9
7
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T26582 | AIM-102 | ||
AIM-102, a nonsteroidal, immune modulating, anti-inflammatory drug, is used potentially for the treatment of allergic asthma. | |||
T82593 | Debotansine | ||
Debotansine是具有免疫调节和抗肿瘤作用的化合物。 | |||
T81114 | Spns2-IN-1 | LPL Receptor | GPCR/G Protein |
Spns2-IN-1,作为一种Spns2依赖性S1P转运(Spns2)的有效抑制剂,其IC50值为1.4±0.3 μM,对免疫反应有着显著影响<sup>[1]。 | |||
T74651 |
L-Inosine
|
||
L-Inosine 是 L-构型形式的 Inosine。Inosine 是一种由腺苷分解代谢产生的内源性嘌呤核苷。Inosine 具有抗炎免疫调节,抗伤害和神经保护作用。 | |||
T80089 |
HCV-1 e2 Protein (554-569) (TFA)
|
||
HCV-1 e2 Protein (554-569) TFA 为丙型肝炎病毒(HCV)e2 蛋白关键抗原区段,含一个假定 N-糖基化位点,该位点早先推测会影响 e2 蛋白的免疫识别。 | |||
T76748 | Foralumab | ||
Foralumab(NI-0401)为口服有效的人源化单克隆抗体,针对CD3进行靶向。其能够调控NSG小鼠体内,由人类造血干细胞重建的人类细胞的免疫反应。 | |||
T74910 | ODN 24888 | ||
ODN 24888 是一种鸟嘌呤修饰的抑制性寡核苷酸 (INH-ODN),对TLR7/TLR9介导的信号通路表现出强烈的抑制作用。ODN 24888 损害 IFN-α 水平和NF-κB 激活,抑制IL-6的释放。ODN 24888 参与免疫和炎症应答,可作为疫苗佐剂使用。 | |||
T76022 |
Chemerin-9 (149-157) (TFA)
|
||
Chemerin-9 (149-157) TFA 作为趋化因子样受体1 (CMKLR1) 的有效激动剂,展现出抗炎活性,并能促进Akt与ERK磷酸化及活性氧生成,进而改善Aβ1-42诱发的记忆障碍。此外,该化合物还参与调节免疫反应、脂肪细胞分化以及糖代谢。 | |||
T37644 |
Bengamide B
|
||
Potent inhibitor of NF-κB activation (IC50 = 85 nM); decreases IκBα phosphorylation. Attenuates LPS-induced nitric oxide production and expression of TNF-α, IL-6 and MCP. Suppresses proliferation of HeLa and HCT116 cells. Anti-inflammatory and antitumor. Hu et al (2007) Regulation of c-Src nonreceptor tyrosine kinase activity by bengamide A through inhibition of methionine aminopeptidases. Chem.Biol. 14 764 PMID:17656313 |Johnson et al (2012) Myxobacteria versus sponge-derived alkaloids: the be... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8689 |
Chloroquine
CQ,氯喹 |
SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy | Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome |
Chloroquine 是一种 Toll 样受体抑制剂,可以抑制自噬。Chloroquine 具有抗疟疾和抗炎活性,广泛用于治疗疟疾和类风湿性关节炎。Chloroquine 还具有抗 SARS-CoV-2 (COVID-19) 活性、抗 HIV-1 活性。 | |||
T0194 |
Chloroquine phosphate
Chloroquine diphosphate,Aralen phosphate,磷酸氯喹,Chingamin phosphate |
SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy | Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome |
Chloroquine phosphate (Aralen phosphate) 是广泛用于疟疾和类风湿性关节炎的抗疟疾和抗炎剂。它是autophagy 和toll-like receptors 抑制剂,有效抑制SARS-CoV-2(COVID-19) 感染 (EC50=1.13 μM)。 | |||
T7544 |
Fucoidan
岩藻多糖 |
Others | Others |
Fucoidan 是一种 α-淀粉酶和 α-葡萄糖苷酶的有效抑制剂,是一种生物特性多糖。 它具有抗凝血,抗肿瘤,抗氧化和抗脂肪特性。 | |||
T15705 |
Laminaran
β-1,3-Glucan |
||
Laminaran 是一种从褐藻中分离出来的 β-1-3-葡聚糖,常作为 Dectin-1 的典型配体,具有抗癌、免疫调节和辐射防护作用。 Laminaran 可被葡糖酶催化。Laminaran 在体内外实验中显示出抗肿瘤活性,可用于预防和治疗癌症。 | |||
T4S1469 |
Cucurbitacin IIb
葫芦素IIB,雪胆素乙 |
Apoptosis; Others | Apoptosis; Others |
Cucurbitacin IIb 是一种雪胆中的活性成分。它阻碍 STAT3,JNK 和 Erk1/2 的磷酸化,提高 IκB 和 NF-κB (p65) 的磷酸化水平,抑制 NF-κB (p65) 的核转位,降低 IκBα 和 TNF-α 的 mRNA 水平。它能够诱导细胞凋亡,具有抗炎作用。 | |||
T7009 |
Soyacerebroside II
|
IL Receptor; Calcium Channel | Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism |
Soyacerebroside II exhibits ionophoretic activity for Ca2+ ion. Soyacerebrosides I and II have modulating the cellular immune response effects, they show obvious inhibitory activity on IL-18 secretion in human peripheral blood mononuclear cells (PBMC). | |||
TN3741 |
Cyclocurcumin
|
TNF; ROS | Apoptosis; Immunology/Inflammation |
Cyclocurcumin, a curcumin derivative, exhibits anticancer, anti-inflammatory, and immune-modulating abilities and is a potential compound for the treatment of rheumatoid arthritis as predicted by the MM-PBSA method. It may have a therapeutic potential as |