Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) 是一种神经保护剂,是一种弱的非麦角类多巴胺受体激动剂。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
1 mg | ¥ 182 | 现货 | ||
5 mg | ¥ 463 | 现货 | ||
10 mg | ¥ 747 | 现货 | ||
25 mg | ¥ 1,580 | 现货 | ||
50 mg | ¥ 2,660 | 现货 | ||
100 mg | ¥ 3,920 | 现货 | ||
200 mg | ¥ 5,580 | 现货 | ||
1 mL * 10 mM (in DMSO) | ¥ 493 | 现货 |
产品描述 | Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine agonist. |
体外活性 | Dextromethorphan has been found to have neuroprotective effects and is being studied for the treatment of amyotrophic lateral sclerosis (ALS). Dexpramipexole reduces mitochondrial reactive oxygen species (ROS) production, inhibits the activation of apoptosis pathways, and improves cell survival in response to various neurotoxins and β-amyloid neurotoxicity. Compared with the S-(-) isomer, dextromethorphan has lower dopamine agonist activity. |
别名 | 普拉克索杂质D, KNS-760704 dihydrochloride, R-(+)-Pramipexole dihydrochloride, 右旋普拉克索二盐酸盐, (R)-Pramipexole dihydrochloride |
分子量 | 284.25 |
分子式 | C10H19Cl2N3S |
CAS No. | 104632-27-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (351.80 mM)
H2O: 100 mg/mL (351.80 mM), Sonication is recommended.
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO / H2O | 1 mM | 3.518 mL | 17.5901 mL | 35.1803 mL | 87.9507 mL |
5 mM | 0.7036 mL | 3.518 mL | 7.0361 mL | 17.5901 mL | |
10 mM | 0.3518 mL | 1.759 mL | 3.518 mL | 8.7951 mL | |
20 mM | 0.1759 mL | 0.8795 mL | 1.759 mL | 4.3975 mL | |
50 mM | 0.0704 mL | 0.3518 mL | 0.7036 mL | 1.759 mL | |
100 mM | 0.0352 mL | 0.1759 mL | 0.3518 mL | 0.8795 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
Dexpramipexole dihydrochloride 104632-27-1 GPCR/G Protein Neuroscience Dopamine Receptor inhibit Inhibitor KNS 760704 Dihydrochloride KNS-760704 Dihydrochloride (R)-Pramipexole KNS760704 普拉克索杂质D KNS-760704 dihydrochloride R-(+)-Pramipexole dihydrochloride R-Pramipexole Dihydrochloride Pramipexole Dexpramipexole 右旋普拉克索二盐酸盐 KNS 760704 Pramipexole Dihydrochloride KNS760704 Dihydrochloride Dexpramipexole Dihydrochloride (R)-Pramipexole dihydrochloride R-Pramipexole KNS-760704 inhibitor