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15

抑制剂 & 化合物

6

天然产物

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Cat. No. Product Name Target Signaling Pathways
T7807 Bendazac

AF-983,Bendazolic acid

Others Others
Bendazac (Bendazolic acid) 是一种氧乙酸,具有抗过敏、抗炎、利胆和抗血脂作用。它能够阻断蛋白质变性,延缓白内障的发生过程。
T0857 Fenipentol

非尼戊醇,1-Phenyl-1-pentanol,1-Phenylpentanol,Pancoral,苯戊醇,1-phenylpentan-1-ol

Lipid Metabolism
Fenipentol (Pancoral) 是一种口服活性的利胆剂,在释放碳酸氢盐和蛋白质的分泌素,胃泌素和胰腺分泌中起重要作用。它也是姜黄成分的合成衍生物,可用作调味品和染料。
T19239 Cicloxilic acid

Cycloxilic acid

Others Others
Cicloxilic acid(Cycloxilic acid) 具有利胆活性,抑制胆汁胆固醇的输出。
T6375 Alibendol

cebera,EB 1856,阿利苯多

Others Others
Alibendol (cebera) 具有促胆汁分泌及抗痉挛的作用。
T1148 Menbutone

孟布酮,Naftobil,Genabilic acid,Genabilin

Others Others
Menbutone (Genabilin) 是一种利胆剂,是氧代丁酸衍生物。
T0353 Osalmid

Oxaphenamide,4'-Hydroxysalicylanilide,羟苯水杨胺,柳胺酚

HBV; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Osalmid (Oxaphenamide) 是一种利胆药物,通过靶向核糖核苷酸还原酶小亚基 M2 来抑制核糖核苷酸还原酶的活性,IC50值为8.23 μM。
T34076 Piprozolin

W3699,W-3699,W 3699

Piprozolin (W 3699) 是一种新型的利胆酸,在慢性实验过程中高剂量显示出轻微的镇痛性。Piprozolin 对氧化系统的某些酶具有轻微的诱导作用。
T34788 Taurolithocholic acid

Lithocholyltaurine,Lithocholic acid taurine conjugate

Taurolithocholic acid is a cholagogue and choleretic.
T69481 Clanobutin

Clanobutin inhibits gluconeogenesis and acts as a choleretic and digestion-stimulating agent.
T23923 Cyclobutyrol

BRN 2209058,BRN-2209058,BRN2209058,Cyclobutyrolum,JL 130

Cyclobutyrol is a choleretic agent. It also inhibits biliary lipid secretion.
T19851 Azintamide

Azinthiamide,Oragalin,Bilipurum,Colerin,BRN 0885011

Azintamide is a choleretic. It has shown effective and safe for dyspepsia symptoms when Domperidone therapy is not satisfactory.
T33580 Nafcaproic acid

DA-808,Acide nafcaproique,Acido nafcaproico,Nafcapronsaeure,DA 808

Nafcaproic acid (DA-808) 是一种合成的胆汁利尿剂。
T71403 Cyclobutyrol sodium salt

Cyclobutyrol sodium salt is a choleretic agent which also inhibits biliary lipid secretion.
T20928 Febuprol

H33,K-10033,H 33,H-33,NSC 30151

Febuprol, a choleretic drug, stimulates bile secretion. In addition, it also has lipid-lowering (lowering blood lipid) and spasmolytic (anticonvulsant) properties.
T30703 Cantabiline sodium

Hymecromone sodium,LM 94 sodium

Cantabiline sodium is a coumarin derivative possessing properties as a spasmolytic, choleretic and light-protective agent. It is also used in analytical chemistry for the determination of NITRIC ACID.

