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Search Results for " a. membranaceus "

1

抑制剂 & 化合物

14

天然产物

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Cat. No. Product Name Target Signaling Pathways
T32320 Julocrotine

Julocrotonine,Julocrotine, (-)-

Julocrotine is a type of glutarimide alkaloid from Croton membranaceus.

化合物

Julocrotine
Cat.No: T32320
Synonym: Julocrotonine,Julocrotine, (-)-
Target:
Cat. No. Product Name Target Signaling Pathways
T3859 Isomucronulatol

7,2'-Dihydroxy-3',4'-dimethoxyisoflavan,7,2'-二羟基-3',4'-二甲氧基异黄烷,异短尖剑豆酚

Others Others
Isomucronulatol (7,2'-Dihydroxy-3',4'-dimethoxyisoflavan) 是一种黄酮类化合物,分离自 A. membranaceus 根。它在体外对 LPS 刺激产生的 IL-12 p40 有抑制作用,具有潜在的抗炎作用。
T3848 7,2′-Dihydroxy-3′,4′-dimethoxyisoflavan 7-O-β-D-glucoside

Isomucronulatol 7-O-glucoside,7,2'-dihydroxy-3',4'-dimethoxyisoflavane-7-O-glucoside,黄芪异黄烷苷

Others Others
7,2′-Dihydroxy-3′,4′-dimethoxyisoflavan 7-O-β-D-glucoside (Isomucronulatol 7-O-glucoside) 是一种具有生物活性的异黄酮,分离自黄芪中。
T6395 Astragaloside A

Astragalin A,黄芪甲苷,Astramembrannin I

Calcium Channel Membrane transporter/Ion channel; Metabolism
Astragaloside A (Astramembrannin I) 是从黄芪中分离得到的初级纯皂苷,已广泛用于心血管疾病的治疗。
T0724 Formononetin

Biochanin B,Flavosil,刺芒柄花素,Formononetol

Apoptosis; FGFR Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
Formononetin (Flavosil) 是一种 FGFR2抑制剂,IC50约为4.31 μM。 它是一种 O-甲基化的异黄酮,是来自黄芪根的植物雌激素,可有效抑制血管生成和肿瘤生长。
T5S0836 Isoastragaloside II

黄芪甲苷VII,Astrasieversianin VII

Others Others
Isoastragaloside II (Astrasieversianin VII) 是一种是从黄芪毛状根培养分离得到的黄芪甲苷。
TN1772 Isoastilbin

Anti-infection; Tyrosinase; Antibacterial Microbiology/Virology; Proteases/Proteasome
Isoastilbin 是Rhizoma Smilacis glabrae 和Astragalus membranaceus 中的二氢黄酮醇糖苷。它抑制酪氨酸酶活性,还抑制葡萄糖基转移酶,IC50值为 54.3 μg/mL。它具有神经保护、抗氧化、抗微生物和抗凋亡活性,可研究阿尔茨海默氏病。
T3925 Astragaloside I

黄芪皂苷I,Cyclosieversioside B,Astrasieversianin IV

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
Astragaloside I (Cyclosieversioside B) 是从黄芪中分离得到天然产物。它可通过 Wnt/β-catenin 信号通路刺激成骨细胞分化,可用于成骨活性研究。
T5575 Cycloastragenol

环黄芪醇,Cyclogalegenol,Astramembrangenin

Epigenetic Reader Domain; Telomerase Chromatin/Epigenetic; DNA Damage/DNA Repair
Cycloastragenol (Astramembrangenin) 是一种三萜皂苷类化合物,是黄芪主要活性成分的水解产物,具有抗氧化、抗炎、抗衰老、抗凋亡和心血管保护作用。它是端粒酶激活剂,可以延长端粒,还能缓解与年龄相关的骨丢失,改善骨微结构和生物力学特性。
TN6967 (R)-Isomucronulatol

