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72

抑制剂 & 化合物

18

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Cat. No. Product Name Target Signaling Pathways
T0396 Pipemidic acid

吡哌酸,Acido pipemidico

Antibacterial; Antibiotic Microbiology/Virology
Pipemidic acid (Acido pipemidico) 是一种新型抗菌剂,对革兰氏阴性菌和某些革兰氏阳性细菌具有活性,可研究肠道、泌尿和胆道感染。
T4201 Avibactam sodium

阿维巴坦,AVE-1330A,阿维巴坦钠,NXL-104

Antibacterial; Antibiotic Microbiology/Virology
Avibactam sodium (NXL-104) 是一种可逆的 β-内酰胺酶抑制剂,抑制 TEM-1,P99和KPC-2 β-内酰胺酶,IC50分别为8、80和38 nM。
T1293 Gatifloxacin

BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin (CG5501) 是一种具有广谱抗菌活性的氟喹诺酮类抗生素。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml) 和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml)。在动物模型中,它有抗细菌性结膜炎作用。
T20711 Hemipyocyanine

1-羟基吩嗪,528-71-2

Amylase Metabolism
Hemipyocyanine (528-71-2) 是一种 α-淀粉酶抑制剂。
T38173 Propargylcholine

Propargylcholine (bromide)

Antibacterial Microbiology/Virology
Propargylcholine (Propargylcholine (bromide)) 是一种炔烃修饰的胆碱类似物,在铜绿假单胞菌中 Dgc 酶催化的二甲基甘氨酸去甲基化水平上抑制胆碱分解代谢。
T65309 S-Methyl methanesulfonothioate

Antibacterial Microbiology/Virology
S-Methyl methanesulfonothioate 是一种生物原料,具有细胞毒性和潜在的抗菌活性,可用于研究铜绿假单胞菌感染。
T67912 PA3552-IN-1

PA3552-IN-1 是一种抗生素佐剂, 可以降低 PA3552 的表达,恢复 MDR 铜绿假单胞菌 DK2 菌株对 Polymyxin B 的敏感性。
T7495 Hexa-D-arginine

Others Others
Hexa-D-arginine 是稳定的furin 抑制剂,能够作用于 furin (Ki:106 nM)、PACE4 (Ki:580 nM)、PC1 (Ki:13.2 nM)。它在体外和体内均可阻断假单胞菌外毒素 A 和炭疽毒素的毒性。
T9119 SU0268

Others Others
SU0268 是有效的 8-8-氧鸟嘌呤 DNA 糖基化酶1的选择性抑制剂,具有调控铜绿假单胞杆菌感染免疫反应的能力。
T38137 3,5-Dimethylbenzaldehyde

Endogenous Metabolite; Antifungal Metabolism; Microbiology/Virology
3,5-Dimethylbenzaldehyde 具有广谱的抗菌活性,对枯草芽孢杆菌、白假丝酵母菌、大肠杆菌、铜绿假单胞菌、金黄色葡萄杆菌和肺炎链球菌具有抑制作用。
T77686 1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone

Antifungal Microbiology/Virology
1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone 具有广谱的抗真菌活性,对白色念珠菌、黑曲霉、铜绿假单胞菌、金黄色葡萄球菌等具有抑制作用。
T78226 Methyl 2-amino-5-bromobenzoate

Methyl 5-Bromoanthranilate

HCV Protease; Antifungal Microbiology/Virology; Proteases/Proteasome
Methyl 2-amino-5-bromobenzoate (Methyl 5-Bromoanthranilate) 是一种丙型肝炎病毒 NS5b RNA 聚合酶抑制剂,具有抗菌活性,可抑制铜绿假单胞菌感染,参与许多毒力因子的产生和生物膜的形成。
TP1050L Murepavadin acetate(944252-63-5 free base)

Antibacterial; Antibiotic Microbiology/Virology
Murepavadin acetate(944252-63-5 free base) 是一种有效且特异性的抗生素,用于治疗由铜绿假单胞菌引起的细菌感染。 Murepavadin acetate 靶向脂多糖转运蛋白 D。
T23858 WCK-5153

WCK 5153,WCK5153

Antibacterial Microbiology/Virology
WCK-5153 是 β-Lactamase 的增强剂和 PBP2 的抑制剂,对铜绿假单胞菌具有抗菌活性。 WCK-5153 可用于治疗由高度耐药的革兰氏阴性病原体引起的严重感染的研究。
T4998L Cefpodoxime (free acid)

