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Cat. No. Product Name Target Signaling Pathways
T2868 Evodiamine

d-Evodiamine,Isoevodiamine,(+)-Evodiamine,吴茱萸碱

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Evodiamine (d-Evodiamine) 是一种生物碱,从萱草的果实中分离得到,具有多种生物活性,包括抗炎,抗肥胖和抗肿瘤。
T2972 Rutaecarpine

Rutacarpine,吴茱萸次碱,Rhetine,Rutecarpine

COX Immunology/Inflammation; Neuroscience
Rutaecarpine (Rhetine) 是从槐木中提取的一种生物碱,是 COX-2的抑制剂,IC50值为0.28 μM。
T2S2335 Dehydroevodiamine

DHED,去氢吴茱萸碱

Others; NF-κB; COX; PGE Synthase; NO Synthase Immunology/Inflammation; Neuroscience; NF-κB; Others
Dehydroevodiamine (DHED) 是从吴茱萸中分离出的一种喹唑啉生物碱,可抑制 LPS 诱导的小鼠巨噬细胞中iNOS、COX-2、PGE2和NF-κB 的表达,对豚鼠心室肌细胞具有抗心律失常作用。
T8207 Evolitrine

Others Others
Evolitrine 是一种来源于Acronychia pedunculata、具有抗炎作用的物质。
TN1121 Evocarpine

Apoptosis; cAMP; Anti-infection; Calcium Channel; Antibacterial Apoptosis; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Evocarpine 是从 Evodiae fructus 分离得到的一种喹诺酮类生物碱,有抗细菌活性。它可通过电压依赖性钙通道抑制 Ca2+内流。
T5721 Dehydroevodiamine hydrochloride

AChE Neuroscience
Dehydroevodiamine hydrochloride 是分离自吴茱萸叶中,能够抑制 AChE。 它能够调节一氧化氮的产生,具有降压和神经保护作用。
TN1752 Hydroxyevodiamine

Others Others
Hydroxyevodiamine is a natural product
TN1173 1-Hydroxyrutaecarpine

Others Others
1-Hydroxyrutaecarpine exhibits cytotoxicities (ED50 values < 4 microg/mL) against P-388 or HT-29 cell lines in vitro.
TN1099 Dihydroevocarpine

MAO; P-gp; Antifection Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
Dihydroevocarpine shows potent anti-Helicobacter pylori activity with the minimum inhibitory concentration (MIC) value of 10-20 microg/ml. Dihydroevocarpine is a moderate modulator of p-glycoprotein (p-gp) activity; it shows more potent inhibitory effects against MAO-B compared to MAO-A.
TN1340 7beta-Hydroxyrutaecarpine

Others Others
7beta-Hydroxyrutaecarpine is a natural product from Euodia ruticarpa.

天然产物

Evodiamine
Cat.No: T2868
Synonym: d-Evodiamine,Isoevodiamine,(+)-Evodiamine,吴茱萸碱
Target: Prostaglandin Receptor
Rutaecarpine
Cat.No: T2972
Synonym: Rutacarpine,吴茱萸次碱,Rhetine,Rutecarpine
Target: COX
Dehydroevodiamine
Cat.No: T2S2335
Synonym: DHED,去氢吴茱萸碱
Target: Others, NF-κB, COX, PGE Synthase, NO Synthase
Evolitrine
Cat.No: T8207
Synonym:
Target: Others
Evocarpine
Cat.No: TN1121
Synonym:
Target: Apoptosis, cAMP, Anti-infection, Calcium Channel, Antibacterial
Dehydroevodiamine hydrochloride
Cat.No: T5721
Synonym:
Target: AChE
Hydroxyevodiamine
Cat.No: TN1752
Synonym:
Target: Others
1-Hydroxyrutaecarpine
Cat.No: TN1173
Synonym:
Target: Others
Dihydroevocarpine
Cat.No: TN1099
Synonym:
Target: MAO, P-gp, Antifection
7beta-Hydroxyrutaecarpine
Cat.No: TN1340
Synonym:
Target: Others
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