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Search Results for " prolactin "

26

抑制剂 & 化合物

2

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
TP1767	Prolactin Releasing Peptide (12-31), human
	Prolactin Releasing Peptide (1-31), human is a high affinity GPR10 ligand that cause the release of the prolactin
TP1769	Prolactin Releasing Peptide (1-31), human
	Prolactin Releasing Peptide (1-31), human is a high affinity GPR10 ligand that cause the release of the prolactin. Human and rat Prolactin Releasing Peptide (1-31) binds to GPR10 with Kis of 1.03 and 0.33 nM, respectively.Prolactin-releasing peptide is a
T81390	Prolactin-Releasing Peptide (1-31) (rat)
	Prolactin-Releasing Peptide (1-31) (rat) 通过减少禁食诱导的大鼠食物摄入，有效提升血浆LH、FSH及睾酮水平。
T81391	Prolactin-Releasing Peptide (12-31), rat
	Prolactin-Releasing Peptide (12-31), rat 为催乳素释放肽的一个段落，对 GPR10 受体具有高度亲和性，并能在转染了 PrRP 受体的 CHOK1 细胞中激发钙离子动员。
T78006	Prolactin Releasing Peptide (1-31), human acetate
	ProlactinReleasing Peptide (1-31), human (acetate) 是一款针对 GPR10 的高亲和力配体，并具备诱导催乳素释放的功能。该肽段与人类和大鼠的 GPR10 结合力极强，Ki 值分别为 1.03 nM 和 0.33 nM，适用于针对下丘脑-垂体轴进行的生物医学研究。
T4008	Metergoline 甲麦角林,Methergoline,Liserdol	Dopamine Receptor; 5-HT Receptor; Sodium Channel	GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
	Metergoline (Methergoline) 是多巴胺激动剂和血清素拮抗剂。它是 h5-HT7受体的高亲和力配体，Ki 为 16 nM。它还是可逆神经 Na+通道抑制剂，用于研究季节性情绪障碍、催乳激素调节。
T7943	Fluphenazine decanoate	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Fluphenazine decanoate 是一种高度连续的多巴胺 D2受体阻滞剂，是一种长效吩噻嗪抗精神病药，用于精神分裂症的研究。
T6956L	Protirelin Acetate(24305-27-9 free base) Thyroliberin Acetate,TRF Acetate,Synthetic thyrotropin-releasing hormone Acetate,Lopremone Acetate,pGlu-His-Pro-NH2 Acetate,TRH Acetate	Thyroid hormone receptor(THR)	Endocrinology/Hormones
	Protirelin Acetate(24305-27-9 free base) (Thyroliberin Acetate) 是一种三肽，可刺激促甲状腺素和催乳素的释放。
TP1022	Protirelin Acetate TSH-RF Acetate,TRH Acetate,TRF Acetate,醋酸普罗瑞林	Thyroid hormone receptor(THR); Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Protirelin Acetate (TRH Acetate) 是高度保守的神经肽，具有促甲状腺激素水平的激素控制作用，及神经调节的能力。
T21649L	GnRH Associated Peptide (GAP) (1-13), human Acetate GnRH Associated Peptide (GAP) (1-13), human Acetate (100111-07-7 Free base)	Others	Others
	GnRH Associated Peptide (GAP) (1-13), human Acetate 被发现是催乳素分泌的有效抑制剂并刺激促性腺激素的释放。用对应于 GAP 序列的肽进行主动免疫导致催乳素分泌大大增加。
TP1310	Neurotensin	Neurotensin Receptor	GPCR/G Protein
	Neurotensin 是一种 13 个氨基酸的神经肽，参与调节促黄体激素和催乳素的释放，并与多巴胺能系统有显着的相互作用。它作为细胞有丝分裂原，作用于各种结肠直肠癌和胰腺癌。
TP1937L1	RFRP-1 (human) acetate(311309-25-8 free base)	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	RFRP-1 (human) acetate(311309-25-8 free base) 是一种有效的内源性 NPFF 受体激动剂（NPFF2 和 NPFF1 的 EC50 值分别为 0.0011 和 29 nM）。它减弱离体大鼠和兔心肌细胞的收缩功能。降低心率、每搏输出量、射血分数和心输出量，并增加大鼠的血浆催乳素水平。 GnIH 同系物。
T25671	Lergotrile LY-79907,LY79907,LY 79907
