52
15
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11992 |
Mefuparib hydrochloride
MPH |
PARP | Chromatin/Epigenetic; DNA Damage/DNA Repair |
Mefuparib hydrochloride induces apoptosis and possesses prominent anticancer activity in vitro and in vivo. Mefuparib hydrochloride (MPH) is an orally active, substrate-competitive and selective PARP1/2 inhibitor with IC50s of 3.2 nM and 1.9 nM, respectively. | |||
T73439 |
MPH-220
|
||
MPH-220是一种口服活性的、选择性骨骼肌myosin-2抑制剂,能够促进肌肉松弛。作为一种抗痉挛药物,它用于研究痉挛和肌肉僵硬。 | |||
T0205 |
Brompheniramine maleate
Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane |
5-HT Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Brompheniramine maleate (Dimotane) 是一种可口服的丙胺类抗组胺剂,具有抗胆碱能和抗抑郁作用,可用于过敏性鼻炎和缓解疼痛的研究。它是一种选择性组胺 H1 受体拮抗剂,Kd 为 6.06 nM。 | |||
T1550 |
Thiamphenicol
甲砜霉素,Dextrosulphenidol,Thiophenicol |
Antibacterial; Antibiotic | Microbiology/Virology |
Thiamphenicol (Dextrosulphenidol) 是 Chloramphenicol 的甲基磺酰基衍生物,是一种广谱抗菌类抗生素。它与 50S 核糖体亚基结合,抑制蛋白质合成并具有抑菌作用 ,特别针对革兰氏阴性,革兰氏阳性需氧和厌氧菌。 | |||
T60080 |
TMPH
2,2,6,6-Tetramethylpiperidin-4-yl heptanoate |
AChR | Neuroscience |
TMPH 是一种 nAChR 抑制剂,可抑制缺乏 α5、α6 或 β3 亚基的 nAChR。 TMPH 可用于关于 nAChR 功能障碍或神经系统疾病的研究。 | |||
T20525 |
Chloramphenicol palmitate
|
Antibacterial; Antibiotic | Microbiology/Virology |
Chloramphenicol palmitate 是一种广谱抗生素,对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。 | |||
T7465 |
4-Methylbenzylidene camphor
Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC |
AChE | Neuroscience |
4-Methylbenzylidene camphor 是有机的樟脑衍生物,应用于化妆品行业,具有保护皮肤抵抗紫外线(特别是紫外线B 辐射)的能力。 | |||
TF0050 | Amphipol A8-35 | ||
Amphipol A8-35 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0050,CAS号为 326856-53-5。 | |||
T25239 |
Chloramphenicol stearate
Eusynthomycin,Chloramphenicol monostearate,Madomicetina |
||
Chloramphenicol stearate is an antibiotic useful for the therapy of numbers of bacterial infections. This includes an eye ointment to treat conjunctivitis. | |||
T10311 |
Amphotericin X1
两性霉素 X1 |
Others | Others |
Amphotericin X1 is a derivative of Amphotericin B with good antifungal activity. Amphotericin X1 inhibits Candida albicans 33/079, Cryptococcus neoformans 451, C.parapsilosis 937A, Aspergillus niger 57A and A.fumigatus (MICs: 1 μg/mL, 1 μg/mL, 8 μg/mL, 2 | |||
T74079 | m-Chloramphenicol | ||
m-Chloramphenicol (m-threo-Chloramphenicol) 是 Chloramphenicol 的一种杂质。Chloramphenicol 是一种广谱抗生素,是细菌蛋白质生物合成的有效抑制剂。 | |||
T75276 | Dexbrompheniramine | ||
Dexbrompheniramine为口服活性H1受体拮抗剂(H1 receptor),具有抗组胺药属性,能够减轻天然化学组胺的作用。该化合物适用于花粉热与荨麻疹的研究。 | |||
T23462 |
TMPH hydrochloride
|
Others | Others |
neuronal nicotinic ACh receptors (nAChRs) antagonist | |||
T72093 |
Thiamphenicol glycinate hydrochloride
甲砜霉素甘氨酸酯盐酸盐 |
||
Thiamphenicol glycinate hydrochloride 是一种广谱抗菌剂,可用于呼吸道感染的研究。 | |||
T74061 | Amphotericin B methyl ester hydrochloride | ||
