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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
TP1148L	Glucagon-like peptide 1 (1-37), human acetate	Glucagon Receptor	GPCR/G Protein
	Glucagon-like peptide 1 (1-37), human acetate 是一种高效的 GLP-1 受体激动剂。
TP1487	Glucagon-Like Peptide (GLP) II, human
	Glucagon-like peptide 2 (GLP-2) is a recently identified intestinal epithelium-specific growth factor that has been shown to reduce the severity of inflammatory disorders of the intestine in rodent models. Currently Glucagon-Like Peptide 2 is used as a po
TP1148	Glucagon-like peptide 1 (1-37), human HuGLP-1
	Glucagon-like peptide 1 (1-37), human is a highly potent agonist of the GLP-1 receptor.Pancreatic hormone synthesized by post-translational processing of proglucagon. Unlike truncated forms of GLP-1, it has no effect on food intake in rats and does not en
TP1147	Glucagon-like peptide 1 (1-37), human TFA HuGLP-1 TFA
	Glucagon-like peptide 1 (1-37), human (TFA) is a highly potent agonist of the GLP-1 receptor, it is a kind of pancreatic hormone synthesized by post-translational processing of proglucagon.
T6203	Saxagliptin BMS-477118,沙克列汀,Onglyza,沙格列汀	Proteasome; DPP-4	Proteases/Proteasome; Ubiquitination
	Saxagliptin (BMS-477118) 是一种选择性，可逆性，竞争性和口服活性的二肽基肽酶 4 (DPP-4) (Ki= 0.6-1.3 nM) 抑制剂。Saxagliptin 能够用于 2 型糖尿病的研究。
T0178	Saxagliptin hydrate 沙格列汀单水化合物,Onglyza hydrate,BMS-477118 hydrate	Proteasome; DPP-4	Proteases/Proteasome; Ubiquitination
	Saxagliptin hydrate (Onglyza hydrate) 是一种选择性，竞争性，可逆性和口服活性的二肽基肽酶 4 (DPP-4) (Ki= 0.6-1.3 nM) 抑制剂。Saxagliptin hydrate 能够用于 2 型糖尿病的研究。
T2316	Omarigliptin MK-3102,奥格列汀	Proteasome; DPP-4	Proteases/Proteasome; Ubiquitination
	Omarigliptin (MK-3102) 是高效选择性 DPP4抑制剂，IC50=为1.6nM。
T80453	GLP-1 (1-36) amide (human, rat) Glucagon-like Peptide 1 (1-36) amide (human, rat)
	GLP-1(1-36) amide (human, rat)（人类及大鼠的胰高血糖素样肽1（1-36）酰胺）是GLP-1(7-36)酰胺的一种分子变体。该化合物能激发[14C]氨基吡啶在大鼠胃壁细胞的酶分散体中积累。
TP1157	GLP-2(1-33)(human) GLP-2 (human),Glucagon-like peptide 2 (human)
	GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.
T82309	GLP-1 (1-36) amide (human, rat) (TFA) Glucagon-like Peptide 1 (1-36) amide (human, rat) (TFA)
	GLP-1(1-36) amide (human, rat) TFA为胰高血糖素样肽1(GLP-1)-(7-36)酰胺的分子变体，能够促进[14C]氨基吡啶在大鼠壁细胞的酶分散体中的积累。
T3984	GLP-1(7-36), amide MKC 253,胰高血糖素样肽-1,Human GLP-1-(7-36)-amide,Glucagon-like Peptide 1 (7-36) amide,Glucagon-Like Peptide (GLP) I (7-36), amide, human,GLP-1(7-36),GLP-1-(7-36)-amide	Glucagon Receptor	GPCR/G Protein
	GLP-1(7-36), amide (MKC 253) 是一种生理性肠降血糖素，能够刺激胰岛素分泌。
T76330	Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide
	Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide 是一种带有生物素标签的Glucagon-like peptide-1-(7-36)，后者为一种具备提升胰岛素释放功能，从而表现出抗糖尿病活性的胃肠道肽。
T76085	Glucagon-Like Peptide 1 (GLP-1) (7-36)-Lys (Biotin), amide, human
	Glucagon-Like Peptide 1 (GLP-1) (7-36)-Lys (Biotin), amide, human 是一种被 C 端标记的生物素化 GLP-1(7-36) 酰胺。