Others Others
Cefpodoxime (free acid) 是一种口服的第三代头孢菌素抗生素。除铜绿假单胞菌、肠球菌和脆弱拟杆菌外,它对大多数革兰氏阳性和革兰氏阴性微生物均有效。
T22269 Benzyldodecyldimethylammonium Chloride Dihydrate

Antibacterial Microbiology/Virology
Benzyldodecyldimethylammonium chloride dihydrate 可以用作杀虫试剂,可以靶向耐药性细菌,如耐甲氧西林金黄色葡萄球菌、耐多药铜绿假单胞菌等,且具有浓度依赖性。
T7858 Ceftezole sodium

Celoslin,Falomesin,头孢替唑钠,Alomen

Anti-infection; Antibacterial; Antibiotic; Glucosidase Metabolism; Microbiology/Virology
Ceftezole sodium (Falomesin) 是一种广谱 cephem 抗生素,具有抑制多种革兰氏阳性菌和革兰氏阴性菌活性。它是一种α-葡萄糖苷酶抑制剂,具有体内抗糖尿病活性。
T60247 Diethylamine NONOate diethylammonium salt

NOC-18 Diethylamine,DEA NONOate diethylamine

Antibiotic Microbiology/Virology
Diethylamine NONOate diethylammonium salt (DEA NONOate diethylamine) 是一种一氧化氮供体,具有抗菌活性,是铜绿假单胞菌生物膜预形成生物膜的分散剂,可抑制大肠杆菌的生长。Diethylamine NONOate diethylammonium salt 可用于离体大鼠心脏的保存。
T124492 Imipenem

N-Formimidoyl thienamycin,MK0787

Antifungal Microbiology/Virology
Imipenem (MK0787) 是一种噻吩霉素衍生物,属于抗生素类,具有抗菌活性,对革兰氏阳性和革兰氏阴性菌具有部分的抑制作用。Imipenem 可用于研究碳青霉烯类非易感性感染和铜绿假单胞菌生物膜感染。
T13789 N-dodecanoyl-L-Homoserine lactone

C12-HSL,十二烷酰-L-高丝氨酸内酯

Others Others
N-dodecanoyl-L-Homoserine lactone (C12-HSL) 是群体感应 (QS) 信号分子的一种。它适配体可用于阻止群体感应,并能够阻碍铜绿假单胞菌 (Pseudomonas aeruginosa) 生物膜的形成。
T35449 α-(difluoromethyl)-DL-Arginine

DFMA,RMI 71897,α-(difluoromethyl)-DL-Arginine

Others Others
α-(difluoromethyl)-DL-Arginine (RMI 71897) 是一种酶激活的、不可逆的大肠杆菌(Ki = 800 μM)、铜绿假单胞菌和肺炎克雷伯菌精氨酸脱羧酶抑制剂。在0.01 mM 时,它已被证明可以防止渗透胁迫诱导的燕麦叶片细胞精氨酸脱羧酶活性和腐胺合成的增加。当α-(difluoromethyl)-DL-Arginine 与多种多胺类似物联用时,能在10 mM 的最低浓度下抑制克氏锥虫在哺乳动物宿主细胞中的生长,并在T 细胞受体α缺陷小鼠模型中阻止小锥虫的生长。
T33857 PA Autoinducer

3O-C12 autoinducer,PA-Autoinducer

PA Autoinducer is a Pseudomonas aeruginosa autoinducer.
T39983 SPR206 acetate

SPR206 acetate is a polymyxin analog that exhibits antibiotic activity against Gram-negative pathogens, including multidrug-resistant (MDR) variants. By interacting with the outer membrane of the bacterium, SPR206 acetate effectively combats bacterial infections. Notably, SPR206 acetate demonstrates significant efficacy with minimum inhibitory concentration (MIC) values of 0.125 mg/L against Pseudomonas aeruginosa Pa14 and Acinetobacter baumannii NCTC13301.
T13788 N-Butanoyl-DL-homoserine lactone

(Rac)-C4-HSL

Others Others
N-Butanoyl-DL-homoserine lactone aptamers blocks qurom sensing and inhibits biofilm formation in Pseudomonas aeruginosa.
T61368 FPI-1602

FPI-1602 is a β-lactamase inhibitor with strong antimicrobial activity against Pseudomonas aeruginosa, Escherichia coli, and Enterobacter species [1].
T39296 DS86760016

