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12

抑制剂 & 化合物

3

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Cat. No. Product Name Target Signaling Pathways
T14981 Clobetasone butyrate

Glucocorticoid Receptor Endocrinology/Hormones
Clobetasone butyrate 是糖皮质类固醇,特别是在皮肤上,具有局部抗炎活性。它可用于改善皮质类固醇反应性症状,如特应性皮炎、牛皮癣。
T2548 Diflorasone

Glucocorticoid Receptor Endocrinology/Hormones
Diflorasone 是一种皮质类固醇激素受体激动剂,具有抗炎和免疫抑制作用。它可通过细胞膜扩散进入细胞,并与细胞质中的糖皮质激素受体结合。它用于研究湿疹、牛皮癣等皮肤病。
T1531 Mometasone furoate

糠酸莫美他松,糠酸莫米松,Sch32088

Glucocorticoid Receptor Endocrinology/Hormones
Mometasone furoate (Sch32088) 是糖皮质激素受体激动剂,具有抗炎和抗过敏作用。它是皮质固醇类试剂,动物模型中,可局部应用于气道炎症、慢性皮肤湿疹、哮喘。
T4966 Ufenamate

氟芬那酸丁酯,Flufenamic acid butyl ester,Butyl flufenamate,氟灭酸丁酯

Others Others
Ufenamate (Flufenamic acid butyl ester) 是一种基于邻氨基苯甲酸的抗炎药。它可用于皮肤疾病研究。
T4502 BISMUTH SUBGALLATE

次没食子酸铋,Dermatol Puder,Bismuth Gallate

Others Others
Bismuth subgallate (Dermatol Puder) 是一种止血剂,可作用于凝血因子 XII ,促使凝血级联的激活,改善纤维蛋白凝块的早期形成。
T77601 (2-{[2-(2-fluorophenoxy)ethyl]sulfanyl}-1H-benzimidazol-1-yl)acetic acid

GPR Endocrinology/Hormones; GPCR/G Protein
(2-{[2-(2-fluorophenoxy)ethyl]sulfanyl}-1H-benzimidazol-1-yl)acetic acid是一种前列腺素类 CRTH2拮抗剂,其IC50< 10 μM,可用于研究鼻炎、慢性阻塞性肺疾病、类风湿性关节炎、湿疹和结膜炎。
T0339 Resorcinol monoacetate

乙醯間二酚(1,3-苯二醇单乙酸酯 ),Resorcin monoacetate

Others Others
Resorcinol monoacetate (Resorcin monoacetate) 是一种防腐剂,及消毒剂,是用于合成其他药品的化学中间体。有用于痤疮,脂溢性皮炎,湿疹,银屑病和其它皮肤病的研究潜力。
T0500 Chloroxine

Capitrol,氯喔星

Antibacterial; Antibiotic Microbiology/Virology
Chloroxine (Capitrol) 是重要的 8-羟基喹啉衍生物之一,有抗细菌,抗真菌,抗原生动物和抗阿米巴虫活性,可研究肠道阿米巴病,还可研究头皮屑和头皮脂溢性皮炎。
T31443 Diethazine HCl

Diethazine hydrochloride,RP2987,Dinezine,RP 2987,RP-2987,Diparcol

Diethazine HCl is a topical corticosteroid product used to help treat eczema, psoriasis, and other skin conditions.
T14154 Alclometasone

7a-​Chloro-​16a-​methyl prednisolone

Alclometasone (7a-Chloro-16a-methyl prednisolone), a glucocorticoid, inhibits leukocytes from releasing pro-inflammatory mediators. It is effective in treating corticosteroid-responsive dermatoses such as atopic dermatitis, psoriasis, allergic dermatitis, and eczema [1].
T72279 Flurandrenolone Acetate

Flurandrenolone Acetate 是一种 Flurandrenolide 的衍生物,Flurandrenolone Acetate 是一种合成糖皮质激素类固醇,可用于湿疹和牛皮癣等皮肤病的研究。
T82074 Immune cell migration-IN-1

