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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T13920L Terlipressin Acetate

Terlipressin diacetate anhydrous,Terlipressin acetate anhydrous,醋酸特利加压素

Vasopressin Receptor GPCR/G Protein
Terlipressin Acetate 是一种高度选择性的加压素 V1 受体激动剂,对氧和葡萄糖剥夺/再氧合 (OGD/R) 诱导的肠上皮细胞损伤 (IEC-6) 具有抗炎和抗氧化作用,可用于肝肾综合征和耐去甲肾上腺素的败血性休克的研究。
T14964 CI 972 anhydrous

CI 972 (anhydrous)

Others Others
CI 972 anhydrous is an inhibitor of purine nucleoside phosphorylase (PNP) (Ki: 0.83 μM) used as a T cell-selective immunosuppressive agent.
T1118L Cefprozil

Cefprozilum,Cefprozilo,Cefzil,Brisoral,Cefprozil anhydrous

Antibacterial; Antibiotic Microbiology/Virology
Cefprozil (Cefzil) 是一种新型头孢菌素类抗生素,具有抗病毒活性,可用于研究免疫系统疾病。
T23232 Remoxipride hydrochloride

Remoxipride Hydrochloride Anhydrous,Roxiam,(S)-Remoxipride Hydrochloride

Dopamine Receptor GPCR/G Protein; Neuroscience
Remoxipride hydrochloride (Roxiam) 是一种选择性的 D2 受体拮抗剂,对 D2 受体、D1 受体和 α1-肾上腺素能受体的 IC50 分别为 1.57 μM、>100 μM 和 42 μM。
T69105 Methyldopa anhydrous

Methyldopa anhydrous is a Central alpha-2 Adrenergic Agonist. The mechanism of action of methyldopa anhydrous is as an Adrenergic alpha2-Agonist.
T6999 Teneligliptin hydrobromide

Teneligliptin hydrobromide anhydrous,MP-513 (hydrobromide)

Others; Proteasome; DPP-4 Others; Proteases/Proteasome; Ubiquitination
Teneligliptin hydrobromide (MP-513(hydrobromide)) 是β2肾上腺素能受体 (β2AR) 阻滞剂,具有抗高血压、抗氧化、清除自由基的活性。
T68603 Mioflazine hydrochloride anhydrous

Mioflazine hydrochloride anhydrous is a nucleoside transport inhibitor that acts on adenosine to improve sleep.
T25004 Advantame anhydrous

Advantame

Advantame anhydrous is a non-caloric sweetener, synthesized from isovanillin and aspartame. The U.S. Food and Drug Administration has approved Advantame for general use in foods and beverages except for meat and poultry as a food additive.
T72004 Azumolene sodium anhydrous

Azumolene sodium anhydrous is a muscle relaxant that inhibits the release of calcium from skeletal muscle sarcoplasmic reticulum. Azumolene inhibits a component of store-operated calcium entry coupled to the skeletal muscle ryanodine receptor. Azumolene, an equipotent dantrolene analog, inhibits a component of SOCE coupled to activation of RyR1 by caffeine and ryanodine, whereas the SOCE component induced by thapsigargin is not affected.
T68319 MBX-8025 lysine anhydrous

MBX-8025 lysine anhydrous is a selective PPAR-delta agonist.
T20165 Alitame anhydrous

CP54802,CP-54802,CP 54802

Alitame anhydrous is a non-nutritive sweetener. It is 2000 times sweeter than sucrose.
T24254 KB-5492 anhydrous

KB-5492,KB5492,KB 5492

KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.
T6349L Sitafloxacin

DU6859,DU 6859,DU 6859A,Sitafloxacin anhydrous,DU-6859,DU6859A,DU-6859A,西他沙星

Sitafloxacin, a new generation of broad-spectrum oral fluoroquinolones, is highly effective against many Gram-positive, Gram-negative, and anaerobic clinical isolates (including strains resistant to other fluoroquinolones).
T11907 Pomaglumetad methionil anhydrous

