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5

抑制剂 & 化合物

25

天然产物

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Cat. No. Product Name Target Signaling Pathways
T12017 Methyllycaconitine citrate

MLA

AChR Neuroscience
Methyllycaconitine citrate (MLA) 是一种可穿过血脑屏障的 α7 神经元烟碱乙酰胆碱受体(α7nAChR)拮抗剂,可用于研究神经系统疾病。
T131546 N-Deacetyllapaconitine

N-Deacetyllapaconitine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131546。
T2806L Lappaconitine HCl

Lappaconitine hydrochloride

Lappaconitine HCl is a centrally acting non-opioid analgesic and class-I antiarrhythmic. It acts by binding to the site-2 receptor and irreversibly blocking hH1 sodium channels.
T131453 Yunaconitine (Vilmorrianine B and other names)

Yunaconitine (Vilmorrianine B and other names) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131453。
T131508 Pseudaconitine

Pseudaconitine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131508。

化合物

Methyllycaconitine citrate
Cat.No: T12017
Synonym: MLA
Target: AChR
N-Deacetyllapaconitine
Cat.No: T131546
Synonym:
Target:
Lappaconitine HCl
Cat.No: T2806L
Synonym: Lappaconitine hydrochloride
Target:
Yunaconitine (Vilmorrianine B and other names)
Cat.No: T131453
Synonym:
Target:
Pseudaconitine
Cat.No: T131508
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN4711 Onitin

Others Others
Onitin shows super-oxide and DPPH free radical scavenging effects.It also exhibits hepatoprotective activity on tacrine-induced cytotoxicity in human liver-derived Hep G2 cells.
TN5342 Onitin 2'-O-glucoside

Onitin 2'-O-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5342,CAS号为 76947-60-9。
T5S1891 Flaconitine

乙酰乌头碱,3-Acetylaconitine,Acetylaconitine

Others; NF-κB NF-κB; Others
Flaconitine (Acetylaconitine) 是一种 NF-κB 抑制剂,是一种生物碱。
T3021 Bulleyaconitine A

草乌甲素,Bulleyaconi cine A

Sodium Channel Membrane transporter/Ion channel
Bulleyaconitine A (Bulleyaconi cine A) 是一种分离自乌头属植物的抗炎活性化合物,也可用于缓解疼痛的研究。
TN3273 8-Deacetylyunaconitine

Others Others
8-Deacetylyunaconitine 是一种源自乌头的二萜生物碱。
T6560 Lappaconitine hydrobromide

氢溴酸高乌甲素,Lappaconite HBr,Allapinine

Others Others
Lappaconitine hydrobromide (Allapinine) 是天然生物碱类化合物,具有抗心律失常作用。
T6S0630 Hypaconitine

P450; TNF Apoptosis; Metabolism
Hypaconitine 是从乌头属种分离的一种高毒性成分,可研究风湿病。
T4S1876 3-Deoxyaconitine

Sodium Channel Membrane transporter/Ion channel
3-Deoxyaconitine 是一种二萜类生物碱,对钠离子通道有激活作用。
T5S1889 Yunaconitine

Guayewuanine B,滇乌头碱

Others Others
Yunaconitine (Guayewuanine B) 是一种乌头类生物碱,具有剧毒。
T5765 ranaconitine

羟基高乌碱,7-羟基高乌甲素

Apoptosis; Others Apoptosis; Others
Ranaconitine 是从高乌头中分离得到的一种二萜生物碱,具有心脏毒性。
T2806 Lappaconitine

高乌甲素,(+)-Lappaconitine

P2X Receptor; Sodium Channel Membrane transporter/Ion channel; Neuroscience
Lappaconitine ((+)-Lappaconitine) 是从高乌头中分离得到的一种天然产物,可用于缓解疼痛的研究。
T6S0627 Mesaconitine

新乌碱,新乌头碱;中乌头碱

TNF Apoptosis
Mesaconitine 是乌头属植物的一种主要活性成分,通过循环 AMP 和刺激中枢 β-肾上腺素能系统具有镇痛活性,还有抗炎活性。
TN1647 Foresaconitine

