SM-1652; Wy-44635) is a Pseudomonas-active cephalosporin. It has a broad spectrum of antibacterial activity.
T34761 Syringomycin A1

Syringomycin A1 is a small cyclic lipodepsinonapeptides produced by the plant bacterium Pseudomonas syringae pv. syringae.
T39983 SPR206 acetate

SPR206 acetate is a polymyxin analog that exhibits antibiotic activity against Gram-negative pathogens, including multidrug-resistant (MDR) variants. By interacting with the outer membrane of the bacterium, SPR206 acetate effectively combats bacterial infections. Notably, SPR206 acetate demonstrates significant efficacy with minimum inhibitory concentration (MIC) values of 0.125 mg/L against Pseudomonas aeruginosa Pa14 and Acinetobacter baumannii NCTC13301.
T26205 Sperabillin C

Sperabillin C is a potent antibacterial antibiotic in vivo isolated from Pseudomonas fluorescens YK-437.
T36599 4-Epianhydrotetracycline hydrochloride

Epianhydrotetracycline (EATC) is a degradation product of the antibiotic tetracycline .1 EATC is active against Pseudomonas, Agrobacterium, Moraxella, Bacillus, and E. coli (MIC50s = 0.75-16 mg/L).
T25514 Hypeptin

Hypeptin is an antibiotic agent from Pseudomonas sp.
T26203 Sperabillin A (free base)

Sperabillin A

Sperabillin A (free base) is a potent antibacterial antibiotic in vivo isolated from Pseudomonas fluorescens YK-437.
T33960 Phaseolotoxin

Phaseolotoxin A

Phaseolotoxin is an exotoxin from Pseudomonas sp.; cleavage of C terminal alanine and homoarginine from phaseolotoxin leaves octicidine.
T34174 Pseudobactin

Ferric pseudobactin

Pseudobactin is a linear hexapeptide fluorescent iron transport agent (siderophore) from plant growth promoter Pseudomonas B10.
T30826 Cgp 31523A

Cgp-31523A,Cgp31523A

CGP 31523a is a new type of aminothiazolyl cephalosporin, which can inhibit Escherichia coli, Klebsiella pneumoniae, Pseudomonas mirabilis, Clostridium diving, Klebsiella acidogenes, Pseudomonas Stuart, Salmonella, and Shigella.
T64422 Murepavadin

Murepavadin is a highly potent, specific, macrocycle Pseudomonas antibiotic for the treatment of bacterial infections caused by Pseudomonas aeruginosa..
T40497 3,4-Dichlorocatechol

3,4-Dichlorocatechol serves as a substrate for the broad-spectrum chlorocatechol 1,2-dioxygenase enzyme found in pseudomonas chlororaphis RW71.
T13788 N-Butanoyl-DL-homoserine lactone

(Rac)-C4-HSL

Others Others
N-Butanoyl-DL-homoserine lactone aptamers blocks qurom sensing and inhibits biofilm formation in Pseudomonas aeruginosa.
T26204 Sperabillin A (HCl)

Sperabillin A (HCl) is a potent antibacterial antibiotic in vivo isolated from Pseudomonas fluorescens YK-437.
T25997 Pseudomonic acid C

Mupirocin calcium impurity B

Pseudomonic acid C is the analogue of Pseudomonic Acid D which is an antibiotic agent from Pseudomonas fluorescens.
T34486 Safracin A

Y-16760

Safracin A 是一种由荧光假单胞菌 A2-2 产生的抗生素。
T34175 Pseudobactin A

Pseudobactin A is a nonfluorescent extracellular siderophore produced by plant growth-promoting bacterium Pseudomonas B10.

