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Search Results for " vasoconstrictor "

67

抑制剂 & 化合物

3

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T13920L	Terlipressin Acetate Terlipressin diacetate anhydrous,Terlipressin acetate anhydrous,醋酸特利加压素	Vasopressin Receptor	GPCR/G Protein
	Terlipressin Acetate 是一种高度选择性的加压素 V1 受体激动剂，对氧和葡萄糖剥夺/再氧合 (OGD/R) 诱导的肠上皮细胞损伤 (IEC-6) 具有抗炎和抗氧化作用，可用于肝肾综合征和耐去甲肾上腺素的败血性休克的研究。
T2568L	Felypressin acetate 2-(L-Phenylalanine)-8-L-lysinevasopressin,醋酸苯赖加压素,PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond),PLV 2,PLV-2	Vasopressin Receptor	GPCR/G Protein
	Felypressin acetate (PLV-2) 是加压素 1 的激动剂，作用于所有精氨酸加压素受体 1AS。 Felypressin acetate 可用于牙科手术。
T2568	Felypressin Octapressin,Felypressin Acetate,PLV-2,H-[Cys-Phe-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2,苯赖加压素	Vasopressin Receptor	GPCR/G Protein
	Felypressin (Octapressin) 是一种加压素 1 激动剂，也是血管收缩剂，可用于牙科手术中。
T21708L	Angiotensin 1/2 + A (2 - 8) Acetate Angiotensin 1/2 + A (2 - 8) Acetate (51833-76-2 Free base)	Others	Others
	Angiotensin 1/2 + A (2 - 8) Acetate 是一种血管收缩剂。
TP2165	Urotensin II, mouse acetate (9047-55-6 free base) Urotensin II, mouse acetate	GPR	Endocrinology/Hormones; GPCR/G Protein
	Urotensin II, mouse acetate (9047-55-6 free base) 是孤儿 GPR14 或 SENR 的内源性配体。它是一种强效血管收缩剂。
TP1737L	Urotensin II (114-124), human acetate Urotensin II (114-124), human acetate(251293-28-4 free base)	GPR	Endocrinology/Hormones; GPCR/G Protein
	Urotensin II (114-124), human acetate(251293-28-4 free base) 是一种 11 个氨基酸残基肽，是一种有效的血管收缩剂和孤儿受体 GPR14 的激动剂。
T0045	Heptaminol hydrochloride 盐酸庚胺醇,RP-2831 hydrochloride	Others	Others
	Heptaminol hydrochloride (RP-2831 hydrochloride) 是一种血管收缩剂，有用于低血压(特别是体位性低血压)的研究潜力。
T12924	Sitaxsentan TBC-11251,IPI 1040	Endothelin Receptor	GPCR/G Protein
	Sitaxsentan (TBC-11251) 是选择性内皮素A (ETA) 受体拮抗剂。内皮素是一种有效的血管收缩剂。Sitaxsentan 阻断内皮素与其受体的结合，从而消除内皮素的有害作用。
T19309L1	Endothelin 1 (swine, human) acetate Endothelin 1 (swine, human) acetate(117399-94-7 free base)	Endothelin Receptor	GPCR/G Protein
	Endothelin 1 (swine, human) acetate(117399-94-7 free base) 是一种合成肽，其序列为人和猪内皮素 1。它是一种有效的内源性血管收缩剂，通过两种类型的受体 ETA 和 ETB 起作用。
TP1049L	Ornipressin Acetate（3397-23-7，free）鸟氨酸加压素,Orpressin,POR-8	Others	Others
	Ornipressin Acetate (POR-8) 是一种有效的血管收缩剂、止血剂和肾脏剂。
T0446	Naphazoline hydrochloride 盐酸萘甲唑啉,Albalon,Rhinantin,Naphazoline HCl	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Naphazoline hydrochloride (Naphazoline HCl) 是一种咪唑啉衍生物，是一种眼血管收缩剂。
T7386	Bretylium tosylate 溴苄乙胺,托西溴苄铵	Others	Others
	Bretylium tosylate 是交感神经和肾上腺素神经的阻断剂，是血管收缩的神经递质突触前释放的抑制剂。
T21445	Naphazoline AK-Con,Naphcon-a,Clear Eyes,All Clear,萘甲唑林	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Naphazoline (Naphcon-a) 是一种具有显着 α 肾上腺素能活性的拟交感神经化合物。萘甲唑啉可用作血管收缩剂，当应用于粘膜时可快速减少肿胀。
T0948	Adrenalone hydrochloride Adrenalone HCl,肾上腺酮盐酸盐,盐酸肾上腺酮	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Adrenalone hydrochloride (Adrenalone HCl) 是一种多巴胺β氧化酶 (dopamine β oxidase) 抑制剂，结构与去甲肾上腺素转运蛋白 (NET) 配体相似，IC50=36.9 μM。它是一种肾上腺素能 (adrenergic) 激动剂，用作局部血管收缩剂和止血剂。
T0279	Metaraminol tartrate 重酒石酸间羟胺,Metaradrine tartrate,Metaraminol bitartrate	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Metaraminol tartrate (Metaradrine tartrate) 是一种 α-肾上腺素能 (α-adrenergic) 激动剂，是一种直接或间接影响肾上腺素受体的拟交感神经胺，其中 α 效应占主导地位，可作为血管加压剂。
T1462	Captopril SQ 14225,甲巯丙脯酸,卡托普利,SQ-14534,SA333	RAAS	Endocrinology/Hormones