Others Others
Foresaconitine is a natural product
T24198 Jesaconitine

BRN0075405,BRN-0075405,BRN 0075405,Diesaconitine

Jesaconitine is an Aconitine analog.
T83445 16-Epipyromesaconitine

16-Epipyromesaconitine为通过Mesaconitine热解产生的天然产物。
TN2919 3-Acetylyunaconitine

Others Others
3-Acetylyunaconitine is a natural product from Aconitum episcopale Levl.
TN4830 Prionitin

Others Others
Prionitin is a natural product from Salvia prionitis Hance.
TN6341 Sachaconitine

黄草乌碱丁,Vilmorrianine D

Sachaconitine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6341,CAS号为 1361-02-0。
TN6115 Lipoaconitine

Lipoaconitine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6115,CAS号为 81941-14-2。
T83455 13-Dehydroxyindaconitine

13-Dehydroxyindaconitine是一种天然生物碱,表现出抗氧化特性。
T6S1879 Indaconitine

Others Others
Indaconitine 可分离自乌头植物根茎。
T11890 Ludaconitine

Others Others
Ludaconitine, isolated from Aconitum spicatum (Bruhl) Stapf, exhibits antileishmanial activity with an IC50 of 36.10 μg/mL.
TN6114 Lipodeoxyaconitine

Lipodeoxyaconitine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6114,CAS号为 244190-83-8。
TN6342 14-O-Acetylsachaconitine

14-O-Acetylsachaconitine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6342,CAS号为 102719-98-2。
TN4713 Onitisin

5-HT Receptor GPCR/G Protein; Neuroscience
Onitisin, onitinoside and onitin can inhibit the contraction of isolated guinea-pig ileum.

天然产物

Onitin
Cat.No: TN4711
Synonym:
Target: Others
Onitin 2'-O-glucoside
Cat.No: TN5342
Synonym:
Target:
Flaconitine
Cat.No: T5S1891
Synonym: 乙酰乌头碱,3-Acetylaconitine,Acetylaconitine
Target: Others, NF-κB
Bulleyaconitine A
Cat.No: T3021
Synonym: 草乌甲素,Bulleyaconi cine A
Target: Sodium Channel
8-Deacetylyunaconitine
Cat.No: TN3273
Synonym:
Target: Others
Lappaconitine hydrobromide
Cat.No: T6560
Synonym: 氢溴酸高乌甲素,Lappaconite HBr,Allapinine
Target: Others
Hypaconitine
Cat.No: T6S0630
Synonym:
Target: P450, TNF
3-Deoxyaconitine
Cat.No: T4S1876
Synonym:
Target: Sodium Channel
Yunaconitine
Cat.No: T5S1889
Synonym: Guayewuanine B,滇乌头碱
Target: Others
ranaconitine
Cat.No: T5765
Synonym: 羟基高乌碱,7-羟基高乌甲素
Target: Apoptosis, Others
Lappaconitine
Cat.No: T2806
Synonym: 高乌甲素,(+)-Lappaconitine
Target: P2X Receptor, Sodium Channel
Mesaconitine
Cat.No: T6S0627
Synonym: 新乌碱,新乌头碱;中乌头碱
Target: TNF
Foresaconitine
Cat.No: TN1647
Synonym:
Target: Others
Jesaconitine
Cat.No: T24198
Synonym: BRN0075405,BRN-0075405,BRN 0075405,Diesaconitine
Target:
16-Epipyromesaconitine
Cat.No: T83445
Synonym:
Target:
3-Acetylyunaconitine
Cat.No: TN2919
Synonym:
Target: Others
Prionitin
Cat.No: TN4830
Synonym:
Target: Others
Sachaconitine
Cat.No: TN6341
Synonym: 黄草乌碱丁,Vilmorrianine D
Target:
Lipoaconitine
Cat.No: TN6115
Synonym:
Target:
13-Dehydroxyindaconitine
Cat.No: T83455
Synonym:
Target:
Indaconitine
Cat.No: T6S1879
Synonym:
Target: Others
Ludaconitine
Cat.No: T11890
Synonym:
Target: Others
Lipodeoxyaconitine
Cat.No: TN6114
Synonym:
Target:
14-O-Acetylsachaconitine
Cat.No: TN6342
Synonym:
Target:
Onitisin
Cat.No: TN4713
Synonym:
Target: 5-HT Receptor
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