化合物

Benzyldodecyldimethylammonium Chloride Dihydrate
Cat.No: T22269
Synonym:
Target: Antibacterial
Pipemidic acid
Cat.No: T0396
Synonym: 吡哌酸,Acido pipemidico
Target: Antibacterial, Antibiotic
Avibactam sodium
Cat.No: T4201
Synonym: 阿维巴坦,AVE-1330A,阿维巴坦钠,NXL-104
Target: Antibacterial, Antibiotic
Gatifloxacin
Cat.No: T1293
Synonym: BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Nandrolone acetate
Cat.No: T38862
Synonym: 19-Nortestosterone 17β-acetate
Target: Others
Moxalactam sodium salt
Cat.No: T6179
Synonym: Latamoxef sodium,6059 S,拉氧头孢钠,Moxalactam Disodium,LY-127935,Antibiotic 6059S,Shiomarin,FestamoxinLy
Target: Antibacterial, Antibiotic
4,5-Dichlorocatechol
Cat.No: T40421
Synonym:
Target: Others
Hemipyocyanine
Cat.No: T20711
Synonym: 1-羟基吩嗪,528-71-2
Target: Amylase
3,5-Dimethylbenzaldehyde
Cat.No: T38137
Synonym:
Target: Endogenous Metabolite, Antifungal
Acid Yellow 9 monosodium salt
Cat.No: T18910
Synonym: Hydrogen 4-aminoazobenzene-3,4'-disulphonate (sodium salt)
Target: Others
S-Methyl methanesulfonothioate
Cat.No: T65309
Synonym:
Target: Antibacterial
Propargylcholine
Cat.No: T38173
Synonym: Propargylcholine (bromide)
Target: Antibacterial
1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone
Cat.No: T77686
Synonym:
Target: Antifungal
PA3552-IN-1
Cat.No: T67912
Synonym:
Target:
Cefoperazone sodium salt
Cat.No: T1218
Synonym: CP 52640-2,头孢哌酮钠,Cefoperazone sodium
Target: Antibacterial, Antibiotic
Hexa-D-arginine
Cat.No: T7495
Synonym:
Target: Others
SU0268
Cat.No: T9119
Synonym:
Target: Others
piperacillin
Cat.No: T8620
Synonym: Pipril,Pipracil,哌拉西林,Pipercillin
Target: Antibacterial
3-hydroxy Stearic Acid
Cat.No: T37681
Synonym: 3-hydroxystearic acid,3-hydroxyoctadecanoic acid
Target:
ROS inducer 1
Cat.No: T77574
Synonym:
Target: ROS, Antibiotic
Murepavadin acetate(944252-63-5 free base)
Cat.No: TP1050L
Synonym:
Target: Antibacterial, Antibiotic
Methyl 2-amino-5-bromobenzoate
Cat.No: T78226
Synonym: Methyl 5-Bromoanthranilate
Target: HCV Protease, Antifungal
Cefpodoxime (free acid)
Cat.No: T4998L
Synonym:
Target: Others
WCK-5153
Cat.No: T23858
Synonym: WCK 5153,WCK5153
Target: Antibacterial
Ceftezole sodium
Cat.No: T7858
Synonym: Celoslin,Falomesin,头孢替唑钠,Alomen
Target: Anti-infection, Antibacterial, Antibiotic, Glucosidase
Cyclo(L-Leu-L-Pro)
Cat.No: T125115
Synonym:
Target: Antifungal
Imipenem
Cat.No: T124492
Synonym: N-Formimidoyl thienamycin,MK0787
Target: Antifungal
Diethylamine NONOate diethylammonium salt
Cat.No: T60247
Synonym: NOC-18 Diethylamine,DEA NONOate diethylamine
Target: Antibiotic
1H-Indole, 3,3'-(2-thienylmethylene)bis[2-methyl-
Cat.No: T77608
Synonym:
Target: Antifungal
N-dodecanoyl-L-Homoserine lactone
Cat.No: T13789
Synonym: C12-HSL,十二烷酰-L-高丝氨酸内酯
Target: Others
α-(difluoromethyl)-DL-Arginine
Cat.No: T35449
Synonym: DFMA,RMI 71897,α-(difluoromethyl)-DL-Arginine
Target: Others
N-decanoyl-L-Homoserine lactone
Cat.No: T37739
Synonym: C10-HSL,N-decanoyl-L-Homoserine lactone
Target: Reactive Oxygen Species, Antibacterial
PA Autoinducer
Cat.No: T33857
Synonym: 3O-C12 autoinducer,PA-Autoinducer
Target:
Cefpiramide sodium
Cat.No: T14923
Synonym: 头孢匹胺钠,SM-1652,Wy-44635
Target: Others
Syringomycin A1
Cat.No: T34761
Synonym:
Target:
SPR206 acetate
Cat.No: T39983
Synonym:
Target:
Sperabillin C
Cat.No: T26205
Synonym:
Target:
4-Epianhydrotetracycline hydrochloride
Cat.No: T36599
Synonym:
Target:
Hypeptin
Cat.No: T25514
Synonym:
Target:
Sperabillin A (free base)
Cat.No: T26203
Synonym: Sperabillin A
Target:
Phaseolotoxin
Cat.No: T33960
Synonym: Phaseolotoxin A
Target:
Pseudobactin
Cat.No: T34174
Synonym: Ferric pseudobactin
Target:
Cgp 31523A
Cat.No: T30826
Synonym: Cgp-31523A,Cgp31523A
Target:
Murepavadin
Cat.No: T64422
Synonym:
Target:
3,4-Dichlorocatechol
Cat.No: T40497
Synonym:
Target:
N-Butanoyl-DL-homoserine lactone
Cat.No: T13788
Synonym: (Rac)-C4-HSL
Target: Others
Sperabillin A (HCl)
Cat.No: T26204
Synonym:
Target:
Pseudomonic acid C
Cat.No: T25997
Synonym: Mupirocin calcium impurity B
Target:
Safracin A
Cat.No: T34486
Synonym: Y-16760
Target:
Pseudobactin A
Cat.No: T34175
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T38373 2-heptyl-3-hydroxy-4(1H)-Quinolone

