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55

抑制剂 & 化合物

9

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
TP1285	Chlorotoxin(linear)
	Chlorotoxin(linear) is a linear 36 amino-acid peptide which can be used in Chlorotoxin related research. Chlorotoxin is a chloride channel blocker which has been found in the venom of the Egyptian scorpion Leiurus quinquestriatus.
T32764	Linear-benzoadenosine diphosphate Lin-benzo-ADP
	Linear-benzoadenosine diphosphate is a nucleotide analog.
T64749	ditridecylamine
	ditridecylamine 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T64749，CAS号为 101012-97-9。
T36049	Linearmycin B
	Linearmycin B is a polyene antibiotic that has been found inStreptomyces.1It induces lysis and degradation ofB. subtilisas a component ofStreptomycesMg1 extract.2 1.Sakuda, S., Guce-Bigol, U., Itoh, M., et al.Novel linear polyene antibiotics: LinearmycinsJ. Chem. Soc., Perkin Trans. 1182315-2319(1996) 2.Stubbendieck, R.M., and Straight, P.D.Escape from lethal bacterial competition through coupled activation of antibiotic resistance and a mobilized subpopulationPLoS Genet.11(12)e1005722(2015)
T36048	Linearmycin A
	Linearmycin A is a polyene antibiotic that has been found inStreptomyces.1It is active against the bacteriaS. aureusandE. coli(MICs = 3.1 and 1.6 μg/disc, respectively), the fungiS. cerevisiaeandC. albicans(MICs = 0.1 and 1.6 μg/disc, respectively), and the plant pathogenic fungusA. nigerin disc assays (MIC = 0.2 μg/disc). Linearmycin A induces lysis and degradation ofB. subtilisas a component ofStreptomycesMg1 extract.2 1.Sakuda, S., Guce-Bigol, U., Itoh, M., et al.Novel linear polyene antibiot...
T25736	Linearolactone
	Linearolactone, isolated from Salvia polystachya, inhibits Entamoeba histolytica and Giardia lamblia.
T25735	Linearol
	Linearol is a diterpene found in Sideritis L. spp. (Lamiaceae) with a broad range of demonstrated properties including antioxidant, anti-inflammatory, and anti-apoptotic activities.
T32216	Isolinearol
	Isolinearol is a secodolastane diterpene.
T60021	ecMetAP-IN-1	Others	Others
	ecMetAP-IN-1 可用作 QSAR 模型，以使用多元线性回归研究蛋氨酸氨基肽酶抑制剂作为抗癌剂。
TP1290	GRGDSP acetate(91037-75-1 free base) GRGDSP TFA	Integrin	Cytoskeletal Signaling
	GRGDSP acetate(91037-75-1 free base) 是一种合成的线性 RGD 肽，是一种整合素抑制剂。
TP1766L	D-γ-Glutamyl-D-glutamic acid acetate D-γ-Glutamyl-D-glutamic acid acetate(4553-17-7 free base)	Others	Others
	D-γ-Glutamyl-D-glutamic acid acetate(4553-17-7 free base) 是一种聚（γ-谷氨酸），由线性链中的 D-和 D-谷氨酸重复单元簇组成。
TP1410	Cecropin A	Antibacterial; Antibiotic	Microbiology/Virology
	Cecropin A 是37个氨基酸组成的线性多肽，表现出抗菌、抗炎和抗肿瘤的功效。
T78557	HOIPIN-1 JTP0819958	NF-κB	NF-κB
	HOIPIN-1 (JTP0819958) 是一种具有选择性和有效性的线性泛素链组装复合物 (LUBAC) 抑制剂（IC50 >2.8 μM）。HOIPIN-1 对LUBAC 介导的 NF-kB 激活有抑制作用。