	Lergotrile is used as an enzyme Inhibitor (Prolactin).
T25671L	Lergotrile mesylate LY83636,LY-83636,LY 83636
	Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.
T24003	Disulergine CM 29717,CH 29717,CH 29-717
	Disulergine is a dopamine receptor agonist. It also prolactin release-inhibiting 8 alpha-amino-ergoline.
T61065	Lisuride
	Lisuride is an orally active agonist of dopamine D2 receptors, classified as an ergot derivative. It is utilized for research purposes relating to Parkinson's disease, migraine, and elevated prolactin levels [1] [2].
T75947	RFRP-1(human) TFA
	RFRP-1(human) TFA, an endogenous NPFF receptor agonist, exhibits potent activity with EC50 values of 0.0011 nM for NPFF2 and 29 nM for NPFF1. It significantly diminishes the contractile function of isolated rat and rabbit cardiac myocytes. Moreover, it decreases heart rate, stroke volume, ejection fraction, and cardiac output, while elevating plasma prolactin levels in rats.
T25443	FW 34569 FW-34-569,FW34569,FW 34-569,FW-34569,FW34-569
	FW 34569 is an enkephalin analogue. It stimulated growth hormones and prolactin release and inhibited the release of cortisol and LH, while FSH remained unchanged.
T68551	Cabergoline diphosphate
	Cabergoline diphosphate is a dopamine D2 receptor agonist used for prolactinoma treatment. Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels.
T77258	Trh-gly
	Trh-gly (TRH-glycine) 是促甲状腺素 (TSH) 释放激素 (TRH) 的前体，可释放促甲状腺素和催乳素。
T8775	Lisuride maleate R-(+)-LISURIDE HYDROGEN MALEATE
	Lisuride maleate is an agonist of Dopamine receptor and anti-Parkinson's agent. Displays high affinity for D2, D3 and D4 receptors along with 5-HT1A. Exhibits some 5-HT2B receptor antagonist properties. Decreases prolactin release; reduces inflammatory me
TP1937	RFRP-1(human) RFRP-1 (human)
	Potent endogenous NPFF receptor agonist (EC50 values are 0.0011 and 29 nM for NPFF2 and NPFF1, respectively). Attenuates contractile function of isolated rat and rabbit cardiac myocytes. Reduces heart rate, stroke volume, ejection fraction and cardiac out
T81598	Org OD 02-0 10-Ethenyl-19-norprogesterone	p38 MAPK	MAPK
	Org OD 02-0（10-Ethenyl-19-norprogesterone）为mPRα（膜孕酮受体α）特异性激动剂，IC50值为33.9 nM。该化合物能够激活MAPK活性，并且能抑制催乳素（PRL）的分泌。
T80114	FA-Ala-Arg	Endogenous Metabolite	Metabolism
	FA-Ala-Arg是一种携带呋喃丙烯酰基的二肽，它能够分解产生精氨酸，并因此提高精氨酸水平，后者可转化为一氧化氮(NO)。该化合物还可增强MCF-7细胞产生NO的能力，并在催乳素(PRL)处理下提升细胞存活率，其中PRL会调节CPD mRNA的表达。
T83756	S1H TFA Site 1-binding Helix
	S1H是一种人造肽类模拟物，模仿人类生长激素的第36至51个氨基酸，且为生长激素受体的拮抗剂。在溶液中呈现α-螺旋结构，并在100和200纳摩尔（nM）的浓度下，能降低SK-MEL-28和MALME-3M黑色素瘤细胞系以及IM-9 B细胞淋巴细胞中，由人类生长激素及泌乳素诱导的STAT5磷酸化。
TP1532	γ-2-MSH (41-58), amide
	Melanocortin (MC) 3-MSH (Melanocyte-Stimulating Hormone) is believed to signal through the MC 3 receptor. It induces a sustained increase in intracellular free calcium levels ([Ca2+]i) in a subpopulation of pituitary cells. Most of the cells responding to