2-heptyl-3-hydroxy-4(1H)-Quinolone,PQS,Pseudomonas Quinolone Signal

Others Others
2-heptyl-3-hydroxy-4(1H)-Quinolone (Pseudomonas Quinolone Signal) 是一种铜绿假单胞菌为应对细胞密度增加而产生的一种法定人数感应信号分子。 它增加了铜绿假单胞菌中lasB 基因的表达,增加代谢物焦蓝蛋白和凝集素PA-IL 的分泌,以及增加铜绿假单胞菌种群的生物膜生产。当使用浓度为40 μM 时,它还会降低铜绿假单胞菌生长介质中的铁含量,并在硫酸铁溶液中充当一种铁螯合剂。
T5780 HYPOCRELLIN B

Apoptosis; Parasite; Antifungal Apoptosis; Microbiology/Virology
Hypocrellin B 是从真菌Hypocrella bambusae 和Shiraia bambusicola 中分离得到的一种感光颜料,可用于癌症光动力研究。它是一个凋亡诱导剂,还拥有抗菌和抗利什曼活性。
T2904 Sclareolide

香紫苏内酯,Norambreinolide

Others; Antibacterial Microbiology/Virology; Others
Sclareolide (Norambreinolide) 是一种从Salvia sclarea 的花中分离得到的天然产物,具有抗菌和细胞毒性作用。
TQ0251 (Z)-2-decenoic acid

(Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid

Others Others
(Z)-2-decenoic acid (cis-dec-2-enoic acid) 是一种由铜绿假单胞菌产生的不饱和脂肪酸。它能够诱导一系列革兰氏阴性细菌(包括铜绿假单胞菌)和革兰氏阳性细菌形成的生物膜发生分散反应。它能够抑制生物膜发育。
T8384 Gatifloxacin hydrochloride

AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。
T3603 Sodium lauryl sulfoacetate

