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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T67784	6-fluorinated-aristeromycin2c
	6-fluorinated-aristeromycin2c 具有抗病毒感染活性，对热病毒、寨卡病毒和Sars 冠状病毒具有抑制作用。
T21404	Fluticasone furoate Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate	Glucocorticoid Receptor	Endocrinology/Hormones
	Fluticasone furoate (Avamys) 是一种合成的三氟化皮质类固醇，衍生自氟替卡松，Kd 为 0.3 nM。Fluticasone furoate 具有有效的抗炎、抗哮喘活性和低全身暴露。Fluticasone furoate 可用作过敏性鼻炎治疗研究的鼻喷雾剂。
T1038	Fludarabine NSC 118218,Fludarabinum,氟达拉宾,氟达拉滨,F-ara-A	Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis; STAT	Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; JAK/STAT signaling; Stem Cells
	Fludarabine (Fludarabinum) 是一种氟化嘌呤类似物，一种核酸合成抑制剂和 STAT1 激活抑制剂。Fludarabine 具有抗肿瘤活性，可以用于治疗白血病和淋巴瘤。
T71011	Perfluorinated SAHA
	Perfluorinated SAHA is an HDAC inhibitor for use in cancer treatment regimens, with demonstrated greater antiproliferative properties than SAHA . PFSAHA has also been shown to have higher selectivity for PA3774, an HDAC-like enzyme from P. aeruginosa, as well as other HDACs, which may prove beneficial for developing novel chemotherapeutic treatments for cancer.
T37720	Difluorinated H2S Fluorescent Probe 1
	Difluorinated H2S probe 1 is a fluorescent probe for hydrogen sulfide (H2S).1It selectively fluoresces in the presence of H2S over Zn2+, Fe3+, S2O32-, ClO-, SO32-, H2O2, NO2-, cysteine (Cys), homocysteine (Hcy), and glutathione (GSH) when used at a concentration of 1 μM. Difluorinated H2S probe 1 displays excitation/emission maxima of 365/450 nm, respectively. 1.Zhang, J., Gao, Y., Kang, X., et al.o,o-Difluorination of aromatic azide yields a fast-response fluorescent probe for H2S detection and...
T7398	ONC212	Apoptosis; GPR	Apoptosis; Endocrinology/Hormones; GPCR/G Protein
	ONC212 是氟化 ONC201 类似物，是有前景的抗癌剂。它也是 GPR132的选择性激动剂，可诱导凋亡。
T36020	Florfenicol amine (hydrochloride)
	Florfenicol amine is a major metabolite of the antibiotic florfenicol, a fluorinated derivative of chloramphenicol that is commonly used in veterinary medicine. The pharmacokinetics of florfenicol and florfenicol amine are commonly studied in edible tissues from domestic animals.
T31224	Piflufolastat DCFPYL	Epigenetic Reader Domain	Chromatin/Epigenetic
	Piflufolastat (DCFPYL) 是一种针对前列腺癌 PSMA 的 PET 显像剂。是一种含氟前列腺特异性膜抗原（PSMA）制剂。Piflufolastat 可用于制备 piflufolastat F 18 (DCFPyL F-18)。
T1428	Trifluridine 曲氟尿苷,NSC 529182,Trifluorothymidine,5-Trifluorothymidine,NSC 75520,曲氟胸苷,Viroptic,Trifluridina	Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis; HSV	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
	Trifluridine (NSC-75520) 是一种氟化胸苷类似物，具有潜在的抗肿瘤活性，还具有抗病毒活性。它掺入 DNA 并抑制胸苷酸合酶，从而抑制 DNA 合成、抑制蛋白质合成和细胞凋亡。
T38404	MJ33 lithium salt	ROS	Immunology/Inflammation
	MJ33 lithium salt 是 NADPH 氧化酶 2 型介导的 ROS 生成抑制剂，是一种氟化磷脂类似物，可抑制过氧化物还蛋白 6 （Prdx6）的磷脂酶 A2 （PLA2）活性，可用于研究急性肺损伤。
T8698	Hydrazinium hydroxide	Others	Others
	Hydrazinium hydroxide 是一种氟化羧酸，已被用于研究酶、激素和其他生物分子的作用机制，也已用于研究各种药物对身体的影响，以及研究环境毒素对身体的作用。
T27342L	Flurocitabine HCl Flurocitabine HCl(37717-21-8 Free base)	Others	Others
	Flurocitabine HCl 是阿糖胞苷的氟化酸酐类似物，在体内部分水解成两种活性抗肿瘤物质 (阿拉伯糖基-氟尿嘧啶 (ara-FC) 和阿拉伯糖基-氟尿嘧啶 (ara-FU))。Flurocitabine HCl 在急性白血病和实体瘤的 I 期研究中具显示出抗肿瘤活性。
T0454	Florfenicol 氟苯尼考,Nuflor,Aquafen	Others	Others
	Florfenicol (Aquafen) 是甲砜霉素的氟化合成类似物。在美国，氟苯尼考目前用于治疗与溶血性曼氏杆菌(巴氏杆菌)、多杀性巴氏杆菌和嗜血嗜血杆菌相关的牛呼吸道疾病(BRD)，以治疗与坏死梭杆菌和黑色素拟杆菌相关的牛趾间痰。
T0454L	Florfenicol SCH-25298,氟苯尼考,(-)-Florfenicol	Antibacterial; Antibiotic	Microbiology/Virology