	Captopril (SA333) 是一种含巯基的，具有口服活性的血管紧张素转换酶(ACE)抑制剂，IC50=0.025 μM，广泛应用于高血压和充血性心力衰竭的研究。Captopril 也是NDM-1抑制剂，IC50=7.9 μM。
T14021	20-HETE 20-hydroxy Arachidonic Acid	Others	Others
	20-HETE (20-hydroxy Arachidonic Acid) is a CYP450 metabolite and a potent vasoconstrictor and it is an endogenous inhibitor of the large-conductance Ca2+-activated K+ channel in renal arterioles. 20-HETE increases NADPH oxidase, ROS, and NF-κB activity, a
T8560	Angiotensin II human acetate Ang II acetate,DRVYIHPF acetate,Angiotensin II acetate,血管紧张素II	Apoptosis; RAAS	Apoptosis; Endocrinology/Hormones
	Angiotensin II human acetate (DRVYIHPF acetate) 是血管收缩剂，是肾素/血管紧张素系统的主要生物活性肽，在调节人类血压中起着核心作用。它刺激交感神经刺激，增加醛固酮生物合成和肾脏活动。它诱导血管平滑肌细胞生长，也诱导细胞凋亡。它通过 LOX-1 依赖的氧化还原敏感途径诱导内皮细胞毛细血管形成。
TP1295	Angiotensin I (human, mouse, rat) Angiotensin 1 Human,血管紧张素 1 (人)	Others	Others
	Angiotensin I (human, mouse, rat) 是血管紧张素Ⅱ的前体物质，在血管紧张素转化酶 (ACE) 的参与下裂解成血管紧张素Ⅱ。
TP1345	Kisspeptin-10, human (TFA)(374675-21-5,FREE)	GPR; Kisspeptin	Endocrinology/Hormones; GPCR/G Protein
	Kisspeptin-10, human (TFA)(374675-21-5,FREE) 是一种有效的血管收缩剂和血管生成抑制剂。 Kisspeptin-10，人类 TFA 通过其受体 GPR54 充当肿瘤转移抑制因子。 Kisspeptin-10-GPR54系统在胚胎肾发育中发挥重要作用。 Kisspeptin-10/GPR54 信号通过 NFATc4 介导的 BMP2 表达诱导成骨细胞分化
T6264	Bosentan Actelion,波生坦,Ro 47-0203,Benzenesulfonamide	Endothelin Receptor	GPCR/G Protein
	Bosentan (Benzenesulfonamide) 是 endothelin-1 (ET)拮抗剂，在人的 SMC 细胞中，它能够作用于 ETA 受体(Ki:4.7 nM)和 ETB 受体(Ki:95 nM)。
T6529	Halobetasol propionate 卤贝他索丙酸酯,Halobetasol Propionate,Ulobetasol propionate,BMY-30056,卤倍他索丙酸酯,CGP-14458	Phospholipase	Metabolism
	Halobetasol propionate (BMY-30056) 是一种在皮肤外使用的合成类固醇，具有抗炎，止痒和收缩血管的活性。
T0871	Noradrenaline bitartrate	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Noradrenaline bitartrate 直接作用于 α 和 β 肾上腺素能受体。它是去甲肾上腺素的酒石酸氢盐，去甲肾上腺素是一种合成苯乙胺，可模拟内源性去甲肾上腺素的拟交感神经作用。临床上，去甲肾上腺素用作外周血管收缩剂，通过其α-肾上腺素能作用导致动脉和静脉床收缩。它还被用作通过其 β-1 肾上腺素能作用介导的强效正性肌力和变时性心脏刺激剂。
T70216	Clonazoline
	Clonazoline is a coronary vasodilator that is an imidazoline sympathomimetic, an alpha-adrenoreceptor agonist. It was used as a nasal decongestant and vasoconstrictor.
T24603	PD-34799-SA PD 34799-SA,PD34799-SA
	PD-34799-SA is an effective inhibitor of vasoconstrictor responses to sympathetic nerve stimulation.
T24541	Norbormide Mcneil 1025,S 6999,MCN 1025,Shoxin,Raticate
	Norbormide is a toxic compound used as a rodenticide. It has several mechanisms of action, acting as a vasoconstrictor and calcium channel blocker.
TP1175	Endothelin-3, human, mouse, rabbit, rat Endothelin 3 (Rat,Human)
	Endothelin-3, human, mouse, rabbit, rat , is a cyclic 21 amino acid peptide. It is an endogenous neuropeptide and potent vasoconstrictor.
T81652	Nordefrin (±)-Cobefri
	Nordefrin ((±)-Cobefri)为Norepinephrine的衍生物，具有血管收缩作用。
TP1522	Angiotensin II (5-8), human
	Angiotensin II (5-8) is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin II
T69670	Clonazoline HCl
	Clonazoline HCl is the salt form of Clonazoline, a coronary vasodilator that is an imidazoline sympathomimetic, an alpha-adrenoreceptor agonist. It was used as a nasal decongestant and vasoconstrictor.
TP1737	Urotensin II (114-124), human
	Urotensin II (114-124), human, is an 11-amino acid residue peptide that exhibits strong vasoconstrictor activity and acts as an agonist for the orphan receptor GPR14.
T76564L	Endothelin-1 (1-31) (Human) acetate
	Endothelin-1 (1-31) (Human) acetate，源自于chymase对大ET-1的选择性水解，是一种有效的血管收缩剂和血压升高剂。
T13920	Terlipressin	Others	Others
	Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells.
T19309	Endothelin 1 (swine, human)	Others	Others
	Endothelin 1 (swine, human), a synthetic peptide mirroring the sequence of both human and swine Endothelin 1, functions as a robust endogenous vasoconstrictor by interacting with two receptor types, ETA and ETB.
TP1661	Angiotensin II (1-4), human TFA
	Angiotensin II is a potent direct vasoconstrictor, causing arteries and veins to constrict, so leading to an increase in blood pressure.
T25199	Cafaminol Cafaminolum,G1,G-1,G 1
	Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant.
TP1049	Ornipressin POR-8,鸟氨酸加压素
	Ornipressin is a vasoconstrictor, haemostatic and renal agent.
TP1396	Kisspeptin-10, human
	Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.
T0279L2	Metaraminol hydrochloride Metaraminol HCl
	Metaraminol hydrochloride, used primarily as a vasoconstrictor in the treatment of HYPOTENSION, is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.
T78063	Endothelin-1 (1-31) (Human) TFA	ERK	MAPK
	Endothelin-1 (1-31) (Human) TFA 是源自chymase对大ET-1选择性水解的一种有效血管收缩剂和血压升高剂。
T37227	(±)8(9)-DiHET
	Epoxide hydrolases convert the EETs into vicinal diols, with the concurrent loss of much of their biological activity. The 8(S),9(R)-EET isomer is metabolized by platelet COX to form 8(S),9(R),11(R)-THETA, a trihydroxy fatty acid which may act as a renal vasoconstrictor.
T76564	Endothelin-1 (1-31) (Human)
	Endothelin-1 (1-31) (Human) 是源于chymase对大ET-1选择性水解而来的有效血管收缩剂和血压升高剂。
TP1415	Urotensin II (114-124), human TFA
	Urotensin II (114-124), human TFA, is an 11-amino acid residue peptide with a strong vasoconstrictor effect. This compound acts as an agonist for the orphan receptor GPR14.
T19631	PD 109488 PD-109488,Quinapril Diketopiperazine,PD109488
	PD 109488 is a metabolite of quinapril and is a derivative of Quinapril that acts as an ACE inhibitor. Inhibition of ACE prevents the conversion of signaling peptide angiotensin I into angiotensin II, which acts as a potent vasoconstrictor. Reduced levels of angiotensin II also reduces the amount of aldosterone that is expressed due to RAAS signaling.
TP2166	Urotensin II, mouse TFA (9047-55-6 free base) Urotensin II, mouse TFA	GPR	Endocrinology/Hormones; GPCR/G Protein
	Urotensin II, mouse TFA is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor.
T75962	Urotensin II, mouse acetate
	Urotensin II, mouse acetate，是孤儿G蛋白偶联受体（GPR14或SENR）的一种内源性配体，具有显著的血管收缩活性并在中枢神经系统中发挥重要功能。
T68825	Doxazosin HCl
	Doxazosin HCl is the salt form of Doxazosin Free Base which acts by inhibiting the postsynaptic alpha(1)-adrenoceptors on vascular smooth muscle. This inhibits the vasoconstrictor effect of circulating and locally released catecholamines (epinephrine and norepinephrine), resulting in peripheral vasodilation.
T36479	Big Endothelin-1 (1-38), human
	Human Big ET-1 comprises residues 53-90 of the endothelin precursor (preproendothelin). Compared to the mature endothelin-1 (hET-1), the peptide show less vasoconstrictor activity in vitro, but similar pressor effects in vivo. Former CAS-number 121014-53-7.
T76081	Endothelin 1 (swine, human), Alexa Fluor 488-labeled
	Endothelin 1 (swine, human), Alexa Fluor 488-labeled 是标记了488 荧光的 Endothelin 1 合成肽。Endothelin 1 (swine, human) 是具有人和猪内皮素 1 序列的合成肽，是有效的内源性血管收缩剂。Endothelin 1 通过两种类型受体 ETA 和 ETB 发挥作用。
T75961	Urotensin II, mouse TFA
	Urotensin II, mouse TFA 为孤儿G蛋白偶联受体GPR14或SENR的内源性配体，具有强效血管收缩作用，并在中枢神经系统中发挥重要角色。