月桂醇磺基乙酸酯钠,鱼腥草,新鱼腥草素钠,Sodium houttuyfonate

NF-κB; MAPK MAPK; NF-κB
Sodium lauryl sulfoacetate (Sodium houttuyfonate) 是一种植物来源的固体阴离子表面活性剂,也是一种具有抗免疫抑制作用的免疫佐剂。
T7283 sodium lauroyl-α-hydroxyethyl sulfonate

鱼腥草

NF-κB; MAPK MAPK; NF-κB
sodium lauroyl-α-hydroxyethyl sulfonate 是抗假单胞菌药物,抑制假单胞菌的毒力相关运动。
T8148 Mupirocin calcium hydrate

莫匹罗星钙,Mupirocin calcium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Mupirocin calcium hydrate 是从Pseudomonas fluorescens 中分离得到的,一种有口服活性的抗生素。它可逆地抑制异亮氨酸转移RNA,并抑制细菌蛋白和RNA 的合成起到抗菌作用。
T5707 3-O-Methylgalangin

3-Methylgalangin,GALANGIN-3-METHYLETHER,高良姜素 3-O-甲醚,高良姜素-3-甲醚

Antibacterial Microbiology/Virology
3-O-Methylgalangin (GALANGIN-3-METHYLETHER) 是一种来源于高良姜根茎的天然黄酮,具有抗菌活性,抑制胰腺脂肪酶。
TN2111 Prunin

Naringenin 7-0-glucoside,柚皮素-7-O-葡萄糖苷

Phosphatase; Anti-infection; Virus Protease Metabolism; Microbiology/Virology
Prunin (Naringenin 7-0-glucoside) 是一种人肠道病毒 A71 抑制剂。它抑制蛋白酪氨酸磷酸酶 1B,IC50值为 5.5 μM。
T3742 3-Methylcatechol

3-甲基苯邻二酚,3-Methylpyrocatechol,2,3-Toluenediol,3-甲基邻苯二酚,2,3-dihydroxytoluene

Others Others
3-Methylcatechol (2,3-Toluenediol) 是由 Pseudomonas putidaMC2 产生,能够用作化学合成中的分子砌块。
T4816 6-Hydroxynicotinic acid

6-Hydroxypyridine-3-carboxylic acid,6-羟基烟酸,2-Hydroxy-5-pyridinecarboxylic acid

Others; Endogenous Metabolite Metabolism; Others
6-Hydroxynicotinic acid (6-Hydroxypyridine-3-carboxylic acid) 用于核磁共振波谱或气相色谱-质谱法诊断尿路感染中的铜绿假单胞菌。在引起尿液感染的常见细菌中,只有铜绿假单胞菌从烟酸中产生6-羟基烟酸。
T8066 Sulbenicillin disodium

磺苄西林钠,Sulbenicillin Sodium

Antibacterial; Antibiotic Microbiology/Virology
Sulbenicillin disodium (Sulbenicillin Sodium) 是 Sulbenicillin 的二钠盐。Sulbenicillin 是一种青霉素抗生素,对Pseudomonas aeruginosa 的许多粘液型和非粘液型菌株具有抗菌活性。
T37341 N-Acetyltyramine

Antibacterial Microbiology/Virology
N-Acetyltyramine 是一种群体感应抑制剂,由溶藻弧菌 M3-10 产生。N-Acetyltyramine 可以抑制C. violaceumATCC 12472 的群体感应。它可以逆转阿霉素耐药白血病 P388 细胞的耐药性。
T1465 Mupirocin

Pseudomonic acid,莫匹罗星,BRL-4910A

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Mupirocin (BRL-4910A) 是从Pseudomonas fluorescens 中分离得到的一种有口服活性的抗生素。它可逆地抑制异亮氨酸转移RNA,并抑制细菌蛋白和RNA 的合成起抗菌作用。
TN3861 Dihydropinosylvin

