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Cat. No. Product Name Target Signaling Pathways
TN2062 Phyllanthin

1,1'-[(2S,3S)-2,3-双(甲氧基甲基)-1,4-丁二基]双[3,4-二甲氧基苯],叶下珠素

NF-κB NF-κB
Phyllanthin 是 Phyllanthus amarus 的一种主要生物活性木脂素成分,具有显著的抗氧化和保肝活性。
TN6623 Phyllanthusiin C

Phyllanthusiin C是一种天然产物,属于使君子科诃子属,其产品编号为 TN6623,CAS号为 142674-52-0。Phyllanthusiin C可用作对照参考。
TN3005 4',4'''-Di-O-methylcupressuflavone

Others Others
4',4'''-Di-O-methylcupressuflavone is a natural product from Phyllanthus niruri Linn.
T38484 Englerin A

(-)-Englerin A

TRP/TRPV Channel Membrane transporter/Ion channel
Englerin A 是一种具有选择性和高效性的 TRPC4 和 TRPC5 通道激动剂,是一种来自东非植物 Phyllanthus engleri 的小分子化合物,具有镇痛、抗炎和抗癌活性。Englerin A 可刺激 TRPC4/C5 阳离子通道以抑制肿瘤细胞系增殖,诱导人肾癌细胞坏死。
TN4660 Niranthin

Anti-infection; HBV; PAFR; Topoisomerase DNA Damage/DNA Repair; GPCR/G Protein; Microbiology/Virology
Niranthin 是一种木脂素,具有广泛的药理活性。它是L. donovaniIB 拓扑异构酶的非竞争性抑制剂,可用于研究耐药利什曼病的治疗。
T6S2099 Geraniin

Antioxidant; TNF Apoptosis; oxidation-reduction
Geraniin 是一种肿瘤坏死因子α释放抑制剂,其IC50值为 43 μM,具有抗肿瘤、抗炎和抗高血糖活性。
TN1757 Hypophyllanthin

叶下珠次素,(7S,8S,9R)-9-(3,4-二甲氧基苯基)-6,7,8,9-四氢-4-甲氧基-7,8-双(甲氧基甲基)萘并[1,2-D]-1,3-二恶茂

Potassium Channel; Calcium Channel; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Hypophyllanthin 是珠子草中的一种木脂素,能直接抑制 P-gp 的活性,具有很强的抗炎活性。
TN1451 Brevifolincarboxylic acid

AhR; Aryl Hydrocarbon Receptor; Glucosidase Immunology/Inflammation; Metabolism
Brevifolincarboxylic acid 是从头状蓼中分离得到的一种天然产物,抑制芳烃受体(AhR)。它是一种 α-葡萄糖苷酶抑制剂,IC50 为 323.46 μM。
T36734 Methyl brevifolincarboxylate

Methyl brevifolincarboxylate (Brevifolincarboxylic acid methyl ester) is a potent influenza virus PB2 cap-binding inhibitor. Methyl brevifolincarboxylate exhibits inhibitory activity against influenza virus A/Puerto Rico/8/34 (H1N1) and A/Aichi/2/68 (H3N2) with IC50s of 27.16 μM and 33.41 μM. Anti-oxidant activity[1][2]. Methyl brevifolincarboxylate exhibits significant DPPH radical scavenging activity with an IC50 value of 8.9 μM. [1]. Wu QY, et al. Chromatographic fingerprint and the simultane...
TN4139 Glochicoccin D

Others Others
Glochicoccin D is a Standard reference.

天然产物

Phyllanthin
Cat.No: TN2062
Synonym: 1,1'-[(2S,3S)-2,3-双(甲氧基甲基)-1,4-丁二基]双[3,4-二甲氧基苯],叶下珠素
Target: NF-κB
Phyllanthusiin C
Cat.No: TN6623
Synonym:
Target:
4',4'''-Di-O-methylcupressuflavone
Cat.No: TN3005
Synonym:
Target: Others
Englerin A
Cat.No: T38484
Synonym: (-)-Englerin A
Target: TRP/TRPV Channel
Niranthin
Cat.No: TN4660
Synonym:
Target: Anti-infection, HBV, PAFR, Topoisomerase
Geraniin
Cat.No: T6S2099
Synonym:
Target: Antioxidant, TNF
Hypophyllanthin
Cat.No: TN1757
Synonym: 叶下珠次素,(7S,8S,9R)-9-(3,4-二甲氧基苯基)-6,7,8,9-四氢-4-甲氧基-7,8-双(甲氧基甲基)萘并[1,2-D]-1,3-二恶茂
Target: Potassium Channel, Calcium Channel, P-gp
Brevifolincarboxylic acid
Cat.No: TN1451
Synonym:
Target: AhR, Aryl Hydrocarbon Receptor, Glucosidase
Methyl brevifolincarboxylate
Cat.No: T36734
Synonym:
Target:
Glochicoccin D
Cat.No: TN4139
Synonym:
Target: Others
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