T8951	JTP 0819958 - HOIPIN-1	IκB/IKK	NF-κB
	JTP 0819958 - HOIPIN-1 是一种选择性线性泛素链组装复合物 (LUBAC) 抑制剂，IC50 为 2.8 μM。 JTP-0819958 在体外抑制 LUBAC 介导的 NF-kB 活化[2]。
TP1432	Enfuvirtide acetate 醋酸恩夫韦地	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	Enfuvirtide acetate 是一种抗HIV-1融合的抑制肽，是一种由 36 个氨基酸组成的线性合成肽。它具有乙酰化的 N 端和羧酰胺 C 端。
T32750	Lignarenone B
	Lignarenone B is a linear polyene extracted from the mantles of the mollusc Scaphander lignaruis.
T40820	Gly6 hydrochloride Hexaglycine hydrochloride
	Gly6 hydrochloride (Hexaglycine hydrochloride) is a linear oligopeptide consisting of six glycine units.
T39278	L-Pentaguluronic acid
	L-Pentaguluronic acid, a linear polysaccharide copolymer, consists predominantly of four units of L-guluronic acid (G).
T70689	MEN-10354
	MEN-10354 is a less potent and less selective NK-2 tachykinin receptor antagonist compared to the linear analog, R 396.
TP1766	D-γ-Glutamyl-D-glutamic acid
	D-γ-Glutamyl-D-glutamic acid is a linear poly(γ-glutamic acid) compound composed of clusters of D-glutamic acid and D-glutamic acid repeating units.
T34174	Pseudobactin Ferric pseudobactin
	Pseudobactin is a linear hexapeptide fluorescent iron transport agent (siderophore) from plant growth promoter Pseudomonas B10.
T25368	Emd 51921 Emd51921,Emd-51921,Emd-51,921,Emd 51,921,Emd 51 921
	Emd 51921 is a linear peptide renin inhibitor.
TP1151	Gly6 Hexaglycine
	Gly6 is a linear peptide with six amino acids.
T38982	L-Tetraguluronic acid
	L-Tetraguluronic acid, a linear polysaccharide copolymer, comprises four units of L-guluronic acid (G).
T34628	SG3199 SG 3199,SG-3199
	SG3199 is a PBD dimer which binds in the minor groove of DNA, and forms covalent DNA interstrand cross-links in naked linear plasmid DNA. SG3199 is potently cytotoxic against a panel of human solid tumour and haematological cancer cell lines.
T39279	L-Hexaguluronic acid
	L-Hexaguluronic acid, a linear polysaccharide copolymer, consists of six units of L-guluronic acid (G).
T21075	Perfluoro(1,3-dimethylcyclohexane) Cyclohexane, perfluoro-1,3-dimethyl-,Hexadecafluoro-1,3-dimethylcyclohexane,Cyclohexane, decafluoro-1,3-bis(trifluoromethyl)-
	Perfluoro-1,3-dimethylcyclohexane is used as a synthesis reagent for amorphous fluorocarbon film preparation by plasma polymerization, and for the hydroformylation of linear terminal alkenes. As a chemically inert compound, it is similar in properties to
T38246	L-Triguluronic acid
	L-Triguluronic acid, a linear polysaccharide copolymer consisting of three L-guluronic acid (G) units, serves as a precursor for Alginate[1]. Alginate, an unbranched polyanionic polysaccharide, has applications in the development of delivery carriers for anti-fungal agents[2].
