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164

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T39387 Xanthine amine congener dihydrochloride

XAC dihydrochloride,Xanthine amine congener dihydrochloride

Xanthine amine congener dihydrochloride (XAC dihydrochloride), a potent antagonist for both Adenosine A1 and A2 receptors, exhibits IC50 values of 1.8 nM for A1 and 114 nM for A2 receptors. Additionally, it functions as a convulsant agent in mouse models.
T23535 Xanthine amine congener

Adenosine Receptor GPCR/G Protein; Neuroscience
Xanthine amine congener 是非选择性的腺苷受体拮抗剂,在小鼠中具有诱发惊厥的作用。
T7865 Danofloxacin

达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine

Others; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Danofloxacin (Danofloxacin free base) free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。
T8747 Levofloxacin hydrochloride

DNA gyrase; Topoisomerase DNA Damage/DNA Repair
Levofloxacin hydrochloride 是一种广谱的第三代氟喹诺酮类抗生素,是氧氟沙星的光学活性 L-异构体,具有抗菌活性。左氧氟沙星通过细菌细胞壁扩散并通过抑制 DNA 促旋酶(细菌拓扑异构酶 II)起作用,这是一种 DNA 复制、RNA 转录和细菌 DNA 修复所需的酶。 DNA 促旋酶活性的抑制导致细菌细胞生长受阻。
T6349L Sitafloxacin

DU6859,DU 6859,DU 6859A,Sitafloxacin anhydrous,DU-6859,DU6859A,DU-6859A,西他沙星

Sitafloxacin, a new generation of broad-spectrum oral fluoroquinolones, is highly effective against many Gram-positive, Gram-negative, and anaerobic clinical isolates (including strains resistant to other fluoroquinolones).
T3117 Marbofloxacin

马波沙星,Marbofloxacine,Zeniquin,Marbocyl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。
T1107 Sarafloxacin hydrochloride

Sarafloxacin HCl,盐酸沙拉沙星,A-56620 (hydrochloride),A-56620 HCl

Antibacterial; Antibiotic Microbiology/Virology
Sarafloxacin hydrochloride (A-56620 (hydrochloride)) 是一种抗菌化合物。
T1466 Nadifloxacin

OPC7251,那氟沙星

Antibacterial; Antibiotic Microbiology/Virology
Nadifloxacin (OPC7251) 是一种对粉刺有效的广谱氟喹诺酮类抗生素。
T7804 Garenoxacin mesylate hydrate

Garenoxacin mesylate [USAN],加雷沙星甲磺酸盐,BMS284756 (Mesylate hydrate)

Antibacterial Microbiology/Virology
Garenoxacin mesylate hydrate (Garenoxacin mesylate [USAN]) 是一种新型口服 des-fluoro(6) 喹诺酮,具有强抗菌活性,抗呼吸道病原体。
T5966 Hexaconazole

己唑醇,(-)-Hexaconazol

Reactive Oxygen Species; Antifungal Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Hexaconazole ((-)-Hexaconazol) 是一种广谱三唑类杀菌剂,通过抑制羊毛甾醇的细胞色素 P450 依赖性 14α-去甲基化来抑制麦角甾醇的生物合成,从而导致真菌细胞膜的破坏和细胞死亡。
T9319 Tosufloxacin

tosufloxacin tosilate,托氟沙星,Ozex,7-(3-Aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid

Others Others
Tosufloxacin (Ozex) 是一种喹诺酮类抗菌剂,是茶碱代谢的有效抑制剂。
T19805 Benoxacor

BRN-4190275,解草酮,BRN 4190275,BRN4190275

Others Others
Benoxacor (BRN-4190275) 是一种惰性农业化学品。它作为一种除草剂安全剂,可保护作物免受除草剂毒性。
T0985 Oxacillin sodium salt

苯唑西林,Oxacillin sodium,Oxabel

Antibacterial; Antibiotic Microbiology/Virology
Oxacillin sodium salt (Oxabel) 是一种青霉素类的窄谱β-内酰胺抗生素,用于耐药葡萄球菌感染。
T0717L Enoxacin

