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Cat. No. | Product Name | Target | Signaling Pathways |
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T7807 |
Bendazac
AF-983,Bendazolic acid |
Others | Others |
Bendazac (Bendazolic acid) 是一种氧乙酸,具有抗过敏、抗炎、利胆和抗血脂作用。它能够阻断蛋白质变性,延缓白内障的发生过程。 | |||
T0857 |
Fenipentol
非尼戊醇,1-Phenyl-1-pentanol,1-Phenylpentanol,Pancoral,苯戊醇,1-phenylpentan-1-ol |
Lipid | Metabolism |
Fenipentol (Pancoral) 是一种口服活性的利胆剂,在释放碳酸氢盐和蛋白质的分泌素,胃泌素和胰腺分泌中起重要作用。它也是姜黄成分的合成衍生物,可用作调味品和染料。 | |||
T19239 |
Cicloxilic acid
Cycloxilic acid |
Others | Others |
Cicloxilic acid(Cycloxilic acid) 具有利胆活性,抑制胆汁胆固醇的输出。 | |||
T6375 |
Alibendol
cebera,EB 1856,阿利苯多 |
Others | Others |
Alibendol (cebera) 具有促胆汁分泌及抗痉挛的作用。 | |||
T1148 |
Menbutone
孟布酮,Naftobil,Genabilic acid,Genabilin |
Others | Others |
Menbutone (Genabilin) 是一种利胆剂,是氧代丁酸衍生物。 | |||
T0353 |
Osalmid
Oxaphenamide,4'-Hydroxysalicylanilide,羟苯水杨胺,柳胺酚 |
HBV; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Osalmid (Oxaphenamide) 是一种利胆药物,通过靶向核糖核苷酸还原酶小亚基 M2 来抑制核糖核苷酸还原酶的活性,IC50值为8.23 μM。 | |||
T34076 |
Piprozolin
W3699,W-3699,W 3699 |
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Piprozolin (W 3699) 是一种新型的利胆酸,在慢性实验过程中高剂量显示出轻微的镇痛性。Piprozolin 对氧化系统的某些酶具有轻微的诱导作用。 | |||
T34788 |
Taurolithocholic acid
Lithocholyltaurine,Lithocholic acid taurine conjugate |
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Taurolithocholic acid is a cholagogue and choleretic. | |||
T69481 |
Clanobutin
|
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Clanobutin inhibits gluconeogenesis and acts as a choleretic and digestion-stimulating agent. | |||
T23923 |
Cyclobutyrol
BRN 2209058,BRN-2209058,BRN2209058,Cyclobutyrolum,JL 130 |
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Cyclobutyrol is a choleretic agent. It also inhibits biliary lipid secretion. | |||
T19851 |
Azintamide
Azinthiamide,Oragalin,Bilipurum,Colerin,BRN 0885011 |
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Azintamide is a choleretic. It has shown effective and safe for dyspepsia symptoms when Domperidone therapy is not satisfactory. | |||
T33580 |
Nafcaproic acid
DA-808,Acide nafcaproique,Acido nafcaproico,Nafcapronsaeure,DA 808 |
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Nafcaproic acid (DA-808) 是一种合成的胆汁利尿剂。 | |||
T71403 | Cyclobutyrol sodium salt | ||
Cyclobutyrol sodium salt is a choleretic agent which also inhibits biliary lipid secretion. | |||
T20928 |
Febuprol
H33,K-10033,H 33,H-33,NSC 30151 |
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Febuprol, a choleretic drug, stimulates bile secretion. In addition, it also has lipid-lowering (lowering blood lipid) and spasmolytic (anticonvulsant) properties. | |||
T30703 |
Cantabiline sodium
Hymecromone sodium,LM 94 sodium |
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Cantabiline sodium is a coumarin derivative possessing properties as a spasmolytic, choleretic and light-protective agent. It is also used in analytical chemistry for the determination of NITRIC ACID. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1285 |
Anethole trithione
茴三硫,Anetholtrithion |
Others; AChR | Neuroscience; Others |
Anethole trithione (Anetholtrithion) 是硫杂环胆碱,是一种胆汁分泌刺激剂,可增强唾液分泌并增加 mAChR 受体,用于口干症的研究。 | |||
T1391 |
4-Methylumbelliferone
Hymecromone,4-MU,胆通 |
Others | Others |
4-Methylumbelliferone (Hymecromone) 是透明质酸生物合成抑制剂,显示出抗肿瘤和抗转移活性。 | |||
T2965 |
Deoxycholic acid
Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic |
Endogenous Metabolite; GPCR19 | GPCR/G Protein; Metabolism |
Deoxycholic acid (Cholanoic Acid) 是 G 蛋白偶联胆汁酸受体 TGR5的激活剂。 | |||
T5736 |
1,3-Dicaffeoylquinic acid
CYNARIN,1,3-二咖啡酰奎宁酸,Cyclohexanecarboxylic acid, 1,3-bis[[3-(3,4-dihydroxyphenyl)-1-oxo-2-propen-1-yl]oxy]-4,5-dihydroxy-, (1S,3R,4R,5R)-,1,3-O-Dicaffeoylquinic acid,1,5-Dicaffeoylquinic acid |
Reactive Oxygen Species; Akt; PI3K | Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB; PI3K/Akt/mTOR signaling |
1,3-Dicaffeoylquinic acid (CYNARIN) 是一种咖啡酰奎宁酸衍生物,具有抗氧化、自由基清除作用。 | |||
T0847 |
Chenodeoxycholic acid
CDCA,鹅去氧胆酸,Chenodiol |
Potassium Channel; FXR; Endogenous Metabolite; Autophagy | Autophagy; Membrane transporter/Ion channel; Metabolism |
Chenodeoxycholic acid (CDCA) 是一种胆汁酸,通常与甘氨酸或牛磺酸结合。它作为清洁剂溶解脂肪以供肠道吸收,并被小肠重新吸收。它被用作利胆剂、利胆泻药,以及预防或溶解胆结石。 | |||
T2202 |
Lithocholic acid
3α-Hydroxy-5β-cholanic acid,石胆酸 |
Apoptosis; Others; FXR; Endogenous Metabolite; Autophagy | Apoptosis; Autophagy; Metabolism; Others |
Lithocholic acid (3α-Hydroxy-5β-cholanic acid) 是由鹅去氧胆酸盐通过细菌作用形成的胆汁酸,通常与甘氨酸或牛磺酸结合,被用作利胆剂。 它作为清洁剂溶解脂肪以供吸收,并且本身被吸收。 |