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Search Results for " ask-1-in-1 "

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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T9697 ASK1-IN-1

ASK Apoptosis
ASK1-IN-1 是一种凋亡信号调节激酶 1(SK1) 抑制剂,具有良好的效价 (细胞IC50=138 nM; BiochemicalIC50=21 nM)。ASK1-IN-1具有中枢神经系统渗透性。
T9377 ASK1-IN-2

Apoptosis; ASK; MAPK Apoptosis; MAPK
ASK1-IN-2 是一种口服有活性的凋亡信号调节激酶 1 抑制剂(IC50:32.8 nM)。它可用于研究溃疡性结肠炎。

化合物

ASK1-IN-1
Cat.No: T9697
Synonym:
Target: ASK
ASK1-IN-2
Cat.No: T9377
Synonym:
Target: Apoptosis, ASK, MAPK
Cat. No. Product Name Target Signaling Pathways
TN4635 Neoechinulin A

NADPH-oxidase; Beta Amyloid; ASK; IκB/IKK; p38 MAPK; TNF; NOS; NF-κB; COX; Prostaglandin Receptor Apoptosis; GPCR/G Protein; Immunology/Inflammation; MAPK; Neuroscience; NF-κB
Neoechinulin A has anti-inflammatory effect against LPS-stimulated RAW264.7 macrophages through inhibition of the NF-κB and p38 MAPK pathways, it may block the phosphorylation of mitogen-activated protein kinase (MAPK) molecule p38, apoptosis signal-regu

天然产物

Neoechinulin A
Cat.No: TN4635
Synonym:
Target: NADPH-oxidase, Beta Amyloid, ASK, IκB/IKK, p38 MAPK, TNF, NOS, NF-κB, COX, Prostaglandin Receptor
TargetMol Loading
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