Amphotericin B methyl ester hydrochloride 是多烯类抗生素 Amphotericin B (A634250) 的甲酯衍生物。Amphotericin B methyl ester hydrochloride 是胆固醇结合物,具有显著的抗真菌活性。Amphotericin B methyl ester hydrochloride 干扰HIV-1颗粒的产生,抑制HIV-1的复制。 | |||
T35651 |
Bromamphenicol
|
||
Bromamphenicol is a dibrominated derivative of the antibiotic chloramphenicol. It inhibits rat liver mitochondrial and E. coli protein synthesis by 90.6 and 98.8%, respectively, when used at a concentration of 93 μM, and inhibits DNA synthesis in human lymphoblastoid cells by 83% at 1 mM. Bromamphenicol can also bind to the major adhesin subunit DraE from E. coli. | |||
T73891 |
Amphotericin A
|
||
Amphotericin A 是一种有效的抗真菌抗生素。 | |||
T64105 |
Voriconazole camphorsulfonate
|
||
Voriconazole (UK-109496) camphorsulfonate 是一种二代广谱的三唑类抗真菌 (antifungal) 化合物,对真菌麦角甾醇的生物合成表现出抑制作用。Voriconazole camphorsulfonate 能够抑制由真菌细胞色素 P450 酶介导的 14-α-羊毛甾醇去甲基化作用,表现出抗真菌效果。 | |||
T65136 |
Camphorquinone
|
||
Camphorquinone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65136,CAS号为 10373-78-1。 | |||
T66682 |
(1R,3S)-(+)-Camphoric acid
|
||
(1R,3S)-(+)-Camphoric acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66682,CAS号为 124-83-4。 | |||
T34895 |
Tocamphyl
Tocanfil,Biliphorin,Gallogen |
||
Tocamphyl is a cholagogic agent that stimulates pancreatic exocrine and bile flow when administered in the duodenum. | |||
T71879 | Proximphan | ||
Proximphan is a cholinesterase or acetylcholinesterase (AChE) inhibitor. It is widely used as an insecticide or pesticide in homes, gardens and agricultural applications and is a synthetic compound. | |||
T71810 |
Thiamphenicol palmitate
|
||
Thiamphenicol palmitate is a Prodrug of Thiamphenicol, inhibiting the 50S subunit of the bacterial ribosome and protein translation. | |||
T20401 |
(-)-Isopinocampheol
l-Isopinocampheol |
||
(-)-Isopinocampheol is a monoterpene and a component of several plant essential oils. It showed dual viricidal activity against herpes simplex virus 1. | |||
T65673 |
(+)-10,2-Camphorsultam
|
||
(+)-10,2-Camphorsultam 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65673,CAS号为 108448-77-7。 | |||
T16903 |
SMPH Crosslinker
|
Others | Others |
SMPH Crosslinker is an alkyl/ether-based PROTAC linker utilized for synthesizing PROTACs[1]. | |||
T66968 |
(1S)-(+)-Camphor-10-sulphonic acid
|
||
(1S)-(+)-Camphor-10-sulphonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66968,CAS号为 3144-16-9。 | |||
T30475 |
Bismuth camphocarbonate
Bi-Valeas,Solmuth,Cardyl,Rectobismutina,Angimuth |
||
Bismuth camphocarbonate is used for herpes zoster. | |||
T30040 |
Amphocil
Amphotericin B cholesteryl sulfate |
||
Amphocil is used to treat patients with invasive fungal infection. | |||
T124353 | Stemphol | ||
Stemphol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124353,CAS号为 70680-20-5。 | |||
T30038 | Amphidinolide F | ||
Amphidinolide F is a new cytotoxic macrolide | |||
T30036 | Amphenidone | ||
Amphenidone is a Tranquilizer. | |||
T25083 |
Amphotalide
RP 6171,RP-6171,RP6171,Schistomide |