化合物

Prolactin Releasing Peptide (12-31), human

Cat.No: TP1767

Prolactin Releasing Peptide (1-31), human

Cat.No: TP1769

Prolactin-Releasing Peptide (1-31) (rat)

Cat.No: T81390

Prolactin-Releasing Peptide (12-31), rat

Cat.No: T81391

Prolactin Releasing Peptide (1-31), human acetate

Cat.No: T78006

Cat.No: T4008

Synonym: 甲麦角林,Methergoline,Liserdol

Target: Dopamine Receptor, 5-HT Receptor, Sodium Channel

Fluphenazine decanoate

Cat.No: T7943

Target: Dopamine Receptor

Protirelin Acetate(24305-27-9 free base)

Cat.No: T6956L

Synonym: Thyroliberin Acetate,TRF Acetate,Synthetic thyrotropin-releasing hormone Acetate,Lopremone Acetate,pGlu-His-Pro-NH2 Acetate,TRH Acetate

Target: Thyroid hormone receptor(THR)

Protirelin Acetate

Cat.No: TP1022

Synonym: TSH-RF Acetate,TRH Acetate,TRF Acetate,醋酸普罗瑞林

Target: Thyroid hormone receptor(THR), Endogenous Metabolite

GnRH Associated Peptide (GAP) (1-13), human Acetate

Cat.No: T21649L

Synonym: GnRH Associated Peptide (GAP) (1-13), human Acetate (100111-07-7 Free base)

Target: Others

Cat.No: TP1310

Target: Neurotensin Receptor

RFRP-1 (human) acetate(311309-25-8 free base)

Cat.No: TP1937L1

Target: Neuropeptide Y Receptor

Cat.No: T25671

Synonym: LY-79907,LY79907,LY 79907

Lergotrile mesylate

Cat.No: T25671L

Synonym: LY83636,LY-83636,LY 83636

Cat.No: T24003

Synonym: CM 29717,CH 29717,CH 29-717

Cat.No: T61065

RFRP-1(human) TFA

Cat.No: T75947

Cat.No: T25443

Synonym: FW-34-569,FW34569,FW 34-569,FW-34569,FW34-569

Cabergoline diphosphate

Cat.No: T68551

Cat.No: T77258

Lisuride maleate

Cat.No: T8775

Synonym: R-(+)-LISURIDE HYDROGEN MALEATE

Cat.No: TP1937

Synonym: RFRP-1 (human)

Cat.No: T81598

Synonym: 10-Ethenyl-19-norprogesterone

Target: p38 MAPK

Cat.No: T80114

Target: Endogenous Metabolite

Cat.No: T83756

Synonym: Site 1-binding Helix

γ-2-MSH (41-58), amide

Cat.No: TP1532

Cat. No.	Product Name	Target	Signaling Pathways
T14853	Cabergoline FCE-21336,卡麦角林	Dopamine Receptor; 5-HT Receptor; Autophagy	Autophagy; GPCR/G Protein; Neuroscience
	Cabergoline (FCE-21336) 是一种麦角衍生的多巴胺 D2亚类受体激动剂，高亲和力作用于D2、D3和5-HT2B 受体，Ki 分别为 0.7、1.5 和 1.2。
T6956	Protirelin Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,Thyroliberin,TRH,普罗瑞林,TRF	Thyroid hormone receptor(THR); Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Protirelin (Thyroliberin) 是高度保守的神经肽，具有促甲状腺激素水平的激素控制作用，及神经调节功能。

天然产物

Cat.No: T14853

Synonym: FCE-21336,卡麦角林

Target: Dopamine Receptor, 5-HT Receptor, Autophagy

Cat.No: T6956

Synonym: Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,Thyroliberin,TRH,普罗瑞林,TRF

Target: Thyroid hormone receptor(THR), Endogenous Metabolite

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