(-)-Isomucronulatol,2H-1-Benzopyran-7-ol

Apoptosis Apoptosis
(R)-Isomucronulatol (2H-1-Benzopyran-7-ol) 是一种可从黄芪、刺槐、虎杖和甘草叶片中提取得到的类黄酮,抑制BMSCs 在TNF-α微环境中的增殖和凋亡。(R)-Isomucronulatol 具有潜在的抗炎活性。
T2973 Astragaloside IV

AST-IV,黄芪甲苷IV,AS-IV,黄芪皂苷 IV

MMP; ERK; Estrogen/progestogen Receptor; JNK Endocrinology/Hormones; MAPK; Proteases/Proteasome
Astragaloside IV (AS-IV) 是从黄芪中分离得到的一种皂苷,抑制ERK1/2和JNK 激活,在乳腺癌细胞 MDA-MB-231 中,下调(MMP)-2和(MMP)-9的信号通路。
TN4561 N-Decyl-4-methoxyaniline

IL Receptor; TNF Apoptosis; Immunology/Inflammation
Methylnissolin is a natural product from A. membranaceus.
TN2748 2''-Acetylastragalin

Others Others
2''-Acetylastragalin is a natural product from Astragalus membranaceus.
T83138 Aloinoside A

Aloinoside A,一种可自黄芪分离的芦荟素,为Aloinoside B的对映异构体,应用于代谢研究的生物标志物。其通过大鼠肠道细菌代谢生成物包括芦荟苷、异芦荟苷及羟基代谢物。
TN2344 Swainsonine

Tridolgosir

Apoptosis; Others; Antibiotic Apoptosis; Microbiology/Virology; Others
Swainsonine (Tridolgosir) 是一种从黄芪中分离出来的一种生物碱,是一种强效和可逆的α-甘露糖苷酶抑制剂。Swainsonine 具有抗肿瘤活性,可诱导细胞凋亡和细胞周期停滞在 G2/M 期。

天然产物

Isomucronulatol
Cat.No: T3859
Synonym: 7,2'-Dihydroxy-3',4'-dimethoxyisoflavan,7,2'-二羟基-3',4'-二甲氧基异黄烷,异短尖剑豆酚
Target: Others
7,2′-Dihydroxy-3′,4′-dimethoxyisoflavan 7-O-β-D-glucoside
Cat.No: T3848
Synonym: Isomucronulatol 7-O-glucoside,7,2'-dihydroxy-3',4'-dimethoxyisoflavane-7-O-glucoside,黄芪异黄烷苷
Target: Others
Astragaloside A
Cat.No: T6395
Synonym: Astragalin A,黄芪甲苷,Astramembrannin I
Target: Calcium Channel
Formononetin
Cat.No: T0724
Synonym: Biochanin B,Flavosil,刺芒柄花素,Formononetol
Target: Apoptosis, FGFR
Isoastragaloside II
Cat.No: T5S0836
Synonym: 黄芪甲苷VII,Astrasieversianin VII
Target: Others
Isoastilbin
Cat.No: TN1772
Synonym:
Target: Anti-infection, Tyrosinase, Antibacterial
Astragaloside I
Cat.No: T3925
Synonym: 黄芪皂苷I,Cyclosieversioside B,Astrasieversianin IV
Target: Wnt/beta-catenin
Cycloastragenol
Cat.No: T5575
Synonym: 环黄芪醇,Cyclogalegenol,Astramembrangenin
Target: Epigenetic Reader Domain, Telomerase
(R)-Isomucronulatol
Cat.No: TN6967
Synonym: (-)-Isomucronulatol,2H-1-Benzopyran-7-ol
Target: Apoptosis
Astragaloside IV
Cat.No: T2973
Synonym: AST-IV,黄芪甲苷IV,AS-IV,黄芪皂苷 IV
Target: MMP, ERK, Estrogen/progestogen Receptor, JNK
N-Decyl-4-methoxyaniline
Cat.No: TN4561
Synonym:
Target: IL Receptor, TNF
2''-Acetylastragalin
Cat.No: TN2748
Synonym:
Target: Others
Aloinoside A
Cat.No: T83138
Synonym:
Target:
Swainsonine
Cat.No: TN2344
Synonym: Tridolgosir
Target: Apoptosis, Others, Antibiotic
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