228
7
Cat. No. | Product Name | Target | Signaling Pathways |
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T14069 |
A-3 hydrochloride
|
CaMK; Casein Kinase; PKA; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Neuroscience; Stem Cells; Tyrosine Kinase/Adaptors |
A-3 hydrochloride 是一种细胞可渗透的、可逆的、ATP 竞争性非选择性拮抗剂。它抑制 PKA 、酪蛋白激酶 II 和肌球蛋白轻链激酶,Ki 值分别为4.3 µM、5.1 µM 和7.4 µM。它还抑制 PKC 和酪蛋白激酶 I 的活性,Ki 分别为 47 µM 和 80 µM。 | |||
T9881 |
Benzoquinamide hydrochloride
3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride |
Others | Others |
Benzoquinamide hydrochloride (3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride) 是一种止吐剂,其增加动脉内压的作用是由于增加了外周血管阻力。 | |||
T35526 |
PI3-Kinase α Inhibitor 2 (hydrochloride)
PI3-Kinase α Inhibitor 2 (hydrochloride) |
||
PI3-Kinase α Inhibitor 2 (hydrochloride) 是一种 PI3-Kinase α 抑制剂。 | |||
T2287 |
PIK-75 hydrochloride
PIK-75 HCl,2-甲基-5-硝基苯磺酸 [(6-溴咪唑并[1,2-a]吡啶-3-基)亚甲基]甲基肼盐酸盐,PIK-75 |
Apoptosis; DNA-PK; PI3K | Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling |
PIK-75 hydrochloride (PIK-75 HCl) 是一种可逆的 DNA-PK 和 p110α-选择性抑制剂,抑制 DNA-PK,p110α和 p110γ,可诱导凋亡。 | |||
T10111 |
3-Deazaadenosine hydrochloride
|
Others; HIV Protease | Microbiology/Virology; Others; Proteases/Proteasome |
3-Deazaadenosine hydrochloride 是 S-腺苷高半胱氨酸水解酶的抑制剂,Ki 值为 3.9 µM。 它具有抗炎、抗增殖和抗 HIV 活性。 | |||
T40002 |
Pomalidomide-C3-NH2 hydrochloride
|
Others; E3 Ligase Ligand-Linker Conjugate | Others; PROTAC |
Pomalidomide-C3-NH2 hydrochloride 包含基于 Pomalidomide 的 cereblon 配体和 1 个 linker,是合成的 E3 连接酶配体-linker 偶联物,可用于 PROTAC 的合成。 | |||
T35839 |
3-Iodothyronamine (hydrochloride)
|
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3-Iodothyronamine is derived from the deiodination and decarboxylation of endogenous thyroxine. It activates the G protein-coupled receptor known as trace amine-associated receptor 1 at nanomolar concentrations whereupon it rapidly influences thyroid hormone actions including body temperature, heart rate, and cardiac output. It has also been reported to function in controlling lipid and glucose utilization, hormonal secretion, and neuronal function, and has been considered for use in chemically-... | |||
T39581 |
PI3K-IN-19 hydrochloride
PI3K-IN-19 hydrochloride |
||
PI3K-IN-19 hydrochloride (WO2017153220, step 5) acts as a phosphatidylinositol-3-kinase (PI3K) inhibitor. | |||
T39662 | CCR4 antagonist 3 hydrochloride | ||
CCR4 antagonist 3 hydrochloride is an orally active, potent and selective CCR4 antagonist. CCR4 antagonist 3, featuring a novel piperidinyl-azetidine motif, has IC 50 s of 22 nM and 50 nM in the calcium flux and CTX assay. CCR4 antagonist 3 has antitumor activity. | |||
T41071 |
NH2-PEG3 hydrochloride
NH2-PEG3 hydrochloride |
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NH2-PEG3 hydrochloride is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells. | |||
T65572 |
3-Azetidinemethanol hydrochloride
|
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3-Azetidinemethanol hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65572,CAS号为 928038-44-2。 | |||
T76073 |
BH3 hydrochloride
|
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BH3 hydrochloride是一种能够穿透血脑屏障的多肽,其机制是通过直接激活促凋亡蛋白Bax/Bak或中和抗凋亡Bcl-2家族蛋白(Bcl-2、Bcl-XL、Bcl-w、mcl1和A-1),从而诱导细胞凋亡。这一作用是通过与BH3结构域的结合实现的。 | |||
T78654 |
MraY-IN-3 hydrochloride
|
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MraY-IN-1(compound 12a)是一种针对细菌转位酶MraY的有效抑制剂,具有140 μM的IC50值。其对Escherichia coli K12、Bacillus subtilis W23和Pseudomonas fluorescens Pf-5展现出抗菌活性,相应的MIC50为7 µg/mL、12 µg/mL和46 µg/mL。MraY-IN-1适用于抗菌药物的研究领域。 | |||