LY2140023

GluR Neuroscience
LY2140023 has the potential for schizophrenia.LY2140023 is an orally active prodrug of LY404039. LY404039 is a selective metabotropic glutamate 2/3 receptor agonist.
T69677 Mitapivat sulfate anhydrous

Mitapivat sulfate anhydrous is an allosteric activator of Pyruvate Kinase (PK) that may be useful in the treatment of Pyruvate Kinase Deficiency.
T71048 Tacrolimus anhydrous 8-epimer

Tacrolimus anhydrous 8-epimer is a new l-pipecolic acid macrolide lactone, an important immunosuppressive drug that blocks T cell proliferation in vitro by inhibiting the generation of several lymphokines, especially IL-2.
T20122 Isoproterenol sulfate anhydrous

Norisodrine,Novodrine,Novodrin,dl-Isoproterenol sulfate,Isoprenaline sulphate,Aleudrin

Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.
T68519 Maropitant citrate anhydrous

Maropitant citrate anhydrous is a neurokinin (NK1) receptor antagonist.
T70755 Fimasartan potassium anhydrous

Fimasartan potassium anhydrous is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure.
T35350 Calcium gluconate monohydrate

Calciofon,Calcium gluconate anhydrous,Calcium D-gluconate,Glucobiogen,Calcarea gluconica

Others Others
Calcium gluconate (Calcarea gluconica, Calcium gluconate anhydrous, Calcium D-gluconate, Calciofon, Glucobiogen)是维持正常神经、肌肉和心脏功能所必需的元素或矿物质。葡萄糖钙可维持体内钙平衡,口服可阻止骨质疏松。
T20897 Cefepime dihydrochloride

Cefepime hydrochloride anhydrous,BMY-28142 dihydrochloride,Cepimax,Axepim,Cefepime HCl

Cefepime dihydrochloride, a broad-spectrum fourth-generation cephalosporin, binds and inactivates penicillin-binding proteins (PBPs) located on the inner membrane of the bacterial cell wall.
T20167 Cilazapril

Ro-34-2848,Ro 34-2848,Cilazapril (anhydrous),Ro34-2848,西拉普利

Cilazapril is an angiotensin-converting enzyme inhibitor. It has been researched for mild to moderate essential hypertension.
T21112 Triprolidine hydrochloride

295 C 51,Pro-Entra,Entra,盐酸曲普利啶,Actidilat,Triprolidine hydrochloride anhydrous,Actidil,Pro-Actidil

Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.
T69273 Mexrenoate potassium

Mexrenoate potassium is a steroidal aldosterone antagonist and antihypertensive.
T28414 Piclozotan

SUN-N-4057,SUN4057,SUNN-4057,SUN-4057,SUNN4057

5-HT Receptor GPCR/G Protein; Neuroscience
Piclozotan (anhydrous) 是一种 5-HT1A 受体激动剂,在短暂的大脑中动脉闭塞(t-MCAO)模型中表现出显着的神经保护活性,可以改善晚期帕金森病患者的运动并发症。
T3289 Amifostine

氨磷汀,Ethyol,WR2721,Gammaphos

Others; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism; Others
Amifostine (Ethyol) 是一种广谱细胞保护剂和辐射防护剂,具有清除自由基的作用。它可选择性保护正常组织免受放射线和化学疗法造成的损害。它是有效的 HIF-α1和 p53诱导剂,可降低肾脏毒性并具有抗血管生成作用。
T0366 Cefadroxil

BL-S 578,头孢羟氨苄

Antibacterial; Antibiotic Microbiology/Virology
Cefadroxil (BL-S 578) 是头孢菌素类广谱抗生素, 有效抑制革兰氏阳性和阴性菌感染。
T65281 Magnesium acetate tetrahydrate

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
Magnesium acetate tetrahydrate 是无水醋酸镁盐的水合形式。Magnesium acetate tetrahydrate 常用来合成其他化合物,可作为电解质补充剂或分子生物学实验中的试剂。
T13647 Dextran sulfate sodium salt (MW 4500-5500)

