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50

抑制剂 & 化合物

16

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0893 Tinidazole

替硝唑,CP12574

Antibacterial; Antibiotic Microbiology/Virology
Tinidazole (CP12574) 是一种对厌氧菌和原生动物具有选择性抗菌活性的 5-硝基咪唑,是一种具有口服活性的抗菌剂。
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T19794 Temafloxacin

替马沙星,Omniflox

Antibiotic Microbiology/Virology
Temafloxacin (Omniflox) 是一种喹诺酮类广谱抗菌剂,对革兰氏阳性菌、革兰氏阴性菌和厌氧菌均有效。
T2279 Tizoxanide

替唑尼特,Desacetyl-nitazoxanide,TIZ

Antiviral; HIV Protease; Antibacterial; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Tizoxanide (Desacetyl-nitazoxanide) 是 Nitazoxanide 活性代谢物,有抗HIV-1的活性。Nitazoxanide 可抗细菌和多种病毒复制。
T5189 Omadacycline

PTK 0796,Amadacycline

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Omadacycline (Amadacycline) 是一种具有口服活性的氨基甲基环素抗菌剂,是四环素类抗生素。它与 30S 核糖体亚基结合,抑制细菌蛋白质合成。它可用于研究急性细菌性皮肤和皮肤结构感染,感染性肺炎和尿路感染。
T4991 Ertapenem sodium

厄他培南钠,MK-826,L-749345,尔他培南钠

Antibacterial; Antibiotic Microbiology/Virology
Ertapenem sodium (MK-826) 是碳青霉烯,是一种 β-内酰胺抗生素,具有广谱抗菌活性。
T0195 Secnidazole

RP-14539,PM-185184,塞克硝唑

Antibiotic; Parasite Microbiology/Virology
Secnidazole (PM-185184) 是一种具有口服活性唑类抗生素,半衰期比甲硝唑更长。它有潜力研究细菌性阴道病。
T12004 Meropenem trihydrate

美罗培南三水合物,SM 7338 trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Meropenem trihydrate (SM 7338 trihydrate) 是一种碳青霉烯抗生素,具有广谱抗菌活性。它对敏感和耐药的杜克氏杆菌 (MIC 值为 0.015-0.12 mg/mL), 淋病奈瑟氏球菌 (MIC 值为 0.02-0.06 mg/mL)和流感嗜血杆菌 (MIC 值为 0.03-0.12 mg/mL) 具有活性。
T1283 Clinafloxacin

克林沙星,PD 127391,CI-960,AM-1091

Antibacterial; Antibiotic Microbiology/Virology
Clinafloxacin (CI-960) 是一种高效广谱氟喹诺酮类抗生素,抑制革兰氏阳性、革兰氏阴性和厌氧病原体。它对金黄色葡萄球菌的 DNA 促旋酶和拓扑异构酶 IV 有抑制作用,IC50值分别为 0.92 µg/ml 和 1.62 µg/ml。
T11013L2 Levorotation nimorazole phosphate ester TFA

Others Others
Levorotation nimorazole phosphate ester TFA 是一种抗厌氧菌和抗原虫感染的试剂。
T11013L1 Dextrorotation nimorazole phosphate ester TFA

Others Others
Dextrorotation nimorazole phosphate ester TFA 是一种抗厌氧菌和抗原虫感染的试剂。
T7466 5-Bromocytosine

Others Others
5-Bromocytosine 可用于在厌氧和需氧条件下合成交联产物。
T3263 (6R,7S)-Cefminox sodium heptahydrate

Meicelin,头孢米诺钠,Cefminox Sodium,Alteporina,Tencef

Antibiotic Microbiology/Virology
(6R,7S)-Cefminox sodium heptahydrate (Meicelin) 是一种 Cefminox sodium heptahydrate 的异构体。它也是一种具有广谱抗菌活性的 β-内酰胺头孢菌素抗生素。
T12096L Morinidazole