依诺沙星,NSC 629661,AT 2266,Pd107779,CI 919

DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Enoxacin (NSC-629661) 是一种可干扰DNA 复制的氟喹诺酮,抑制细菌 DNA 促旋酶 (IC50=126 µg/ml) 和拓扑异构酶 IV (IC50=26.5 µg/ml)。它是特异性癌症生长抑制剂,可有效抑制革兰氏阳性和阴性细菌。
T1293 Gatifloxacin

BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin (CG5501) 是一种具有广谱抗菌活性的氟喹诺酮类抗生素。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml) 和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml)。在动物模型中,它有抗细菌性结膜炎作用。
T1031 Cloxacillin sodium monohydrate

Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物

Antibacterial; Antibiotic Microbiology/Virology
Cloxacillin sodium monohydrate (Cloxacillin Sodium) 有抗菌作用,对Staphylococcus aureus25923 的最小抑菌浓度为256 mg/L。
T1001 Dicloxacillin Sodium hydrate

Dicloxacillin sodium salt monohydrate,双氯西林钠,Dicloxacillin sodium monohydrate

Antibacterial; Antibiotic Microbiology/Virology
Dicloxacillin Sodium hydrate 是一种青霉素类窄谱β内酰胺抗生素,可研究革兰氏阳性菌感染。
TQ0221 Rufloxacin hydrochloride

MF-934 hydrochloride,盐酸芦氟沙星

Antibacterial Microbiology/Virology
Rufloxacin hydrochloride (MF-934 hydrochloride) 是一种氟喹诺酮类抗菌剂,可抑制拓扑异构酶。 Rufloxacin hydrochloride 抑制人单核细胞中的 B 细胞分化。
T1640 Ciprofloxacin

Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Ciprofloxacin (Bay-09867) 是一种有高抗菌活性的氟喹诺酮类抗生素。
T16015 Maxacalcitol

马沙骨化醇,22-Oxacalcitriol

Others Others
Maxacalcitol (22-Oxacalcitriol) 是非血钙维生素 D3的一种类似物,是 VDR 样受体的配体。
T0425L Pefloxacin Mesylate Dihydrate

Pefloxacinium mesylate dihydrate,1589 RB,甲磺酸培氟沙星二水合物

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate Dihydrate (1589 RB) 是一种抗菌素,能通过抑制DNA 旋转酶阻断细菌DNA 复制。
T6349 Sitafloxacin Hydrate

西他沙星水合物,DU-6859a,DU6859a hydrate

Antibacterial; Antibiotic Microbiology/Virology
Sitafloxacin Hydrate (DU-6859a) 是一种口服有效的氟喹诺酮类抗生素,在体外可对抗广泛的革兰氏阳性和阴性细菌有活性。Sitafloxacin 可研究呼吸道感染和尿路感染。
T10987 Decarboxy Moxifloxacin

Others Others
Decarboxy Moxifloxacin 是一种莫西沙星的脱羧化合物。Moxifloxacin 是一种能够口服的 8-甲氧基喹诺酮类抗菌药物,可用于急性细菌性鼻窦炎,慢性支气管炎的急性细菌性加重和感染性肺炎。
T20774 Sarafloxacin

A-56620,A 56620,A56620,沙拉沙星

Antibacterial; Antibiotic Microbiology/Virology
Sarafloxacin (A56620) 对革兰氏阳性菌和革兰氏阴性菌具有抗菌活性。
T1451 Levofloxacin hydrate

左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin hydrate (Cravit hydrate) 是抗生素化合物,抑制细菌DNA 旋转酶活性。
T4063 Delafloxacin

ABT492,WQ-3034,德拉沙星,RX-3341

Antibacterial; Antibiotic Microbiology/Virology
Delafloxacin (WQ-3034) 是一种广谱氟喹诺酮类抗生素,抑制耐药性的金黄色葡萄球菌,肺炎链球菌和肺炎克雷伯菌。
T8142 Difloxacin hydrochloride

Difloxacin HCl,盐酸二氟沙星

Antibacterial; Antibiotic Microbiology/Virology
Difloxacin hydrochloride (Difloxacin HCl) 是一种广谱抗菌药物。它干扰 DNA 促旋酶和拓扑异构酶 IV 的活性,抑制细菌 DNA 促旋酶并显示出浓度依赖性的杀菌作用。
T5006 Flucloxacillin sodium