DS86760016 is a highly effective inhibitor of leucyl-tRNA synthetase (LeuRS), demonstrating potent activity against multidrug-resistant (MDR) Gram-negative bacteria including Escherichia coli, Klebsiella pneumoniae, and Pseudomonas aeruginosa. Notably, DS86760016 effectively inhibits LeuRS enzymes derived from Escherichia coli, Pseudomonas aeruginosa, and Acinetobacter baumannii, exhibiting IC50 values of 0.38 μM, 0.62 μM, and 0.16 μM, respectively.
T64422 Murepavadin

Murepavadin is a highly potent, specific, macrocycle Pseudomonas antibiotic for the treatment of bacterial infections caused by Pseudomonas aeruginosa..
T37912 Furanone C-30

Synthetic furanone bacterial quorum sensing inhibitor. Inhibits virulence factor expression in Pseudomonas aeruginosa and increases bacterial susceptibility to antibiotics in vitro. Also inhibits bacterial quorum sensing in vivo and promotes bacterial clearance in a mouse pulmonary infection model. Hentzer et al (2003) Attenuation of Pseudomonas aeruginosa virulence by quorum sensing inhibitors. EMBO J. 22 3803 PMID:12881415
T15142 Vebufloxacin

OPC7241,Flumenique,DM8966

Antibacterial Microbiology/Virology
Vebufloxacin (OPC-7251) shows potent antibacterial activity against gram-positive and -negative bacteria, including Staphylococcus aureus and Pseudomonas aeruginosa. It has potent activity characteristically against Propionibacterium acnes.
T77029 Gremubamab

Gremubamab (MEDI3902) 是一种人源化 IgG1kappa 抗PcrV/Psl 单克隆抗体。Gremubamab 结合 PA PcrV 蛋白和 Psl 胞外多糖 Gremubamab 具有研究铜绿假单胞菌感染的潜力。
T25136 Aztreonam lysine

Corus 1020,Corus1020,Corus-1020,Aztreonam lysinate

Aztreonam lysine is an inhaled anti-pseudomonal treatment for people who have pulmonary Pseudomonas aeruginosa infection with cystic fibrosis (CF).
T10944 D13-9001

Others Others
The KD values of D13-9001 in Escherichia coli and Pseudomonas aeruginosa were 1.15μM and 3.57μM, respectively. D13-9001 has antibiotic activity. It is an effective AcrB (AcrAB-TolC efflux pump subunit) and MexB (MexAB-OprM efflux pump subunit) inhibitor.
T61169 PqsR-IN-1

PqsR-IN-1 (Compound 18) is a potent inhibitor of PqsR, which is a transcriptional regulator involved in the quorum sensing mechanism of Pseudomonas aeruginosa. This compound effectively reduces the production of pyocyanin and exhibits minimal cytotoxicity [1].
T79004 ATP synthase inhibitor 2 TFA

ATP synthase inhibitor2 (Compound 22) TFA 为针对铜绿假单胞菌 (PA) ATP synthase 的抑制剂,具IC50值为10 μg/mL,在浓度达到128 μg/mL 时能够全面阻断铜绿假单胞菌 (PA) ATP的合成活性。
T61305 LasR-IN-3

LasR-IN-3, a chemical compound, acts as an inhibitor of LasR in Pseudomonas aeruginosa. It induces structural instability in LasR and causes complete dissociation of its functioning dimeric form [1].
T73531 SABA1

SABA1 具有抗菌活性,比如铜绿假单胞菌和大肠杆菌,其对大肠杆菌的IC50值为 4.0 µM。
T78537 Cefetamet pivoxyl

Ro 15-8075 free base

Antibiotic Microbiology/Virology
Cefetamet pivoxyl为头孢类抗生素,能抑制355种肠道病原体Keime、革兰氏阴性菌(ausgenommenPseudomonas aeruginosa)及嗜肺军团菌。
T62624 LpxA-IN-1

LpxA-IN-1 是一种新型的 UDP-N-乙酰氨基葡萄糖酰基转移酶 (LpxA)抑制剂(IC502 nM)。LpxA-IN-1 具有抑制 Pseudomonas aeruginosa(MIC 8 μg/mL)的活性。
T77184 Rivabazumab