TP2100	Avexitide Exendin-3 (9-39) amide,Exendin (9-39),艾塞那肽	Glucagon Receptor	GPCR/G Protein
	Avexitide (Exendin-3 (9-39) amide) 是一种特异竞争性的glucagon-like peptide-1 (GLP-1)受体拮抗剂。
T8355	Exenatide Exendin-4,Extendin-4	Glucagon Receptor	GPCR/G Protein
	Exenatide (Extendin-4) 是一种胰高血糖素样蛋白 1 (GLP-1) 受体激动剂。
T76559	Survodutide BI 456906	Glucagon Receptor	GPCR/G Protein
	Survodutide (BI 456906) 是一种胰高血糖素和胰高血糖素样肽 1 (GLP-1) 受体 (GLP Receptor) 双重激动剂,可降低 HbA1c16 型糖尿病的体重。
TP1103	Cotadutide acetate MEDI0382 acetate,Cotadutide acetate (1686108-82-6 Free base)	Glucagon Receptor	GPCR/G Protein
	Cotadutide acetate (MEDI0382 acetate) 是一种有效的胰高血糖素样肽-1 (GLP-1) 和胰高血糖素受体肽双重激动剂，EC50 分别为 6.9 pM 和 10.2 pM。
T12431	PF-06882961	Glucagon Receptor	GPCR/G Protein
	PF-06882961 是一种口服生物可利用的胰高血糖素样肽-1 受体 (GLP-1R) 激动剂。
T60047L	V-0219 hydrochloride V-0219 hydrochloride（878453-71-5 Free base）	Glucagon Receptor	GPCR/G Protein
	V-0219 hydrochloride 是一种具有口服活性的 glucagon-like peptide-1 receptor (GLP-1R) 正向别构调节剂 (PAM)。V-0219 能被用于肥胖相关糖尿病的研究。
T19850L	Semaglutide Acetate 索玛鲁肽醋酸盐,Semaglutide Acetate(910463-68-2 Free base)	Glucagon Receptor	GPCR/G Protein
	Semaglutide Acetate 是胰高血糖素样肽 1 (GLP-1) 受体的激动剂，可用于治疗 2 型糖尿病的研究。
T8876	PF-06882961 Tris UNII-2HJV78O0SS	Glucagon Receptor	GPCR/G Protein
	PF-06882961 Tris (UNII-2HJV78O0SS) 是一种口服生物可利用的胰高血糖素样肽-1 受体 (GLP-1R) 激动剂。
TP1469	Lixisenatide acetate (320367-13-3 free base) Lixisenatide acetate	Glucagon Receptor	GPCR/G Protein
	Lixisenatide acetate 是一种胰高血糖素样肽 1 受体的激动剂，可用于研究 2 型糖尿病。
T36579	GLP-1R Agonist DMB	Glucagon Receptor	GPCR/G Protein
	GLP-1R Agonist DMB 是胰高血糖素样肽1受体的激动剂（GLP-1R；重组人受体的 KB＝26.3nM）。
T11408	Orforglipron LY3502970,GLP-1 receptor agonist 1	Glucagon Receptor	GPCR/G Protein
	Orforglipron (LY3502970; GLP-1 receptor agonist 1) 是一种可口服的胰高血糖素样肽 (GLP-1) 受体激动剂，可用于研究成人肥胖和1型糖尿病。
TP1976L	Oxyntomodulin acetate	Glucagon Receptor	GPCR/G Protein
	Oxyntomodulin acetate 是一种 37 个氨基酸的肽激素，是一种胰高血糖素样肽 1 (GLP-1) 受体激动剂。
TP2100L	Avexitide acetate Exendin 9-39 acetate,Avexitide acetate（133514-43-9 Free base）	Glucagon Receptor	GPCR/G Protein
	Avexitide acetate (exendin 9-39）是一种有效的胰高血糖素样肽 1 受体 (GLP-1R) 拮抗剂，可用于研究肥胖后低血糖。
T76279	Retatrutide LY3437943	Glucagon Receptor	GPCR/G Protein
	Retatrutide (LY3437943) 是胰高血糖素受体、葡萄糖依赖性促胰岛素多肽受体和胰高血糖素样肽-1 受体三重激动剂,对GCGR、GIPR 和 GLP-1R 具有抑制作用。Retatrutide 可用研究肥胖症。
T3967	Exendin-4 艾塞那肽,Exenatide,Exenatide Acetate	Glucagon Receptor	GPCR/G Protein
	Exendin-4 (Exenatide) 是一种长效的 glucagon-likepeptide-1 受体激动剂(IC50: 3.22 nM)，是一种由 39 个氨基酸组成的多肽。
T76279L1	Retatrutide sodium salt Retatrutide sodium salt(2381089-83-2 free base),LY3437943 sodium salt	Glucagon Receptor	GPCR/G Protein
	Retatrutide sodium salt 是一种有效的胰高血糖素受体 (GCGR)、葡萄糖依赖性促胰岛素多肽受体 (GIPR) 和胰高血糖素样肽-1 受体 (GLP-1R) 的三重激动剂肽。Retatrutide sodium salt 可用于研究2型糖尿病和肥胖症。
T63166L	(S, R)-LSN 3318839 (S, R)-LSN 3318839(Isomer-2764704-18-7)	Glucagon Receptor	GPCR/G Protein