山药

Anti-infection Microbiology/Virology
Dihydropinosylvin 是一种植物抗毒素,对枝孢枝孢菌、Botryodiplodia theobromae、黑曲霉和石化青霉具有抗真菌活性,对蜡状芽孢杆菌、金黄色葡萄球菌、铜绿假单胞菌和大肠杆菌也有很强的抗菌活性。双色高粱幼苗的种子和根伸长。
T4716 Pyrrole-2-carboxylic acid

吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline

Endogenous Metabolite Metabolism
Pyrrole-2-carboxylic acid (Minaline) 是一种天然生物碱类,从海洋细菌Pelomonas puraquaesp. Nov 中分离得到。
TN2760 2-Hydroxy-1,8-cineole

Antifection Microbiology/Virology
1. 2-endo-Hydroxy-1,8-cineole shows antimicrobial and bactericidal activities against against test bacteria (Staphylococcus aureus, Escherichia coli, and Pseudomonas fluorescens) .<BR/>
T1255L Tobramycin Sulfate

Dartobcin,Nebcine,Tobraneg,Tobrasix

Tobramycin Sulfate is a broad-spectrum antibiotic. It is effective against gram-negative bacteria. It especially potent against the Pseudomonas species.
TN4851 Pterodondiol

Antifection Microbiology/Virology
Pterodondiol has moderate activity against bacteria including Staphylococcus aureus, Pseudomonas aeruginosa, Bacillus subtilis, Mycobacteium phlei and Bacillus circulans.
TN6688 Cyclo(Ala-Tyr)

Cyclo(Val-Tyr) is a product from the culture of Pseudomonas putida.
TN1203 2,3,8-Tri-O-methylellagic acid

2,3,8-三邻甲基鞣花酸

Antifection Microbiology/Virology
2,3,8-tri-O-Methyl ellagic acid has antimicrobial activity agaist Vibro cholera, Staphylococcus aureus, Klebsiella pneumoniae, Pseudomonas aeruginosa, Bacillus cereus, Escherichia coli.
TN5229 Vibralactone B

Antifection Microbiology/Virology
Vibralactone B shows antibacterial activity, it can inhibit significantly the growth of E. coli and Pseudomonas aeruginosa, with MBC values of 50 and 100 ug/mL, respectively.
TN2420 Protoanemonin

Antibacterial Microbiology/Virology
Protoanemonin is a naturally occurring compound which may be isolated from plants of the family Ranunculaceae. Protoanemonin can also be produced by Pseudomonas sp.
TN4579 Monomethylsulochrin

Antifection Microbiology/Virology
Monomethylsulochrin shows antimicrobial activity against Escherichia coli, Pseudomonas aeruginosa, Bacillus subtilis and Staphylococcus aureus. It shows moderately inhibitory effects on the human bacterial pathogen Helicobacter pylori with the MIC value of 28.9+/-0.1 microM.
T72250 4aα,7α,7aα-Nepetalactone

4aα,7α,7aα-Nepetalactone 具有抗菌 (antibacterial) 活性,抑制Escherichia coli,Pseudomonas aeruginosa,Staphylococcus aureus,Salmonella typhi 和Enterococcus faecalis。
TN4852 Pterodontic acid

Antifection Microbiology/Virology
Pterodontic acid and pterodondiol showed moderate activity against bacteria including Staphylococcus aureus, Pseudomonas aeruginosa, Bacillus subtilis.
T75442 Galloyl-bis-HHDP glucose

Galloyl-bis-HHDP glucose (HeT) 是一种鞣花单宁,对绿色假单胞菌具有植物保护作用。
TN2392 9,17-Octadecadiene-12,14-diyne-1,11,16-triol

Antifection Microbiology/Virology
9,17-Octadecadiene-12,14-diyne-1,11,16-triol shows antibacterial activity against Bacillus subtilis and Pseudomonas fluorescens, antifungal activity against Cladosporium cucumerinum, moiluscicidal activity against Biomphalaria glabrata at low concentratio
TN2032 Pachypodol