Antibacterial Microbiology/Virology
Morinidazole 具有抗菌活性,可用于厌氧菌引起的阑尾炎、盆腔炎等细菌感染研究。
T1037 Doripenem monohydrate

多尼培南(一水合物),S 4661 monohydrate,Doripenem Hydrate,S-4661

Antibacterial; Antibiotic Microbiology/Virology
Doripenem monohydrate (S 4661 monohydrate) 是广谱β-内酰胺抗生素,它对革兰氏阳性,阴性和厌氧菌有抗菌作用。
T6706 Ticarcillin sodium

Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Ticarcillin sodium (Aerugipen hydrate) 主要用于抗革兰氏阴性菌, 也能用于研究嗜麦芽感染。
T12022 Metronidazole Benzoate

Benzoyl metronidazole

Antibacterial Microbiology/Virology
Metronidazole Benzoate (Benzoyl metronidazole) 是甲硝唑和苯甲酸衍生物,具有抗菌,抗寄生虫,抗滴虫等作用,常用于治疗由厌氧菌引起的感染。
T11427 Antibacterial compound 2

Antifungal Microbiology/Virology
Antibacterial compound 2 是一种有效的抗菌剂,对许多人类兽医病原体有效,对多重耐药葡萄球菌、肠球菌和链球菌,以及厌氧菌有抑制作用。
T67826 Alalevonadifloxacin

DNA gyrase; Topoisomerase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Alalevonadifloxacin 是一种DNA 回旋酶和DNA 拓扑异构酶抑制剂,是一种喹诺酮类针对Mrsa 的新型抗菌化合物。Alalevonadifloxacin 对治疗细菌性革兰氏阳性、革兰氏阴性和厌氧性感染有潜在作用。
T7043 Cefotetan

头孢替坦,Apacef

Antibacterial; Antibiotic Microbiology/Virology
Cefotetan (Apacef) 是一种半合成的头霉素抗生素,能抑制细胞壁合成发挥杀菌作用。
T4501 Ceftizoxime

头孢唑肟,Epocelin

Antibacterial; Antibiotic Microbiology/Virology
Ceftizoxime (Epocelin) 是一种强效抗菌剂,它通过干扰细菌细胞壁合成和抑制肽聚糖的交联起作用。它对广谱的 β-内酰胺酶具有高度抗性,并且对多种需氧和厌氧的革兰氏阳性和革兰氏阴性微生物均有效。
T4103 (L)-Sodium lactate

L-乳酸钠,Sodium L-Lactate

Others Others
(L)-Sodium lactate (Sodium L-Lactate) 是由乳酸脱氢酶从丙酮酸中产生的。它在无氧糖酵解过程中或增殖活跃的细胞中产生。 它在人和动物的血液和肌肉液中少量存在。剧烈运动后,肌肉和血液中的乳酸浓度会增加。 它也存在于肝脏、肾脏、胸腺、人羊水以及其他器官和体液中。
T32949 Luminamicin

Luminamicin is active against anaerobic bacteria, especially Clostridium sp.; isolated from actinomycete strain OMR-59.
T26449 A 80556

A-80556,A80556

A 80556, a fluoroquinolone antibiotic, has potent antibacterial activity against gram-positive, gram-negative, and anaerobic organisms.
T33899 PD 131628

PD131628,PD-131628

PD 131628 is a novel fluoroquinolone that is a bioactive form of PD 131112 or CI-990 for use against anaerobic bacteria.
T31590 E 4441

E-4441,E4441

E 4441 is a third-generation difluoroquinolone, which has good activity against G(+) aerobic bacteria and anaerobic bacteria in vitro and in vivo.
T11013 Dextrorotation nimorazole phosphate ester

Others Others
Dextrorotation nimorazole phosphate ester is an anti-anaerobic and anti-parasitic agent. D-morpholine ornidazole organic phosphate is a newly developed, highly efficient, well-tolerated fourth-generation nitroimidazole derivative. Objective: Antibacterial
T6349L Sitafloxacin