T78097L	Mazdutide acetate（2259884-03-0 free base） Mazdutide acetate（2259884-03-0 free base）,OXM-3 acetate,LY-3305677 acetate,IBI-362 acetate	Glucagon Receptor	GPCR/G Protein
	Mazdutide acetate 是一种高效的胰高血糖素样肽 (GLP-1R) 与胰高血糖素受体 (GCGR) 的共激动剂，是一种胃泌酸调节素类似物。Mazdutide acetate可刺激小鼠胰岛的胰岛素分泌，可用于研究肥胖和 2 型糖尿病 (T2D) 。
T15387	GLP-1R Antagonist 1	Glucagon Receptor	GPCR/G Protein
	GLP-1R Antagonist 1 (compound 5d) 是口服有效的、能透过中枢神经系统的，胰高血糖素样肽 1 受体 (GLP-1R) 的非竞争性抑制，其 IC50 值为 650 nM。
T19850	Semaglutide 索玛鲁肽,司美格鲁肽,索马鲁肽	Glucagon Receptor	GPCR/G Protein
	Semaglutide 是人胰高血糖素样肽-1受体激动剂，是一种人胰高血糖素样肽-1 的长效类似物。它有用于 2 型糖尿病研究的潜力。
T63166	LSN3318839 LSN-3318839,LSN 3318839	Glucagon Receptor	GPCR/G Protein
	LSN3318839 是一种有效且可口服的胰高血糖素样肽-1受体（GLP-1R）变构调节剂。LSN3318839可增强GLP-1R的G蛋白偶联信号传导，可用来降低血糖。
TP1111	Tirzepatide LY-3298176	Glucagon Receptor	GPCR/G Protein
	Tirzepatide (LY-3298176) 是葡萄糖依赖性多肽 (GIP) 和胰高血糖素样肽-1 (GLP-1) 受体双重激动剂，具有神经保护活性，可改善血压并降低低密度脂蛋白（LDL）胆固醇和甘油三酯，可以用于研究糖尿病和肥胖症。
T11407	GLP-1 receptor agonist 2	Others	Others
	GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist.
T39820	Dapiglutide ZP7570
	Dapiglutide (ZP7570) is a long-acting dual agonist of glucagon-like peptide-1 receptor (GLP-1R) and glucagon-like peptide-2 receptor (GLP-2R) that holds potential for short bowel syndrome (SBS) research.
T70279	Cotadutide
	Cotadutide is a dual receptor agonist that modifies the activity of glucagon and glucagon-like peptide-1 (GLP-1).
T24620	PF-06372222 PF-0637222,PF0637222,PF 0637222
	PF-06372222 is a small-molecule negative allosteric modulator of the glucagon receptor (GCGR). PF-06372222 is also an antagonist for glucagon-like peptide-1 receptor GLP-1R, which inhibits glucagon secretion and glucose-dependent insulin secretion.
T120347	6751-0002
	Glucagon-like peptide 1 receptor, Potency: 2238.7 nM
T32343	JWU-A021 JWU A021
	JWU-A021 is a particularly potent stimulant of glucagon-like peptides-1 (GLP-1) secretion in vivo.
T36072	Skyrin Endothianin,Rhodophyscin
	Skyrin is a fungal metabolite characterized by a bisanthraquinone structure. It interferes with glucagon signaling through adenylate cyclase without binding to the glucagon receptor. At 10 μM, skyrin reduces both glucagon-stimulated cAMP production and glycogenolysis. It does not interfere with epinephrine or glucagon-like peptide 1 effects on these parameters.[1] Reference：[1]. Parker, J.C., McPherson, R.K., Andrews, K.M., et al. Effects of skyrin, a receptor-selective glucagon antagonist, in r...
T12878	Semaglutide TFA (910463-68-2 free base) Semaglutide TFA	Glucagon Receptor	GPCR/G Protein
	Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
T13091	Taspoglutide R1583,BIM51077,ITM077	Others	Others
	Taspoglutide is a long-acting glucagon-like peptide 1 (GLP-1) receptor agonist(EC50 value of 0.06 nM),and for treatment of type 2 diabetes
TP2209	Xenin-8	Others	Others
	neurotensin-like peptide that modulate pancreatic insulin and glucagon secretion/effects
T76234	Ecnoglutide
	Ecnoglutide (XW003) 是胰高血糖素样肽 1(GLP-1)受体激动剂。
T40374	Pal-Glu(OSu)-OH
	Pal-Glu(OSu)-OH is a side chain specific to Liraglutide, which is a glucagon-like peptide-1 (GLP-1) receptor agonist employed in type 2 diabetes mellitus research.
T11406	TT-OAD2 free base	Others	Others
	TT-OAD2 free base has the potential for diabetes treatment. TT-OAD2 free base is a non-peptide glucagon-like peptide-1 (GLP-1) receptor agonist with an EC50 of 5 nM.
T76237	Utreglutide
	Utreglutide 是一种有效的胰高血糖素样肽 1(GLP-1)受体激动剂。
T36428	PACAP-related Peptide (human) (trifluoroacetate salt)	PACAP	GPCR/G Protein
	PACAP-related peptide (PRP) is an endogenous 29-amino acid peptide that belongs to the secretin/glucagon superfamily of peptides, which includes secretin , glucagon , glucagon-like peptide-1 , GLP-2 , and pituitary adenylate cyclase-activating polypeptide . It is expressed in normal human pancreas and adrenal gland tissue and in some tumors that produce vasoactive intestinal peptide (VIP). PRP (1-29) is secreted by CHO-K1 cells that express human recombinant preproPACAP.