Immune cell migration-IN-1(compound 2)是一种抑制免疫细胞迁移的有效化合物,适用于干眼病、湿疹、皮炎和牛皮癣等疾病研究。

化合物

Clobetasone butyrate
Cat.No: T14981
Synonym:
Target: Glucocorticoid Receptor
Diflorasone
Cat.No: T2548
Synonym:
Target: Glucocorticoid Receptor
Mometasone furoate
Cat.No: T1531
Synonym: 糠酸莫美他松,糠酸莫米松,Sch32088
Target: Glucocorticoid Receptor
Ufenamate
Cat.No: T4966
Synonym: 氟芬那酸丁酯,Flufenamic acid butyl ester,Butyl flufenamate,氟灭酸丁酯
Target: Others
BISMUTH SUBGALLATE
Cat.No: T4502
Synonym: 次没食子酸铋,Dermatol Puder,Bismuth Gallate
Target: Others
(2-{[2-(2-fluorophenoxy)ethyl]sulfanyl}-1H-benzimidazol-1-yl)acetic acid
Cat.No: T77601
Synonym:
Target: GPR
Resorcinol monoacetate
Cat.No: T0339
Synonym: 乙醯間二酚(1,3-苯二醇单乙酸酯 ),Resorcin monoacetate
Target: Others
Chloroxine
Cat.No: T0500
Synonym: Capitrol,氯喔星
Target: Antibacterial, Antibiotic
Diethazine HCl
Cat.No: T31443
Synonym: Diethazine hydrochloride,RP2987,Dinezine,RP 2987,RP-2987,Diparcol
Target:
Alclometasone
Cat.No: T14154
Synonym: 7a-​Chloro-​16a-​methyl prednisolone
Target:
Flurandrenolone Acetate
Cat.No: T72279
Synonym:
Target:
Immune cell migration-IN-1
Cat.No: T82074
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4558 Trioxsalen

三甲沙林,Trimethylpsoralen,Trioxysalen,Trisoralen

DNA Alkylator/Crosslinker; DHFR Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Trioxsalen (Trioxysalen) 是一种呋喃香豆素和补骨脂素衍生物,与 UV-A 一起用于光疗治疗白癜风和手部湿疹。它是一种光化学 DNA 交联剂,可用于激光激活定位的基因组链间交联可视化。
TN2063 Physalin B

NSC-287088

Apoptosis; NF-κB; Akt; PI3K; Nrf2; NOD Apoptosis; Cytoskeletal Signaling; Immunology/Inflammation; NF-κB; PI3K/Akt/mTOR signaling
Physalin B 是茄科植物的主要活性化合物之一,具有广泛的生物活性,可用于治疗炎症湿疹和疱疹等疾病。Physalin B 通过激活 PI3K/Akt 通路抑制 NF-κB 和 NLRP3,从而改善脂多糖诱导的急性肺损伤造成的炎症反应。Physalin B 通过激活 Nrf2 通路抑制 PDGF-BB 诱导的 VSMC 增殖、迁移和表型转化。Physalin B 通过抑制 LAP2α-HDAC1 介导的胶质瘤相关癌基因 1 的去乙酰化和肝星状细胞活化来发挥抗肿瘤活性。
T40859 5-Hydroxy-8-methoxypsoralen

5-Hydroxyxanthotoxin,5-Hydroxy-8-methoxypsoralen

5-Hydroxy-8-methoxypsoralen (5-Hydroxyxanthotoxin) is a metabolite derived from Xanthotoxin, which acts as a potent tricyclic furocoumarin suicide inhibitor of CYP (cytochrome P-450). It is employed as an agent for the treatment of psoriasis, eczema, vitiligo, and certain cutaneous Lymphomas, in combination with phototherapy involving exposure to sunlight.

天然产物

Trioxsalen
Cat.No: T4558
Synonym: 三甲沙林,Trimethylpsoralen,Trioxysalen,Trisoralen
Target: DNA Alkylator/Crosslinker, DHFR
Physalin B
Cat.No: TN2063
Synonym: NSC-287088
Target: Apoptosis, NF-κB, Akt, PI3K, Nrf2, NOD
5-Hydroxy-8-methoxypsoralen
Cat.No: T40859
Synonym: 5-Hydroxyxanthotoxin,5-Hydroxy-8-methoxypsoralen
Target:
TargetMol Loading
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