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Search Results for " 盐酸多巴胺 "

6

抑制剂 & 化合物

5

天然产物

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Cat. No. Product Name Target Signaling Pathways
T12352 Oxidopamine hydrochloride

6-Hydroxydopamine hydrochloride,6-OHDA hydrochloride,6-羟基多巴胺盐酸盐

Mitophagy; Dopamine Receptor; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) 是一种神经递质多巴胺拮抗剂,可选择性地破坏多巴胺能神经元,是一种广泛使用的神经毒素。
T13512 5-Hydroxydopamine hydrochloride

Antifungal Microbiology/Virology
5-Hydroxydopamine hydrochloride 是人体尿液中的一种天然胺,对卢克斯普受体的 IC50 值为 22 µM 。5-Hydroxydopamine hydrochloride 具有潜在的抗菌活性和抗癌活性。
T12352L Oxidopamine hydrobromide

6-Hydroxydopamine hydrobromide,6-羟基多巴胺氢溴酸盐,6-OHDA hydrobromide

Mitophagy; Dopamine Receptor; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Oxidopamine hydrobromide (6-OHDA hydrobromide) 是一种神经递质多巴胺拮抗剂,可选择性地破坏多巴胺能神经元,是一种广泛使用的神经毒素。
T23234 Rimcazole dihydrochloride

Others Others
Rimcazole dihydrochloride 是 Rimcazole 的盐酸盐,是一种σ受体拮抗剂。Rimcazole dihydrochloride 还与多巴胺转运蛋白结合,抑制多巴胺的摄取。
T6188 Desvenlafaxine succinate hydrate

O-Desmethylvenlafaxine succinate hydrate,WY 45233 Succinate,琥珀酸去甲文拉法辛,Desvenlafaxine Succinate

5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Desvenlafaxine succinate hydrate (WY 45233 Succinate) 是 Venlafaxine 主要代谢物的丁二酸盐形式,在人多巴胺转运体上显示弱的结合亲和力。它是具有口服活性的、能透过血脑屏障的5-HT 和 去甲肾上腺素再摄取的抑制剂,对 hSERT 和 hNET 的IC50值分别为47.3 nM 和531.3 nM。
T1580 Desvenlafaxine

去甲文拉法辛,WY 45233 Succinate,O-Desmethylvenlafaxine

5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Desvenlafaxine (O-Desmethylvenlafaxine) 是 Venlafaxine 主要代谢物的丁二酸盐形式,在人多巴胺转运体上显示弱的结合亲和力。它是一种具有口服活性的、能透过血脑屏障的5-HT 和去甲肾上腺素再摄取的抑制剂,对 hSERT 和 hNET 的IC50值分别为 47.3 nM 和 531.3 nM。

化合物

Oxidopamine hydrochloride
Cat.No: T12352
Synonym: 6-Hydroxydopamine hydrochloride,6-OHDA hydrochloride,6-羟基多巴胺盐酸盐
Target: Mitophagy, Dopamine Receptor, Autophagy
5-Hydroxydopamine hydrochloride
Cat.No: T13512
Synonym:
Target: Antifungal
Oxidopamine hydrobromide
Cat.No: T12352L
Synonym: 6-Hydroxydopamine hydrobromide,6-羟基多巴胺氢溴酸盐,6-OHDA hydrobromide
Target: Mitophagy, Dopamine Receptor, Autophagy
Rimcazole dihydrochloride
Cat.No: T23234
Synonym:
Target: Others
Desvenlafaxine succinate hydrate
Cat.No: T6188
Synonym: O-Desmethylvenlafaxine succinate hydrate,WY 45233 Succinate,琥珀酸去甲文拉法辛,Desvenlafaxine Succinate
Target: 5-HT Receptor, Serotonin Transporter, Norepinephrine
Desvenlafaxine
Cat.No: T1580
Synonym: 去甲文拉法辛,WY 45233 Succinate,O-Desmethylvenlafaxine
Target: 5-HT Receptor, Serotonin Transporter, Norepinephrine
Cat. No. Product Name Target Signaling Pathways
T1644 Dopamine hydrochloride