T64404 |
3-Aminobutanenitrile hydrochloride
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3-Aminobutanenitrile hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64404,CAS号为 50840-31-8。 | |||
T36108 |
YW3-56 (hydrochloride) (technical grade)
YW3-56 (hydrochloride) (technical grade) |
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YW3-56 is an inhibitor of protein arginine deiminase 2 (PAD2) and PAD4 (IC50s = 0.5-1 and 1-5 μM, respectively).1It inhibits the growth of U2OS osteosarcoma cells (IC50= ~2.5 μM) in a p53-dependent mannerviainduction of SESN2 and subsequent inhibition of mTORC1. YW3-56 (10 mg/kg) reduces tumor growth in an S-180 murine sarcoma tumor model. It also inhibits tumor growth in the 1883 MDA-MB-231 breast cancer bone metastasis mouse xenograft model.2 1.Wang, Y., Li, P., Wang, S., et al.Anticancer pept... | |||
T65208 |
3-Piperazinobenzisothiazole hydrochloride
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3-Piperazinobenzisothiazole hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65208,CAS号为 87691-88-1。 | |||
T65970 |
Ethyl 3-aminopropanoate hydrochloride
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Ethyl 3-aminopropanoate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65970,CAS号为 4244-84-2。 | |||
T39894 |
Thalidomide-4-C3-NH2 hydrochloride
Thalidomide-4-C3-NH2 hydrochloride |
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Thalidomide-4-C3-NH2 hydrochloride is a Thalidomide-derived cereblon ligand utilized for the recruitment of CRBN protein. This compound can be linked to the ligand for protein using a linker to create PROTACs. | |||
T70960 |
Maprotiline-d3 hydrochloride
|
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Maprotiline-d3 is intended for use as an internal standard for the quantification of maprotiline by GC- or LC-MS. Maprotiline is a tricyclic antidepressant. It binds to the norepinephrine transporter (NET) and is selective for NET over the serotonin and dopamine transporters. Maprotiline also binds to the serotonin (5-HT) receptor subtype 5-HT2A, as well as histamine H1, muscarinic acetylcholine, α1-adrenergic, and dopamine D2 receptors. In vivo, maprotiline inhibits norepinephrine reuptake in r... | |||
T64061 | Mps1-IN-3 hydrochloride | ||
Mps1-IN-3 hydrochloride 是一种有效的、选择性的 Mps1 抑制剂 (IC50: 50 nM)。Mps1-IN-3 hydrochloride 对胶质母细胞瘤细胞的增殖表现出抑制作用,并在原位异种移植瘤模型中可有效地使胶质母细胞瘤对长春新碱敏感。 | |||
T66829 |
3-(Chloromethyl)pyridine hydrochloride
|
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3-(Chloromethyl)pyridine hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66829,CAS号为 6959-48-4。 | |||
T63850 |
FGFR2-IN-3 hydrochloride
|
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FGFR2-IN-3 hydrochloride 是一种选择性的、口服具有活力的 FGFR2 抑制剂。 | |||
T39953 |
Pomalidomide-amino-PEG3-NH2 hydrochloride
Pomalidomide-amino-PEG3-NH2 hydrochloride |
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Pomalidomide-amino-PEG3-NH2 hydrochloride is a synthetic conjugate compound incorporating the cereblon ligand from Pomalidomide and a linker commonly utilized in PROTAC technology. This compound functions as an E3 ligase ligand-linker conjugate in biochemical reactions. | |||
T66004 |
Azetidin-3-ol hydrochloride
|
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Azetidin-3-ol hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66004,CAS号为 18621-18-6。 | |||
T64231 | 3,6-DMAD hydrochloride | ||
3,6-DMAD hydrochloride 是一种未折叠蛋白质应答 (IRE1α-XBP1) 通路的抑制剂。 | |||
