10
1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1939 |
DMOG
Dimethyloxalylglycine,Dimethyloxallyl Glycine,Dimethyloxaloylglycine,二甲基草酰甘氨酸 |
HIF/HIF Prolyl-Hydroxylase; HIF; Autophagy | Angiogenesis; Autophagy; Chromatin/Epigenetic; Metabolism |
DMOG (Dimethyloxalylglycine) 是 α-酮戊二酸辅因子的拮抗剂,是一种 HIF 脯氨酰羟化酶抑制剂,可导致蛋白HIF-1α的积聚和稳定,诱导细胞自噬。它是一种促血管生成剂,在结肠炎和腹泻动物模型中起保护作用。 | |||
T0424 |
Bismuth Subsalicylate
Bismuth subsalicylat,Bismuth(III) salicylate basic,Bismuth oxysalicylate,碱式水杨酸铋,次水杨酸铋 |
COX; PGE Synthase | Immunology/Inflammation; Neuroscience |
Bismuth Subsalicylate (Bismuth subsalicylat) 是口服抗酸和止泻试剂。它能够抑制体内前列腺素合成,抑制胃和肠道黏膜炎症反应。它广泛用于研究腹泻疾病,如恶心、消化不良、腹泻等。 | |||
T10755L |
Celgosivir
MX3253,MBI 3253,6 O-butanoyl castanospermine,MDL 28574 |
Glucosidase | Metabolism |
Celgosivir (6 O-butanoyl castanospermine) 是 α-葡萄糖苷酶 I (α-glucosidase I) 抑制剂,在体外实验中的 IC50 值为 1.27 μM。 | |||
T10591L |
(R)-BPO-27
|
CFTR; Autophagy | Autophagy; Membrane transporter/Ion channel |
(R)-BPO-27 是一种具有口服活性和高效性的 ATP 竞争性 CFTR 抑制剂(IC50:4 nM),可用于研究腹泻和多囊肾。 | |||
T68025 |
Zoliprofen
|
Others | Others |
Zoliprofen 是一种一种高效的且可口服的非甾体抗炎剂,具有抗炎、解热和镇痛活性,对角叉菜素、制霉菌素、刀豆球蛋白A 诱导的大鼠爪水肿,以及抗大鼠兔血清诱导的骨折或背皮水肿具有抑制作用。Zoliprofen 在大鼠和兔子中对胶原蛋白或花生四烯酸引起的血小板聚集方面比布洛芬和非诺洛芬有效20倍。Zoliprofen 对小鼠内毒素诱导的腹泻和花生四烯酸诱导的兔急性死亡抑制作用显著。 | |||
T10755 |
Celgosivir hydrochloride
MX3253 hydrochloride,MBI 3253 hydrochloride,MDL 28574 hydrochloride |
Others | Others |
Celgosivir hydrochloride (MBI 3253 hydrochloride) is an α-glucosidase I inhibitor and inhibits bovine viral diarrhoea virus (BVDV) (IC50: 1.27 μM). | |||
T60288 |
3′-Deoxyuridine
|
||
3′-Deoxyuridine 是一种潜在的抗癌剂和抗病毒剂。3′-Deoxyuridine 抑制牛腹泻病毒 (BVDV) 的产生。 | |||
T95359 |
Compound F0433-0067
|
||
hiCE inhibitor-1是一种磺胺衍生物,是一种选择性的人体肠道酶 (hiCE) 抑制剂,Ki 值为 53.3 nM。hiCE inhibitor-1可用于改善 Irinotecan 引起的腹泻。 | |||
T32171 |
Iodoalphionic acid
NSC 11854,NSC-11854,Pheniodolum,NSC11854,Tenamid |
||
Iodoalphionic acid is the contrast medium for gallbladder examination. It is rarely found in the colon and can rarely masked the gallbladder. The density of the shadow from Iodoalphionic acid was greater than that produced by iodophthalein. It was reliabl | |||
T14382 |
AZD7687
|
Others | Others |
AZD7687 is a potent and selective DGAT1 inhibitor with an IC50 value of 80 nM (hDGAT1). IC50 value: 80 nM [1] Target: DGAT1 in vitro: Plasma AZD7687 exposure was measured repeatedly. AZD7687 markedly reduced postprandial TAG excursion with a steep concent |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1788 |
Isookanin
|
Amylase | Metabolism |
Isookanin 在多种疾病领域有研究价值,包括肿瘤,皮疹,蛇和昆虫叮咬,糖尿病,腹泻。它可作为抗病毒剂对抗 HSV 和水痘带状疱疹病毒。它也具有抗氧化特性。 |