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52

抑制剂 & 化合物

15

天然产物

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Cat. No. Product Name Target Signaling Pathways
T11992 Mefuparib hydrochloride

MPH

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Mefuparib hydrochloride induces apoptosis and possesses prominent anticancer activity in vitro and in vivo. Mefuparib hydrochloride (MPH) is an orally active, substrate-competitive and selective PARP1/2 inhibitor with IC50s of 3.2 nM and 1.9 nM, respectively.
T73439 MPH-220

MPH-220是一种口服活性的、选择性骨骼肌myosin-2抑制剂,能够促进肌肉松弛。作为一种抗痉挛药物,它用于研究痉挛和肌肉僵硬。
T0205 Brompheniramine maleate

Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane

5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Brompheniramine maleate (Dimotane) 是一种可口服的丙胺类抗组胺剂,具有抗胆碱能和抗抑郁作用,可用于过敏性鼻炎和缓解疼痛的研究。它是一种选择性组胺 H1 受体拮抗剂,Kd 为 6.06 nM。
T1550 Thiamphenicol

甲砜霉素,Dextrosulphenidol,Thiophenicol

Antibacterial; Antibiotic Microbiology/Virology
Thiamphenicol (Dextrosulphenidol) 是 Chloramphenicol 的甲基磺酰基衍生物,是一种广谱抗菌类抗生素。它与 50S 核糖体亚基结合,抑制蛋白质合成并具有抑菌作用 ,特别针对革兰氏阴性,革兰氏阳性需氧和厌氧菌。
T60080 TMPH

2,2,6,6-Tetramethylpiperidin-4-yl heptanoate

AChR Neuroscience
TMPH 是一种 nAChR 抑制剂,可抑制缺乏 α5、α6 或 β3 亚基的 nAChR。 TMPH 可用于关于 nAChR 功能障碍或神经系统疾病的研究。
T20525 Chloramphenicol palmitate

Antibacterial; Antibiotic Microbiology/Virology
Chloramphenicol palmitate 是一种广谱抗生素,对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。
T7465 4-Methylbenzylidene camphor

Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC

AChE Neuroscience
4-Methylbenzylidene camphor 是有机的樟脑衍生物,应用于化妆品行业,具有保护皮肤抵抗紫外线(特别是紫外线B 辐射)的能力。
TF0050 Amphipol A8-35

Amphipol A8-35 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0050,CAS号为 326856-53-5。
T25239 Chloramphenicol stearate

Eusynthomycin,Chloramphenicol monostearate,Madomicetina

Chloramphenicol stearate is an antibiotic useful for the therapy of numbers of bacterial infections. This includes an eye ointment to treat conjunctivitis.
T10311 Amphotericin X1

两性霉素 X1

Others Others
Amphotericin X1 is a derivative of Amphotericin B with good antifungal activity. Amphotericin X1 inhibits Candida albicans 33/079, Cryptococcus neoformans 451, C.parapsilosis 937A, Aspergillus niger 57A and A.fumigatus (MICs: 1 μg/mL, 1 μg/mL, 8 μg/mL, 2
T74079 m-Chloramphenicol

m-Chloramphenicol (m-threo-Chloramphenicol) 是 Chloramphenicol 的一种杂质。Chloramphenicol 是一种广谱抗生素,是细菌蛋白质生物合成的有效抑制剂。
T75276 Dexbrompheniramine

Dexbrompheniramine为口服活性H1受体拮抗剂(H1 receptor),具有抗组胺药属性,能够减轻天然化学组胺的作用。该化合物适用于花粉热与荨麻疹的研究。
T23462 TMPH hydrochloride

Others Others
neuronal nicotinic ACh receptors (nAChRs) antagonist
T72093 Thiamphenicol glycinate hydrochloride

甲砜霉素甘氨酸酯盐酸盐

Thiamphenicol glycinate hydrochloride 是一种广谱抗菌剂,可用于呼吸道感染的研究。
T74061 Amphotericin B methyl ester hydrochloride