T62442 |
MY33-3 hydrochloride
|
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MY33-3 hydrochloride 是一种有效的、选择性的蛋白酪氨酸磷酸酶 RPTPβ/ζ 抑制剂 (IC50~0.1 μM)。MY33-3 hydrochloride 对 PTP-1B 具有抑制作用 (IC50~0.7 μM)。MY33-3 hydrochloride 能够降低乙醇消耗,缓解 Sevoflurane 引起的神经炎症和认知功能障碍。 | |||
T60831 | AChE/BChE-IN-3 hydrochloride | ||
AChE/BChE-IN-3 (BMC-1) hydrochloride 是 AChE 和 BChE 的双重抑制剂。AChE/BChE-IN-3 对马血清 BChE (eqBChE) 和电鳗 AChE (elAChE) 的 IC50值分别为 0.383 μM 和 6.08 μM。 | |||
T73711 |
Atomoxetine-d3 hydrochloride
|
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Atomoxetine-d3 hydrochloride 是氘代标记的Atomoxetine hydrochloride。Atomoxetine hydrochloride 是去甲肾上腺素重吸收抑制剂,与人NET,SERT 和DAT 的放射性配体结合的 Ki 分别为5,77和1451 nM。 | |||
T78653 | NS2B/NS3-IN-3 hydrochloride | Virus Protease | Microbiology/Virology |
NS2B/NS3-IN-3 hydrochloride为Flavivirus NS2B-NS3蛋白酶的专一性抑制剂。 | |||
T66061 |
(S)-3-Aminobutanoic acid hydrochloride
|
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(S)-3-Aminobutanoic acid hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66061,CAS号为 58610-41-6。 | |||
T67574 |
3-Chloro-L-alanine Hydrochloride
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3-Chloro-L-alanine Hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67574,CAS号为 51887-89-9。 | |||
T65152 | Ethyl azetidine-3-carboxylate hydrochloride | ||
Ethyl azetidine-3-carboxylate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65152,CAS号为 405090-31-5。 | |||
T66088 |
(S)-3-Aminohexanedioic acid hydrochloride
|
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(S)-3-Aminohexanedioic acid hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66088,CAS号为 61884-74-0。 | |||
T65646 |
Methyl azetidine-3-carboxylate hydrochloride
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Methyl azetidine-3-carboxylate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65646,CAS号为 100202-39-9。 | |||
T40105 |
Pomalidomide-PEG3-C2-NH2 hydrochloride
Pomalidomide-PEG3-C2-NH2 hydrochloride,Cereblon Ligand-Linker Conjugates 5 hydrochloride,E3ligaseLigand-LinkerConjugates30hydrochloride |
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Pomalidomide-PEG3-C2-NH2 hydrochloride, also known as Cereblon Ligand-Linker Conjugate 5, is a chemically synthesized E3 ligase ligand-linker conjugate. This compound incorporates a cereblon ligand based on Pomalidomide and a linker commonly employed in PROTAC technology. | |||
T64497 |
Methyl-D3-amine hydrochloride
|
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Methyl-D3-amine hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64497,CAS号为 7436-22-8。 | |||
T77880 | 3-Azido-D-alanine hydrochloride | ||
3-Azido-D-alanine hydrochloride是盐酸D-丙氨酸(D-alanine)的叠氮基改性形式,适用于点击化学标记。 | |||
T81142 | SNIPER(TACC3)-1 hydrochloride | SNIPERs | PROTAC |
SNIPERTACC3-1 hydrochloride 是一种基于IAPE3连接酶的化合物,其机制是针对泛素-蛋白酶体系统,靶向性地降解TACC3蛋白,从而诱导癌细胞死亡。 | |||
T81141 | SNIPER(TACC3)-2 hydrochloride | SNIPERs | PROTAC |
SNIPER(TACC3)-2 hydrochloride 是一个基于IAPE3配体的小分子化合物,其作用机制为通过泛素-蛋白酶体系统靶向降解TACC3蛋白,从而诱导癌细胞死亡。 | |||
T64915 |
Methyl 2-amino-3-phenylpropanoate hydrochloride
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Methyl 2-amino-3-phenylpropanoate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64915,CAS号为 5619-07-8。 | |||
T83114 |
Angiopep-Bim BH3 hydrochloride
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Angiopep-Bim BH3 hydrochloride,一种可穿透血脑屏障的多肽,用于探究中枢神经系统通透性的研究。 | |||
T67646 |
Methyl 2-amino-3-chloropropanoate hydrochloride
|