Rivabazumab 是一种抗铜绿假单胞菌 pcrV 重组抗体。
T82944 ATP Synthesis-IN-2

ATP Synthesis-IN-2 (Compound 5) 是一种有效的ATP合成活性抑制剂,对Pseudomonas aeruginosa (PA) 表现出抗菌活性,其IC50值为0.7 μg/mL。
T68438 APO-6619

APO-6619 is an iron chelator which was shown to inhibit growth of the following bacterial strains: Acinetobacter baumannii, Pseudomonas aeruginosa, Staphylococcus aureus, Klebsiella pneumoniae, and Escherichia coli. APO-6619 may be useful as a non-traditional treatment of bacterial infections.
T60610 LasR-IN-4

LasR-IN-4 是 LasR 的有效抑制剂,可抑制铜绿假单胞菌及其生物膜的形成、绿脓素和鼠李糖脂的产生。
T80254 Elafin(human)

Elafin,亦称为ESI(elafin-specific inhibitor)或SKALP(skin anti-leucoprotease),为一种低分子量抑制剂,专一性地抑制肺部中性粒细胞中的HNE(人中性粒细胞弹性蛋白酶)和proteinase 3。同时,Elafin对Pseudomonas aeruginosa和Staphylococcus aureus亦具有抗生素效果。
T80527 D-K6L9

D-K6L9表现出针对囊性纤维化患者中的P. aeruginosa具有抗菌(antimicrobial)及抗生物膜效应,能稳定抵抗囊性纤维化痰中的蛋白酶降解,且不诱发细菌耐药性。
TP1638 OV-1, sheep

This alpha-helical antimicrobial OV-1 ovispirin peptide derived from SMAP29 peptide.It was found to inhibit several antibiotic-resistant bacterial strains including mucoid and nonmucoid Pseudomonas aeruginosa.
T61353 PqsR-IN-2

PqsR-IN-2 (Compound 19) is a highly potent inhibitor of PqsR, the transcriptional regulator responsible for quorum sensing in Pseudomonas aeruginosa. It effectively suppresses pyocyanin production without causing significant cytotoxicity, making it a promising compound for therapeutic applications [1].
T64315 VP-4509

VP-4509 是一种抗耐甲氧西林金黄色葡萄球菌 (MRSA) 剂 (MIC: 49.3 μM)。VP-4509 对革兰氏阴性细菌铜绿假单胞菌 (ATCC9027) 表现出高抗菌效果。
T77185 Rivabazumab pegol

Rivabazumab pegol为II期聚乙二醇化Fab, 是针对PcrV蛋白的抗体, 用于研究慢性铜绿假单胞菌感染。
T78535 trans-Clopenthixol dihydrochloride

(E)-Clopenthixol dihydrochloride

Parasite Microbiology/Virology
trans-Clopenthixol ((E)-Clopenthixol) diHCl为一种抗生素,具备抗菌性质但不具有镇静效果。该化合物能够用于抑制体外铜绿假单胞菌与恶性疟原虫。
T61649 ATP synthase inhibitor 2

ATP synthase inhibitor2 是一个铜绿假单胞菌 (PA)ATP synthase 抑制剂 (IC50=10 μg/mL),在 128 μg/mL 时可完全抑制铜绿假单胞菌 (PA) 的 ATP 合成活性。