||
Amphotalide is an anthelminthic agent. | |||
T71443 | Amphidinolide D | ||
Amphidinolide D is a powerful activator of actomyosin ATPase enhances skeletal muscle contraction. | |||
T10309 |
Amphethinile
Amphetinile,CRC 82-07 |
Others | Others |
Amphethinile is an anti-tubulin agent. The Ka of Amphethinile with tubulin is 1.3 μM. | |||
T61234 |
Stemphyperylenol
|
||
Stemphyperylenol exhibits potent antifungal activity against Alternaria solani, a plant pathogen, with a minimum inhibitory concentration (MIC) value of 1.57 μM. | |||
T30037 |
Amphidinolide C
|
||
Amphidinolide C is a potent cytotoxic 25-membered macrolide from marine dinoflagellate Amphidinium sp. | |||
T34715 |
Stemphyloxin I
Deacyl-FR 225654 |
||
Stemphyloxin I is a phytotoxin from Stemphylium botryosum. | |||
T24401 |
L-erythro-Chloramphenicol
L(+)-erythro-Chloramphenicol |
||
L-erythro-Chloramphenicol functions as a potent inhibitor of electron transport. | |||
T131515 |
Picroside II (Amphicoside)
|
||
Picroside II (Amphicoside) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131515。 | |||
T30041 |
Amphoglucamine
|
||
Amphoglucamine is used in the combined chemotherapy of viral diseases. | |||
T65131 |
(+/-)-10-Camphorsulfonic Acid
|
||
(+/-)-10-Camphorsulfonic Acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65131,CAS号为 5872-08-2。 | |||
T31396 |
Dexbrompheniramine maleate
D-Brompheniramine,Brompheniramine d-,Dexbrompheniraminum,Disophrol,Drixoral |
||
Dexbrompheniramine is an antihistamine with anticholinergic properties. It is used to treat allergic diseases such as hay fever or urticaria. It can compete with histamine for H1 receptor sites on effector cells of the gastrointestinal tract, blood vessel | |||
T66944 | (1R)-(-)-10-Camphorsulfonic acid | ||
(1R)-(-)-10-Camphorsulfonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66944,CAS号为 35963-20-3。 | |||
T20818 |
Propetamphos
Deadmag,Safrotin S 200 |
||
Propetamphos, an organophosphate pesticide, can effectively control cockroaches, flies, mosquitoes, and other pests. It is also effective for cattle lice. | |||
T10310 |
Amphotericin B methyl ester
|
Others | Others |
Amphotericin B methyl ester is the derivative of the antibiotic Amphotericin B. Amphotericin B methyl ester is the cholesterol-binding compound that possesses significant antifungal activity. It disrupts HIV-1 particle production and potently inhibits HIV | |||
T60843 |
Brompheniramine
|
||
Brompheniramine ((±)-Brompheniramine) 是具有口服活性的烷基胺类抗组胺药。Brompheniramine 是组胺 H1 受体的选择性拮抗剂 (Kd = 6.06 nM)。Brompheniramine 可用于过敏性鼻炎,它具有抗胆碱能、抗抑郁和麻醉作用。Brompheniramine 可阻断钙离子通道、钠离子通道和 hERG 通道,IC50分别为 16.12 μM, 21.26 μM 和 0.90 μM。 | |||
T124427 |
Camphans?ure (+)-
|
||
Camphans?ure (+)- 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124427,CAS号为 67111-66-4。 | |||
T30039 |
Amphimedine
|
||
Amphimedine is a Pyridoacridine Marine Alkaloid. | |||
T34757 |
Symphytine
|
||