T31487	Dimethicone 350 Polysilane,Dimeticonum,Dimethicone,Ophtasiloxane,Dimeticona
	Dimethicone 350 is a silicone oil consisting of a mixture of fully methylated linear siloxane polymers end-blocking with trimethylsiloxy units. Commonly used in skin and hair products.
T34817	Tetrabutylphosphonium cation Tetra-n-butylphosphonium,J279H,Tetrabutylphosphonium ion,Tetrabutylphosphonium,Phosphonium, tetrabutyl-
	Tetrabutylphosphonium cation is a light orange solid and is the salt of the liphilic tetrabutylammonium cation and linear tribromide anion.
T40802	Poloxamer 188
	Poloxamer 188, a nonionic linear copolymer possessing surfactant properties, demonstrates anti-thrombotic, anti-inflammatory, and cytoprotective activities across different tissue injury models.
T29077	Urolinin nWWK-Tyr(3-NO2)-Abu
	Urolinin is a linear peptidic Urotensin-II Receptor Agonist with low nanomolar potency as well as improved metabolic stability. Urolinin is a hexameric UIIR agonist with an EC50 of 4.75 nM and a metabolic stability of 1319 min, 6.3-fold higher than wild-t
T75844	BIM-23056 TFA
	BIM23056 TFA为线性八肽类化合物，作为sst3与sst5生长抑素受体的有效拮抗剂，其Ki值分别为10.8和5.7。
T83487	[Pmp1,Tyr(OEt)2] AVP
	[Pmp1,Tyr(OEt)2] AVP为环状加压素(AVP)的线性拮抗剂，具备相似结构。
TP1171	Apraglutide TFA (1295353-98-8 free base) Apraglutide TFA,FE 203799e (TFA)
	Apraglutide TFA (FE 203799 TFA), a synthetic 33-amino-acid peptide and a long-acting GLP-2 analogue, enhances adaptation and linear intestinal growth in a neonatal piglet model of short bowel syndrome with total resection of the ileum.
T24697	R 396 Acleu-asp-gln-trp-phe-glynh2,速激肽拮抗剂多肽	Neurokinin receptor	GPCR/G Protein; Neuroscience
	R 396 (Acleu-asp-gln-trp-phe-glynh2) 是一种线性六肽，也是一种 NK-2 速激肽受体拮抗剂。
T38731	Intoplicine dimesylate RP 60475 dimesylate
	Intoplicine (RP 60475) dimesylate is a DNA topoisomerase I and II inhibitor belonging to the 7H-benzo[e]pyrido[4,3-b]indole series. It exhibits a strong affinity for DNA (K A = 2 x 10^5 /M), resulting in increased linear DNA length.
T36783	BPIQ-II (hydrochloride)
	BPIQ-II is a linear imidazoloquinazoline that potently inhibits the tyrosine kinase activity of the epidermal growth factor receptor (EGFR; IC50 = 8 pM). It is selective for EGFR over an assortment of other tyrosine and serine/threonine kinases. Cellular studies indicate that BPIQ-II can enter cells and very selectively shut down EGF-stimulated signal transmission by binding competitively at the ATP site of EGFR.
T82633	Cys-Asp-Pro-Gly-Tyr-Ile-Gly-Ser-Arg-NH2
	Cys-Asp-Pro-Gly-Tyr-Ile-Gly-Ser-Arg-NH2是源自层粘连蛋白B1链的线性肽，能够干预肿瘤细胞对基底膜的附着与侵袭，且表现出抗血管生成活性。
T83671	CCP-biotin Peptide (non-cyclized) Citrullinated Filaggrin (Q447H, S449C, G459R, E460G, S462C) (R455) (447-467)-biotin Peptide (non-cyclized),Cyclic Citrullinated Peptide-biotin Peptide (non-cyclized)
