购物车

搜索结果

Search Results for " fgfr1 inhibitor-6 "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T63816 FGFR1 inhibitor-6

FGFR1 inhibitor-6FGFR1 的有效抑制剂 (IC50: 16.31 nM),具有细胞毒活性。FGFR1 inhibitor-6 能够将细胞周期阻滞在前 G1 和 G2/M 期并诱导细胞凋亡 (apoptosis) 。
T4318 EOC317

ACTB-1003,ACTB1003,ACTB 1003

VEGFR; FGFR; Tie-2 Angiogenesis; Tyrosine Kinase/Adaptors
EOC317 (ACTB-1003) 是一种口服可用的激酶抑制剂,能够抑制 FGFR1 (IC50:6 nM),VEGFR2 (IC50:2 nM) 和 Tie-2 (IC50:4 nM)。
T36680 SM1-71

Serine/threonin kinase; MAPK; LIM Kinase; TGF-beta/Smad; AAK1 (AP2 associated kinase 1) Cell Cycle/Checkpoint; MAPK; Metabolism; Neuroscience; Stem Cells
SM1-71 是一种有效的多靶点丙烯酰胺修饰的 TAK1 抑制剂,抑制 MKNK2、MAP2K1/2/3/4/6/7、GAK、AAK1、BMP2K、MAP3K7、MAPKAPK5、GSK3A/B、MAPK1/3、SRC、YES1FGFR1、ZAK (MLTK)、MAP3K1、LIMK1 和 RSK2。SM1-71 可作为激酶探针,具有抗癌活性,抑制多种癌细胞系的增殖。
T13156L TG 100572 Hydrochloride

VEGFR; FGFR; PDGFR; Src Angiogenesis; Tyrosine Kinase/Adaptors
TG 100572 Hydrochloride 是一种多靶点激酶抑制剂,能够抑制受体酪氨酸激酶和Src 激酶。
T13156 TG 100572

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
TG 100572 is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 nM for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src, Yes, respectively).
T13157L TG 100801 Hydrochloride

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
TG 100801 Hydrochloride is a prodrug to treat age-related macular degeneration. TG 100572 is a inhibitor of multi-targeted kinase(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src,

化合物

FGFR1 inhibitor-6
Cat.No: T63816
Synonym:
Target:
EOC317
Cat.No: T4318
Synonym: ACTB-1003,ACTB1003,ACTB 1003
Target: VEGFR, FGFR, Tie-2
SM1-71
Cat.No: T36680
Synonym:
Target: Serine/threonin kinase, MAPK, LIM Kinase, TGF-beta/Smad, AAK1 (AP2 associated kinase 1)
TG 100572 Hydrochloride
Cat.No: T13156L
Synonym:
Target: VEGFR, FGFR, PDGFR, Src
TG 100572
Cat.No: T13156
Synonym:
Target: VEGFR
TG 100801 Hydrochloride
Cat.No: T13157L
Synonym:
Target: VEGFR
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