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Cat. No. Product Name Target Signaling Pathways
T78830 FGFR1 inhibitor 7

FGFR Angiogenesis; Tyrosine Kinase/Adaptors
FGFR1 inhibitor7(compound 5),作为一种FGFR1络氨酸激酶抑制剂,具有0.33 nM的IC50。它对多种人癌细胞系显示出广谱的细胞毒性,能在2.1 μM的IC50抑制MOLT3细胞系。
T15185 Lucitanib

E-3810,德立替尼

VEGFR; FGFR Angiogenesis; Tyrosine Kinase/Adaptors
Lucitanib (E-3810) 是 VEGFR 和 FGFR 的双重抑制剂,有效和选择性地抑制VEGFR1 (IC50:7 nM),VEGFR2 (IC50:25 nM),VEGFR3 (IC50:10 nM),FGFR1 (IC50:17.5 nM),FGFR2 (IC50:82.5 nM)。
T36680 SM1-71

Serine/threonin kinase; MAPK; LIM Kinase; TGF-beta/Smad; AAK1 (AP2 associated kinase 1) Cell Cycle/Checkpoint; MAPK; Metabolism; Neuroscience; Stem Cells
SM1-71 是一种有效的多靶点丙烯酰胺修饰的 TAK1 抑制剂,抑制 MKNK2、MAP2K1/2/3/4/6/7、GAK、AAK1、BMP2K、MAP3K7、MAPKAPK5、GSK3A/B、MAPK1/3、SRC、YES1FGFR1、ZAK (MLTK)、MAP3K1、LIMK1 和 RSK2。SM1-71 可作为激酶探针,具有抗癌活性,抑制多种癌细胞系的增殖。
T13156L TG 100572 Hydrochloride

VEGFR; FGFR; PDGFR; Src Angiogenesis; Tyrosine Kinase/Adaptors
TG 100572 Hydrochloride 是一种多靶点激酶抑制剂,能够抑制受体酪氨酸激酶和Src 激酶。
T78832 FGFR1 inhibitor-9

FGFR Angiogenesis; Tyrosine Kinase/Adaptors
FGFR1inhibitor-9(Compound 9),一种FGFR1抑制剂(IC50为0.85 nM),可与FGFR1的ATP结合袋发生结合,并展现出抗癌活性。
T13156 TG 100572

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
TG 100572 is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 nM for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src, Yes, respectively).
T13157L TG 100801 Hydrochloride

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
TG 100801 Hydrochloride is a prodrug to treat age-related macular degeneration. TG 100572 is a inhibitor of multi-targeted kinase(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src,

化合物

FGFR1 inhibitor 7
Cat.No: T78830
Synonym:
Target: FGFR
Lucitanib
Cat.No: T15185
Synonym: E-3810,德立替尼
Target: VEGFR, FGFR
SM1-71
Cat.No: T36680
Synonym:
Target: Serine/threonin kinase, MAPK, LIM Kinase, TGF-beta/Smad, AAK1 (AP2 associated kinase 1)
TG 100572 Hydrochloride
Cat.No: T13156L
Synonym:
Target: VEGFR, FGFR, PDGFR, Src
FGFR1 inhibitor-9
Cat.No: T78832
Synonym:
Target: FGFR
TG 100572
Cat.No: T13156
Synonym:
Target: VEGFR
TG 100801 Hydrochloride
Cat.No: T13157L
Synonym:
Target: VEGFR
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