化合物

Pipemidic acid
Cat.No: T0396
Synonym: 吡哌酸,Acido pipemidico
Target: Antibacterial, Antibiotic
Avibactam sodium
Cat.No: T4201
Synonym: 阿维巴坦,AVE-1330A,阿维巴坦钠,NXL-104
Target: Antibacterial, Antibiotic
Gatifloxacin
Cat.No: T1293
Synonym: BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Hemipyocyanine
Cat.No: T20711
Synonym: 1-羟基吩嗪,528-71-2
Target: Amylase
Propargylcholine
Cat.No: T38173
Synonym: Propargylcholine (bromide)
Target: Antibacterial
S-Methyl methanesulfonothioate
Cat.No: T65309
Synonym:
Target: Antibacterial
PA3552-IN-1
Cat.No: T67912
Synonym:
Target:
Hexa-D-arginine
Cat.No: T7495
Synonym:
Target: Others
SU0268
Cat.No: T9119
Synonym:
Target: Others
3,5-Dimethylbenzaldehyde
Cat.No: T38137
Synonym:
Target: Endogenous Metabolite, Antifungal
1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)-pyridinone
Cat.No: T77686
Synonym:
Target: Antifungal
Methyl 2-amino-5-bromobenzoate
Cat.No: T78226
Synonym: Methyl 5-Bromoanthranilate
Target: HCV Protease, Antifungal
Murepavadin acetate(944252-63-5 free base)
Cat.No: TP1050L
Synonym:
Target: Antibacterial, Antibiotic
WCK-5153
Cat.No: T23858
Synonym: WCK 5153,WCK5153
Target: Antibacterial
Cefpodoxime (free acid)
Cat.No: T4998L
Synonym:
Target: Others
Benzyldodecyldimethylammonium Chloride Dihydrate
Cat.No: T22269
Synonym:
Target: Antibacterial
Ceftezole sodium
Cat.No: T7858
Synonym: Celoslin,Falomesin,头孢替唑钠,Alomen
Target: Anti-infection, Antibacterial, Antibiotic, Glucosidase
Diethylamine NONOate diethylammonium salt
Cat.No: T60247
Synonym: NOC-18 Diethylamine,DEA NONOate diethylamine
Target: Antibiotic
Imipenem
Cat.No: T124492
Synonym: N-Formimidoyl thienamycin,MK0787
Target: Antifungal
N-dodecanoyl-L-Homoserine lactone
Cat.No: T13789
Synonym: C12-HSL,十二烷酰-L-高丝氨酸内酯
Target: Others
α-(difluoromethyl)-DL-Arginine
Cat.No: T35449
Synonym: DFMA,RMI 71897,α-(difluoromethyl)-DL-Arginine
Target: Others
PA Autoinducer
Cat.No: T33857
Synonym: 3O-C12 autoinducer,PA-Autoinducer
Target:
SPR206 acetate
Cat.No: T39983
Synonym:
Target:
N-Butanoyl-DL-homoserine lactone
Cat.No: T13788
Synonym: (Rac)-C4-HSL
Target: Others
FPI-1602
Cat.No: T61368
Synonym:
Target:
DS86760016
Cat.No: T39296
Synonym:
Target:
Murepavadin
Cat.No: T64422
Synonym:
Target:
Furanone C-30
Cat.No: T37912
Synonym:
Target:
Vebufloxacin
Cat.No: T15142
Synonym: OPC7241,Flumenique,DM8966
Target: Antibacterial
Gremubamab
Cat.No: T77029
Synonym:
Target:
Aztreonam lysine
Cat.No: T25136
Synonym: Corus 1020,Corus1020,Corus-1020,Aztreonam lysinate
Target:
D13-9001
Cat.No: T10944
Synonym:
Target: Others
PqsR-IN-1
Cat.No: T61169
Synonym:
Target:
ATP synthase inhibitor 2 TFA
Cat.No: T79004
Synonym:
Target:
LasR-IN-3
Cat.No: T61305
Synonym:
Target:
SABA1
Cat.No: T73531
Synonym:
Target:
Cefetamet pivoxyl
Cat.No: T78537
Synonym: Ro 15-8075 free base
Target: Antibiotic
LpxA-IN-1
Cat.No: T62624
Synonym:
Target:
Rivabazumab
Cat.No: T77184
Synonym:
Target:
ATP Synthesis-IN-2
Cat.No: T82944
Synonym:
Target:
APO-6619
Cat.No: T68438
Synonym:
Target:
LasR-IN-4
Cat.No: T60610
Synonym:
Target:
Elafin(human)
Cat.No: T80254
Synonym:
Target:
D-K6L9
Cat.No: T80527
Synonym:
Target:
OV-1, sheep
Cat.No: TP1638
Synonym:
Target:
PqsR-IN-2
Cat.No: T61353
Synonym:
Target:
VP-4509
Cat.No: T64315
Synonym:
Target:
Rivabazumab pegol
Cat.No: T77185
Synonym:
Target:
trans-Clopenthixol dihydrochloride
Cat.No: T78535
Synonym: (E)-Clopenthixol dihydrochloride
Target: Parasite
ATP synthase inhibitor 2
Cat.No: T61649
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5780 HYPOCRELLIN B

Apoptosis; Parasite; Antifungal Apoptosis; Microbiology/Virology
Hypocrellin B 是从真菌Hypocrella bambusae 和Shiraia bambusicola 中分离得到的一种感光颜料,可用于癌症光动力研究。它是一个凋亡诱导剂,还拥有抗菌和抗利什曼活性。
T2904 Sclareolide