氟氯西林钠,floxacillin sodium

Antibacterial; Antibiotic Microbiology/Virology
Flucloxacillin sodium (floxacillin sodium) 是一种高活性抗生素,抑制革兰氏阳性和革兰氏阴性菌。
T9066 Merafloxacin

CI 934

SARS-CoV Microbiology/Virology
Merafloxacin (CI 934) 是一种氟喹诺酮类抗菌药物,也被确定为 SARS-CoV-2 的 1 PRF 抑制剂。它对革兰氏阳性菌和革兰氏阴性菌具有体外活性。
T5394 Prulifloxacin

AF 3012,Pruvel,NM441,普卢利沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Prulifloxacin (NM441) 是一种口服有效的氟喹诺酮抗生素 ,对革兰氏阳性和阴性细菌具有广泛活性。它是噻唑喹啉羧酸衍生物 Ulifloxacin 的前药。它有潜力用于下尿路感染和慢性支气管炎。
T9680 Irloxacin

Antibacterial Microbiology/Virology
Irloxacin 是一种口服活性的喹诺酮类抗菌剂,在酸性条件下具有更强大的活性。在体外,Irloxacin 对革兰氏阳性菌和革兰氏阴性菌都具有良好的抗菌谱。
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T0425 Pefloxacin Mesylate

Pefloxacinium mesylate,甲磺酸培氟沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate (Pefloxacinium mesylate) 是一种抗菌化合物,可抑制DNA 旋转酶阻断DNA 复制。
T0292 Orbifloxacin

CP-104354,奥比沙星

Antibacterial; Antibiotic Microbiology/Virology
Orbifloxacin (CP-104354) 是一种可用于犬类的氟喹诺酮类合成广谱抗生素。
T12649 Ibafloxacine

S25930,Ibafloxacin,R835

Antifungal Microbiology/Virology
Ibafloxacine (R835) 是一种氟喹诺酮类抗生素,专门用于兽类,对巴氏杆菌显示出良好的抑菌效果。
T8835 Tosufloxacin hydrochloride

A-61827 hydrochloride,盐酸妥舒沙星,T-3262 hydrochloride

Antibacterial Microbiology/Virology
Tosufloxacin hydrochloride 是一种氟喹诺酮类抗菌剂,用于治疗细菌感染。 Tosufloxacin hydrochloride 也是一种细菌 Topo(DNA 促旋酶,拓扑异构酶)抑制剂。
T1283 Clinafloxacin

克林沙星,PD 127391,CI-960,AM-1091

Antibacterial; Antibiotic Microbiology/Virology
Clinafloxacin (CI-960) 是一种高效广谱氟喹诺酮类抗生素,抑制革兰氏阳性、革兰氏阴性和厌氧病原体。它对金黄色葡萄球菌的 DNA 促旋酶和拓扑异构酶 IV 有抑制作用,IC50值分别为 0.92 µg/ml 和 1.62 µg/ml。
T0902 Ofloxacin

DL8280,菲宁达,Hoe-280,氧氟沙星,Floxin,Tarivid,Oxaldin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Ofloxacin (Oxaldin) 是可抑制细菌DNA 旋转酶的一种氟喹诺酮类抗生素。
T1492 Gemifloxacin mesylate

LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate

DNA gyrase; Topoisomerase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Gemifloxacin mesylate (Gemifloxacin mesylate) 是一种喹诺酮类口服广谱抗菌剂,可研究轻中度肺炎和慢性支气管炎的急性细菌性发作。
T1095 Sparfloxacin

AT-4140,PD 131501,Zagam,司帕沙星,CI-978

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Sparfloxacin (CI-978) 是一种氟喹诺酮类抗菌素。
T0717 Enoxacin hydrate

CI-919 hydrate,Enoxacin Sesquihydrate,依诺沙星半水合物,AT-2266 hydrate,依诺沙星倍半水合物

DNA gyrase; DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Enoxacin hydrate (AT-2266 hydrate) 是氟喹诺酮,可干扰DNA 复制,抑制细菌 DNA 促旋酶 (IC50=126 µg/ml) 和拓扑异构酶 IV (IC50=26.5 µg/ml)。它是特异性癌症生长抑制剂,抑制革兰氏阳性和阴性细菌。
T0331 Moxifloxacin hydrochloride

盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Moxifloxacin hydrochloride (BAY12-8039 HCl) 是一种口服有效的 8-甲氧基喹诺酮类抗菌药物,可研究感染性肺炎,急性细菌性鼻窦炎和慢性支气管炎的急性细菌性加重。
T0331L Moxifloxacin

Avelox,Moxeza,莫西沙星

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Moxifloxacin (Avelox) 是一种8-甲氧基喹诺酮类口服有效抗菌药物,用于急性细菌性鼻窦炎,慢性支气管炎的急性细菌性加重和感染性肺炎的研究。
T17254 Amifloxacin

Win49375,氨氟沙星

Antibacterial Microbiology/Virology
Amifloxacin (Win49375) 是有效的喹诺酮类抗菌剂。
T16789 Rosoxacin

罗索沙星,Acrosoxacin

Antibacterial; Antibiotic Microbiology/Virology
Rosoxacin (Acrosoxacin) 是具有口服活性的喹诺酮类抗生素,具有广谱的抗菌活性,抑制革兰氏阴性菌,包括淋病奈瑟氏球菌(MIC90=0.03 mg/ml)。它在尿路感染中有应用的潜能。
T0250 Ciprofloxacin monohydrochloride

Bay-09867 (hydrochloride),Ciprofloxacin HCl,盐酸环丙沙星,环丙沙星盐酸盐,Ciprofloxacin hydrochloride

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Ciprofloxacin monohydrochloride (Bay-09867 hydrochloride) 是一种高抗菌活性的氟喹诺酮类抗生素。
T16475 Pexacerfont

BMS-562086

CRFR GPCR/G Protein
Pexacerfont (BMS-562086) 是一种选择性的促肾上腺皮质激素释放因子 (CRF1) 受体拮抗剂,作用于人 CRF1 受体,IC50 为 6.1±0.6 nM。
T1733 Ciprofloxacin EP IMpurity A

Q-Acid,Fluoroquinolonic Acid,环丙羧酸,Ciprofloxacin Impurity A

Antibiotic Microbiology/Virology
Ciprofloxacin EP IMpurity A (Fluoroquinolonic Acid) 是一种抗生素和抗菌剂。
T6622 Oxacillin sodium monohydrate

苯唑西林钠一水合物,Stapenor monohydrate,苯唑青霉素钠,Sodium oxacillin monohydrate,Methicillin,Bactocill monohydrate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Oxacillin sodium monohydrate (Stapenor monohydrate) 是一种抗生素,可研究耐药性葡萄球菌感染,类似 Flucloxacillin。
T13231L Trovafloxacin mesylate

Others; DNA/RNA Synthesis; Topoisomerase; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Trovafloxacin是一种广谱氟喹诺酮类抗生素,可阻断 DNA 促旋酶 (DNA gyrase) 和拓扑异构酶 IV (topoisomerase IV) 的活性,也是一种有效的特异性 pannexin 1 通道抑制剂 (PANX1, IC50 = 4 μM)。