	CCP-biotin Peptide（非环化）是一种生物素化且非环化的圆形瓜氨酸化肽（CCP）版本。该序列对应于人类filaggrin的447-467氨基酸，但包含Q447H、S449C、G459R、E460G和S462C的替换，并在455位的精氨酸处发生了瓜氨酸化。CCP-biotin Peptide（非环化）旨在用于检测可能与线性肽结合的抗瓜氨酸自身抗体。
T75673	L-Diguluronic acid disodium
	L-Diguluronic acid disodium 是由两个 L-Guluronic acid 单元直接连接形成的直链多糖共聚物，主要应用于海藻酸的合成。作为无支链的聚阴离子多糖，它在抗真菌试剂载体的研究中也有其用途。
T76550	CooP
	CooP为一种针对线性胶质母细胞瘤的九肽，与胶质母细胞瘤细胞及其相关血管系统中的乳腺来源生长抑制剂/脂肪酸结合蛋白3 (FABP3) 发生结合。该化合物主要应用于化学疗法和多种纳米粒子的靶向递送。
T79925	T4 UvsX Recombinase	DNA/RNA Synthesis	Cell Cycle/Checkpoint; DNA Damage/DNA Repair
	T4 UvsX Recombinase 促进双链DNA模板上DNA复制的启动，通过催化模板DNA与同源单链DNA引物间的突触形成。此酶显著增强了T4 DNA聚合酶全酶在线性单链DNA模板上进行的回跳（发夹引物）DNA合成反应。
T74567	Phospholipid-PEG-Biotin (MW 10000)
	Phospholipid-PEG-Biotin (MW 10000)与Phospholipid-PEG-Biotin (MW 3400)均为磷脂与生物素通过线性PEG连接剂桥接形成的聚乙二醇衍生物。Phospholipid-PEG-Biotin (MW 3400) 能与亲和抗体相互作用，用于脂质体和细胞表面的修饰以及胰岛细胞的移植。
T36681	Sorafenib N-oxide
	Sorafenib N-oxide is an active metabolite of sorafenib , an inhibitor of Raf-1, B-RAF, and receptor tyrosine kinases. Sorafenib N-oxide inhibits FLT3 that contains the internal tandem duplication mutation (FLT3-ITD; Kd = 70 nM) and inhibits proliferation of MV4-11 acute myeloid leukemia (AML) cells expressing FLT3-ITD (IC50 = 25.8 nM). It is selective for AML cell lines containing FLT3-ITD over lines containing wild-type FLT3 (IC50s = 3.9-13.3 μM). Sorafenib N-oxide is also a linear-mixed inhibi...
T36523	Extracellular Death Factor
	Programmed cell death in bacteria is dependent on a system of cell-to-cell communication termed quorum sensing. Extracellular death factor (EDF) is a linear pentapeptide that communicating cells produce and release, which upon reaching a sufficient concentration activates the cell death pathway in a subset of cells. It is sensitive to extreme pH, high temperatures, and other stressful conditions. At 2.5 ng/ml, EDF has been shown to facilitate mazEF-mediated cell death, significantly reducing pop...
T74565	Phospholipid-PEG-Biotin (MW 3400)
	Phospholipid-PEG-Biotin (MW 3400) 为一种通过线性PEG链接剂桥接磷脂和生物素的磷脂聚乙二醇衍生物。该化合物能够与亲和抗体进行相互作用，并可用于脂质体及细胞表面的修饰，也适用于胰岛细胞移植。
T74568	Phospholipid-PEG-Biotin (MW 20000)
	Phospholipid-PEG-Biotin (MW 20000) 与 Phospholipid-PEG-Biotin (MW 3400) 均为磷脂和生物素通过线性 PEG 连接剂桥接形成的磷脂聚乙二醇衍生物。其中，Phospholipid-PEG-Biotin (MW 3400) 能与亲和抗体进行相互作用，并可用于修饰脂质体、细胞表面及胰岛细胞移植。
T76001	Apraglutide TFA
	Apraglutide TFA (FE 203799 TFA) 是一种合成的、含33个氨基酸的肽类药物，为长效GLP-2类似物。它能在全回肠切除后导致的新生短肠综合征小猪中增强适应性和线性肠生长。
T76523	HCV Core Protein (107-114)
	HCVCore Protein (107-114) 是主要线性 HCV 核心区域中免疫原性极低的残基。HCVCore Protein (107-114) 被鉴定为 101-118 区域内的结合位点，其包含基因型 Ⅰ/Ⅱ 和基因型 Ⅲ/Ⅵ 之间不同的两个残基。HCVCore Protein (107-114) 可能是传播 HCV 血清型的潜在位点。