香紫苏内酯,Norambreinolide

Others; Antibacterial Microbiology/Virology; Others
Sclareolide (Norambreinolide) 是一种从Salvia sclarea 的花中分离得到的天然产物,具有抗菌和细胞毒性作用。
TQ0251 (Z)-2-decenoic acid

(Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid

Others Others
(Z)-2-decenoic acid (cis-dec-2-enoic acid) 是一种由铜绿假单胞菌产生的不饱和脂肪酸。它能够诱导一系列革兰氏阴性细菌(包括铜绿假单胞菌)和革兰氏阳性细菌形成的生物膜发生分散反应。它能够抑制生物膜发育。
T8384 Gatifloxacin hydrochloride

AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。
T38373 2-heptyl-3-hydroxy-4(1H)-Quinolone

2-heptyl-3-hydroxy-4(1H)-Quinolone,PQS,Pseudomonas Quinolone Signal

Others Others
2-heptyl-3-hydroxy-4(1H)-Quinolone (Pseudomonas Quinolone Signal) 是一种铜绿假单胞菌为应对细胞密度增加而产生的一种法定人数感应信号分子。 它增加了铜绿假单胞菌中lasB 基因的表达,增加代谢物焦蓝蛋白和凝集素PA-IL 的分泌,以及增加铜绿假单胞菌种群的生物膜生产。当使用浓度为40 μM 时,它还会降低铜绿假单胞菌生长介质中的铁含量,并在硫酸铁溶液中充当一种铁螯合剂。
T4816 6-Hydroxynicotinic acid

6-Hydroxypyridine-3-carboxylic acid,6-羟基烟酸,2-Hydroxy-5-pyridinecarboxylic acid

Others; Endogenous Metabolite Metabolism; Others
6-Hydroxynicotinic acid (6-Hydroxypyridine-3-carboxylic acid) 用于核磁共振波谱或气相色谱-质谱法诊断尿路感染中的铜绿假单胞菌。在引起尿液感染的常见细菌中,只有铜绿假单胞菌从烟酸中产生6-羟基烟酸。
T5707 3-O-Methylgalangin

3-Methylgalangin,GALANGIN-3-METHYLETHER,高良姜素 3-O-甲醚,高良姜素-3-甲醚

Antibacterial Microbiology/Virology
3-O-Methylgalangin (GALANGIN-3-METHYLETHER) 是一种来源于高良姜根茎的天然黄酮,具有抗菌活性,抑制胰腺脂肪酶。
TN2111 Prunin

Naringenin 7-0-glucoside,柚皮素-7-O-葡萄糖苷

Phosphatase; Anti-infection; Virus Protease Metabolism; Microbiology/Virology
Prunin (Naringenin 7-0-glucoside) 是一种人肠道病毒 A71 抑制剂。它抑制蛋白酪氨酸磷酸酶 1B,IC50值为 5.5 μM。
T37341 N-Acetyltyramine

Antibacterial Microbiology/Virology
N-Acetyltyramine 是一种群体感应抑制剂,由溶藻弧菌 M3-10 产生。N-Acetyltyramine 可以抑制C. violaceumATCC 12472 的群体感应。它可以逆转阿霉素耐药白血病 P388 细胞的耐药性。
T8066 Sulbenicillin disodium

磺苄西林钠,Sulbenicillin Sodium

Antibacterial; Antibiotic Microbiology/Virology
Sulbenicillin disodium (Sulbenicillin Sodium) 是 Sulbenicillin 的二钠盐。Sulbenicillin 是一种青霉素抗生素,对Pseudomonas aeruginosa 的许多粘液型和非粘液型菌株具有抗菌活性。
TN3861 Dihydropinosylvin

山药

Anti-infection Microbiology/Virology
Dihydropinosylvin 是一种植物抗毒素,对枝孢枝孢菌、Botryodiplodia theobromae、黑曲霉和石化青霉具有抗真菌活性,对蜡状芽孢杆菌、金黄色葡萄球菌、铜绿假单胞菌和大肠杆菌也有很强的抗菌活性。双色高粱幼苗的种子和根伸长。
TN1203 2,3,8-Tri-O-methylellagic acid

2,3,8-三邻甲基鞣花酸

Antifection Microbiology/Virology
2,3,8-tri-O-Methyl ellagic acid has antimicrobial activity agaist Vibro cholera, Staphylococcus aureus, Klebsiella pneumoniae, Pseudomonas aeruginosa, Bacillus cereus, Escherichia coli.
TN4851 Pterodondiol

