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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TF0106 |
Cholesteryl Hemisuccinate Tris Salt
|
Apoptosis | Apoptosis |
Cholesteryl Hemisuccinate Tris Salt 是一种具有保肝和抗癌活性的酸性胆固醇酯,是一种含有柴胡皂苷-d的二棕榈酰磷脂酰胆碱脂质体中的膜稳定剂,可增强顺铂的抗癌功效。Cholesteryl hemisuccinate 具有抗肿瘤活性,抑制肿瘤生长,抑制对乙酰氨基酚 (AAP) 的肝毒性,预防 AAP 诱导的肝细胞凋亡。Cholesteryl hemisuccinate 可保护啮齿动物免受对乙酰氨基酚、阿霉素、四氯化碳、氯仿和半乳糖胺的毒性作用。 | |||
T67509 |
Cholesteryl Hemisuccinate
Cholesterol hydrogen succinate |
Apoptosis; DNA/RNA Synthesis; Topoisomerase | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Cholesteryl Hemisuccinate (Cholesterol hydrogen succinate) 是一种经常使用在极性溶液中具有高溶解度的胆固醇类似物 ,具有保肝、抗癌和抑制肿瘤生长的作用。Cholesteryl Hemisuccinate 抑制对乙酰氨基酚 的肝毒性,并防止 AAP 诱导的肝细胞凋亡 和坏死 。Cholesteryl Hemisuccinate 抑制 DNA 聚合酶 和 DNA 拓扑异构酶 ,从而抑制 DNA 复制和修复以及细胞分裂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2768 |
Saikosaponin A
柴胡皂苷A,柴胡皂苷 A |
NF-κB; Antibacterial; Liver X Receptor | Metabolism; Microbiology/Virology; NF-κB |
Saikosaponin A 是银柴胡中的主要活性成分,有抗炎活性,可上调 LXRα的表达。 | |||
TN1186 |
11(α)-Methoxysaikosaponin F
11 α-甲氧基柴胡皂苷 F,11alpha-Methoxysaikosaponin F,11(Α)甲氧基柴胡皂苷F |
Others | Others |
11alpha-Methoxysaikosaponin F is a natural product | |||
T3913 |
Saikosaponin D
|
Estrogen Receptor/ERR; NF-κB; Antibacterial; STAT | Endocrinology/Hormones; JAK/STAT signaling; Microbiology/Virology; NF-κB; Stem Cells |
Saikosaponin D 是一种从柴胡中分离到的三萜皂苷类天然产物,具有抗炎,抗菌,抗肿瘤,抗过敏作用。它抑制 selectin,STAT3和 NF-kB 的活性,活化estrogen receptor-β。 | |||
T3912 |
Saikosaponin B1
柴胡皂苷B1,柴胡皂苷 B1 |
Others | Others |
Saikosaponin B1 是柴胡的生物活性成分,具有抗癌作用。它能够靶向SMO 抑制 Hedgehog 通路,显著抑制髓母细胞瘤模型中的肿瘤生长。 | |||
T3914 |
Saikosaponin C
柴胡皂苷C,柴胡皂苷 C |
Beta Amyloid; Caspase | Apoptosis; Neuroscience; Proteases/Proteasome |
Saikosaponin C 是一种柴胡中的活性成分,能够抑制 Aβ1-40 和 Aβ1-42 的释放,抑制异常 tau 蛋白的磷酸化,但对 BACE1 的活性和表达无作用。它在阿尔滋海默症中主要靶作用于amyloid beta 和tau 蛋白。 | |||
T16838 |
Saikogenin A
|
Proteasome; DPP-4 | Proteases/Proteasome; Ubiquitination |
Saikogenin A 是一种二肽基肽酶 IV 抑制剂,可从中药柴胡中提取。 | |||
TN1014 |
Saikosaponin E
|
Others | Others |
Saikosaponin E 是一种从柴胡中分离出来的天然产物。 | |||
TN6864 |
Prosaikogenin F
(2R,3R,4S,5R,6R)-2-{[(1S,2R,4S,5R,8R,9S,10R,13S,14R,17S,18R)-2-hydroxy-9-(hydroxymethyl)-4,5,9,13,20,20-hexamethyl-24-oxahexacyclo[15.5.2.01,1?.0?,1?.0?,1?.0?,13]tetracos-15-en-10-yl]oxy}-6-methyloxane-3,4,5-triol,前柴胡皂苷F |