化合物

Chlorotoxin(linear)

Cat.No: TP1285

Linear-benzoadenosine diphosphate

Cat.No: T32764

Synonym: Lin-benzo-ADP

ditridecylamine

Cat.No: T64749

Linearmycin B

Cat.No: T36049

Linearmycin A

Cat.No: T36048

Linearolactone

Cat.No: T25736

Cat.No: T25735

Cat.No: T32216

Cat.No: T60021

Target: Others

GRGDSP acetate(91037-75-1 free base)

Cat.No: TP1290

Synonym: GRGDSP TFA

Target: Integrin

D-γ-Glutamyl-D-glutamic acid acetate

Cat.No: TP1766L

Synonym: D-γ-Glutamyl-D-glutamic acid acetate(4553-17-7 free base)

Target: Others

Cat.No: TP1410

Target: Antibacterial, Antibiotic

Cat.No: T78557

Synonym: JTP0819958

Target: NF-κB

JTP 0819958 - HOIPIN-1

Cat.No: T8951

Target: IκB/IKK

Enfuvirtide acetate

Cat.No: TP1432

Synonym: 醋酸恩夫韦地

Target: HIV Protease

Cat.No: T32750

Gly6 hydrochloride

Cat.No: T40820

Synonym: Hexaglycine hydrochloride

L-Pentaguluronic acid

Cat.No: T39278

Cat.No: T70689

D-γ-Glutamyl-D-glutamic acid

Cat.No: TP1766

Cat.No: T34174

Synonym: Ferric pseudobactin

Cat.No: T25368

Synonym: Emd51921,Emd-51921,Emd-51,921,Emd 51,921,Emd 51 921

Cat.No: TP1151

Synonym: Hexaglycine

L-Tetraguluronic acid

Cat.No: T38982

Cat.No: T34628

Synonym: SG 3199,SG-3199

L-Hexaguluronic acid

Cat.No: T39279

Perfluoro(1,3-dimethylcyclohexane)

Cat.No: T21075

Synonym: Cyclohexane, perfluoro-1,3-dimethyl-,Hexadecafluoro-1,3-dimethylcyclohexane,Cyclohexane, decafluoro-1,3-bis(trifluoromethyl)-

L-Triguluronic acid

Cat.No: T38246

Dimethicone 350

Cat.No: T31487

Synonym: Polysilane,Dimeticonum,Dimethicone,Ophtasiloxane,Dimeticona

Tetrabutylphosphonium cation

Cat.No: T34817

Synonym: Tetra-n-butylphosphonium,J279H,Tetrabutylphosphonium ion,Tetrabutylphosphonium,Phosphonium, tetrabutyl-

Cat.No: T40802

Cat.No: T29077

Synonym: nWWK-Tyr(3-NO2)-Abu

Cat.No: T75844

[Pmp1,Tyr(OEt)2] AVP

Cat.No: T83487

Apraglutide TFA (1295353-98-8 free base)

Cat.No: TP1171

Synonym: Apraglutide TFA,FE 203799e (TFA)

Cat.No: T24697

Synonym: Acleu-asp-gln-trp-phe-glynh2,速激肽拮抗剂多肽

Target: Neurokinin receptor

Intoplicine dimesylate

Cat.No: T38731

Synonym: RP 60475 dimesylate

BPIQ-II (hydrochloride)

Cat.No: T36783

Cys-Asp-Pro-Gly-Tyr-Ile-Gly-Ser-Arg-NH2

Cat.No: T82633

CCP-biotin Peptide (non-cyclized)

Cat.No: T83671

Synonym: Citrullinated Filaggrin (Q447H, S449C, G459R, E460G, S462C) (R455) (447-467)-biotin Peptide (non-cyclized),Cyclic Citrullinated Peptide-biotin Peptide (non-cyclized)

L-Diguluronic acid disodium

Cat.No: T75673

Cat.No: T76550

T4 UvsX Recombinase

Cat.No: T79925

Target: DNA/RNA Synthesis

Phospholipid-PEG-Biotin (MW 10000)

Cat.No: T74567

Sorafenib N-oxide

Cat.No: T36681

Extracellular Death Factor

Cat.No: T36523

Phospholipid-PEG-Biotin (MW 3400)

Cat.No: T74565

Phospholipid-PEG-Biotin (MW 20000)

Cat.No: T74568

Apraglutide TFA

Cat.No: T76001

HCV Core Protein (107-114)