	Florfenicol (SCH-25298) 是一种常见得兽用抗生素，能用于研究牛呼吸疾病，在水产养殖业中可以用来控制鲶鱼肠道败血病，也可诱导鸡蛋早期胚胎死亡，LC50 值为 1.07 μg/g。
T6501	Fludarabine Phosphate NSC 312887 Phosphate,fludara Phosphate,F-ara-A (NSC 312887) Phosphate,F-ara-AMP,磷酸氟达拉滨	Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis	Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
	Fludarabine Phosphate (NSC 312887 Phosphate) 是一种腺苷和脱氧腺苷类似物，与 dATP 竞争，并入到 DNA，可以抑制 DNA 聚合酶 α、核糖核苷酸还原酶和 DNA 引发酶，从而中断 DNA 合成并抑制肿瘤细胞生长。
T1666	Fludrocortisone acetate 9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,醋酸氟氢可的松,9α-fluorocortisol acetate	Glucocorticoid Receptor; Autophagy	Autophagy; Endocrinology/Hormones
	Fludrocortisone acetate (9α-Fludrocortisone acetate) 是一种合成的盐皮质激素，可减少尿液中钠丢失量，也用于增加血压，有用于阿狄森氏病的研究潜力。
T20814	Loratadine specified impurity F 11-Fluoro dihydroloratadine
	Loratadine specified impurity F is a fluorinated analog of Loratadine.
T33930	Perfluidone SB1528,SB 1528,Destun,SB-1528,WL 43423
	Perfluidone is a a fluorinated arylalkylsulphonamide plant growth regulator and herbicide.
T28154	Nemonoxacin Malate TG-873870,TG873870,TG 873870
	Nemonoxacin is a non-fluorinated quinolone antibiotic.
T35067	VM4-037 F-18 (F18)Vm-4-037,VM4037 F-18,VM4 037 F-18
	VM4-037 F-18 is a fluorinated PET imaging agent used for carbonic anhydrase IX.
T7594	Vinflunine
	Vinflunine is a new vinca alkaloid uniquely fluorinated with the properties of mitotic-arresting and tubulin-interacting activity.
T39363	2,4-Difluororesorcinol
	2,4-Difluororesorcinol is a fluorinated building block.
T25424	Flopristin RPR-132552,RPR-132552A,RPR 132552,RPR 132552A
	Flopristin, a semi-synthetic antibiotic of the streptogramin A class, is a fluorinated derivative of pristinamycin IIB.
T37318	Fluo-3FF (potassium salt)
	Fluo-3FF is a fluorescent calcium indicator. It is a di-fluorinated analog of Fluo-3 that displays about a 100-fold lower affinity than Fluo-3 for calcium (Kds = 42 and 0.4 μM, respectively). Low affinity calcium indicators are particularly useful for studying compartments with high concentrations of calcium, such as endoplasmic reticulum, where high affinity dyes will be insensitive to luminal fluctuations. Fluo-3FF has excitation/emission maxima of approximately 506 and 526 nm, respectively.
T6722	Vinflunine Tartrate	Microtubule Associated	Cytoskeletal Signaling
	Vinflunine Tartrate 是一种独特的新型长春花生物碱，具有抑制有丝分裂和微管蛋白相互作用活性的特性。
T21079	Decafluorobenzophenone Perfluorobenzophenone
	Decafluorobenzophenone is used in the synthesis of fluorinated acridones and acridines. Decafluorobenzophenone alcoholic solution generates radical anion and ketyl which can be studied by electron spin resonance spectra. It undergoes photolysis to form ke
T37037	Vinflunine ditartrate
	Vinflunine ditartrate, a fluorinated microtubule inhibitor and member of the Vinca alkaloids family, exhibits anti-angiogenic, vascular-disrupting, and anti-metastatic properties. It presents a potential avenue for studying transitional cell carcinoma of the urothelial tract, non-small cell lung cancer, and breast carcinoma[1][2].
T83830	2'-Deoxy-2'-fluoroadenosine-5'-O-triphosphate sodium 2′-fluoro-2′-deoxy ATP,AfTP,2'-fluoro dATP
	2'-Deoxy-2'-fluoroadenosine-5'-O-triphosphate是ATP的一种氟代衍生物，ATP是细胞代谢必需的能量底物。它抑制E. coli RNA聚合酶(Ki = 200 µM)。
T74786	BIBD-124
	BIBD-124 通过与淀粉样蛋白 (Aβ) 斑块结合，展现出优异的亲和力，其 IC50 值达到了 9.51 nM。作为一种放射性示踪剂，[18F]BIBD-124 能够针对 Aβ 斑块进行高效的标记。
T78879	CXCR4-IN-2	CXCR	Autophagy; GPCR/G Protein; Immunology/Inflammation
	CXCR4-IN-2（compound A1）是一款具有抗癌活性的双功能氟化小分子，是CXCR4的强效抑制剂。它对小鼠结直肠癌(CRC)细胞展现出显著的细胞毒性（IC50：60 μg/mL；72小时）和抗增殖能力，能够引导细胞在G2/M期发生阻滞并诱导细胞凋亡(apoptosis)。