DSS,Dextran sulfate sodium salt (MW 4500-5500),硫酸葡聚糖钠盐

Apoptosis; HIV Protease Apoptosis; Microbiology/Virology; Proteases/Proteasome
Dextran sulfate sodium salt (MW 4500-5500) 是一种脱水葡萄糖的聚合物,分子量范围是4500-5500。Dextran sulfate sodium salt (MW 4500-5500) 通过阻止病毒吸附到宿主细胞中来抑制人免疫缺陷病毒的复制。Dextran sulfate sodium salt (MW 4500-5500) 是常用的炎症性肠病造模药物,可通过硫酸基团引起的高负电荷破坏肠黏膜屏障完整性,从而导致肠屏障受损,巨噬细胞功能失调以及菌群紊乱等现象。
TNU0778 2’-O-Methy-2,5’-anhydro-5-methyluridine

2'-O-Methy-2,5'-anhydro-5-methyluridine is a anhydrous nucleoside; 2'-O-Methyl nucleoside.
TNU0779 2’-O-Methyl-2,5’-anhydrouridine

2'-O-Methyl-2,5'-anhydrouridine is a anhydrous nucleoside; 2'-O-Methyl nucleoside.
TNU0709 2,5’-Anhydro-uridine

2’-Deoxy nucleoside; Anhydrous nucleoside
T1005 Amoxicillin

Amoxycillin,阿莫西林

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin (Amoxycillin) 是一种具有广谱抗菌活性和良好口服吸收的抗生素。
T72272 Glibenclamide potassium

Glyburide potassium

Glibenclamide (Glyburide) potassium 是 Glibenclamide 的钾盐形式。Glibenclamid potassium 以无水和水合物形式存在,与纯 Glibenclamide 相比具有更高的溶解度。
TMIH-0088 Amoxicillin-d4

Amoxicillin-d4 是 Amoxicillin 的氘代化合物。Amoxicillin 的 CAS 号为 26787-78-0。Amoxicillin是一种具有广谱抗菌活性和良好口服吸收的抗生素。
T71066 Cidofovir sodium

Cidofovir sodium is the salt form of Cidofovir, a Cytomegalovirus Nucleoside Analog DNA Polymerase Inhibitor that is an injectable antiviral medication primarily used as a treatment for cytomegalovirus (CMV) retinitis in people with AIDS. The mechanism of action of cidofovir is as a DNA Polymerase Inhibitor. The chemical classification of cidofovir anhydrous is Nucleoside Analog.

