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9
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0442 |
Bucetin
3-Hydroxy-p-butyrophenetidide,布西丁,羟丁酰胺苯醚 |
Others | Others |
Bucetin (3-Hydroxy-p-butyrophenetidide) 是解热化合物,可用于研究疼痛的缓解。 | |||
T1501 |
Rifabutin
LM-427,Ansamycin,利福布汀,利福布丁 |
HSP; DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology |
Rifabutin (LM-427) 是半合成的安莎霉素抗生素,抑制 DNA 依赖性 RNA 聚合酶,有抗分枝杆菌作用。 | |||
T1584 |
Terbutaline Sulfate
Terbutaline hemisulfate,硫酸叔丁宁按,硫酸特布他林 |
Antibacterial; Adrenergic Receptor; Antibiotic | GPCR/G Protein; Microbiology/Virology; Neuroscience |
Terbutaline Sulfate (Terbutaline hemisulfate) 是一种具有口服活性的 β2-肾上腺素能受体激动剂,是班布特罗的活性代谢物。它可研究哮喘。 | |||
T1350 |
4-Butoxyphenol
4-正丁氧基苯酚,P-Butoxyphenol |
Others | Others |
4-Butoxyphenol (P-Butoxyphenol) 是一种在科学和工业领域有广泛应用的酚类化合物。它经常用于合成其他化合物,如4-丁氧基苯乙酸和4-丁氧基苯乙腈;还用于合成药物,如布洛芬和萘普生。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T22308 |
Dimboa
2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one,丁布 |
Others; Antibacterial; Antibiotic; Antifungal | Microbiology/Virology; Others |
Dimboa (2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one) 是抗生素,是禾本科植物化学防御系统的一部分。 它对许多已研究的细菌和真菌菌株具有生长抑制特性。它表现出强大的自由基清除活性和较弱的铁 (III) 离子还原活性和有抗氧化活性。 | |||
T6S1529 |
Cynarin
Cyclohexanecarboxylic acid, 1,3-bis[[3-(3,4-dihydroxyphenyl)-1-oxo-2-propen-1-yl]oxy]-4,5-dihydroxy-, (1R,3R,4S,5R)-,Cynarine,1,5-Dicaffeoylquinic acid,洋蓟素,金银花 |
Antioxidant; Antiviral; Influenza Virus; Reactive Oxygen Species | Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction |
Cynarin (1,5-Dicaffeoylquinic acid) 是一种抗窒息剂,具有抗氧化、抗组胺和抗病毒等多种生物活性。 | |||
TN5254 |
Wighteone
Erythrinin B,6-Isopentenylgenistein |
Antifungal | Microbiology/Virology |
Wighteone (Erythrinin B) 是一种从 Genista ephedroides 中提取出来的小分子化合物,具有潜在的抗真菌和抗癌活性,对 EGFR L858R/T790M 突变非小细胞肺癌具有抗肿瘤作用。。 | |||
TN1918 |
Medicarpin
美迪紫檀素 |
Apoptosis; BCL; ROS; JNK | Apoptosis; Immunology/Inflammation; MAPK |
Medicarpin 是从紫花苜蓿中分离出的一种类黄酮。它通过调节 P-gp 介导的药物外流,诱导白血病 P388 细胞凋亡并克服多药耐药性。 | |||
TN3834 |
Derrone
|
Antifection | Microbiology/Virology |
Derrone may be interesting antimicrobial agents to be used against infectious diseases caused by many pathogens. It is also a novel Aurora kinase inhibitor, it can significantly inhibit the formation and growth of MCF7 tumor spheroids. | |||
T2805 |
Chlorogenic Acid
NSC-407296,3-O-Caffeoylquinic acid,Heriguard,绿原酸 |
Others; Influenza Virus; Reactive Oxygen Species; HIF/HIF Prolyl-Hydroxylase; Endogenous Metabolite; Antibacterial | Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Others |
Chlorogenic Acid (NSC-407296) 是咖啡和茶中的主要酚类化合物。它具有多种生物作用。 | |||
T6S0214 |
dl-Maackiain
(+)-Maackiain,高丽槐素,Demethylpterocarpin |
Apoptosis; Parasite | Apoptosis; Microbiology/Virology |
dl-Maackiain (Demethylpterocarpin) 是分离自Maackia amurensis Rupr.et Maxim 的一种杀幼虫剂,针对埃及伊蚊,其LD50为 21.95 μg/ ml。 | |||
TN3397 | Alpinumisoflavone | ERK; LDL; NF-κB; MEK; MAPK; Antifection | MAPK; Metabolism; Microbiology/Virology; NF-κB |
Alpinumisoflavone has atheroprotective effects, may result from their ability to upregulate mechanisms promoting HDL-cholesterol and bile acid formation, it is endowed with estrogenic properties accounting, at least in part, for E. lysistemon effects. Alp | |||
TN3668 |
cis-Miyabenol C
|
Others | Others |
cis-Miyabenol C exhibits antioxidative activities and shows strong hyaluronidase inhibitory effects. cis-Miyabenol C also has ecdysteroid antagonist activity. |