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21

抑制剂 & 化合物

9

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0863 Idoxuridine

IDU,碘苷,SKF 14287,5-Iodo-2′-deoxyuridine,NSC 39661,5-IUdR,Dendrid

Antifection; HSV Microbiology/Virology
Idoxuridine (Dendrid) 是一种抑制病毒 DNA 合成的脱氧尿苷类似物,用作抗病毒剂。
T7886 Nidufexor

FXR; Autophagy Autophagy; Metabolism
Nidufexor 是一种可口服的法尼醇 X 受体激动剂,可研究非酒精性脂肪性肝炎。
T17232 Vidupiprant

AMG 853

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Vidupiprant (AMG 853) 是一种有效的 CRTH2 和前列腺素 D 受体双重拮抗剂,在人源血浆中的 IC50 分别为 8 nM 和 35 nM。 Vidupiprant 可用于治疗哮喘的研究。
T11286 Fiduxosin

A 185980.1,ABT 980

Adrenergic Receptor GPCR/G Protein; Neuroscience
Fiduxosin 是一种具有选择性和有效性的 α1-adrenoceptor 拮抗剂,对 α1a-adrenoceptor,α1b-adrenoceptor 和 α1d-adrenoceptor 有抑制作用,Ki 值分别为 0.160 nM,24.9 nM 和 0.920 nM。Fiduxosin 可用于治疗良性前列腺增生。
T14298 Rimiducid

Apoptosis; Others; Fatty Acid Synthase Apoptosis; Metabolism; Others
Rimiducid 是一种可渗透脂质的他克莫司类似物,是一种二聚剂,通过交联 FKBP 结构域起作用。它将 Caspase 9 自杀开关二聚化并迅速诱导细胞凋亡。
T6088 Anidulafungin

LY303366,Eraxis,Ecalta,阿尼芬净

Others; Antibiotic; Antifungal Microbiology/Virology; Others
Anidulafungin (Ecalta) 是一种半合成的新棘球白素,具有抗真菌作用。
T69927 Fiduxosin hydrochloride

Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.
T36370 4-Methylumbelliferyl-α-L-Iduronide (free acid)

4-Methylumbelliferyl-α-L-iduronide (free acid) is a fluorogenic substrate for α-L-iduronidase, an enzyme found in cell lysosomes that is involved in the degradation of glycosaminoglycans such as dermatan sulfate and heparin sulfate. 4-Methylumbelliferyl-α-L-iduronide is cleaved by α-L-iduronidase to release the fluorescent moiety 4-methylumbelliferyl (4-MU). 4-MU fluorescence is pH-dependent with excitation maxima of 320 and 360 nm at low (1.97-6.72) and high (7.12-10.3) pH, respectively, and an...
T74706 Vidutolimod

Vidutolimod 是一种CpG-A 类寡核苷酸,是TLR9的激动剂。Vidutolimod 激活浆细胞样树突状细胞(pDCs)并触发IFNα的释放,导致抗肿瘤免疫作用。
T74421 Pemvidutide

Pemvidutide 是一种GLP-1R/GCGR 双重激动剂,可导致体重、肝脏脂肪和血清脂质的显著降低。Pemvidutide 可用于非酒精性脂肪性肝炎 (NASH) 和肥胖症的研究。
T37560 Nidulin

Nidulin is a depsidone originally isolated from A. nidulans. It is active against the bacteria M. tuberculosis and M. ranoe, as well as the fungi T. tonsurans and M. audouini. It also inhibits the growth of methicillin-resistant S. aureus (MRSA; MIC = 4 μg/ml) and has larvicidal activity toward Artemia (LC50 = 2.8 μg/ml). Nidulin is cytotoxic to MOLT-3 cells (IC50 = 21.2 μM) but not HuCCA-1, HepG2, or A549 cells (IC50s = >112.7 μM). It inhibits aromatase with an IC50 value of 11.2 μM.
T125124 Nidurufin

Nidurufin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125124,CAS号为 28458-23-3。
T32138 Iduronate 2-sulfate

Iduronate 2-sulfate is a sulfatase enzyme related to Hunter syndrome.
T76980 Tidutamab

Tidutamab (XmAb-18087) 是一种具有完整 Fc 结构域的人源化及亲和优化双特异性抗体(bsAb),旨在通过SSTR2和CD3两个靶点特异性结合来延长血清半衰期,通过激活T细胞介导的细胞毒性(RTcC)机制,有效消除SSTR+肿瘤细胞。
T78658 Pemvidutide TFA

Pemvidutide (TFA) 是一款针对GLP-1R/GCGR的双重激动剂,有助于显著降低体重、肝脏脂肪以及血清脂质水平。该化合物主要适用于非酒精性脂肪性肝炎(NASH)和肥胖症的研究领域。
T36541 Nornidulin

Nornidulin is a depsidone originally isolated from A. nidulans that has antibacterial activity against M. tuberculosis and M. ranoe as well as antifungal activity against T. tonsurans and M. audouini. It also inhibits the growth of methicillin-resistant S. aureus (MRSA; MIC = 2 μg/ml) and has larvicidal activity toward Artemia (LC50 = 1.7 μg/ml). Nornidulin has cytotoxic activity in MOLT-3 cells (IC50 = 35.7 μM) but not HuCCA-1, HepG2, or A549 cells (IC50s = >116.4 μM).
T125076 Hispidulin 7-glucuronide

Hispidulin 7-glucuronide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125076,CAS号为 31105-76-7。
T32925 Luciduline