化合物

Terlipressin Acetate

Cat.No: T13920L

Synonym: Terlipressin diacetate anhydrous,Terlipressin acetate anhydrous,醋酸特利加压素

Target: Vasopressin Receptor

Felypressin acetate

Cat.No: T2568L

Synonym: 2-(L-Phenylalanine)-8-L-lysinevasopressin,醋酸苯赖加压素,PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond),PLV 2,PLV-2

Target: Vasopressin Receptor

Cat.No: T2568

Synonym: Octapressin,Felypressin Acetate,PLV-2,H-[Cys-Phe-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2,苯赖加压素

Target: Vasopressin Receptor

Angiotensin 1/2 + A (2 - 8) Acetate

Cat.No: T21708L

Synonym: Angiotensin 1/2 + A (2 - 8) Acetate (51833-76-2 Free base)

Target: Others

Urotensin II, mouse acetate (9047-55-6 free base)

Cat.No: TP2165

Synonym: Urotensin II, mouse acetate

Target: GPR

Urotensin II (114-124), human acetate

Cat.No: TP1737L

Synonym: Urotensin II (114-124), human acetate(251293-28-4 free base)

Target: GPR

Heptaminol hydrochloride

Cat.No: T0045

Synonym: 盐酸庚胺醇,RP-2831 hydrochloride

Target: Others

Cat.No: T12924

Synonym: TBC-11251,IPI 1040

Target: Endothelin Receptor

Endothelin 1 (swine, human) acetate

Cat.No: T19309L1

Synonym: Endothelin 1 (swine, human) acetate(117399-94-7 free base)

Target: Endothelin Receptor

Ornipressin Acetate（3397-23-7，free）

Cat.No: TP1049L

Synonym: 鸟氨酸加压素,Orpressin,POR-8

Target: Others

Naphazoline hydrochloride

Cat.No: T0446

Synonym: 盐酸萘甲唑啉,Albalon,Rhinantin,Naphazoline HCl

Target: Adrenergic Receptor

Bretylium tosylate

Cat.No: T7386

Synonym: 溴苄乙胺,托西溴苄铵

Target: Others

Cat.No: T21445

Synonym: AK-Con,Naphcon-a,Clear Eyes,All Clear,萘甲唑林

Target: Adrenergic Receptor

Adrenalone hydrochloride

Cat.No: T0948

Synonym: Adrenalone HCl,肾上腺酮盐酸盐,盐酸肾上腺酮

Target: Adrenergic Receptor

Metaraminol tartrate

Cat.No: T0279

Synonym: 重酒石酸间羟胺,Metaradrine tartrate,Metaraminol bitartrate

Target: Adrenergic Receptor

Cat.No: T1462

Synonym: SQ 14225,甲巯丙脯酸,卡托普利,SQ-14534,SA333

Target: RAAS

Cat.No: T14021

Synonym: 20-hydroxy Arachidonic Acid

Target: Others

Angiotensin II human acetate

Cat.No: T8560

Synonym: Ang II acetate,DRVYIHPF acetate,Angiotensin II acetate,血管紧张素II

Target: Apoptosis, RAAS

Angiotensin I (human, mouse, rat)