Cat.No: T76523

Cat. No.	Product Name	Target	Signaling Pathways
T4S1659	Xanthotoxol 8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,花椒毒酚,8-Hydroxypsoralene	Reactive Oxygen Species; 5-HT Receptor; Endogenous Metabolite	GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
	Xanthotoxol (Psoralen) 是一种具有生物活性的线性呋喃香豆素，具有很强的抗炎、抗氧化、5-HT 拮抗和神经保护作用等药理活性。
T19355	Heparan Sulfate 硫酸乙酰肝素,硫酸类肝素	FGFR; Wnt/beta-catenin; Endogenous Metabolite	Angiogenesis; Cytoskeletal Signaling; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
	Heparan sulfate 是一种复杂的线性多糖。Heparan sulfate 作为硫酸乙酰肝素蛋白聚糖的一部分出现，在细胞外基质和细胞表面表达丰富。
T1130	Gramicidin 短杆菌肽,Gramicidinum,Gramicidine,Gramicidina	MRP; Antibacterial; Antibiotic	Immunology/Inflammation; Microbiology/Virology
	Gramicidin (Gramicidine) 是一种抗菌肽。它通过组装成膜中的通道，增加其对阳离子的渗透性。
T1715	Chitosan (MW 150000) 壳聚糖,Chitosan,Poly(D-glucosamine),Deacetylated chitin	Antibacterial; Antifungal	Microbiology/Virology
	Chitosan (MW 150000) (Deacetylated chitin) 是衍生自几丁质的聚阳离子线性多糖。它无毒，具有低致敏性，生物相容性和可生物降解性。它还具有抗肿瘤，抗细菌，抗真菌和抗氧化活性。
T4794	Glutaric acid	Endogenous Metabolite	Metabolism
	Glutaric acid 是一种 C5 二羧酸，是色氨酸和赖氨酸分解代谢途径中的中间体。Glutaric acid 影响周细胞的收缩性和迁移。Glutaric acid 是 I 型戊二酸尿症的生物指标。
T2864	Lycopene 番茄红素,ψ,ψ-Carotene	Reactive Oxygen Species; ROS	Immunology/Inflammation; Metabolism; NF-κB
	Lycopene (ψ,ψ-Carotene) 是一种番茄及其产品和其他红色水果和蔬菜中天然存在的类胡萝卜素，具有抗氧化活性。
T75974	Cecropin A TFA
	Cecropin A TFA 是由 37 个氨基酸残基构成的线性抗菌肽，从 Hyalaphora cecropiapupae 得到，具有抗菌、抗炎和抗癌作用。
T38245	L-Diguluronic acid
	L-Diguluronic acid, a linear polysaccharide copolymer consisting of two L-guluronic acid (G) units, serves as a precursor for Alginate[1], a categorically unbranched polyanionic polysaccharide. Alginate finds application in the development of antifungal agent delivery carriers[2].
T75647	Nostosin G
	Nostosin G 是一种独特的线性肽，含有 3 个亚基，4-羟基苯乳酸 (Hpla)，高酪氨酸 (Hty) 和精氨酸。Nostosin G 具有有效的胰蛋白酶抑制特性，其 IC50值为 0.1 μM。

天然产物

Cat.No: T4S1659

Synonym: 8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,花椒毒酚,8-Hydroxypsoralene

Target: Reactive Oxygen Species, 5-HT Receptor, Endogenous Metabolite

Heparan Sulfate

Cat.No: T19355

Synonym: 硫酸乙酰肝素,硫酸类肝素

Target: FGFR, Wnt/beta-catenin, Endogenous Metabolite

Cat.No: T1130

Synonym: 短杆菌肽,Gramicidinum,Gramicidine,Gramicidina

Target: MRP, Antibacterial, Antibiotic

Chitosan (MW 150000)

Cat.No: T1715

Synonym: 壳聚糖,Chitosan,Poly(D-glucosamine),Deacetylated chitin

Target: Antibacterial, Antifungal

Cat.No: T4794

Target: Endogenous Metabolite

Cat.No: T2864

Synonym: 番茄红素,ψ,ψ-Carotene

Target: Reactive Oxygen Species, ROS

Cat.No: T75974

L-Diguluronic acid

Cat.No: T38245

Cat.No: T75647

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