Amphotericin B methyl ester hydrochloride 是多烯类抗生素 Amphotericin B (A634250) 的甲酯衍生物。Amphotericin B methyl ester hydrochloride 是胆固醇结合物,具有显著的抗真菌活性。Amphotericin B methyl ester hydrochloride 干扰HIV-1颗粒的产生,抑制HIV-1的复制。
T35651 Bromamphenicol

Bromamphenicol is a dibrominated derivative of the antibiotic chloramphenicol. It inhibits rat liver mitochondrial and E. coli protein synthesis by 90.6 and 98.8%, respectively, when used at a concentration of 93 μM, and inhibits DNA synthesis in human lymphoblastoid cells by 83% at 1 mM. Bromamphenicol can also bind to the major adhesin subunit DraE from E. coli.
T73891 Amphotericin A

Amphotericin A 是一种有效的抗真菌抗生素。
T64105 Voriconazole camphorsulfonate

Voriconazole (UK-109496) camphorsulfonate 是一种二代广谱的三唑类抗真菌 (antifungal) 化合物,对真菌麦角甾醇的生物合成表现出抑制作用。Voriconazole camphorsulfonate 能够抑制由真菌细胞色素 P450 酶介导的 14-α-羊毛甾醇去甲基化作用,表现出抗真菌效果。
T65136 Camphorquinone

Camphorquinone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65136,CAS号为 10373-78-1。
T66682 (1R,3S)-(+)-Camphoric acid

(1R,3S)-(+)-Camphoric acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66682,CAS号为 124-83-4。
T34895 Tocamphyl

Tocanfil,Biliphorin,Gallogen

Tocamphyl is a cholagogic agent that stimulates pancreatic exocrine and bile flow when administered in the duodenum.
T71879 Proximphan

Proximphan is a cholinesterase or acetylcholinesterase (AChE) inhibitor. It is widely used as an insecticide or pesticide in homes, gardens and agricultural applications and is a synthetic compound.
T71810 Thiamphenicol palmitate

Thiamphenicol palmitate is a Prodrug of Thiamphenicol, inhibiting the 50S subunit of the bacterial ribosome and protein translation.
T20401 (-)-Isopinocampheol

l-Isopinocampheol

(-)-Isopinocampheol is a monoterpene and a component of several plant essential oils. It showed dual viricidal activity against herpes simplex virus 1.
T65673 (+)-10,2-Camphorsultam

(+)-10,2-Camphorsultam 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65673,CAS号为 108448-77-7。
T16903 SMPH Crosslinker

Others Others
SMPH Crosslinker is an alkyl/ether-based PROTAC linker utilized for synthesizing PROTACs[1].
T66968 (1S)-(+)-Camphor-10-sulphonic acid

(1S)-(+)-Camphor-10-sulphonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66968,CAS号为 3144-16-9。
T30475 Bismuth camphocarbonate

Bi-Valeas,Solmuth,Cardyl,Rectobismutina,Angimuth

Bismuth camphocarbonate is used for herpes zoster.
T30040 Amphocil

Amphotericin B cholesteryl sulfate

Amphocil is used to treat patients with invasive fungal infection.
T124353 Stemphol

Stemphol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124353,CAS号为 70680-20-5。
T30038 Amphidinolide F

Amphidinolide F is a new cytotoxic macrolide
T30036 Amphenidone

Amphenidone is a Tranquilizer.
T25083 Amphotalide

RP 6171,RP-6171,RP6171,Schistomide

Amphotalide is an anthelminthic agent.
T71443 Amphidinolide D

Amphidinolide D is a powerful activator of actomyosin ATPase enhances skeletal muscle contraction.
T10309 Amphethinile

Amphetinile,CRC 82-07

Others Others
Amphethinile is an anti-tubulin agent. The Ka of Amphethinile with tubulin is 1.3 μM.
T61234 Stemphyperylenol

Stemphyperylenol exhibits potent antifungal activity against Alternaria solani, a plant pathogen, with a minimum inhibitory concentration (MIC) value of 1.57 μM.
T30037 Amphidinolide C

Amphidinolide C is a potent cytotoxic 25-membered macrolide from marine dinoflagellate Amphidinium sp.
T34715 Stemphyloxin I

Deacyl-FR 225654

Stemphyloxin I is a phytotoxin from Stemphylium botryosum.
T24401 L-erythro-Chloramphenicol

