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抑制剂 & 化合物

9

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0442 Bucetin

3-Hydroxy-p-butyrophenetidide,布西丁,羟丁酰胺苯醚

Others Others
Bucetin (3-Hydroxy-p-butyrophenetidide) 是解热化合物,可用于研究疼痛的缓解。
T1501 Rifabutin

LM-427,Ansamycin,利福布汀,利福布丁

HSP; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Rifabutin (LM-427) 是半合成的安莎霉素抗生素,抑制 DNA 依赖性 RNA 聚合酶,有抗分枝杆菌作用。
T1584 Terbutaline Sulfate

Terbutaline hemisulfate,硫酸叔丁宁按,硫酸特布他林

Antibacterial; Adrenergic Receptor; Antibiotic GPCR/G Protein; Microbiology/Virology; Neuroscience
Terbutaline Sulfate (Terbutaline hemisulfate) 是一种具有口服活性的 β2-肾上腺素能受体激动剂,是班布特罗的活性代谢物。它可研究哮喘。
T1350 4-Butoxyphenol

4-正丁氧基苯酚,P-Butoxyphenol

Others Others
4-Butoxyphenol (P-Butoxyphenol) 是一种在科学和工业领域有广泛应用的酚类化合物。它经常用于合成其他化合物,如4-丁氧基苯乙酸和4-丁氧基苯乙腈;还用于合成药物,如布洛芬和萘普生。

化合物

Bucetin
Cat.No: T0442
Synonym: 3-Hydroxy-p-butyrophenetidide,布西丁,羟丁酰胺苯醚
Target: Others
Rifabutin
Cat.No: T1501
Synonym: LM-427,Ansamycin,利福布汀,利福布丁
Target: HSP, DNA/RNA Synthesis, Antibacterial, Antibiotic
Terbutaline Sulfate
Cat.No: T1584
Synonym: Terbutaline hemisulfate,硫酸叔丁宁按,硫酸特布他林
Target: Antibacterial, Adrenergic Receptor, Antibiotic
4-Butoxyphenol
Cat.No: T1350
Synonym: 4-正丁氧基苯酚,P-Butoxyphenol
Target: Others
Cat. No. Product Name Target Signaling Pathways
T22308 Dimboa

2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one,丁布

Others; Antibacterial; Antibiotic; Antifungal Microbiology/Virology; Others
Dimboa (2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one) 是抗生素,是禾本科植物化学防御系统的一部分。 它对许多已研究的细菌和真菌菌株具有生长抑制特性。它表现出强大的自由基清除活性和较弱的铁 (III) 离子还原活性和有抗氧化活性。
T6S1529 Cynarin

Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1R,​3R,​4S,​5R)​-,Cynarine,1,5-Dicaffeoylquinic acid,洋蓟素,金银花

Antioxidant; Antiviral; Influenza Virus; Reactive Oxygen Species Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction
Cynarin (1,5-Dicaffeoylquinic acid) 是一种抗窒息剂,具有抗氧化、抗组胺和抗病毒等多种生物活性。
TN5254 Wighteone

Erythrinin B,6-Isopentenylgenistein

Antifungal Microbiology/Virology
Wighteone (Erythrinin B) 是一种从 Genista ephedroides 中提取出来的小分子化合物,具有潜在的抗真菌和抗癌活性,对 EGFR L858R/T790M 突变非小细胞肺癌具有抗肿瘤作用。。
TN1918 Medicarpin

美迪紫檀素

Apoptosis; BCL; ROS; JNK Apoptosis; Immunology/Inflammation; MAPK
Medicarpin 是从紫花苜蓿中分离出的一种类黄酮。它通过调节 P-gp 介导的药物外流,诱导白血病 P388 细胞凋亡并克服多药耐药性。
TN3834 Derrone

Antifection Microbiology/Virology
Derrone may be interesting antimicrobial agents to be used against infectious diseases caused by many pathogens. It is also a novel Aurora kinase inhibitor, it can significantly inhibit the formation and growth of MCF7 tumor spheroids.
T2805 Chlorogenic Acid

NSC-407296,3-O-Caffeoylquinic acid,Heriguard,绿原酸

Others; Influenza Virus; Reactive Oxygen Species; HIF/HIF Prolyl-Hydroxylase; Endogenous Metabolite; Antibacterial Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Others
Chlorogenic Acid (NSC-407296) 是咖啡和茶中的主要酚类化合物。它具有多种生物作用。
T6S0214 dl-Maackiain

(+)-Maackiain,高丽槐素,Demethylpterocarpin

Apoptosis; Parasite Apoptosis; Microbiology/Virology
dl-Maackiain (Demethylpterocarpin) 是分离自Maackia amurensis Rupr.et Maxim 的一种杀幼虫剂,针对埃及伊蚊,其LD50为 21.95 μg/ ml。
TN3397 Alpinumisoflavone

ERK; LDL; NF-κB; MEK; MAPK; Antifection MAPK; Metabolism; Microbiology/Virology; NF-κB
Alpinumisoflavone has atheroprotective effects, may result from their ability to upregulate mechanisms promoting HDL-cholesterol and bile acid formation, it is endowed with estrogenic properties accounting, at least in part, for E. lysistemon effects. Alp
TN3668 cis-Miyabenol C

Others Others
cis-Miyabenol C exhibits antioxidative activities and shows strong hyaluronidase inhibitory effects. cis-Miyabenol C also has ecdysteroid antagonist activity.

天然产物

Dimboa
Cat.No: T22308
Synonym: 2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one,丁布
Target: Others, Antibacterial, Antibiotic, Antifungal
Cynarin
Cat.No: T6S1529
Synonym: Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1R,​3R,​4S,​5R)​-,Cynarine,1,5-Dicaffeoylquinic acid,洋蓟素,金银花
Target: Antioxidant, Antiviral, Influenza Virus, Reactive Oxygen Species
Wighteone
Cat.No: TN5254
Synonym: Erythrinin B,6-Isopentenylgenistein
Target: Antifungal
Medicarpin
Cat.No: TN1918
Synonym: 美迪紫檀素
Target: Apoptosis, BCL, ROS, JNK
Derrone
Cat.No: TN3834
Synonym:
Target: Antifection
Chlorogenic Acid
Cat.No: T2805
Synonym: NSC-407296,3-O-Caffeoylquinic acid,Heriguard,绿原酸
Target: Others, Influenza Virus, Reactive Oxygen Species, HIF/HIF Prolyl-Hydroxylase, Endogenous Metabolite, Antibacterial
dl-Maackiain
Cat.No: T6S0214
Synonym: (+)-Maackiain,高丽槐素,Demethylpterocarpin
Target: Apoptosis, Parasite
Alpinumisoflavone
Cat.No: TN3397
Synonym:
Target: ERK, LDL, NF-κB, MEK, MAPK, Antifection
cis-Miyabenol C
Cat.No: TN3668
Synonym:
Target: Others
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