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Search Results for " pi4 "

Targets Recommended: PI4K PI4K

15

抑制剂 & 化合物

4

重组蛋白

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Cat. No.	Product Name	Target	Signaling Pathways
TQ0009	UCB9608	PI4K	PI3K/Akt/mTOR signaling
	UCB9608 是选择性、可口服的 PI4KIIIβ 抑制剂，IC50=11 nM，对其选择性高于 PI3KC2 α，β 和 γ。它能够增加代谢稳定性，具有良好的药代动力学特征，是一种免疫抑制剂。
T16967	T-00127_HEV1	PI4K	PI3K/Akt/mTOR signaling
	T-00127_HEV1 是有效的phosphatidylinositol 4-kinase III beta 抑制剂，IC50为 60 nM。
T12454	PI-273	Apoptosis; PI4K	Apoptosis; PI3K/Akt/mTOR signaling
	PI-273 是一种可逆的特异性磷脂酰肌醇 4-激酶抑制剂，IC50为 0.47 μM。它可抑制乳腺癌细胞的增殖，阻断细胞周期并诱导细胞凋亡。
T16125	MMV390048	Parasite; PI4K	Microbiology/Virology; PI3K/Akt/mTOR signaling
	MMV390048 是一种抗疟药，是一种新型化学疟原虫 PI4K 抑制剂。它与疟原虫 PI4K 的 ATP 结合位点结合，不与除人类 PIP4K2C 外的其他恶性疟原虫和人类激酶结合。
T16530	BF738735	Antiviral; PI4K	Immunology/Inflammation; PI3K/Akt/mTOR signaling
	BF738735 是有效的磷脂酰肌醇 4-激酶 IIIβ 抑制剂，IC50为 5.7 nM。
T12468	PI4KIIIbeta-IN-10	PI3K; PI4K	PI3K/Akt/mTOR signaling
	PI4KIIIbeta-IN-10 是PI4KIIIβ抑制剂，IC50=3.6 nM。
T12469	PI4KIIIbeta-IN-9	PI3K; PI4K	PI3K/Akt/mTOR signaling
	PI4KIIIbeta-IN-9 是一种 PI4KIIIβ抑制剂，其 IC50=7 nM。它也抑制 PI3Kδ (IC50:125 nM) 和 PI3Kγ (IC50:1046 nM)。
T2616	PIK-93 PIK 93	ATM/ATR; DNA-PK; Virus Protease; PI3K; Carbonic Anhydrase; PI4K; mTOR; HSV	DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; PI3K/Akt/mTOR signaling
	PIK-93 是一种合成的PI4KIIIβ抑制剂，IC50值为 19 nM，同时可抑制PI3Kγ和PI3Kα的活性，IC50值分别为 16 nM 和 39 nM。
T5421	KDU691	Parasite; PI4K	Microbiology/Virology; PI3K/Akt/mTOR signaling
	KDU691 是一种咪唑吡嗪类药物，对血阶段的裂殖体、配子体和肝期具有较强的抗寄生虫活性，它是 PI4K 抑制剂，选择性抑制双氢青蒿素预处理的恶性疟原虫。
T4220	BQR-695 BQR695,NVP-BQR695	PI3K; Parasite; PI4K	Microbiology/Virology; PI3K/Akt/mTOR signaling
	BQR-695 (NVP-BQR695) 是一种磷脂酰肌醇 4-激酶抑制剂，对于人类和疟原虫 PI4KIIIβ 的 IC50值分别为 80 和 3.5 nM。
T27499	GSK-A1	HCV Protease; PI4K	Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
	GSK-A1 是 III 型磷脂酰肌醇 4-激酶 PI4KA 选择性抑制剂，pIC50为 8.5-9.8，抑制 PtdIns(4,5)P2 再合成，IC50约为 3 nM。GSK-A1有效降低 PtdIns(4)P 的水平，而对 PtdIns(4,5)P2 没影响。GSK-A1在抗丙型肝炎病毒方面有研究的潜力。
T19840	GSK-F1 PI4KA inhibitor-F1	PI4K	PI3K/Akt/mTOR signaling
	GSK-F1 (PI4KA inhibitor-F1) 是一种新型强效 PI4KA 抑制剂。
T12467	PI4KIII beta inhibitor 3	PI3K	PI3K/Akt/mTOR signaling
	PI4KIII beta inhibitor 3 is a novel and high effective inhibitor of PI4KIIIβ (IC50 of 5.7 nM).
T64106	PI4KIIIbeta-IN-11
	PI4KIIIbeta-IN-11 是一种 PI4KIIIβ 抑制剂 (平均 pIC50=9.1)，能够用于研究 RNA 病毒和恶性疟原虫引起的疾病。
T61971	CHMFL-PI4K-127
	CHMFL-PI4K-127 (compound 15g) 是具有口服活性、高选择性的PfPI4K(恶性疟原虫 PI4K 激酶)抑制剂（IC50= 0.9 nM）。CHMFL-PI4K-127 对 3D7 恶性疟原虫表现出较强的抑制活性（EC50= 25.1 nM）。CHMFL-PI4K-127 具有抗疟疾作用。