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Methyl 2-amino-3-chloropropanoate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67646,CAS号为 33646-31-0。 | |||
T41354 |
3-Nitrophenylhydrazine-13C6 hydrochloride
|
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T65408 | Propyl (3-(dimethylamino)propyl)carbamate hydrochloride | ||
Propyl (3-(dimethylamino)propyl)carbamate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T65408。 | |||
T66126 |
(S)-2-Amino-3-hydroxypropanamide hydrochloride
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(S)-2-Amino-3-hydroxypropanamide hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66126,CAS号为 65414-74-6。 | |||
T66437 |
(S)-Methyl 2-amino-3-(3-hydroxyphenyl)propanoate hydrochloride
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(S)-Methyl 2-amino-3-(3-hydroxyphenyl)propanoate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66437,CAS号为 34260-72-5。 | |||
T64466 |
(S)-Isopropyl 2-amino-3-hydroxypropanoate hydrochloride
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(S)-Isopropyl 2-amino-3-hydroxypropanoate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64466,CAS号为 37592-53-3。 | |||
T65367 | 3-Chloro-N-methylpropan-1-amine hydrochloride | ||
3-Chloro-N-methylpropan-1-amine hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65367,CAS号为 97145-88-5。 | |||
T67573 |
(S)-Methyl 2-amino-3-chloropropanoate hydrochloride
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(S)-Methyl 2-amino-3-chloropropanoate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67573,CAS号为 112346-82-4。 | |||
T65241 |
2-(Chloromethyl)-4-(3-methoxypropoxy)-3-methylpyridine hydrochloride
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2-(Chloromethyl)-4-(3-methoxypropoxy)-3-methylpyridine hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65241,CAS号为 153259-31-5。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T4710 |
3-Methoxytyramine hydrochloride
3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride),3-O-甲基多巴胺盐酸盐 |
Others; Endogenous Metabolite; Drug Metabolite | Metabolism; Others |
3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) 是多巴胺的无活性代谢物,能够活化痕量胺相关受体1 。 | |||
T4755 |
2,3-Diaminopropanoic acid hydrochloride
DL-2,3-Diaminopropionic acid monohydroch,3-Amino-DL-alanine monohydrochloride,DL-2,3-二胺基丙酸盐酸盐 |
Others; Endogenous Metabolite | Metabolism; Others |
2,3-Diaminopropanoic acid hydrochloride (3-Amino-DL-alanine monohydrochloride) 是内源性代谢产物的一种。 | |||
TN7062L |
Bufotenidine hydrochloride(487-91-2 Free base)
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Bufotenidine hydrochloride(487-91-2 Free base) 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN7062L,CAS号为 40581-89-3。 | |||
T4429 |
Rauwolscine hydrochloride
Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) 是一种高选择性的 α2 adrenergic 受体拮抗剂,Ki=12 nM。 | |||
T8787 |
Drotaverine hydrochloride
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PDE | Metabolism |
Drotaverine hydrochloride 是磷酸二酯酶 4 (PDE4)的抑制剂,也是 L 型电压依赖钙通道(L-VDCC)的阻滞剂,可阻断3',5'-环腺苷单磷酸的降解。它在体内有抗痉挛效果,但无抗胆碱能的效果。 | |||
T73856 |
Anagyrine hydrochloride
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Anagyrine ((-)-Anagyrine) hydrochloride 是一种存在于Lupinus albus 中的喹啉类生物碱。Anagyrine hydrochloride 可与毒蕈碱和烟碱乙酰胆碱受体 (AChR) 结合,IC50值分别为 132 和 2096 µM。Anagyrine hydrochloride 是一种有效的nAChR 脱敏剂,Anagyrine hydrochloride 可以直接脱敏nAChR,不需要代谢。 | |||
T5143 |
Corynoxine hydrochloride(6877-32-3(free base))
|
Autophagy | Autophagy |
Corynoxine hydrochloride(6877-32-3(free base)) 是一种天然羟吲哚生物碱,可在不同的神经元细胞系(包括 N2a 和 SHSY-5Y 细胞)中诱导自噬。 |