霍香黃酮醇

Antifection Microbiology/Virology
Pachypodol has antibacterial and antifungal activities against Bacillus subtilis, Staphylococcus aureus, Staphylococcus faecalis, Echerichia coli, Pseudomonas aeruginosa, Candida albicans, Candida krusei and Candida galabrata.
T75467 Asperglaucin A

Asperglaucin A 代表一种不寻常的类苯酞衍生物。Asperglaucin A 对两种植物病原体Pseudomonas syringae pv actinidae(Psa) 和Bacillus cereus 具有有效的抗菌活性,MIC 值为 6.25 μM。
TN3400 Altechromone A

Antifection Microbiology/Virology
Altechromone A has antimicrobial activity, it is active against Bacillus subtilis, Escherichia coli, Pseudomonas fluorescens and Candida albicans with the MICs of 3.9, 3.9, 1.8, and 3.9 ug/ml, respectively.
TN4838 Pseurotin A

Antifection Microbiology/Virology
Pseurotin A has immunosuppressive activity, it inhibits immunoglobulin E(IgE) production in vitro.It shows a moderate effect against the phytopathogenic bacteria Erwinia carotovora and Pseudomonas syringae, with IC50 values of 220 and 112 microg ml(-1), r
T75600 Coronatine

Coronatine 是丁香假单胞菌产生的一种植物生长调节剂。Coronatine 模拟生物活性茉莉酸 (jasmonic acid) 缀合物或高等植物的 octadecanoid 信号分子使植物出现致病症状。Coronatine 通过激活抑制水杨酸 (Salicylic acid) 积累的信号级联,促进植物中丁香假单胞菌的毒力。
T75468 Asperglaucin B

Asperglaucin B 是一种来自真菌Aspergillus chevalieriSQ-8 的烷基化水杨醛衍生物,具有抗菌活性。Asperglaucin B 对两种植物病原体Pseudomonas syringae pv actinidae(Psa)和Bacillus cereus 显示出有效的抗菌活性,MIC 值为 6.25 μM。
TN2495 1,4,7-Eudesmanetriol

Antifection Microbiology/Virology
1α,4β,7β-Eudesmanetriol and 1β,4β,7β-Eudesmanetriol can inhibit growth of Pseudomonas stutzeri with a MIC value of 117 uM, they also show remarkable activities against acetylcholinesterase enzyme with IC50 values ranging between 25 and 26 uM.
T83862 Bactobolin A hydrochloride

BN-183B

Bactobolin A 是一种最初从 Pseudomonas 中分离出的微生物代谢产物,具有抗生素和抗癌活性。它对 S. aureus、S. epidermidis、S. faecalis、B. anthracis、B. subtilis、E. coli、S. typhi 和 S. dysenteriae 活跃(MICs = 0.1-12.5 µg/ml)。在体内,bactobolin A (0.25-4 mg/kg) 提高了 L1210 小鼠白血病模型的存活率。