DU6859,DU 6859,DU 6859A,Sitafloxacin anhydrous,DU-6859,DU6859A,DU-6859A,西他沙星

Sitafloxacin, a new generation of broad-spectrum oral fluoroquinolones, is highly effective against many Gram-positive, Gram-negative, and anaerobic clinical isolates (including strains resistant to other fluoroquinolones).
T3052L Sancycline HCl

6-Demethyl-6-deoxytetracycline,GS-2147,GS2147,GS 2147,NSC 51812 (as hydrochloride),Bonomycin

Sancycline is a semi-synthetic tetracycline antibiotic that is more active than tetracycline against 339 strains of anaerobic bacteria (MIC90s = 1 and 32 μg/ml, respectively).
T38322 A-54556B

A-54556B is a natural acyldepsipeptide (ADEP) antibiotic isolated from the fermentation broth of S. hawaiiensis. Like the closely related ADEP, A-54556A , A-54556B is effective against Gram-positive bacteria, including penicillin-resistant S. aureus. A-54556B is also effective against many strains of anaerobic bacteria.
T21400 Cefotetan disodium

YM09330,YM-09330,ICI-156834,ICI 156834,YM 09330,Cefotetan Sodium,ICI156834

Cefotetan Sodium, a second-generation cephalosporin, cephamycin antibiotic, is active against a wide range of both aerobic and anaerobic gram-negative and gram-positive bacteria. Cefotetan disrupts the cell wall synthesis by binding to penicillin-binding
T9233 Metronidazole acetic acid

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Metronidazole acetic acid 是 Metronidazole 的代谢产物,在细菌中具有诱变活性。Metronidazole 是硝基咪唑类抗生素,杀螨剂和抗原生动物剂。
T74332 Rifasutenizol

Rifasutenizol (TNP-2198)为一种有效的口服生物利用度高的双靶向抗菌剂,对微需氧菌和厌氧菌病原体展现出强大的活性。
T37186 D-(-)-Citramalic Acid (lithium salt)

D-(-)-Citramalic acid (lithium salt) is a biochemical intermediate involved in the anaerobic metabolism of glutamate through the methylaspartate pathway of C. tetanomorphum. It also plays various roles in other aspects of bacterial metabolism.
T70418 TLN-232

TLN-232, also known as CAP-232, is a synthetic cyclic heptapeptide with potential antineoplastic activity. Pyruvate kinase (PK) inhibitor TLN-232 targets pyruvate kinase M2 (M2PK), which may disrupt tumor cell anaerobic glycolysis. M2PK is a dimeric isoform of PK and the predominant PK isoform found in tumor cells.
T76114 Diaphorase

Diaphorase 能从厌氧污泥生物中获得。Diaphorase 通过脱硝作用,催化六氢-1,3,5-三硝基-1,3,5-三嗪 (RDX) 的生物转化。
T6471 Dicloxacillin Sodium

Veracillin,双氯西林,BRL1702 Sodium,BRL1702,Sodium dicloxacillin,双氯西林钠

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Dicloxacillin Sodium (BRL1702 Sodium) 是一种青霉素类窄谱β内酰胺抗生素, 用于革兰氏阳性菌感染的研究。它对β-内酰胺酶产生的微生物有抗菌作用。
T40605 N-(2-Hydroxyethyl)oxamic acid

N-(2-hydroxyethyl)-oxamic acid, a compound derived from the reduction of Metronidazole, can result from either chemical processes or through interaction with intestinal bacteria. Metronidazole itself is a nitroimidazole antibiotic with a broad range of efficacy against protozoans, as well as both Gram-negative and Gram-positive anaerobic bacteria.
T73902 Desacetylcefotaxime

Desacetylcefotaxime, Cefotaxime的一种体内代谢物,具有类似其母体化合物对多种需氧和厌氧细菌的体外抗菌活性。
T38321 A-39183A