化合物

Terlipressin Acetate
Cat.No: T13920L
Synonym: Terlipressin diacetate anhydrous,Terlipressin acetate anhydrous,醋酸特利加压素
Target: Vasopressin Receptor
CI 972 anhydrous
Cat.No: T14964
Synonym: CI 972 (anhydrous)
Target: Others
Cefprozil
Cat.No: T1118L
Synonym: Cefprozilum,Cefprozilo,Cefzil,Brisoral,Cefprozil anhydrous
Target: Antibacterial, Antibiotic
Remoxipride hydrochloride
Cat.No: T23232
Synonym: Remoxipride Hydrochloride Anhydrous,Roxiam,(S)-Remoxipride Hydrochloride
Target: Dopamine Receptor
Methyldopa anhydrous
Cat.No: T69105
Synonym:
Target:
Teneligliptin hydrobromide
Cat.No: T6999
Synonym: Teneligliptin hydrobromide anhydrous,MP-513 (hydrobromide)
Target: Others, Proteasome, DPP-4
Mioflazine hydrochloride anhydrous
Cat.No: T68603
Synonym:
Target:
Advantame anhydrous
Cat.No: T25004
Synonym: Advantame
Target:
Azumolene sodium anhydrous
Cat.No: T72004
Synonym:
Target:
MBX-8025 lysine anhydrous
Cat.No: T68319
Synonym:
Target:
Alitame anhydrous
Cat.No: T20165
Synonym: CP54802,CP-54802,CP 54802
Target:
KB-5492 anhydrous
Cat.No: T24254
Synonym: KB-5492,KB5492,KB 5492
Target:
Sitafloxacin
Cat.No: T6349L
Synonym: DU6859,DU 6859,DU 6859A,Sitafloxacin anhydrous,DU-6859,DU6859A,DU-6859A,西他沙星
Target:
Pomaglumetad methionil anhydrous
Cat.No: T11907
Synonym: LY2140023
Target: GluR
Mitapivat sulfate anhydrous
Cat.No: T69677
Synonym:
Target:
Tacrolimus anhydrous 8-epimer
Cat.No: T71048
Synonym:
Target:
Isoproterenol sulfate anhydrous
Cat.No: T20122
Synonym: Norisodrine,Novodrine,Novodrin,dl-Isoproterenol sulfate,Isoprenaline sulphate,Aleudrin
Target:
Maropitant citrate anhydrous
Cat.No: T68519
Synonym:
Target:
Fimasartan potassium anhydrous
Cat.No: T70755
Synonym:
Target:
Calcium gluconate monohydrate
Cat.No: T35350
Synonym: Calciofon,Calcium gluconate anhydrous,Calcium D-gluconate,Glucobiogen,Calcarea gluconica
Target: Others
Cefepime dihydrochloride
Cat.No: T20897
Synonym: Cefepime hydrochloride anhydrous,BMY-28142 dihydrochloride,Cepimax,Axepim,Cefepime HCl
Target:
Cilazapril
Cat.No: T20167
Synonym: Ro-34-2848,Ro 34-2848,Cilazapril (anhydrous),Ro34-2848,西拉普利
Target:
Triprolidine hydrochloride
Cat.No: T21112
Synonym: 295 C 51,Pro-Entra,Entra,盐酸曲普利啶,Actidilat,Triprolidine hydrochloride anhydrous,Actidil,Pro-Actidil
Target:
Mexrenoate potassium
Cat.No: T69273
Synonym:
Target:
Piclozotan
Cat.No: T28414
Synonym: SUN-N-4057,SUN4057,SUNN-4057,SUN-4057,SUNN4057
Target: 5-HT Receptor
Amifostine
Cat.No: T3289
Synonym: 氨磷汀,Ethyol,WR2721,Gammaphos
Target: Others, HIF/HIF Prolyl-Hydroxylase
Cefadroxil
Cat.No: T0366
Synonym: BL-S 578,头孢羟氨苄
Target: Antibacterial, Antibiotic
Magnesium acetate tetrahydrate
Cat.No: T65281
Synonym:
Target: Endogenous Metabolite, Antibacterial
Dextran sulfate sodium salt (MW 4500-5500)
Cat.No: T13647
Synonym: DSS,Dextran sulfate sodium salt (MW 4500-5500),硫酸葡聚糖钠盐
Target: Apoptosis, HIV Protease
2’-O-Methy-2,5’-anhydro-5-methyluridine
Cat.No: TNU0778
Synonym:
Target:
2’-O-Methyl-2,5’-anhydrouridine
Cat.No: TNU0779
Synonym:
Target:
2,5’-Anhydro-uridine
Cat.No: TNU0709
Synonym:
Target:
Amoxicillin
Cat.No: T1005
Synonym: Amoxycillin,阿莫西林
Target: Antibacterial, Antibiotic
Glibenclamide potassium
Cat.No: T72272
Synonym: Glyburide potassium
Target:
Amoxicillin-d4
Cat.No: TMIH-0088
Synonym:
Target:
Cidofovir sodium
Cat.No: T71066
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2O2798 D-(+)-Trehalose

Ergot Sugar,D-Trehalose,Mycose,D-(+)-Trehalose Anhydrous,D-海藻糖,Trehalose

Others; Endogenous Metabolite Metabolism; Others
D-(+)-Trehalose (Mycose) 来源于自Saccharomyces cerevisiae,常用作食品成分和药物赋形剂。

天然产物

D-(+)-Trehalose
Cat.No: T2O2798
Synonym: Ergot Sugar,D-Trehalose,Mycose,D-(+)-Trehalose Anhydrous,D-海藻糖,Trehalose
Target: Others, Endogenous Metabolite
TargetMol Loading
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