化合物

Cat.No: TQ0009

Target: PI4K

Cat.No: T16967

Target: PI4K

Cat.No: T12454

Target: Apoptosis, PI4K

Cat.No: T16125

Target: Parasite, PI4K

Cat.No: T16530

Target: Antiviral, PI4K

PI4KIIIbeta-IN-10

Cat.No: T12468

Target: PI3K, PI4K

PI4KIIIbeta-IN-9

Cat.No: T12469

Target: PI3K, PI4K

Cat.No: T2616

Synonym: PIK 93

Target: ATM/ATR, DNA-PK, Virus Protease, PI3K, Carbonic Anhydrase, PI4K, mTOR, HSV

Cat.No: T5421

Target: Parasite, PI4K

Cat.No: T4220

Synonym: BQR695,NVP-BQR695

Target: PI3K, Parasite, PI4K

Cat.No: T27499

Target: HCV Protease, PI4K

Cat.No: T19840

Synonym: PI4KA inhibitor-F1

Target: PI4K

PI4KIII beta inhibitor 3

Cat.No: T12467

Target: PI3K

PI4KIIIbeta-IN-11

Cat.No: T64106

Cat.No: T61971

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPJ-00931	Serpin A4 Protein, Human, Recombinant (His) Kallistatin,Peptidase Inhibitor 4,KST,Kallikrein In...	Human	HEK293 Cells
	Serpin Peptidase Inhibitor, Clade A (α-1 Antiproteinase, Antitrypsin), Member 4 (Serpin A4) is a member of the Serpin family. Serpin A4 exists as a monomer and some homodimers. Serpin A4 is expressed by the liver and secreted in plasma. Serpin A4 is a regulator of vascular homeostasis capable of controlling a wide spectrum of biological actions in the cardiovascular and renal systems. It can inhibit intracellular reactive oxygen species formation in cultured cardiac and renal cells. In addition,...
TMPY-00623	Serpin A1d Protein, Mouse, Recombinant PI4,serine (or cysteine) peptidase inhibit...	Mouse	HEK293 Cells
	Serpin A1d Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 44.1 kDa and the accession number is XP_003945711.1.
TMPY-00621	Serpin A1d Protein, Mouse, Recombinant (His) AI118301,Serpin A1d,Spi1-4,PI...	Mouse	HEK293 Cells
	Serpin A1d Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 44.9 kDa and the accession number is XP_003945711.1.
TMPY-00619	Serpin A1d Protein, Mouse, Recombinant (hFc) Spi1-4,PI4,Serpi	Mouse	HEK293 Cells
	Serpin A1d Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 70.2 kDa and the accession number is XP_003945711.1.

重组蛋白

Serpin A4 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00931

Species: Human

Expression System: HEK293 Cells

Serpin A1d Protein, Mouse, Recombinant

Cat.No: TMPY-00623

Species: Mouse

Expression System: HEK293 Cells

Serpin A1d Protein, Mouse, Recombinant (His)

Cat.No: TMPY-00621

Species: Mouse

Expression System: HEK293 Cells

Serpin A1d Protein, Mouse, Recombinant (hFc)

Cat.No: TMPY-00619

Species: Mouse

Expression System: HEK293 Cells

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