A-39183A is an active component of the A-39183 antibiotic complex produced by aerobic fermentation of Streptomyces NRRL 12049. It has activity against penicillin-resistant S. aureus 3055 and S. faecalis X66 (MICs = 32 and 32 μg/ml, respectively) and a variety of Gram-positive and Gram-negative anaerobic bacteria (MICs = 16-128 μg/ml) in an agar dilution assay.
T67987 ecenofloxacin

Ecenofloxacin 是一种氟喹诺酮类抗菌药物,对革兰氏阳性、革兰氏阴性和厌氧生物具有有效的抗菌活性。
T34548 SC 28538

SC28538,SC-28538

SC 28538是一种5-硝基咪唑衍生物。它已被证明对脆弱芽孢杆菌、产气荚膜梭菌、阴道滴虫、胎儿滴虫、人型疟原虫和淋病奈瑟菌具有活性。在与284株厌氧菌的比较研究中,SC 28538的活性与甲硝唑或奥硝唑相同。
T75285 Metronidazole hydrochloride

Metronidazole hydrochloride (SC 326421) 是一种有口服活性的硝基咪唑抗生素,适用于厌氧微生物感染的研究。该化合物能穿越血脑屏障,长期服用可能引发炎症和骨骼肌收缩问题。
T78124 SF2312 ammonium

Antibiotic Microbiology/Virology
SF2312铵是SF2312的铵盐形式,后者为一种膦酸盐类抗生素兼烯醇酶抑制剂。该化合物可从放线菌小单孢菌分离而得,在缺氧环境中活性显著。SF2312对ENO1基因缺失的神经胶质瘤细胞显示出选择性毒杀作用。
T75286 Sitafloxacin hydrochloride

Sitafloxacin (DU6859a) hydrochloride 是一款有效的口服活性氟喹诺酮类抗生素,它对广泛的革兰氏阳性细菌、革兰氏阴性细菌(包括厌氧菌)及非典型病原体都显示出抗菌活性。该化合物主要用于研究呼吸道感染和尿路感染。
T75287 Sitafloxacin monohydrate

Sitafloxacin monohydrate (DU6859a) 是一种具有广谱的抗菌活性,并对多种革兰氏阳性和革兰氏阴性细菌(包括厌氧菌)以及非典型病原体有效的口服活性氟喹诺酮类抗生素。它主要用于研究呼吸道感染和尿路感染。
T73804 Botulinum toxin type B

Botulinum toxin type B是用于颈部肌张力障碍研究的抗原特异性肉毒毒素。该毒素为厌氧细菌肉毒梭菌产生的外毒素,其机制是通过抑制乙酰胆碱在神经肌肉接头的释放,从而导致注射部位肌肉的松弛性麻痹或减弱。
T75308 Secnidazole hemihydrate

Secnidazole (RP-14539) hemihydrate是一种具有口服活性的唑类抗生素及咪唑缓释剂,能够抑制黏质沙雷菌毒力,并类似于酰基高丝氨酸内酯地减缓QS导致的铜绿假单胞菌发病。在体外,Secnidazole hemihydrate对多种厌氧革兰氏阴性和革兰氏阳性细菌显示出抗菌活性。此化合物在阿米巴病、贾第虫病和细菌性阴道炎等疾病研究中有应用潜力。
T65598 Cefminox sodium

Cefminox (Sodium) is a new cephamycin antibiotic possessing a D-amino acid moiety derived from D-cysteine at the C-7B side chain. Cefminox is active against a wide range of bacteria, especially Gram-negative and anaerobic bacteria. Cefminox shows excellent in vivo efficacy (ED50) which is higher than would be expected from its in vitro activity (MIC). Moreover, cefminox possesses more potent activity in suppression of bacterial regrowth than other cephems[1]. Cefminox (Sodium) was the most activ...
T37880 OPC-167832

OPC-167832 is a potent and orally active dprE1 Inhibitor with an IC50 of 0.258 μM. OPC-167832 has antituberculosis activity and can be used for the research of tuberculosis caused by Mycobacterium tuberculosis[1]. OPC-167832 exhibits very low MICs against laboratory strains of M. tuberculosis H37Rv (MIC: 0.0005 μg/ml) and Kurono (MIC: 0.0005 μg/ml) and strains with monoresistance to rifampin (RIF), isoniazid (INH), ethambutol (EMB), streptomycin (STR), and pyrazinamide (PZA) (MIC: 0.00024-0.001 ...

