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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T1939 DMOG

Dimethyloxalylglycine,Dimethyloxallyl Glycine,Dimethyloxaloylglycine,二甲基草酰甘氨酸

HIF/HIF Prolyl-Hydroxylase; HIF; Autophagy Angiogenesis; Autophagy; Chromatin/Epigenetic; Metabolism
DMOG (Dimethyloxalylglycine) 是 α-酮戊二酸辅因子的拮抗剂,是一种 HIF 脯氨酰羟化酶抑制剂,可导致蛋白HIF-1α的积聚和稳定,诱导细胞自噬。它是一种促血管生成剂,在结肠炎和腹泻动物模型中起保护作用。
T0424 Bismuth Subsalicylate

Bismuth subsalicylat,Bismuth(III) salicylate basic,Bismuth oxysalicylate,碱式水杨酸铋,次水杨酸铋

COX; PGE Synthase Immunology/Inflammation; Neuroscience
Bismuth Subsalicylate (Bismuth subsalicylat) 是口服抗酸和止泻试剂。它能够抑制体内前列腺素合成,抑制胃和肠道黏膜炎症反应。它广泛用于研究腹泻疾病,如恶心、消化不良、腹泻等。
T10755L Celgosivir

MX3253,MBI 3253,6 O-butanoyl castanospermine,MDL 28574

Glucosidase Metabolism
Celgosivir (6 O-butanoyl castanospermine) 是 α-葡萄糖苷酶 I (α-glucosidase I) 抑制剂,在体外实验中的 IC50 值为 1.27 μM。
T10591L (R)-BPO-27

CFTR; Autophagy Autophagy; Membrane transporter/Ion channel
(R)-BPO-27 是一种具有口服活性和高效性的 ATP 竞争性 CFTR 抑制剂(IC50:4 nM),可用于研究腹泻和多囊肾。
T68025 Zoliprofen

Others Others
Zoliprofen 是一种一种高效的且可口服的非甾体抗炎剂,具有抗炎、解热和镇痛活性,对角叉菜素、制霉菌素、刀豆球蛋白A 诱导的大鼠爪水肿,以及抗大鼠兔血清诱导的骨折或背皮水肿具有抑制作用。Zoliprofen 在大鼠和兔子中对胶原蛋白或花生四烯酸引起的血小板聚集方面比布洛芬和非诺洛芬有效20倍。Zoliprofen 对小鼠内毒素诱导的腹泻和花生四烯酸诱导的兔急性死亡抑制作用显著。
T10755 Celgosivir hydrochloride

MX3253 hydrochloride,MBI 3253 hydrochloride,MDL 28574 hydrochloride

Others Others
Celgosivir hydrochloride (MBI 3253 hydrochloride) is an α-glucosidase I inhibitor and inhibits bovine viral diarrhoea virus (BVDV) (IC50: 1.27 μM).
T60288 3′-Deoxyuridine

3′-Deoxyuridine 是一种潜在的抗癌剂和抗病毒剂。3′-Deoxyuridine 抑制牛腹泻病毒 (BVDV) 的产生。
T95359 Compound F0433-0067

hiCE inhibitor-1是一种磺胺衍生物,是一种选择性的人体肠道酶 (hiCE) 抑制剂,Ki 值为 53.3 nM。hiCE inhibitor-1可用于改善 Irinotecan 引起的腹泻。
T32171 Iodoalphionic acid

NSC 11854,NSC-11854,Pheniodolum,NSC11854,Tenamid

Iodoalphionic acid is the contrast medium for gallbladder examination. It is rarely found in the colon and can rarely masked the gallbladder. The density of the shadow from Iodoalphionic acid was greater than that produced by iodophthalein. It was reliabl
T14382 AZD7687

Others Others
AZD7687 is a potent and selective DGAT1 inhibitor with an IC50 value of 80 nM (hDGAT1). IC50 value: 80 nM [1] Target: DGAT1 in vitro: Plasma AZD7687 exposure was measured repeatedly. AZD7687 markedly reduced postprandial TAG excursion with a steep concent

化合物

DMOG
Cat.No: T1939
Synonym: Dimethyloxalylglycine,Dimethyloxallyl Glycine,Dimethyloxaloylglycine,二甲基草酰甘氨酸
Target: HIF/HIF Prolyl-Hydroxylase, HIF, Autophagy
Bismuth Subsalicylate
Cat.No: T0424
Synonym: Bismuth subsalicylat,Bismuth(III) salicylate basic,Bismuth oxysalicylate,碱式水杨酸铋,次水杨酸铋
Target: COX, PGE Synthase
Celgosivir
Cat.No: T10755L
Synonym: MX3253,MBI 3253,6 O-butanoyl castanospermine,MDL 28574
Target: Glucosidase
(R)-BPO-27
Cat.No: T10591L
Synonym:
Target: CFTR, Autophagy
Zoliprofen
Cat.No: T68025
Synonym:
Target: Others
Celgosivir hydrochloride
Cat.No: T10755
Synonym: MX3253 hydrochloride,MBI 3253 hydrochloride,MDL 28574 hydrochloride
Target: Others
3′-Deoxyuridine
Cat.No: T60288
Synonym:
Target:
Compound F0433-0067
Cat.No: T95359
Synonym:
Target:
Iodoalphionic acid
Cat.No: T32171
Synonym: NSC 11854,NSC-11854,Pheniodolum,NSC11854,Tenamid
Target:
AZD7687
Cat.No: T14382
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN1788 Isookanin

Amylase Metabolism
Isookanin 在多种疾病领域有研究价值,包括肿瘤,皮疹,蛇和昆虫叮咬,糖尿病,腹泻。它可作为抗病毒剂对抗 HSV 和水痘带状疱疹病毒。它也具有抗氧化特性。

天然产物

Isookanin
Cat.No: TN1788
Synonym:
Target: Amylase
TargetMol Loading
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