Symphytine is a natural inducer of hepatic tumors. Symphytine interacts with DNA in liver endothelial cells and hepatocytes, resulting in DNA damage, mutation induction, and cancer development. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8258 |
Chloramphenicol succinate sodium
Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠 |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Chloramphenicol succinate sodium 是 Chloramphenicol 的前药,具有血液学毒性。它是琥珀酸脱氢酶的竞争底物和抑制剂。 | |||
TMS2262 |
(-)-CAMPHOR
L-Camphor,左旋樟脑 |
Others | Others |
(-)-CAMPHOR (L-Camphor) 是樟脑的手性中间体,在食品中用作风味添加剂和甜味剂。 | |||
T1205 |
Chloramphenicol
Chlornitromycin,Levomycetin,Chloromycetin,氯霉素 |
ribosome; HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic | Chromatin/Epigenetic; Metabolism; Microbiology/Virology |
Chloramphenicol (Chloromycetin) 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。 | |||
T7959 |
(+)-ISOPINOCAMPHEOL
|
Others | Others |
(+)-ISOPINOCAMPHEOL 是一种天然产物。 | |||
T20191 |
(-)-Camphoric acid
(-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)- |
GluR | Neuroscience |
(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体,樟脑酸可诱导 GluR 表达。 | |||
T2952 |
Camphor
樟脑,(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa |
Influenza Virus; TRP/TRPV Channel | Membrane transporter/Ion channel; Microbiology/Virology |
Camphor (2-Camphanone) 是一种双环单萜酮,广泛存在于植物中,尤其是樟脑。 它是一种激动剂,局部用作皮肤止痒剂和抗感染剂,具有抗病毒,镇咳和抗癌活性。 | |||
T0882 |
(+)-Camphor
D-(+)-Camphor,D-Camphor,(+)-樟脑,(1R)-(+)-Camphor |
Antibacterial; TRP/TRPV Channel | Membrane transporter/Ion channel; Microbiology/Virology |
(+)-Camphor (D-Camphor) 是一种食品添加剂,在医学上可用作防腐剂。 | |||
T25240 |
Chloramphenicol succinate
Paraxin succinate,Kemicetine succinate,CPSA |
||
Chloramphenicol succinate is an inactive precursor of chloramphenicol. It is used for parenteral administration of chloramphenicol. | |||
T82002 |
Juniper camphor
|
||
Juniper camphor为倍半萜烯类化合物,可通过分馏樟脑蓝油的高沸点馏分进行分离。 | |||
TN4450 |
Longistylumphylline A
|
Others | Others |
Longistylumphylline A是一种天然产物,属于交让木科虎皮楠属,其产品编号为 TN4450,CAS号为 857672-34-5。Longistylumphylline A可用作对照参考。 | |||
TN4667 |
Norcamphor
|
Others | Others |
Norcamphor 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4667,CAS号为 497-38-1。 | |||
TN5908 |
Symphonone I
|
||
Symphonone I 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5908,CAS号为 1235774-18-1。 | |||
T1067 |
Amphotericin B
NSC 527017,两性霉素B |
Antibiotic; Antifungal | Microbiology/Virology |
Amphotericin B (NSC-527017) 是一种多烯类抗真菌剂,对许多真菌物种具有广谱活性。Amphotericin B 不可逆地结合麦角甾醇,破坏细胞膜完整性,从而起到抗真菌活性。 | |||
T38588 |
Amphotericin B trihydrate
|
||
Amphotericin B trihydrate, a polyene antibiotic, is derived from Streptomyces nodosus fermenter cultures. It exhibits antileishmanial properties. | |||
TN2432 |
6-hydroxyl kaempherol-3,6-O-diglucosyl-7-O-Glucuronic acid
|
Others | Others |
6-hydroxyl kaempherol-3,6-O-diglucosyl-7-O-Glucuronic acid is a natural product from Carthamus tinctorius Linn. |