化合物

Tinidazole
Cat.No: T0893
Synonym: 替硝唑,CP12574
Target: Antibacterial, Antibiotic
Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Temafloxacin
Cat.No: T19794
Synonym: 替马沙星,Omniflox
Target: Antibiotic
Tizoxanide
Cat.No: T2279
Synonym: 替唑尼特,Desacetyl-nitazoxanide,TIZ
Target: Antiviral, HIV Protease, Antibacterial, Autophagy
Omadacycline
Cat.No: T5189
Synonym: PTK 0796,Amadacycline
Target: ribosome, Antibacterial, Antibiotic
Ertapenem sodium
Cat.No: T4991
Synonym: 厄他培南钠,MK-826,L-749345,尔他培南钠
Target: Antibacterial, Antibiotic
Secnidazole
Cat.No: T0195
Synonym: RP-14539,PM-185184,塞克硝唑
Target: Antibiotic, Parasite
Meropenem trihydrate
Cat.No: T12004
Synonym: 美罗培南三水合物,SM 7338 trihydrate
Target: Antibacterial, Antibiotic
Clinafloxacin
Cat.No: T1283
Synonym: 克林沙星,PD 127391,CI-960,AM-1091
Target: Antibacterial, Antibiotic
Levorotation nimorazole phosphate ester TFA
Cat.No: T11013L2
Synonym:
Target: Others
Dextrorotation nimorazole phosphate ester TFA
Cat.No: T11013L1
Synonym:
Target: Others
5-Bromocytosine
Cat.No: T7466
Synonym:
Target: Others
(6R,7S)-Cefminox sodium heptahydrate
Cat.No: T3263
Synonym: Meicelin,头孢米诺钠,Cefminox Sodium,Alteporina,Tencef
Target: Antibiotic
Morinidazole
Cat.No: T12096L
Synonym:
Target: Antibacterial
Doripenem monohydrate
Cat.No: T1037
Synonym: 多尼培南(一水合物),S 4661 monohydrate,Doripenem Hydrate,S-4661
Target: Antibacterial, Antibiotic
Ticarcillin sodium
Cat.No: T6706
Synonym: Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen
Target: Others, Antibacterial, Antibiotic
Metronidazole Benzoate
Cat.No: T12022
Synonym: Benzoyl metronidazole
Target: Antibacterial
Antibacterial compound 2
Cat.No: T11427
Synonym:
Target: Antifungal
Alalevonadifloxacin
Cat.No: T67826
Synonym:
Target: DNA gyrase, Topoisomerase, Antibacterial
Cefotetan
Cat.No: T7043
Synonym: 头孢替坦,Apacef
Target: Antibacterial, Antibiotic
Ceftizoxime
Cat.No: T4501
Synonym: 头孢唑肟,Epocelin
Target: Antibacterial, Antibiotic
(L)-Sodium lactate
Cat.No: T4103
Synonym: L-乳酸钠,Sodium L-Lactate
Target: Others
Luminamicin
Cat.No: T32949
Synonym:
Target:
A 80556
Cat.No: T26449
Synonym: A-80556,A80556
Target:
PD 131628
Cat.No: T33899
Synonym: PD131628,PD-131628
Target:
E 4441
Cat.No: T31590
Synonym: E-4441,E4441
Target:
Dextrorotation nimorazole phosphate ester
Cat.No: T11013
Synonym:
Target: Others
Sitafloxacin
Cat.No: T6349L
Synonym: DU6859,DU 6859,DU 6859A,Sitafloxacin anhydrous,DU-6859,DU6859A,DU-6859A,西他沙星
Target:
Sancycline HCl
Cat.No: T3052L
Synonym: 6-Demethyl-6-deoxytetracycline,GS-2147,GS2147,GS 2147,NSC 51812 (as hydrochloride),Bonomycin
Target:
A-54556B
Cat.No: T38322
Synonym:
Target:
Cefotetan disodium
Cat.No: T21400
Synonym: YM09330,YM-09330,ICI-156834,ICI 156834,YM 09330,Cefotetan Sodium,ICI156834
Target:
Metronidazole acetic acid
Cat.No: T9233
Synonym:
Target: Antibacterial, Antibiotic, Parasite
Rifasutenizol
Cat.No: T74332
Synonym:
Target:
D-(-)-Citramalic Acid (lithium salt)
Cat.No: T37186
Synonym:
Target:
TLN-232
Cat.No: T70418
Synonym:
Target:
Diaphorase
Cat.No: T76114
Synonym:
Target:
Dicloxacillin Sodium
Cat.No: T6471
Synonym: Veracillin,双氯西林,BRL1702 Sodium,BRL1702,Sodium dicloxacillin,双氯西林钠
Target: Others, Antibacterial, Antibiotic
N-(2-Hydroxyethyl)oxamic acid
Cat.No: T40605
Synonym:
Target:
Desacetylcefotaxime
Cat.No: T73902
Synonym:
Target:
A-39183A
Cat.No: T38321
Synonym:
Target:
ecenofloxacin
Cat.No: T67987
Synonym:
Target:
SC 28538
Cat.No: T34548
Synonym: SC28538,SC-28538
Target:
Metronidazole hydrochloride
Cat.No: T75285
Synonym:
Target:
SF2312 ammonium
Cat.No: T78124
Synonym:
Target: Antibiotic
Sitafloxacin hydrochloride
Cat.No: T75286
Synonym:
Target:
Sitafloxacin monohydrate
Cat.No: T75287
Synonym:
Target:
Botulinum toxin type B
Cat.No: T73804
Synonym:
Target:
Secnidazole hemihydrate
Cat.No: T75308
Synonym:
Target:
Cefminox sodium
Cat.No: T65598
Synonym:
Target:
OPC-167832
Cat.No: T37880
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1079 Metronidazole