化合物

6-fluorinated-aristeromycin2c

Cat.No: T67784

Fluticasone furoate

Cat.No: T21404

Synonym: Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate

Target: Glucocorticoid Receptor

Cat.No: T1038

Synonym: NSC 118218,Fludarabinum,氟达拉宾,氟达拉滨,F-ara-A

Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis, STAT

Perfluorinated SAHA

Cat.No: T71011

Difluorinated H2S Fluorescent Probe 1

Cat.No: T37720

Cat.No: T7398

Target: Apoptosis, GPR

Florfenicol amine (hydrochloride)

Cat.No: T36020

Cat.No: T31224

Synonym: DCFPYL

Target: Epigenetic Reader Domain

Cat.No: T1428

Synonym: 曲氟尿苷,NSC 529182,Trifluorothymidine,5-Trifluorothymidine,NSC 75520,曲氟胸苷,Viroptic,Trifluridina

Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis, HSV

MJ33 lithium salt

Cat.No: T38404

Target: ROS

Hydrazinium hydroxide

Cat.No: T8698

Target: Others

Flurocitabine HCl

Cat.No: T27342L

Synonym: Flurocitabine HCl(37717-21-8 Free base)

Target: Others

Cat.No: T0454

Synonym: 氟苯尼考,Nuflor,Aquafen

Target: Others

Cat.No: T0454L

Synonym: SCH-25298,氟苯尼考,(-)-Florfenicol

Target: Antibacterial, Antibiotic

Fludarabine Phosphate

Cat.No: T6501

Synonym: NSC 312887 Phosphate,fludara Phosphate,F-ara-A (NSC 312887) Phosphate,F-ara-AMP,磷酸氟达拉滨

Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis

Fludrocortisone acetate

Cat.No: T1666

Synonym: 9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,醋酸氟氢可的松,9α-fluorocortisol acetate

Target: Glucocorticoid Receptor, Autophagy

Loratadine specified impurity F

Cat.No: T20814

Synonym: 11-Fluoro dihydroloratadine

Cat.No: T33930

Synonym: SB1528,SB 1528,Destun,SB-1528,WL 43423

Nemonoxacin Malate

Cat.No: T28154

Synonym: TG-873870,TG873870,TG 873870

Cat.No: T35067

Synonym: (F18)Vm-4-037,VM4037 F-18,VM4 037 F-18

Cat.No: T7594

2,4-Difluororesorcinol

Cat.No: T39363

Cat.No: T25424

Synonym: RPR-132552,RPR-132552A,RPR 132552,RPR 132552A

Fluo-3FF (potassium salt)

Cat.No: T37318

Vinflunine Tartrate

Cat.No: T6722

Target: Microtubule Associated

Decafluorobenzophenone

Cat.No: T21079

Synonym: Perfluorobenzophenone

Vinflunine ditartrate

Cat.No: T37037

2'-Deoxy-2'-fluoroadenosine-5'-O-triphosphate sodium

Cat.No: T83830

Synonym: 2′-fluoro-2′-deoxy ATP,AfTP,2'-fluoro dATP

Cat.No: T74786

Cat.No: T78879

Target: CXCR

Cat. No.	Product Name	Target	Signaling Pathways
T0986	Flucytosine 5-Fluorocytosine,Ro 2-9915,5-氟胞嘧啶,Fluorocytosine,NSC 103805	DNA/RNA Synthesis; Antibiotic; Antifungal	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
	Flucytosine (NSC 103805) 是抗真菌化合物。

天然产物

Cat.No: T0986

Synonym: 5-Fluorocytosine,Ro 2-9915,5-氟胞嘧啶,Fluorocytosine,NSC 103805

Target: DNA/RNA Synthesis, Antibiotic, Antifungal

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