化合物

Bendazac
Cat.No: T7807
Synonym: AF-983,Bendazolic acid
Target: Others
Fenipentol
Cat.No: T0857
Synonym: 非尼戊醇,1-Phenyl-1-pentanol,1-Phenylpentanol,Pancoral,苯戊醇,1-phenylpentan-1-ol
Target: Lipid
Cicloxilic acid
Cat.No: T19239
Synonym: Cycloxilic acid
Target: Others
Alibendol
Cat.No: T6375
Synonym: cebera,EB 1856,阿利苯多
Target: Others
Menbutone
Cat.No: T1148
Synonym: 孟布酮,Naftobil,Genabilic acid,Genabilin
Target: Others
Osalmid
Cat.No: T0353
Synonym: Oxaphenamide,4'-Hydroxysalicylanilide,羟苯水杨胺,柳胺酚
Target: HBV, DNA/RNA Synthesis
Piprozolin
Cat.No: T34076
Synonym: W3699,W-3699,W 3699
Target:
Taurolithocholic acid
Cat.No: T34788
Synonym: Lithocholyltaurine,Lithocholic acid taurine conjugate
Target:
Clanobutin
Cat.No: T69481
Synonym:
Target:
Cyclobutyrol
Cat.No: T23923
Synonym: BRN 2209058,BRN-2209058,BRN2209058,Cyclobutyrolum,JL 130
Target:
Azintamide
Cat.No: T19851
Synonym: Azinthiamide,Oragalin,Bilipurum,Colerin,BRN 0885011
Target:
Nafcaproic acid
Cat.No: T33580
Synonym: DA-808,Acide nafcaproique,Acido nafcaproico,Nafcapronsaeure,DA 808
Target:
Cyclobutyrol sodium salt
Cat.No: T71403
Synonym:
Target:
Febuprol
Cat.No: T20928
Synonym: H33,K-10033,H 33,H-33,NSC 30151
Target:
Cantabiline sodium
Cat.No: T30703
Synonym: Hymecromone sodium,LM 94 sodium
Target:
Cat. No. Product Name Target Signaling Pathways
T1285 Anethole trithione

茴三硫,Anetholtrithion

Others; AChR Neuroscience; Others
Anethole trithione (Anetholtrithion) 是硫杂环胆碱,是一种胆汁分泌刺激剂,可增强唾液分泌并增加 mAChR 受体,用于口干症的研究。
T1391 4-Methylumbelliferone

Hymecromone,4-MU,胆通

Others Others
4-Methylumbelliferone (Hymecromone) 是透明质酸生物合成抑制剂,显示出抗肿瘤和抗转移活性。
T2965 Deoxycholic acid

Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid (Cholanoic Acid) 是 G 蛋白偶联胆汁酸受体 TGR5的激活剂。
T5736 1,3-Dicaffeoylquinic acid

CYNARIN,1,3-二咖啡酰奎宁酸,Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1S,​3R,​4R,​5R)​-,1,3-O-Dicaffeoylquinic acid,1,5-Dicaffeoylquinic acid

Reactive Oxygen Species; Akt; PI3K Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
1,3-Dicaffeoylquinic acid (CYNARIN) 是一种咖啡酰奎宁酸衍生物,具有抗氧化、自由基清除作用。
T0847 Chenodeoxycholic acid

CDCA,鹅去氧胆酸,Chenodiol

Potassium Channel; FXR; Endogenous Metabolite; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism
Chenodeoxycholic acid (CDCA) 是一种胆汁酸,通常与甘氨酸或牛磺酸结合。它作为清洁剂溶解脂肪以供肠道吸收,并被小肠重新吸收。它被用作利胆剂、利胆泻药,以及预防或溶解胆结石。
T2202 Lithocholic acid

3α-Hydroxy-5β-cholanic acid,石胆酸

Apoptosis; Others; FXR; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism; Others
Lithocholic acid (3α-Hydroxy-5β-cholanic acid) 是由鹅去氧胆酸盐通过细菌作用形成的胆汁酸,通常与甘氨酸或牛磺酸结合,被用作利胆剂。 它作为清洁剂溶解脂肪以供吸收,并且本身被吸收。

天然产物

Anethole trithione
Cat.No: T1285
Synonym: 茴三硫,Anetholtrithion
Target: Others, AChR
4-Methylumbelliferone
Cat.No: T1391
Synonym: Hymecromone,4-MU,胆通
Target: Others
Deoxycholic acid
Cat.No: T2965
Synonym: Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic
Target: Endogenous Metabolite, GPCR19
1,3-Dicaffeoylquinic acid
Cat.No: T5736
Synonym: CYNARIN,1,3-二咖啡酰奎宁酸,Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1S,​3R,​4R,​5R)​-,1,3-O-Dicaffeoylquinic acid,1,5-Dicaffeoylquinic acid
Target: Reactive Oxygen Species, Akt, PI3K
Chenodeoxycholic acid
Cat.No: T0847
Synonym: CDCA,鹅去氧胆酸,Chenodiol
Target: Potassium Channel, FXR, Endogenous Metabolite, Autophagy
Lithocholic acid
Cat.No: T2202
Synonym: 3α-Hydroxy-5β-cholanic acid,石胆酸
Target: Apoptosis, Others, FXR, Endogenous Metabolite, Autophagy
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