L(+)-erythro-Chloramphenicol

L-erythro-Chloramphenicol functions as a potent inhibitor of electron transport.
T131515 Picroside II (Amphicoside)

Picroside II (Amphicoside) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131515。
T30041 Amphoglucamine

Amphoglucamine is used in the combined chemotherapy of viral diseases.
T65131 (+/-)-10-Camphorsulfonic Acid

(+/-)-10-Camphorsulfonic Acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65131,CAS号为 5872-08-2。
T31396 Dexbrompheniramine maleate

D-Brompheniramine,Brompheniramine d-,Dexbrompheniraminum,Disophrol,Drixoral

Dexbrompheniramine is an antihistamine with anticholinergic properties. It is used to treat allergic diseases such as hay fever or urticaria. It can compete with histamine for H1 receptor sites on effector cells of the gastrointestinal tract, blood vessel
T66944 (1R)-(-)-10-Camphorsulfonic acid

(1R)-(-)-10-Camphorsulfonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66944,CAS号为 35963-20-3。
T20818 Propetamphos

Deadmag,Safrotin S 200

Propetamphos, an organophosphate pesticide, can effectively control cockroaches, flies, mosquitoes, and other pests. It is also effective for cattle lice.
T10310 Amphotericin B methyl ester

Others Others
Amphotericin B methyl ester is the derivative of the antibiotic Amphotericin B. Amphotericin B methyl ester is the cholesterol-binding compound that possesses significant antifungal activity. It disrupts HIV-1 particle production and potently inhibits HIV
T60843 Brompheniramine

Brompheniramine ((±)-Brompheniramine) 是具有口服活性的烷基胺类抗组胺药。Brompheniramine 是组胺 H1 受体的选择性拮抗剂 (Kd = 6.06 nM)。Brompheniramine 可用于过敏性鼻炎,它具有抗胆碱能、抗抑郁和麻醉作用。Brompheniramine 可阻断钙离子通道、钠离子通道和 hERG 通道,IC50分别为 16.12 μM, 21.26 μM 和 0.90 μM。
T124427 Camphans?ure (+)-

Camphans?ure (+)- 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124427,CAS号为 67111-66-4。
T30039 Amphimedine

Amphimedine is a Pyridoacridine Marine Alkaloid.
T34757 Symphytine

Symphytine is a natural inducer of hepatic tumors. Symphytine interacts with DNA in liver endothelial cells and hepatocytes, resulting in DNA damage, mutation induction, and cancer development.

