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6

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T22889 KF38789

KF 38789

Others Others
KF38789 特异性的抑制P-selectinPSGL-1结合。它对 U937 细胞与 P-selectin 免疫球蛋白 G 嵌合蛋白 (P-selectin-Ig) 的结合具有抑制作用 (IC50:1.97 μM) 。
T16676 PSI-697

P-Selectin Inhibitor

Others Others
PSI-697 is an inhibitor of oral P-selectin (IC50: 125 μM).
T1893 Parmodulin 2

ML 161

Protease-activated Receptor GPCR/G Protein
Parmodulin 2 (ML 161) 是一种蛋白酶激活受体 1(PAR1) 变构抑制剂,IC50为 0.26 μM。它是蛋白酶激活受体 1 (PAR1) 介导的血小板活化的抑制剂,可以抑制体外血小板聚集和体内血小板血栓形成。
T14573 Bimosiamose disodium

TBC-1269Z

Integrin Cytoskeletal Signaling
Bimosiamose disodium has anti-inflammatory effects[1]. Bimosiamose disodium (TBC-1269Z) is a nonoligosaccharide pan-selectin inhibitor with IC50s of 88 μM, 20 μM, and 86 μM for E-selectin, P-selectin, and L-selectin, respectively.
T24144 HMCEF

HMCEF is a P-selectin inhibitor that acts by intercalating into calf thymus DNA, cutting off DNA pBR22. It also inhibits the proliferation of cancer cells.
T39121 Odatroltide

DHDMIQK(KAP),Odatroltide

Odatroltide is a nanoscale P-selectin inhibitor that serves as a nano-delivery system for 6,7-dihydroxyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid and KPAK to specifically target the thrombus.

化合物

KF38789
Cat.No: T22889
Synonym: KF 38789
Target: Others
PSI-697
Cat.No: T16676
Synonym: P-Selectin Inhibitor
Target: Others
Parmodulin 2
Cat.No: T1893
Synonym: ML 161
Target: Protease-activated Receptor
Bimosiamose disodium
Cat.No: T14573
Synonym: TBC-1269Z
Target: Integrin
HMCEF
Cat.No: T24144
Synonym:
Target:
Odatroltide
Cat.No: T39121
Synonym: DHDMIQK(KAP),Odatroltide
Target:
Cat. No. Product Name Target Signaling Pathways
T3S0645 N-trans-Feruloyltyramine

Feruloyltyramine,N-Feruloyltyramine,Moupinamide,N-反式阿魏酰酪胺

Others; COX Immunology/Inflammation; Neuroscience; Others
N-trans-Feruloyltyramine (Feruloyltyramine) 是从大麻中分离得到的一种生物碱,是COX1和COX2的抑制剂,具有抗氧化和抗炎活性。
T4S0498 Glaucocalyxin A

蓝萼甲素,Wangzaozin B,Leukamenin F

Apoptosis; Akt; Caspase; PI3K Apoptosis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Glaucocalyxin A (Leukamenin F) 是来自日本黑纹病菌的一种对映型月桂基二萜,具有抗肿瘤作用。它通过调节PI3K/Akt 信号通路抑制 GLI1 的核易位,诱导骨肉瘤凋亡。

天然产物

N-trans-Feruloyltyramine
Cat.No: T3S0645
Synonym: Feruloyltyramine,N-Feruloyltyramine,Moupinamide,N-反式阿魏酰酪胺
Target: Others, COX
Glaucocalyxin A
Cat.No: T4S0498
Synonym: 蓝萼甲素,Wangzaozin B,Leukamenin F
Target: Apoptosis, Akt, Caspase, PI3K
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