天然产物

2-heptyl-3-hydroxy-4(1H)-Quinolone
Cat.No: T38373
Synonym: 2-heptyl-3-hydroxy-4(1H)-Quinolone,PQS,Pseudomonas Quinolone Signal
Target: Others
HYPOCRELLIN B
Cat.No: T5780
Synonym:
Target: Apoptosis, Parasite, Antifungal
Sclareolide
Cat.No: T2904
Synonym: 香紫苏内酯,Norambreinolide
Target: Others, Antibacterial
(Z)-2-decenoic acid
Cat.No: TQ0251
Synonym: (Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid
Target: Others
Gatifloxacin hydrochloride
Cat.No: T8384
Synonym: AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐
Target: Topoisomerase, Antibacterial, Antibiotic
Sodium lauryl sulfoacetate
Cat.No: T3603
Synonym: 月桂醇磺基乙酸酯钠,鱼腥草,新鱼腥草素钠,Sodium houttuyfonate
Target: NF-κB, MAPK
sodium lauroyl-α-hydroxyethyl sulfonate
Cat.No: T7283
Synonym: 鱼腥草
Target: NF-κB, MAPK
Mupirocin calcium hydrate
Cat.No: T8148
Synonym: 莫匹罗星钙,Mupirocin calcium
Target: Others, Antibacterial, Antibiotic
3-O-Methylgalangin
Cat.No: T5707
Synonym: 3-Methylgalangin,GALANGIN-3-METHYLETHER,高良姜素 3-O-甲醚,高良姜素-3-甲醚
Target: Antibacterial
Prunin
Cat.No: TN2111
Synonym: Naringenin 7-0-glucoside,柚皮素-7-O-葡萄糖苷
Target: Phosphatase, Anti-infection, Virus Protease
3-Methylcatechol
Cat.No: T3742
Synonym: 3-甲基苯邻二酚,3-Methylpyrocatechol,2,3-Toluenediol,3-甲基邻苯二酚,2,3-dihydroxytoluene
Target: Others
6-Hydroxynicotinic acid
Cat.No: T4816
Synonym: 6-Hydroxypyridine-3-carboxylic acid,6-羟基烟酸,2-Hydroxy-5-pyridinecarboxylic acid
Target: Others, Endogenous Metabolite
Sulbenicillin disodium
Cat.No: T8066
Synonym: 磺苄西林钠,Sulbenicillin Sodium
Target: Antibacterial, Antibiotic
N-Acetyltyramine
Cat.No: T37341
Synonym:
Target: Antibacterial
Mupirocin
Cat.No: T1465
Synonym: Pseudomonic acid,莫匹罗星,BRL-4910A
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Dihydropinosylvin
Cat.No: TN3861
Synonym: 山药
Target: Anti-infection
Pyrrole-2-carboxylic acid
Cat.No: T4716
Synonym: 吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline
Target: Endogenous Metabolite
2-Hydroxy-1,8-cineole
Cat.No: TN2760
Synonym:
Target: Antifection
Tobramycin Sulfate
Cat.No: T1255L
Synonym: Dartobcin,Nebcine,Tobraneg,Tobrasix
Target:
Pterodondiol
Cat.No: TN4851
Synonym:
Target: Antifection
Cyclo(Ala-Tyr)
Cat.No: TN6688
Synonym:
Target:
2,3,8-Tri-O-methylellagic acid
Cat.No: TN1203
Synonym: 2,3,8-三邻甲基鞣花酸
Target: Antifection
Vibralactone B
Cat.No: TN5229
Synonym:
Target: Antifection
Protoanemonin
Cat.No: TN2420
Synonym:
Target: Antibacterial
Monomethylsulochrin
Cat.No: TN4579
Synonym:
Target: Antifection
4aα,7α,7aα-Nepetalactone
Cat.No: T72250
Synonym:
Target:
Pterodontic acid
Cat.No: TN4852
Synonym:
Target: Antifection
Galloyl-bis-HHDP glucose
Cat.No: T75442
Synonym:
Target:
9,17-Octadecadiene-12,14-diyne-1,11,16-triol
Cat.No: TN2392
Synonym:
Target: Antifection
Pachypodol
Cat.No: TN2032
Synonym: 霍香黃酮醇
Target: Antifection
Asperglaucin A
Cat.No: T75467
Synonym:
Target:
Altechromone A
Cat.No: TN3400
Synonym:
Target: Antifection
Pseurotin A
Cat.No: TN4838
Synonym:
Target: Antifection
Coronatine
Cat.No: T75600
Synonym:
Target:
Asperglaucin B
Cat.No: T75468
Synonym:
Target:
1,4,7-Eudesmanetriol
Cat.No: TN2495
Synonym:
Target: Antifection
Bactobolin A hydrochloride
Cat.No: T83862
Synonym: BN-183B
Target:
共116条,每页50条 1 2 3
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