Flagyl,Metronidazol,甲硝唑,Anagiardil

Apoptosis; NADPH; Hydrogenase; Antibacterial; Antibiotic; Parasite; Antifection Apoptosis; Metabolism; Microbiology/Virology
Metronidazole (Metronidazol) 是一种合成的硝基咪唑衍生物,具有抗原生动物和抗菌活性。
T3982 Vulpinic Acid

狐衣酸,Vulpic acid,Pulvinic acid methyl ester

Others Others
Vulpinic Acid (Pulvinic acid methyl ester) 是地衣代谢物,可降低人脐静脉内皮细胞 (HUVEC) 中 H2O2诱导的ROS,氧化应激和氧化应激相关损伤,可作用于厌氧菌、葡萄球菌及肠球菌。它对脉粥样硬化的研究具有潜在的价值。
T0224 Meropenem

美罗培南,SM 7338

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Meropenem (SM 7338) 是一种具有广谱抗菌活性的碳青霉烯抗生素,对敏感和耐药的淋病奈瑟氏球菌,流感嗜血杆菌和杜克氏杆菌的 MIC 值分别为 0.02-0.06 mg/mL,0.03-0.12 mg/mL 和 0.015-0.12 mg/mL。
T1205 Chloramphenicol

Chlornitromycin,Levomycetin,Chloromycetin,氯霉素

ribosome; HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Chloramphenicol (Chloromycetin) 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。
T2719 Succinic acid