化合物

Glucagon-like peptide 1 (1-37), human acetate

Cat.No: TP1148L

Target: Glucagon Receptor

Glucagon-Like Peptide (GLP) II, human

Cat.No: TP1487

Glucagon-like peptide 1 (1-37), human

Cat.No: TP1148

Synonym: HuGLP-1

Glucagon-like peptide 1 (1-37), human TFA

Cat.No: TP1147

Synonym: HuGLP-1 TFA

Cat.No: T6203

Synonym: BMS-477118,沙克列汀,Onglyza,沙格列汀

Target: Proteasome, DPP-4

Saxagliptin hydrate

Cat.No: T0178

Synonym: 沙格列汀单水化合物,Onglyza hydrate,BMS-477118 hydrate

Target: Proteasome, DPP-4

Cat.No: T2316

Synonym: MK-3102,奥格列汀

Target: Proteasome, DPP-4

GLP-1 (1-36) amide (human, rat)

Cat.No: T80453

Synonym: Glucagon-like Peptide 1 (1-36) amide (human, rat)

GLP-2(1-33)(human)

Cat.No: TP1157

Synonym: GLP-2 (human),Glucagon-like peptide 2 (human)

GLP-1 (1-36) amide (human, rat) (TFA)

Cat.No: T82309

Synonym: Glucagon-like Peptide 1 (1-36) amide (human, rat) (TFA)

GLP-1(7-36), amide

Cat.No: T3984

Synonym: MKC 253,胰高血糖素样肽-1,Human GLP-1-(7-36)-amide,Glucagon-like Peptide 1 (7-36) amide,Glucagon-Like Peptide (GLP) I (7-36), amide, human,GLP-1(7-36),GLP-1-(7-36)-amide

Target: Glucagon Receptor

Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide

Cat.No: T76330

Glucagon-Like Peptide 1 (GLP-1) (7-36)-Lys (Biotin), amide, human

Cat.No: T76085

Cat.No: TP2100

Synonym: Exendin-3 (9-39) amide,Exendin (9-39),艾塞那肽

Target: Glucagon Receptor

Cat.No: T8355

Synonym: Exendin-4,Extendin-4

Target: Glucagon Receptor

Cat.No: T76559

Synonym: BI 456906

Target: Glucagon Receptor

Cotadutide acetate

Cat.No: TP1103

Synonym: MEDI0382 acetate,Cotadutide acetate (1686108-82-6 Free base)