盐酸多巴胺,Dopamine HCl,ASL279

Ferroptosis; Dopamine Receptor; 5-HT Receptor; Endogenous Metabolite Apoptosis; GPCR/G Protein; Metabolism; Neuroscience
Dopamine hydrochloride (ASL279) 是在脑黑质、脑腹侧被盖区和下丘脑中产生的一种天然儿茶酚胺,由二羟基苯丙氨酸脱羧形成,是去甲肾上腺素和肾上腺素的前体。它通过 D2 多巴胺受体来诱导 VEGFR2 的内吞作用,有促进血管生成活性。
T4710 3-Methoxytyramine hydrochloride

3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride),3-O-甲基多巴胺盐酸盐

Others; Endogenous Metabolite; Drug Metabolite Metabolism; Others
3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) 是多巴胺的无活性代谢物,能够活化痕量胺相关受体1 。
T8149 Dobutamine hydrochloride

盐酸多巴酚丁胺,Dobutamine (hydrochloride)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Dobutamine hydrochloride (Dobutamine(hydrochloride)) 是一种合成的儿茶酚胺,可作用于肾上腺素能受体α1-AR、β1-AR 和β2-AR,是一种选择性的 β1-AR 受体激动剂,对 α1-AR 和 β2-AR 作用相对较弱。它能够增加心输出量,矫正低灌注。
T6871 L-Glutamic acid monosodium salt

Monosodium glutamate,谷氨酸单钠盐,Glutacyl,Glutavene,L-谷氨酸单钠盐,Ajinomoto,MSG

Apoptosis; Ferroptosis; GluR; iGluR Apoptosis; Membrane transporter/Ion channel; Neuroscience
L-Glutamic acid monosodium salt (MSG) 作为兴奋性氨基酸神经递质,是谷氨酸盐受体所有亚型的激动剂,对多巴胺从神经末梢释放的过程有激动作用。
T2A2497 L-Glutamic acid

谷氨酸,(S)-Glutamic acid,glutamic acid,(+)-L-Glutamic acid,Aciglut,L-谷氨酸,glutacid,Glutaminol

Apoptosis; Ferroptosis; Endogenous Metabolite; iGluR Apoptosis; Membrane transporter/Ion channel; Metabolism; Neuroscience
L-Glutamic acid (Glutaminol) 作为一种兴奋性氨基酸神经递质,为谷氨酸盐受体所有亚型的激动剂,对多巴胺从神经末梢释放的过程有激动作用。

天然产物

Dopamine hydrochloride
Cat.No: T1644
Synonym: 盐酸多巴胺,Dopamine HCl,ASL279
Target: Ferroptosis, Dopamine Receptor, 5-HT Receptor, Endogenous Metabolite
3-Methoxytyramine hydrochloride
Cat.No: T4710
Synonym: 3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride),3-O-甲基多巴胺盐酸盐
Target: Others, Endogenous Metabolite, Drug Metabolite
Dobutamine hydrochloride
Cat.No: T8149
Synonym: 盐酸多巴酚丁胺,Dobutamine (hydrochloride)
Target: Adrenergic Receptor
L-Glutamic acid monosodium salt
Cat.No: T6871
Synonym: Monosodium glutamate,谷氨酸单钠盐,Glutacyl,Glutavene,L-谷氨酸单钠盐,Ajinomoto,MSG
Target: Apoptosis, Ferroptosis, GluR, iGluR
L-Glutamic acid
Cat.No: T2A2497
Synonym: 谷氨酸,(S)-Glutamic acid,glutamic acid,(+)-L-Glutamic acid,Aciglut,L-谷氨酸,glutacid,Glutaminol
Target: Apoptosis, Ferroptosis, Endogenous Metabolite, iGluR
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