Asuccin,Amber acid,琥珀酸,1,2-Ethanedicarboxylic acid,Wormwood acid,Butanedioic acid,1,4-Butandioic Acid

Endogenous Metabolite Metabolism
Succinic acid (1,2-Ethanedicarboxylic acid) 是无氧代谢的发酵产物,也是三羧酸循环的中间产物。
T8302 Ceftiofur

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur 是一种半合成抗生素,对家畜的各种革兰氏阳性和革兰氏阴性菌、好氧菌和厌氧菌均有抗菌活性。
TN6952 Hexadecane

n-Hexadecane

Hexadecane (n-Hexadecane) 可作为真菌的碳源,与厌氧生物生物降解有关。Hexadecane 在豚鼠皮肤实验中抑制皮肤过度角质化。
T4845 L-Lactic acid

2-HYDROXYPROPIONIC ACID,L-乳酸,L-(+)-Lactic acid,(S)-2-Hydroxypropanoic acid

Endogenous Metabolite; Antibacterial; Antibiotic Metabolism; Microbiology/Virology
L-Lactic acid ((S)-2-Hydroxypropanoic acid) 属于天然产物,由丙酮酸的无氧糖酵解产生。L-Lactic acid 是组织缺氧的敏感指标,可作为危重病人的血流动力学指标。
T3950 Tridecanoic acid

n-Tridecoic Acid,n-Tridecanoic Acid,十三酸,Tridecylic Acid

Others; Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology; Others
Tridecanoic acid (Tridecylic Acid) 是一种存在于乳制品中的 13 碳饱和脂肪酸,也是正十六烷厌氧生物降解的产物。 它是磷脂酶 A2 的底物,可作为抗粘剂和抗生物膜剂,用于研究细菌感染。它抑制大肠杆菌的持久性和生物膜形成。
T8074 Esafosfan trisodium

Fosfructose trisodium,D-果糖-1,6-二磷酸三钠盐,D-Fructose-1,6-diphosphate trisodium salt octahydrate,FDP trisodium,Diphosphofructose trisodium

Others; Endogenous Metabolite Metabolism; Others
Esafosfan trisodium (FDP trisodium) 是一种细胞保护性的天然糖磷酸盐,用于镰状细胞性贫血,心血管缺血和哮喘的研究。Fosfructose trisodium 通过刺激无氧糖酵解起作用,其在缺血条件下产生三磷酸腺苷。
T3228 Fosfructose

D-fructose-1,6-diphosphate,Betulanonaprenol,4937-84-2,Diphosphofructose,二磷酸果糖,Fructose 1,6-diphosphate,D-fructofuranose 1,6-bisphosphate,Esafosfan

Others; Endogenous Metabolite Metabolism; Others
D-fructose-1,6-diphosphate 是一种细胞保护性的天然糖磷酸盐,Fosfructose 通过刺激无氧糖酵解起作用,其在缺血条件下产生三磷酸腺苷,有潜力用于心血管缺血,镰状细胞性贫血和哮喘的研究。
T20643 Cefoxitin

Rephoxitin,Cefoxitinum

Cell wall; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology
Cefoxitin (Rephoxitin) 是一种广谱的、可口服的第二代头孢霉素类抗生素。Cefoxitin 干扰细菌细胞壁的合成。其活性谱包括革兰氏阴性和革兰氏阳性菌,通常用于腹腔感染、盆腔感染和某些类型的妇科感染等腹部,对厌氧菌具有高效性。
T4838 (S)-Malic acid

L-(-)-Malic acid,(S)-(-)-HYDROXYSUCCINIC ACID,(S)-2-Hydroxysuccinic acid,L-苹果酸

Others; Endogenous Metabolite Metabolism; Others
(S)-Malic acid ((S)-2-Hydroxysuccinic acid) 是天然存在的二羧酸,是水果酸甜味的来源,常用作食品添加剂。
T28764 SF2312