化合物

Xanthine amine congener dihydrochloride
Cat.No: T39387
Synonym: XAC dihydrochloride,Xanthine amine congener dihydrochloride
Target:
Xanthine amine congener
Cat.No: T23535
Synonym:
Target: Adenosine Receptor
Danofloxacin
Cat.No: T7865
Synonym: 达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine
Target: Others, DNA/RNA Synthesis, Antibacterial, Antibiotic
Levofloxacin hydrochloride
Cat.No: T8747
Synonym:
Target: DNA gyrase, Topoisomerase
Sitafloxacin
Cat.No: T6349L
Synonym: DU6859,DU 6859,DU 6859A,Sitafloxacin anhydrous,DU-6859,DU6859A,DU-6859A,西他沙星
Target:
Marbofloxacin
Cat.No: T3117
Synonym: 马波沙星,Marbofloxacine,Zeniquin,Marbocyl
Target: Topoisomerase, Antibacterial, Antibiotic
Sarafloxacin hydrochloride
Cat.No: T1107
Synonym: Sarafloxacin HCl,盐酸沙拉沙星,A-56620 (hydrochloride),A-56620 HCl
Target: Antibacterial, Antibiotic
Nadifloxacin
Cat.No: T1466
Synonym: OPC7251,那氟沙星
Target: Antibacterial, Antibiotic
Garenoxacin mesylate hydrate
Cat.No: T7804
Synonym: Garenoxacin mesylate [USAN],加雷沙星甲磺酸盐,BMS284756 (Mesylate hydrate)
Target: Antibacterial
Hexaconazole
Cat.No: T5966
Synonym: 己唑醇,(-)-Hexaconazol
Target: Reactive Oxygen Species, Antifungal
Tosufloxacin
Cat.No: T9319
Synonym: tosufloxacin tosilate,托氟沙星,Ozex,7-(3-Aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid
Target: Others
Benoxacor
Cat.No: T19805
Synonym: BRN-4190275,解草酮,BRN 4190275,BRN4190275
Target: Others
Oxacillin sodium salt
Cat.No: T0985
Synonym: 苯唑西林,Oxacillin sodium,Oxabel
Target: Antibacterial, Antibiotic
Enoxacin
Cat.No: T0717L
Synonym: 依诺沙星,NSC 629661,AT 2266,Pd107779,CI 919
Target: DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic
Gatifloxacin
Cat.No: T1293
Synonym: BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Cloxacillin sodium monohydrate
Cat.No: T1031
Synonym: Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物
Target: Antibacterial, Antibiotic
Dicloxacillin Sodium hydrate
Cat.No: T1001
Synonym: Dicloxacillin sodium salt monohydrate,双氯西林钠,Dicloxacillin sodium monohydrate
Target: Antibacterial, Antibiotic
Rufloxacin hydrochloride
Cat.No: TQ0221
Synonym: MF-934 hydrochloride,盐酸芦氟沙星
Target: Antibacterial
Ciprofloxacin
Cat.No: T1640
Synonym: Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867
Target: Topoisomerase, Antibacterial, Antibiotic
Maxacalcitol
Cat.No: T16015
Synonym: 马沙骨化醇,22-Oxacalcitriol
Target: Others
Pefloxacin Mesylate Dihydrate
Cat.No: T0425L
Synonym: Pefloxacinium mesylate dihydrate,1589 RB,甲磺酸培氟沙星二水合物
Target: Topoisomerase, Antibacterial, Antibiotic
Sitafloxacin Hydrate
Cat.No: T6349
Synonym: 西他沙星水合物,DU-6859a,DU6859a hydrate
Target: Antibacterial, Antibiotic
Decarboxy Moxifloxacin
Cat.No: T10987
Synonym:
Target: Others
Sarafloxacin
Cat.No: T20774
Synonym: A-56620,A 56620,A56620,沙拉沙星
Target: Antibacterial, Antibiotic
Levofloxacin hydrate
Cat.No: T1451
Synonym: 左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Delafloxacin
Cat.No: T4063
Synonym: ABT492,WQ-3034,德拉沙星,RX-3341
Target: Antibacterial, Antibiotic
Difloxacin hydrochloride
Cat.No: T8142
Synonym: Difloxacin HCl,盐酸二氟沙星
Target: Antibacterial, Antibiotic
Flucloxacillin sodium
Cat.No: T5006
Synonym: 氟氯西林钠,floxacillin sodium
Target: Antibacterial, Antibiotic
Merafloxacin
Cat.No: T9066
Synonym: CI 934
Target: SARS-CoV
Prulifloxacin
Cat.No: T5394
Synonym: AF 3012,Pruvel,NM441,普卢利沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Irloxacin
Cat.No: T9680
Synonym:
Target: Antibacterial
Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Pefloxacin Mesylate
Cat.No: T0425
Synonym: Pefloxacinium mesylate,甲磺酸培氟沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Orbifloxacin
Cat.No: T0292
Synonym: CP-104354,奥比沙星
Target: Antibacterial, Antibiotic
Ibafloxacine
Cat.No: T12649
Synonym: S25930,Ibafloxacin,R835
Target: Antifungal
Tosufloxacin hydrochloride
Cat.No: T8835
Synonym: A-61827 hydrochloride,盐酸妥舒沙星,T-3262 hydrochloride
Target: Antibacterial
Clinafloxacin
Cat.No: T1283
Synonym: 克林沙星,PD 127391,CI-960,AM-1091
Target: Antibacterial, Antibiotic
Ofloxacin
Cat.No: T0902
Synonym: DL8280,菲宁达,Hoe-280,氧氟沙星,Floxin,Tarivid,Oxaldin
Target: Topoisomerase, Antibacterial, Antibiotic
Gemifloxacin mesylate
Cat.No: T1492
Synonym: LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate
Target: DNA gyrase, Topoisomerase, Antibacterial
Sparfloxacin
Cat.No: T1095
Synonym: AT-4140,PD 131501,Zagam,司帕沙星,CI-978
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Enoxacin hydrate
Cat.No: T0717
Synonym: CI-919 hydrate,Enoxacin Sesquihydrate,依诺沙星半水合物,AT-2266 hydrate,依诺沙星倍半水合物
Target: DNA gyrase, DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic
Moxifloxacin hydrochloride
Cat.No: T0331
Synonym: 盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl
Target: Topoisomerase, Antibacterial, Antibiotic
Moxifloxacin
Cat.No: T0331L
Synonym: Avelox,Moxeza,莫西沙星
Target: Others, Antibacterial, Antibiotic
Amifloxacin
Cat.No: T17254
Synonym: Win49375,氨氟沙星
Target: Antibacterial
Rosoxacin
Cat.No: T16789
Synonym: 罗索沙星,Acrosoxacin
Target: Antibacterial, Antibiotic
Ciprofloxacin monohydrochloride
Cat.No: T0250
Synonym: Bay-09867 (hydrochloride),Ciprofloxacin HCl,盐酸环丙沙星,环丙沙星盐酸盐,Ciprofloxacin hydrochloride
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Pexacerfont
Cat.No: T16475
Synonym: BMS-562086
Target: CRFR
Ciprofloxacin EP IMpurity A
Cat.No: T1733
Synonym: Q-Acid,Fluoroquinolonic Acid,环丙羧酸,Ciprofloxacin Impurity A
Target: Antibiotic
Oxacillin sodium monohydrate
Cat.No: T6622
Synonym: 苯唑西林钠一水合物,Stapenor monohydrate,苯唑青霉素钠,Sodium oxacillin monohydrate,Methicillin,Bactocill monohydrate
Target: Others, Antibacterial, Antibiotic
Trovafloxacin mesylate
Cat.No: T13231L
Synonym:
Target: Others, DNA/RNA Synthesis, Topoisomerase, Antibacterial
Cat. No. Product Name Target Signaling Pathways
T5029 Oxaceprol