Antifection Microbiology/Virology
Pterodondiol has moderate activity against bacteria including Staphylococcus aureus, Pseudomonas aeruginosa, Bacillus subtilis, Mycobacteium phlei and Bacillus circulans.
TN4579 Monomethylsulochrin

Antifection Microbiology/Virology
Monomethylsulochrin shows antimicrobial activity against Escherichia coli, Pseudomonas aeruginosa, Bacillus subtilis and Staphylococcus aureus. It shows moderately inhibitory effects on the human bacterial pathogen Helicobacter pylori with the MIC value of 28.9+/-0.1 microM.
TN4852 Pterodontic acid

Antifection Microbiology/Virology
Pterodontic acid and pterodondiol showed moderate activity against bacteria including Staphylococcus aureus, Pseudomonas aeruginosa, Bacillus subtilis.
TN5229 Vibralactone B

Antifection Microbiology/Virology
Vibralactone B shows antibacterial activity, it can inhibit significantly the growth of E. coli and Pseudomonas aeruginosa, with MBC values of 50 and 100 ug/mL, respectively.
TN2032 Pachypodol

霍香黃酮醇

Antifection Microbiology/Virology
Pachypodol has antibacterial and antifungal activities against Bacillus subtilis, Staphylococcus aureus, Staphylococcus faecalis, Echerichia coli, Pseudomonas aeruginosa, Candida albicans, Candida krusei and Candida galabrata.
T72250 4aα,7α,7aα-Nepetalactone

4aα,7α,7aα-Nepetalactone 具有抗菌 (antibacterial) 活性,抑制Escherichia coli,Pseudomonas aeruginosa,Staphylococcus aureus,Salmonella typhi 和Enterococcus faecalis。

天然产物

HYPOCRELLIN B
Cat.No: T5780
Synonym:
Target: Apoptosis, Parasite, Antifungal
Sclareolide
Cat.No: T2904
Synonym: 香紫苏内酯,Norambreinolide
Target: Others, Antibacterial
(Z)-2-decenoic acid
Cat.No: TQ0251
Synonym: (Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid
Target: Others
Gatifloxacin hydrochloride
Cat.No: T8384
Synonym: AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐
Target: Topoisomerase, Antibacterial, Antibiotic
2-heptyl-3-hydroxy-4(1H)-Quinolone
Cat.No: T38373
Synonym: 2-heptyl-3-hydroxy-4(1H)-Quinolone,PQS,Pseudomonas Quinolone Signal
Target: Others
6-Hydroxynicotinic acid
Cat.No: T4816
Synonym: 6-Hydroxypyridine-3-carboxylic acid,6-羟基烟酸,2-Hydroxy-5-pyridinecarboxylic acid
Target: Others, Endogenous Metabolite
3-O-Methylgalangin
Cat.No: T5707
Synonym: 3-Methylgalangin,GALANGIN-3-METHYLETHER,高良姜素 3-O-甲醚,高良姜素-3-甲醚
Target: Antibacterial
Prunin
Cat.No: TN2111
Synonym: Naringenin 7-0-glucoside,柚皮素-7-O-葡萄糖苷
Target: Phosphatase, Anti-infection, Virus Protease
N-Acetyltyramine
Cat.No: T37341
Synonym:
Target: Antibacterial
Sulbenicillin disodium
Cat.No: T8066
Synonym: 磺苄西林钠,Sulbenicillin Sodium
Target: Antibacterial, Antibiotic
Dihydropinosylvin
Cat.No: TN3861
Synonym: 山药
Target: Anti-infection
2,3,8-Tri-O-methylellagic acid
Cat.No: TN1203
Synonym: 2,3,8-三邻甲基鞣花酸
Target: Antifection
Pterodondiol
Cat.No: TN4851
Synonym:
Target: Antifection
Monomethylsulochrin
Cat.No: TN4579
Synonym:
Target: Antifection
Pterodontic acid
Cat.No: TN4852
Synonym:
Target: Antifection
Vibralactone B
Cat.No: TN5229
Synonym:
Target: Antifection
Pachypodol
Cat.No: TN2032
Synonym: 霍香黃酮醇
Target: Antifection
4aα,7α,7aα-Nepetalactone
Cat.No: T72250
Synonym:
Target:
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