SF-2312,SF 2312

SF2312 is an enolase inhibitor produced by the actinomycete Micromonospora, which is active under anaerobic conditions.
T25579 Kijanimicin

Kijanimicin sodium salt

Kijanimicin is an antitumor and antibiotic. It is a unique, large acid enol antibiotic and possesses an unusual in vitro spectrum of activity against some Gram-positive and anaerobic microorganisms. It has also shown interesting activity against malaria i
T1277 Lincomycin hydrochloride

Lincomycin HCl,NSC 70731,盐酸林可霉素,U10149A

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Lincomycin hydrochloride (U10149A) 是由林可链霉菌产生的抗生素,对革兰氏阳性球菌和厌氧菌具有活性。

天然产物

Metronidazole
Cat.No: T1079
Synonym: Flagyl,Metronidazol,甲硝唑,Anagiardil
Target: Apoptosis, NADPH, Hydrogenase, Antibacterial, Antibiotic, Parasite, Antifection
Vulpinic Acid
Cat.No: T3982
Synonym: 狐衣酸,Vulpic acid,Pulvinic acid methyl ester
Target: Others
Meropenem
Cat.No: T0224
Synonym: 美罗培南,SM 7338
Target: Others, Antibacterial, Antibiotic
Chloramphenicol
Cat.No: T1205
Synonym: Chlornitromycin,Levomycetin,Chloromycetin,氯霉素
Target: ribosome, HIF/HIF Prolyl-Hydroxylase, Antibacterial, Antibiotic
Succinic acid
Cat.No: T2719
Synonym: Asuccin,Amber acid,琥珀酸,1,2-Ethanedicarboxylic acid,Wormwood acid,Butanedioic acid,1,4-Butandioic Acid
Target: Endogenous Metabolite
Ceftiofur
Cat.No: T8302
Synonym:
Target: Antibacterial, Antibiotic
Hexadecane
Cat.No: TN6952
Synonym: n-Hexadecane
Target:
L-Lactic acid
Cat.No: T4845
Synonym: 2-HYDROXYPROPIONIC ACID,L-乳酸,L-(+)-Lactic acid,(S)-2-Hydroxypropanoic acid
Target: Endogenous Metabolite, Antibacterial, Antibiotic
Tridecanoic acid
Cat.No: T3950
Synonym: n-Tridecoic Acid,n-Tridecanoic Acid,十三酸,Tridecylic Acid
Target: Others, Endogenous Metabolite, Antibacterial
Esafosfan trisodium
Cat.No: T8074
Synonym: Fosfructose trisodium,D-果糖-1,6-二磷酸三钠盐,D-Fructose-1,6-diphosphate trisodium salt octahydrate,FDP trisodium,Diphosphofructose trisodium
Target: Others, Endogenous Metabolite
Fosfructose
Cat.No: T3228
Synonym: D-fructose-1,6-diphosphate,Betulanonaprenol,4937-84-2,Diphosphofructose,二磷酸果糖,Fructose 1,6-diphosphate,D-fructofuranose 1,6-bisphosphate,Esafosfan
Target: Others, Endogenous Metabolite
Cefoxitin
Cat.No: T20643
Synonym: Rephoxitin,Cefoxitinum
Target: Cell wall, Antibacterial, Antibiotic
(S)-Malic acid
Cat.No: T4838
Synonym: L-(-)-Malic acid,(S)-(-)-HYDROXYSUCCINIC ACID,(S)-2-Hydroxysuccinic acid,L-苹果酸
Target: Others, Endogenous Metabolite
SF2312
Cat.No: T28764
Synonym: SF-2312,SF 2312
Target:
Kijanimicin
Cat.No: T25579
Synonym: Kijanimicin sodium salt
Target:
Lincomycin hydrochloride
Cat.No: T1277
Synonym: Lincomycin HCl,NSC 70731,盐酸林可霉素,U10149A
Target: ribosome, Antibacterial, Antibiotic
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