Target: Glucagon Receptor

Cat.No: T12431

Target: Glucagon Receptor

V-0219 hydrochloride

Cat.No: T60047L

Synonym: V-0219 hydrochloride（878453-71-5 Free base）

Target: Glucagon Receptor

Semaglutide Acetate

Cat.No: T19850L

Synonym: 索玛鲁肽醋酸盐,Semaglutide Acetate(910463-68-2 Free base)

Target: Glucagon Receptor

PF-06882961 Tris

Cat.No: T8876

Synonym: UNII-2HJV78O0SS

Target: Glucagon Receptor

Lixisenatide acetate (320367-13-3 free base)

Cat.No: TP1469

Synonym: Lixisenatide acetate

Target: Glucagon Receptor

GLP-1R Agonist DMB

Cat.No: T36579

Target: Glucagon Receptor

Cat.No: T11408

Synonym: LY3502970,GLP-1 receptor agonist 1

Target: Glucagon Receptor

Oxyntomodulin acetate

Cat.No: TP1976L

Target: Glucagon Receptor

Avexitide acetate

Cat.No: TP2100L

Synonym: Exendin 9-39 acetate,Avexitide acetate（133514-43-9 Free base）

Target: Glucagon Receptor

Cat.No: T76279

Synonym: LY3437943

Target: Glucagon Receptor

Cat.No: T3967

Synonym: 艾塞那肽,Exenatide,Exenatide Acetate

Target: Glucagon Receptor

Retatrutide sodium salt

Cat.No: T76279L1

Synonym: Retatrutide sodium salt(2381089-83-2 free base),LY3437943 sodium salt

Target: Glucagon Receptor

(S, R)-LSN 3318839

Cat.No: T63166L

Synonym: (S, R)-LSN 3318839(Isomer-2764704-18-7)

Target: Glucagon Receptor

Mazdutide acetate（2259884-03-0 free base）

Cat.No: T78097L

Synonym: Mazdutide acetate（2259884-03-0 free base）,OXM-3 acetate,LY-3305677 acetate,IBI-362 acetate

Target: Glucagon Receptor

GLP-1R Antagonist 1

Cat.No: T15387

Target: Glucagon Receptor

Cat.No: T19850

Synonym: 索玛鲁肽,司美格鲁肽,索马鲁肽

Target: Glucagon Receptor

Cat.No: T63166

Synonym: LSN-3318839,LSN 3318839

Target: Glucagon Receptor

Cat.No: TP1111

Synonym: LY-3298176

Target: Glucagon Receptor

GLP-1 receptor agonist 2

Cat.No: T11407

Target: Others

Cat.No: T39820

Synonym: ZP7570

Cat.No: T70279

Cat.No: T24620

Synonym: PF-0637222,PF0637222,PF 0637222

Cat.No: T120347

Cat.No: T32343

Synonym: JWU A021

Cat.No: T36072

Synonym: Endothianin,Rhodophyscin

Semaglutide TFA (910463-68-2 free base)

Cat.No: T12878

Synonym: Semaglutide TFA

Target: Glucagon Receptor

Cat.No: T13091

Synonym: R1583,BIM51077,ITM077

Target: Others

Cat.No: TP2209

Target: Others

Cat.No: T76234

Pal-Glu(OSu)-OH

Cat.No: T40374

TT-OAD2 free base

Cat.No: T11406

Target: Others

Cat.No: T76237

PACAP-related Peptide (human) (trifluoroacetate salt)

Cat.No: T36428

Target: PACAP

Cat. No.	Product Name	Target	Signaling Pathways
T37526	2-Oleoylglycerol 2-Oleoyl Glycerol,2-OG,2-Monoolein	GPR	Endocrinology/Hormones; GPCR/G Protein
	2-Oleoylglycerol 是一种存在于棕榈仁、葵花籽和米糠中的脂质。2-Oleoylglycerol 可当作一种 GPR119 激动剂，具有神经保护作用，可诱导胰高血糖素样肽 1 (GLP-1) 分泌。2-Oleoylglycerol 可用于非酒精性脂肪性肝炎造模。

天然产物

2-Oleoylglycerol

Cat.No: T37526

Synonym: 2-Oleoyl Glycerol,2-OG,2-Monoolein

Target: GPR

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