Cat.No: TP1295

Synonym: Angiotensin 1 Human,血管紧张素 1 (人)

Target: Others

Kisspeptin-10, human (TFA)(374675-21-5,FREE)

Cat.No: TP1345

Target: GPR, Kisspeptin

Cat.No: T6264

Synonym: Actelion,波生坦,Ro 47-0203,Benzenesulfonamide

Target: Endothelin Receptor

Halobetasol propionate

Cat.No: T6529

Synonym: 卤贝他索丙酸酯,Halobetasol Propionate,Ulobetasol propionate,BMY-30056,卤倍他索丙酸酯,CGP-14458

Target: Phospholipase

Noradrenaline bitartrate

Cat.No: T0871

Target: Adrenergic Receptor

Cat.No: T70216

Cat.No: T24603

Synonym: PD 34799-SA,PD34799-SA

Cat.No: T24541

Synonym: Mcneil 1025,S 6999,MCN 1025,Shoxin,Raticate

Endothelin-3, human, mouse, rabbit, rat

Cat.No: TP1175

Synonym: Endothelin 3 (Rat,Human)

Cat.No: T81652

Synonym: (±)-Cobefri

Angiotensin II (5-8), human

Cat.No: TP1522

Clonazoline HCl

Cat.No: T69670

Urotensin II (114-124), human

Cat.No: TP1737

Endothelin-1 (1-31) (Human) acetate

Cat.No: T76564L

Cat.No: T13920

Target: Others

Endothelin 1 (swine, human)

Cat.No: T19309

Target: Others

Angiotensin II (1-4), human TFA

Cat.No: TP1661

Cat.No: T25199

Synonym: Cafaminolum,G1,G-1,G 1

Cat.No: TP1049

Synonym: POR-8,鸟氨酸加压素

Kisspeptin-10, human

Cat.No: TP1396

Metaraminol hydrochloride

Cat.No: T0279L2

Synonym: Metaraminol HCl

Endothelin-1 (1-31) (Human) TFA

Cat.No: T78063

Target: ERK

Cat.No: T37227

Endothelin-1 (1-31) (Human)

Cat.No: T76564

Urotensin II (114-124), human TFA

Cat.No: TP1415

Cat.No: T19631

Synonym: PD-109488,Quinapril Diketopiperazine,PD109488

Urotensin II, mouse TFA (9047-55-6 free base)

Cat.No: TP2166

Synonym: Urotensin II, mouse TFA

Target: GPR

Urotensin II, mouse acetate

Cat.No: T75962

Cat.No: T68825

Big Endothelin-1 (1-38), human

Cat.No: T36479

Endothelin 1 (swine, human), Alexa Fluor 488-labeled

Cat.No: T76081

Urotensin II, mouse TFA

Cat.No: T75961

Cat. No.	Product Name	Target	Signaling Pathways
T1287	Synephrine 辛弗林,Oxedrine	Endogenous Metabolite; Adrenergic Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Synephrine (Oxedrine) 是来自 Citrus aurantium 的α-adrenergic 和β-adrenergic 激动剂，是一种生物碱。它也是一种拟交感神经化合物，能够用于减肥。
T7040	Angiotensin II human DRVYIHPF,Angiotensin II,Hypertensin II,血管紧张素Ⅱ,Ang II,血管紧张素II	Apoptosis; RAAS	Apoptosis; Endocrinology/Hormones
	Angiotensin II human (Ang II) 是一种生物活性肽，一种血管收缩剂。Angiotensin II 可以与 AT1R 和 AT2R 相互作用，调节人类血压，刺激交感神经，增加醛固酮生物合成和肾脏活动。
TN6575	Pilosidine
	Pilosidine has vasoconstrictor activity, it showed facilitating effect on adrenaline evoked contractions in rabbit aorta isolated preparations.

天然产物

Cat.No: T1287

Synonym: 辛弗林,Oxedrine

Target: Endogenous Metabolite, Adrenergic Receptor

Angiotensin II human

Cat.No: T7040

Synonym: DRVYIHPF,Angiotensin II,Hypertensin II,血管紧张素Ⅱ,Ang II,血管紧张素II

Target: Apoptosis, RAAS

Cat.No: TN6575

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