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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T0378 Oxybuprocaine hydrochloride

Risedronic Acid,Oxybuprocaine HCl,奥布卡因盐酸盐

Sodium Channel Membrane transporter/Ion channel
Oxybuprocaine hydrochloride (Oxybuprocaine HCl) 是可逆的钠通道阻断剂,可防止角膜,结膜和巩膜中疼痛神经的冲动传播。Oxybuprocaine hydrochloride 专用于眼科与耳鼻喉科。
T0924 Benzocaine

苯唑卡因,苯佐卡因

Others; MRP; Sodium Channel Immunology/Inflammation; Membrane transporter/Ion channel; Others
Benzocaine 作用电压门控 Na+通道的共同受体,+30 mV 下的 IC50为0.8 mM。
T0222 Proparacaine hydrochloride

盐酸丙美卡因,Proparacaine HCl,Proxymetacaine Hydrochloride

Apoptosis; Sodium Channel Apoptosis; Membrane transporter/Ion channel
Proparacaine hydrochloride (Proparacaine HCl) 是 Lidocaine 的衍生物,具有糖皮质激素样活性和免疫调节作用。
T0802 Procaine hydrochloride

Novocaine HCl,Procaine HCl,盐酸普鲁卡因

Histone Demethylase; 5-HT Receptor; DNA/RNA Synthesis; Sodium Channel; NMDAR; AChR Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Procaine hydrochloride (Novocaine HCl) 是DNA 脱甲基剂,是一种苯甲酸衍生物,具有局部麻醉和抗心律失常特性。
T6782 Benzocaine hydrochloride

Benzocaine HCl,Ethyl p-aminobenzoate hydrochloride,Ethyl 4-aminobenzoate hydrochloride

Sodium Channel Membrane transporter/Ion channel
Benzocaine hydrochloride (Ethyl 4-aminobenzoate hydrochloride) 是一种表面麻醉剂,通过阻止脉冲沿神经纤维和神经末梢传递而起作用。

化合物

Oxybuprocaine hydrochloride
Cat.No: T0378
Synonym: Risedronic Acid,Oxybuprocaine HCl,奥布卡因盐酸盐
Target: Sodium Channel
Benzocaine
Cat.No: T0924
Synonym: 苯唑卡因,苯佐卡因
Target: Others, MRP, Sodium Channel
Proparacaine hydrochloride
Cat.No: T0222
Synonym: 盐酸丙美卡因,Proparacaine HCl,Proxymetacaine Hydrochloride
Target: Apoptosis, Sodium Channel
Procaine hydrochloride
Cat.No: T0802
Synonym: Novocaine HCl,Procaine HCl,盐酸普鲁卡因
Target: Histone Demethylase, 5-HT Receptor, DNA/RNA Synthesis, Sodium Channel, NMDAR, AChR
Benzocaine hydrochloride
Cat.No: T6782
Synonym: Benzocaine HCl,Ethyl p-aminobenzoate hydrochloride,Ethyl 4-aminobenzoate hydrochloride
Target: Sodium Channel
Cat. No. Product Name Target Signaling Pathways
T0894 Thiamine hydrochloride

盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride

Apoptosis; HBV; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology
Thiamine hydrochloride (Vitamin B1) 是一种必需的微量营养素,是许多中枢代谢酶的辅因子。

天然产物

Thiamine hydrochloride
Cat.No: T0894
Synonym: 盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride
Target: Apoptosis, HBV, Endogenous Metabolite
TargetMol Loading
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