Luciduline is a bioactive chemical.
T125725 Hispidulin 7-O-neohesperidoside

Hispidulin 7-O-neohesperidoside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125725。
T36111 L-Iduronic acid sodium salt

L-Iduronic acid sodium salt 是一种单糖,是肝素、硫酸乙酰肝素和硫酸皮肤素等糖胺聚糖 (GAG) 的重要成分。
T124577 Beta-D-glucopyranosiduronic acid

Beta-D-glucopyranosiduronic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124577。

化合物

Idoxuridine
Cat.No: T0863
Synonym: IDU,碘苷,SKF 14287,5-Iodo-2′-deoxyuridine,NSC 39661,5-IUdR,Dendrid
Target: Antifection, HSV
Nidufexor
Cat.No: T7886
Synonym:
Target: FXR, Autophagy
Vidupiprant
Cat.No: T17232
Synonym: AMG 853
Target: Prostaglandin Receptor
Fiduxosin
Cat.No: T11286
Synonym: A 185980.1,ABT 980
Target: Adrenergic Receptor
Rimiducid
Cat.No: T14298
Synonym:
Target: Apoptosis, Others, Fatty Acid Synthase
Anidulafungin
Cat.No: T6088
Synonym: LY303366,Eraxis,Ecalta,阿尼芬净
Target: Others, Antibiotic, Antifungal
Fiduxosin hydrochloride
Cat.No: T69927
Synonym:
Target:
4-Methylumbelliferyl-α-L-Iduronide (free acid)
Cat.No: T36370
Synonym:
Target:
Vidutolimod
Cat.No: T74706
Synonym:
Target:
Pemvidutide
Cat.No: T74421
Synonym:
Target:
Nidulin
Cat.No: T37560
Synonym:
Target:
Nidurufin
Cat.No: T125124
Synonym:
Target:
Iduronate 2-sulfate
Cat.No: T32138
Synonym:
Target:
Tidutamab
Cat.No: T76980
Synonym:
Target:
Pemvidutide TFA
Cat.No: T78658
Synonym:
Target:
Nornidulin
Cat.No: T36541
Synonym:
Target:
Hispidulin 7-glucuronide
Cat.No: T125076
Synonym:
Target:
Luciduline
Cat.No: T32925
Synonym:
Target:
Hispidulin 7-O-neohesperidoside
Cat.No: T125725
Synonym:
Target:
L-Iduronic acid sodium salt
Cat.No: T36111
Synonym:
Target:
Beta-D-glucopyranosiduronic acid
Cat.No: T124577
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TQ0201 Hispidulin

Dinatin

Pim Chromatin/Epigenetic; JAK/STAT signaling
Hispidulin 是存在于豚草中的一种黄酮,是Pim-1抑制剂,IC50值为2.71 μM。
T3932 Viscidulin I

Others Others
Viscidulin I 存在于黄芩中,是一种天然产物。
TN2302 Viscidulin III

Ganhuangenin

Glucosidase Metabolism
Viscidulin III (Ganhuangenin) 存在于黄芩中,可作为α-葡萄糖苷酶抑制剂。
TN4216 Hispidulin 4'-O-β-D-glucopyranoside

Hispidulin 4'-O-beta-D-glucopyranoside

Others Others
Hispidulin 4'-O-β-D-glucopyranoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4216,CAS号为 244285-12-9。
T38928 Oleanolic acid-3-O-glucosyl(1-2)xylyl(1-3)glucosiduronic acid

Oleanolic acid-3-O-glucosyl(1-2)xylyl(1-3)glucosiduronic acid is a naturally occurring triterpene saponin.
TN5239 Viscidulin III tetraacetate

Others Others
Viscidulin III tetraacetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5239,CAS号为 96684-81-0。
TN6645 Lucidumol A

Lucidumol A has relatively good effect against aldose reductase with IC50 of 19.1uM. Lucidumol A has cytotoxic activity, it reduced cell growth in three human carcinoma cells (Caco-2, HepG2, and HeLa cells) dose dependently with LC50s from 20.87 to 84.36
TN5238 Viscidulin II

IL Receptor; TNF Apoptosis; Immunology/Inflammation
Viscidulin II can be potential therapeutic agents against P. acnes-induced skin inflammation, it can significantly suppress P. acnes-induced IL-8 and IL-1β production in THP-1 cells, concomitant intradermal injection of viscidulin II with P. acnes can effectively attenuate P. acnes-induced ear swelling, and decrease the production of IL-6 and tumor necrosis factor-α in ear homogenates.
TN6939 Lucidumoside C

Lucidumoside C is a natural product.

天然产物

Hispidulin
Cat.No: TQ0201
Synonym: Dinatin
Target: Pim
Viscidulin I
Cat.No: T3932
Synonym:
Target: Others
Viscidulin III
Cat.No: TN2302
Synonym: Ganhuangenin
Target: Glucosidase
Hispidulin 4'-O-β-D-glucopyranoside
Cat.No: TN4216
Synonym: Hispidulin 4'-O-beta-D-glucopyranoside
Target: Others
Oleanolic acid-3-O-glucosyl(1-2)xylyl(1-3)glucosiduronic acid
Cat.No: T38928
Synonym:
Target:
Viscidulin III tetraacetate
Cat.No: TN5239
Synonym:
Target: Others
Lucidumol A
Cat.No: TN6645
Synonym:
Target:
Viscidulin II
Cat.No: TN5238
Synonym:
Target: IL Receptor, TNF
Lucidumoside C
Cat.No: TN6939
Synonym:
Target:
TargetMol Loading
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