Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN2062 |
Phyllanthin
1,1'-[(2S,3S)-2,3-双(甲氧基甲基)-1,4-丁二基]双[3,4-二甲氧基苯],叶下珠素 |
NF-κB | NF-κB |
Phyllanthin 是 Phyllanthus amarus 的一种主要生物活性木脂素成分,具有显著的抗氧化和保肝活性。 | |||
TN6623 | Phyllanthusiin C | ||
Phyllanthusiin C是一种天然产物,属于使君子科诃子属,其产品编号为 TN6623,CAS号为 142674-52-0。Phyllanthusiin C可用作对照参考。 | |||
TN3005 |
4',4'''-Di-O-methylcupressuflavone
|
Others | Others |
4',4'''-Di-O-methylcupressuflavone is a natural product from Phyllanthus niruri Linn. | |||
T38484 |
Englerin A
(-)-Englerin A |
TRP/TRPV Channel | Membrane transporter/Ion channel |
Englerin A 是一种具有选择性和高效性的 TRPC4 和 TRPC5 通道激动剂,是一种来自东非植物 Phyllanthus engleri 的小分子化合物,具有镇痛、抗炎和抗癌活性。Englerin A 可刺激 TRPC4/C5 阳离子通道以抑制肿瘤细胞系增殖,诱导人肾癌细胞坏死。 | |||
TN4660 |
Niranthin
|
Anti-infection; HBV; PAFR; Topoisomerase | DNA Damage/DNA Repair; GPCR/G Protein; Microbiology/Virology |
Niranthin 是一种木脂素,具有广泛的药理活性。它是L. donovaniIB 拓扑异构酶的非竞争性抑制剂,可用于研究耐药利什曼病的治疗。 | |||
T6S2099 |
Geraniin
|
Antioxidant; TNF | Apoptosis; oxidation-reduction |
Geraniin 是一种肿瘤坏死因子α释放抑制剂,其IC50值为 43 μM,具有抗肿瘤、抗炎和抗高血糖活性。 | |||
TN1757 |
Hypophyllanthin
叶下珠次素,(7S,8S,9R)-9-(3,4-二甲氧基苯基)-6,7,8,9-四氢-4-甲氧基-7,8-双(甲氧基甲基)萘并[1,2-D]-1,3-二恶茂 |
Potassium Channel; Calcium Channel; P-gp | Membrane transporter/Ion channel; Metabolism; Neuroscience |
Hypophyllanthin 是珠子草中的一种木脂素,能直接抑制 P-gp 的活性,具有很强的抗炎活性。 | |||
TN1451 |
Brevifolincarboxylic acid
|
AhR; Aryl Hydrocarbon Receptor; Glucosidase | Immunology/Inflammation; Metabolism |
Brevifolincarboxylic acid 是从头状蓼中分离得到的一种天然产物,抑制芳烃受体(AhR)。它是一种 α-葡萄糖苷酶抑制剂,IC50 为 323.46 μM。 | |||
T36734 |
Methyl brevifolincarboxylate
|
||
Methyl brevifolincarboxylate (Brevifolincarboxylic acid methyl ester) is a potent influenza virus PB2 cap-binding inhibitor. Methyl brevifolincarboxylate exhibits inhibitory activity against influenza virus A/Puerto Rico/8/34 (H1N1) and A/Aichi/2/68 (H3N2) with IC50s of 27.16 μM and 33.41 μM. Anti-oxidant activity[1][2]. Methyl brevifolincarboxylate exhibits significant DPPH radical scavenging activity with an IC50 value of 8.9 μM. [1]. Wu QY, et al. Chromatographic fingerprint and the simultane... | |||
TN4139 |
Glochicoccin D
|
Others | Others |
Glochicoccin D is a Standard reference. |