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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T8773 MID-1

Others; IGF-1R Others; Tyrosine Kinase/Adaptors
MID-1 是 MG53-IRS-1 相互作用的抑制剂,能够破坏 MG53 与 IRS-1 的分子缔合,并消除 MG53 诱导的 IRS-1 泛素化和骨骼肌降解,升高 IRS-1 表达水平,增加胰岛素信号传导和葡萄糖摄取。
T75151 Aganirsen

Aganirsen 是一种反义寡核苷酸(25个核苷酸),抑制胰岛素受体底物1 (IRS-1)。

化合物

MID-1
Cat.No: T8773
Synonym:
Target: Others, IGF-1R
Aganirsen
Cat.No: T75151
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0760 Cholesterol

Cholesterin,Cholesteryl alcohol,胆固醇

Estrogen Receptor/ERR; MRP; Endogenous Metabolite; ROR Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Cholesterol (Cholesteryl alcohol) 属于天然产物,是哺乳动物中的主要固醇,是一种雌激素相关受体 α (ERRα) 的激动剂。Cholesterol 广泛存在于动物的细胞膜,也是合成几种重要荷尔蒙及胆酸的材料。
T4S1545 Licarin B

(-)-Licarin B,Licarine B,(-)-利卡灵B

transporter; Antibacterial; PPAR DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Licarin B (Licarine B) 是来源于肉豆蔻种子的一种天然产物,是 NO 生成抑制剂,可通过激活 IRS-1/PI3K/AKT 通路中的PPARγ和GLUT4 改善胰岛素敏感性。
TL0014 Pinusolide

ERK; p38 MAPK; Calcium Channel; Lipoxygenase; PAFR; Caspase; JNK; AMPK Apoptosis; Chromatin/Epigenetic; GPCR/G Protein; MAPK; Membrane transporter/Ion channel; Metabolism; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Pinusolide is a platelet activating factor ( PAF) antagonist, it may prove of therapeutic value in the treatment of hypotension, it has antileukemic potential, and could be used to treat neurodegenerative diseases. Pinusolide attenuates blockade of insulin signaling by enhancing IRS-1 tyrosine phosphorylation by the activating the AMPK pathway, indicates the targeting of AMPK represents a new therapeutic strategy for hyperglycemia-induced insulin resistance and type 2 diabetes.

天然产物

Cholesterol
Cat.No: T0760
Synonym: Cholesterin,Cholesteryl alcohol,胆固醇
Target: Estrogen Receptor/ERR, MRP, Endogenous Metabolite, ROR
Licarin B
Cat.No: T4S1545
Synonym: (-)-Licarin B,Licarine B,(-)-利卡灵B
Target: transporter, Antibacterial, PPAR
Pinusolide
Cat.No: TL0014
Synonym:
Target: ERK, p38 MAPK, Calcium Channel, Lipoxygenase, PAFR, Caspase, JNK, AMPK
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