Others | Others |
Prosaikogenin F ((2R,3R,4S,5R,6R)-2-{[(1S,2R,4S,5R,8R,9S,10R,13S,14R,17S,18R)-2-hydroxy-9-(hydroxymethyl)-4,5,9,13,20,20-hexamethyl-24-oxahexacyclo[15.5.2.01,1?.0?,1?.0?,1?.0?,13]tetracos-15-en-10-yl]oxy}-6-methyloxane-3,4,5-triol) 是一种单糖苷,具有溶血和抗癌特性。 | |||
T3810 |
Saikosaponin B2
柴胡皂苷 B2,柴胡皂甙 B2 |
Others; HCV Protease | Microbiology/Virology; Others; Proteases/Proteasome |
Saikosaponin B2 是从柴胡根中分离得到的一种活性成分,可抑制 HCV 病毒感染的侵入,有抗癌作用。 | |||
T8209 |
Saikosaponin b3
柴胡皂苷b3 |
Others | Others |
Saikosaponin b3 是从 Bupleurum falcatum L. 的根中分离得到的。Saikosaponin b3 抑制 ACTH 诱导的脂肪细胞中的脂肪分解并具有镇痛作用。 | |||
T8210 |
Saikosaponin B4
|
Others | Others |
Saikosaponin B4 是一种柴胡皂苷,分离自柴胡的根。Saikosaponin B4选择性地抑制 ACTH 诱导的脂解作用。 | |||
TN2170 |
Saikosaponin G
|
Others | Others |
Saikosaponin G is a natural product | |||
TN6859 |
Saikogenin F
(1S,2S,4S,5R,8R,9R,10S,13S,14R,17S,18R)-9-(hydroxymethyl)-4,5,9,13,20,20-hexamethyl-24-oxahexacyclo[15.5.2.01,1?.0?,1?.0?,1?.0?,13]tetracos-15-ene-2,10-diol |
Others | Others |
Saikogenin F ((1S,2S,4S,5R,8R,9R,10S,13S,14R,17S,18R)-9-(hydroxymethyl)-4,5,9,13,20,20-hexamethyl-24-oxahexacyclo[15.5.2.01,1?.0?,1?.0?,1?.0?,13]tetracos-15-ene-2,10-diol) 是一种具有抗癌活性的天然产物。 | |||
TN2172 | Saikosaponin I | Antifection | Microbiology/Virology |
Saikosaponin I shows strong inhibition activity against influenza virus WSN33. | |||
TN2171 | Saikosaponin H | Others | Others |
Saikosaponin H is a natural product from Bupleurum chinense. | |||
T8174 |
Saikosaponin F
柴胡皂苷F,柴胡皂苷 F |
Others | Others |
Saikosaponin F 是一种柴胡中的天然成分。 | |||
T41137 |
Prosaikogenin A
|
||
Prosaikogenin A, a triterpene saponin extracted from Clinopodium chinense, exhibits notable platelet aggregation promotion activity, indicated by an EC 50 value of 12.2 μM. | |||
TN1149 |
6''-O-acetylsaikosaponin A
|
Others | Others |
6''-O-Acetylsaikosaponin A 是一种分离自柴胡根中的乙酰柴胡皂苷,表现出一定的破骨细胞抑制活性。 | |||
T41138 |
Prosaikogenin H
|
||
Prosaikogenin H, an intestinal metabolite derived from saikosaponin, exhibits weak hemolytic activity. | |||
TN5968 |
6″-O-Acetylsaikosaponin b3
6″-O-乙酰基柴胡皂苷b3 |
||
6″-O-Acetylsaikosaponin b3 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5968,CAS号为 104109-34-4。 | |||
T83463 |
11(α)-Hydroxynepasaikosaponin k
|
||
11(α)-Hydroxynepasaikosaponin k(HOSSc)是B. scorzonerifolium Willd中的一种柴胡皂苷。 |