化合物

Mefuparib hydrochloride
Cat.No: T11992
Synonym: MPH
Target: PARP
MPH-220
Cat.No: T73439
Synonym:
Target:
Brompheniramine maleate
Cat.No: T0205
Synonym: Dimotane,马来酸溴苯那敏,Rolabromophen,Brompheniramine hydrogen maleate,Dimetane
Target: 5-HT Receptor, Histamine Receptor
Thiamphenicol
Cat.No: T1550
Synonym: 甲砜霉素,Dextrosulphenidol,Thiophenicol
Target: Antibacterial, Antibiotic
TMPH
Cat.No: T60080
Synonym: 2,2,6,6-Tetramethylpiperidin-4-yl heptanoate
Target: AChR
Chloramphenicol palmitate
Cat.No: T20525
Synonym:
Target: Antibacterial, Antibiotic
4-Methylbenzylidene camphor
Cat.No: T7465
Synonym: Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC
Target: AChE
Amphipol A8-35
Cat.No: TF0050
Synonym:
Target:
Chloramphenicol stearate
Cat.No: T25239
Synonym: Eusynthomycin,Chloramphenicol monostearate,Madomicetina
Target:
Amphotericin X1
Cat.No: T10311
Synonym: 两性霉素 X1
Target: Others
m-Chloramphenicol
Cat.No: T74079
Synonym:
Target:
Dexbrompheniramine
Cat.No: T75276
Synonym:
Target:
TMPH hydrochloride
Cat.No: T23462
Synonym:
Target: Others
Thiamphenicol glycinate hydrochloride
Cat.No: T72093
Synonym: 甲砜霉素甘氨酸酯盐酸盐
Target:
Amphotericin B methyl ester hydrochloride
Cat.No: T74061
Synonym:
Target:
Bromamphenicol
Cat.No: T35651
Synonym:
Target:
Amphotericin A
Cat.No: T73891
Synonym:
Target:
Voriconazole camphorsulfonate
Cat.No: T64105
Synonym:
Target:
Camphorquinone
Cat.No: T65136
Synonym:
Target:
(1R,3S)-(+)-Camphoric acid
Cat.No: T66682
Synonym:
Target:
Tocamphyl
Cat.No: T34895
Synonym: Tocanfil,Biliphorin,Gallogen
Target:
Proximphan
Cat.No: T71879
Synonym:
Target:
Thiamphenicol palmitate
Cat.No: T71810
Synonym:
Target:
(-)-Isopinocampheol
Cat.No: T20401
Synonym: l-Isopinocampheol
Target:
(+)-10,2-Camphorsultam
Cat.No: T65673
Synonym:
Target:
SMPH Crosslinker
Cat.No: T16903
Synonym:
Target: Others
(1S)-(+)-Camphor-10-sulphonic acid
Cat.No: T66968
Synonym:
Target:
Bismuth camphocarbonate
Cat.No: T30475
Synonym: Bi-Valeas,Solmuth,Cardyl,Rectobismutina,Angimuth
Target:
Amphocil
Cat.No: T30040
Synonym: Amphotericin B cholesteryl sulfate
Target:
Stemphol
Cat.No: T124353
Synonym:
Target:
Amphidinolide F
Cat.No: T30038
Synonym:
Target:
Amphenidone
Cat.No: T30036
Synonym:
Target:
Amphotalide
Cat.No: T25083
Synonym: RP 6171,RP-6171,RP6171,Schistomide
Target:
Amphidinolide D
Cat.No: T71443
Synonym:
Target:
Amphethinile
Cat.No: T10309
Synonym: Amphetinile,CRC 82-07
Target: Others
Stemphyperylenol
Cat.No: T61234
Synonym:
Target:
Amphidinolide C
Cat.No: T30037
Synonym:
Target:
Stemphyloxin I
Cat.No: T34715
Synonym: Deacyl-FR 225654
Target:
L-erythro-Chloramphenicol
Cat.No: T24401
Synonym: L(+)-erythro-Chloramphenicol
Target:
Picroside II (Amphicoside)
Cat.No: T131515
Synonym:
Target:
Amphoglucamine
Cat.No: T30041
Synonym:
Target:
(+/-)-10-Camphorsulfonic Acid
Cat.No: T65131
Synonym:
Target:
Dexbrompheniramine maleate
Cat.No: T31396
Synonym: D-Brompheniramine,Brompheniramine d-,Dexbrompheniraminum,Disophrol,Drixoral
Target:
(1R)-(-)-10-Camphorsulfonic acid
Cat.No: T66944
Synonym:
Target:
Propetamphos
Cat.No: T20818
Synonym: Deadmag,Safrotin S 200
Target:
Amphotericin B methyl ester
Cat.No: T10310
Synonym:
Target: Others
Brompheniramine
Cat.No: T60843
Synonym:
Target:
Camphans?ure (+)-
Cat.No: T124427
Synonym:
Target:
Amphimedine
Cat.No: T30039
Synonym:
Target:
Symphytine
Cat.No: T34757
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T8258 Chloramphenicol succinate sodium

Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Chloramphenicol succinate sodium 是 Chloramphenicol 的前药,具有血液学毒性。它是琥珀酸脱氢酶的竞争底物和抑制剂。
TMS2262 (-)-CAMPHOR

L-Camphor,左旋樟脑

Others Others
(-)-CAMPHOR (L-Camphor) 是樟脑的手性中间体,在食品中用作风味添加剂和甜味剂。
T1205 Chloramphenicol

Chlornitromycin,Levomycetin,Chloromycetin,氯霉素

ribosome; HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Chloramphenicol (Chloromycetin) 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。
T7959 (+)-ISOPINOCAMPHEOL

Others Others
(+)-ISOPINOCAMPHEOL 是一种天然产物。
T20191 (-)-Camphoric acid

(-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-

GluR Neuroscience
(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体,樟脑酸可诱导 GluR 表达。
T2952 Camphor