奥沙西罗,N-Acetyl-L-hydroxyproline,N-乙酰-L-4-羟基脯氨酸

Others Others
Oxaceprol (N-Acetyl-L-hydroxyproline) 是一种可口服的、具有显著抗炎作用的 L-脯氨酸衍生物,常用于研究骨关节炎和类风湿性关节炎。
T6567 Levofloxacin

Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin (Fluoroquinolone) 是合成的氟喹诺酮类抗生素,有抑制细菌DNA 旋转酶的超螺旋活性的作用,能阻止DNA 复制。
T8130 Ciprofloxacin hydrochloride monohydrate

Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan

Antibacterial; Antibiotic Microbiology/Virology
Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) 是一种具有高效抗菌活性的氟喹诺酮类抗生素。
TN6751 1-HEXACOSANOL

NPC1L1; AMPK Chromatin/Epigenetic; Membrane transporter/Ion channel; PI3K/Akt/mTOR signaling
1-HEXACOSANOL 激活 AMPK 和肝脏自噬并抑制 SREBP2,导致降胆固醇活性和肝脏脂肪变性的改善。
T8384 Gatifloxacin hydrochloride

AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。
T7095 Hexacosanoic acid

二十六酸,Cerotic acid

Endogenous Metabolite Metabolism
Hexacosanoic acid 是长链脂肪酸,与多种疾病有关(如肾上腺脑白质营养不良,肾上腺髓鞘病和动脉粥样硬化)。
T8046 Tosufloxacin tosylate hydrate

Tosufloxacin p-Toluenesulfonate Hydrate,A-61827 tosylate hydrate,对甲苯磺酸妥舒沙星水合物,T-3262 Tosylate Hydrate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Tosufloxacin tosylate hydrate (A-61827 tosylate hydrate) 是一个氟喹诺酮类抗菌剂。
T1306 Norfloxacin

氟哌酸,MK-0366,诺氟沙星

DNA gyrase; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Norfloxacin (MK-0366) 是广谱抗生素,能通过结合DNA 旋转酶抑制革兰氏阳性和阴性菌。
T1276 Danofloxacin mesylate