樟脑,(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa

Influenza Virus; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology
Camphor (2-Camphanone) 是一种双环单萜酮,广泛存在于植物中,尤其是樟脑。 它是一种激动剂,局部用作皮肤止痒剂和抗感染剂,具有抗病毒,镇咳和抗癌活性。
T0882 (+)-Camphor

D-(+)-Camphor,D-Camphor,(+)-樟脑,(1R)-(+)-Camphor

Antibacterial; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology
(+)-Camphor (D-Camphor) 是一种食品添加剂,在医学上可用作防腐剂。
T25240 Chloramphenicol succinate

Paraxin succinate,Kemicetine succinate,CPSA

Chloramphenicol succinate is an inactive precursor of chloramphenicol. It is used for parenteral administration of chloramphenicol.
T82002 Juniper camphor

Juniper camphor为倍半萜烯类化合物,可通过分馏樟脑蓝油的高沸点馏分进行分离。
TN4450 Longistylumphylline A

Others Others
Longistylumphylline A是一种天然产物,属于交让木科虎皮楠属,其产品编号为 TN4450,CAS号为 857672-34-5。Longistylumphylline A可用作对照参考。
TN4667 Norcamphor

Others Others
Norcamphor 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4667,CAS号为 497-38-1。
TN5908 Symphonone I

Symphonone I 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5908,CAS号为 1235774-18-1。
T1067 Amphotericin B

NSC 527017,两性霉素B

Antibiotic; Antifungal Microbiology/Virology
Amphotericin B (NSC-527017) 是一种多烯类抗真菌剂,对许多真菌物种具有广谱活性。Amphotericin B 不可逆地结合麦角甾醇,破坏细胞膜完整性,从而起到抗真菌活性。
T38588 Amphotericin B trihydrate

Amphotericin B trihydrate, a polyene antibiotic, is derived from Streptomyces nodosus fermenter cultures. It exhibits antileishmanial properties.
TN2432 6-hydroxyl kaempherol-3,6-O-diglucosyl-7-O-Glucuronic acid

Others Others
6-hydroxyl kaempherol-3,6-O-diglucosyl-7-O-Glucuronic acid is a natural product from Carthamus tinctorius Linn.

天然产物

Chloramphenicol succinate sodium
Cat.No: T8258
Synonym: Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠
Target: Others, Antibacterial, Antibiotic
(-)-CAMPHOR
Cat.No: TMS2262
Synonym: L-Camphor,左旋樟脑
Target: Others
Chloramphenicol
Cat.No: T1205
Synonym: Chlornitromycin,Levomycetin,Chloromycetin,氯霉素
Target: ribosome, HIF/HIF Prolyl-Hydroxylase, Antibacterial, Antibiotic
(+)-ISOPINOCAMPHEOL
Cat.No: T7959
Synonym:
Target: Others
(-)-Camphoric acid
Cat.No: T20191
Synonym: (-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-
Target: GluR
Camphor
Cat.No: T2952
Synonym: 樟脑,(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa
Target: Influenza Virus, TRP/TRPV Channel
(+)-Camphor
Cat.No: T0882
Synonym: D-(+)-Camphor,D-Camphor,(+)-樟脑,(1R)-(+)-Camphor
Target: Antibacterial, TRP/TRPV Channel
Chloramphenicol succinate
Cat.No: T25240
Synonym: Paraxin succinate,Kemicetine succinate,CPSA
Target:
Juniper camphor
Cat.No: T82002
Synonym:
Target:
Longistylumphylline A
Cat.No: TN4450
Synonym:
Target: Others
Norcamphor
Cat.No: TN4667
Synonym:
Target: Others
Symphonone I
Cat.No: TN5908
Synonym:
Target:
Amphotericin B
Cat.No: T1067
Synonym: NSC 527017,两性霉素B
Target: Antibiotic, Antifungal
Amphotericin B trihydrate
Cat.No: T38588
Synonym:
Target:
6-hydroxyl kaempherol-3,6-O-diglucosyl-7-O-Glucuronic acid
Cat.No: TN2432
Synonym:
Target: Others
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