甲磺酸达氟沙星,CP 76136-27

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Danofloxacin mesylate (CP 76136-27) 是一种兽医用氟喹诺酮类抗菌素。
TN2753 2-Deacetyltaxachitriene A

Others Others
2-Deacetyltaxachitriene A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2753,CAS号为 214769-96-7。
TN7016 Hexacosane

Hexacosane is a natural product.
TN5102 Taxachitriene A

Others Others
Taxachitriene A is a natural product from the Chinese yew Taxus chinensis.
TN5104 Taxacin

Others Others
Taxacin shows strong inhibitory effects on platelet aggregation induced by arachidonic acid (IC(50):21.9 microM). Taxacin can suppress the superoxide generation induced by N-formyl-methionyl-leucyl-phenylalanine (fMLP) and arachidonic acid (AA) in a conce
TN2380 Glycerol 1-(26-hydroxyhexacosanoate)

Others Others
Glycerol 1-(26-hydroxyhexacosanoate) has weak activities antiplasmodial
TN5816 Glyceryl hexacosanoate

Glyceryl hexacosanoate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5816,CAS号为 127098-14-0。
TMA0245 Hexacosyl (E)-ferulate

Others Others
Hexacosyl (E)-ferulate displays significant antioxidant activity in the DPPH assay (RC50 = 0.0976 mg/mL). It also might be a chemotaxonomic marker in the genus Echinops.
TN5103 Taxachitriene B

Others Others
Taxachitriene B is a natural product from the Chinese yew Taxus chinensis.
TN3103 5-Acetyltaxachitriene A

Others Others
5-Acetyltaxachitriene A is a natural product from Taxus mairei.
TN2609 13-Deacetyltaxachitriene A

Others Others
13-Deacetyltaxachitriene A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2609,CAS号为 239800-99-8。

天然产物

Oxaceprol
Cat.No: T5029
Synonym: 奥沙西罗,N-Acetyl-L-hydroxyproline,N-乙酰-L-4-羟基脯氨酸
Target: Others
Levofloxacin
Cat.No: T6567
Synonym: Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin
Target: Topoisomerase, Antibacterial, Antibiotic
Ciprofloxacin hydrochloride monohydrate
Cat.No: T8130
Synonym: Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan
Target: Antibacterial, Antibiotic
1-HEXACOSANOL
Cat.No: TN6751
Synonym:
Target: NPC1L1, AMPK
Gatifloxacin hydrochloride
Cat.No: T8384
Synonym: AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐
Target: Topoisomerase, Antibacterial, Antibiotic
Hexacosanoic acid
Cat.No: T7095
Synonym: 二十六酸,Cerotic acid
Target: Endogenous Metabolite
Tosufloxacin tosylate hydrate
Cat.No: T8046
Synonym: Tosufloxacin p-Toluenesulfonate Hydrate,A-61827 tosylate hydrate,对甲苯磺酸妥舒沙星水合物,T-3262 Tosylate Hydrate
Target: Others, Antibacterial, Antibiotic
Norfloxacin
Cat.No: T1306
Synonym: 氟哌酸,MK-0366,诺氟沙星
Target: DNA gyrase, Topoisomerase, Endogenous Metabolite, Antibacterial, Antibiotic
Danofloxacin mesylate
Cat.No: T1276
Synonym: 甲磺酸达氟沙星,CP 76136-27
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
2-Deacetyltaxachitriene A
Cat.No: TN2753
Synonym:
Target: Others
Hexacosane
Cat.No: TN7016
Synonym:
Target:
Taxachitriene A
Cat.No: TN5102
Synonym:
Target: Others
Taxacin
Cat.No: TN5104
Synonym:
Target: Others
Glycerol 1-(26-hydroxyhexacosanoate)
Cat.No: TN2380
Synonym:
Target: Others
Glyceryl hexacosanoate
Cat.No: TN5816
Synonym:
Target:
Hexacosyl (E)-ferulate
Cat.No: TMA0245
Synonym:
Target: Others
Taxachitriene B
Cat.No: TN5103
Synonym:
Target: Others
5-Acetyltaxachitriene A
Cat.No: TN3103
Synonym:
Target: Others
13-Deacetyltaxachitriene A
Cat.No: TN2609
Synonym:
Target: Others
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