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33

抑制剂 & 化合物

8

天然产物

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Cat. No. Product Name Target Signaling Pathways
T8365 Methenamine Hippurate

Antibacterial Microbiology/Virology
Methenamine hippurate 是一种口服活性尿液广谱抗菌剂。它对大多数常见的尿路病原体有效。
T7533 Taurolidine

Apoptosis; Others; Antibacterial; Antibiotic Apoptosis; Microbiology/Virology; Others
Taurolidine 是一种广谱抗菌剂,用于预防中心静脉导管相关感染。它具有抗真菌和抗肿瘤作用。
T1440 Ethacridine lactate monohydrate

乳酸依沙吖啶一水物,利凡诺

Antibacterial; Antibiotic Microbiology/Virology
Ethacridine lactate monohydrate 是一种聚 (ADP-核糖) 糖基水解酶 (PARG) 抑制剂,有抗金黄色葡萄球菌和其他革兰氏阳性球菌的活性。它也是抗菌剂和流产剂。
T0314 Hexylresorcinol

己雷锁辛,4-己基间苯二酚,4-Hexylresorcinol

Apoptosis; Tyrosinase; Antibacterial; Parasite Apoptosis; Microbiology/Virology; Proteases/Proteasome
Hexylresorcinol (4-Hexylresorcinol) 是在植物中发现的一种天然产物,具有抗菌、驱虫、防腐和抗肿瘤活性。它是一种可逆、非竞争性的 α-葡萄糖苷酶抑制剂,有抗 DNA 氧化损伤的保护作用。它可诱导鳞癌细胞凋亡。
T7887 8-Hydroxyquinoline hemisulfate

8-羟基喹啉硫酸盐,Oxyquinoline sulfate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
8-Hydroxyquinoline hemisulfate (Oxyquinoline sulfate) 是一种单质子双齿螯合剂,具有温和的抑菌、驱虫和杀螨作用。
T5967 Ethacridine lactate

乳酸依沙吖啶,Acrinol,6,9-DIAMINO-2-ETHOXYACRIDINE LACTATE

Others; Antibacterial Microbiology/Virology; Others
Ethacridine lactate (Acrinol) 是一种聚 (ADP-核糖) 糖水解酶 (PARG) 抑制剂,也是一种抗菌剂和流产剂。它有抗金黄色葡萄球菌和其他革兰氏阳性球菌的活性。
T1253 Chlorindanol

7-Chloro-4-indanol,Lanesta,Clorindanol,4-氯-7-羟基氢化茚,7-氯-4-羟基氢化茚

Others Others
Chlorindanol (Lanesta) 是新型的防腐剂。
T0328 Hexetidine

NSC-17764,海克替啶

Antibacterial; Antifungal Microbiology/Virology
Hexetidine (NSC-17764) 是一种口服活性的抗菌抗真菌试剂,可用于口腔感染的相关研究。
T19027 Methyl Blue

Others Others
Methyl blue 是一种三氨基三苯甲烷染料。它在多色染色法中被广泛用作抗菌染料,并能够应用于组织学和微生物学染色溶液。它已被用作研究各种催化剂对染料光降解影响的模型。
T10295 Amantanium bromide

金刚溴铵,Amantanil bromidum

Others Others
Amantanium bromide (Amantanil bromidum) 是一种季铵抗菌/抗真菌剂,可用作手术防腐剂以及粘液和皮肤感染的局部治疗。
T0497 Cetrimonium bromide

Lauroseptol,Cetyltrimethylammonium Bromide,西曲溴铵,CTAB

Antibiotic Microbiology/Virology
Cetrimonium bromide (Lauroseptol) 是局部消毒剂 Cetrimide 的组成部分之一,是一种阳离子季胺盐表面活性剂。
T4502 BISMUTH SUBGALLATE

次没食子酸铋,Dermatol Puder,Bismuth Gallate

Others Others
Bismuth subgallate (Dermatol Puder) 是一种止血剂,可作用于凝血因子 XII ,促使凝血级联的激活,改善纤维蛋白凝块的早期形成。
T22408 Proflavine

吡啶-3,6-二胺,3,6-Diaminoacridine

Antibacterial Microbiology/Virology
Proflavine (3,6-Diaminoacridine) 是吖啶染料,可用作抗菌剂。它是 DNA 嵌入剂,能够阻滞Kir3.2孔。它用作与 Kir3.2 相关的神经系统疾病的研究。
T0404 8-Hydroxyquinoline

Hydroxyquinoline,8-Quinolinol,羟基喹啉,Oxine,8-羟基喹啉,8-Oxychinolin

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
8-Hydroxyquinoline (8-Quinolinol) 是单质子二齿螯合剂, 也是转录抑制剂,防腐剂,消毒剂和杀虫剂。
T0438 Proflavine Hemisulfate

3,6-Diaminoacridine hemisulfate,Proflavin hemisulfate,硫酸原黄素

Others; Potassium Channel; DNA; Thrombin; Antibacterial; Autophagy Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology; Others; Proteases/Proteasome
Proflavine Hemisulfate (3,6-Diaminoacridine hemisulfate) 是一种 DNA 嵌入剂,也是一种吖啶染料。它是抗菌剂,也可作为 Kir3.2孔阻滞剂,可研究与 Kir3.2 相关的神经系统疾病。
T6439 Cetylpyridinium Chloride

西吡氯铵,Cetamium,Pristacin,Hexadecylpyridinium Chloride

Others; HBV; Antibacterial Microbiology/Virology; Others
Cetylpyridinium Chloride (Hexadecylpyridinium Chloride) 是阳离子季铵,是一种广谱抗菌剂。它有效抑制 HBV 衣壳装配,IC50为 2.5 μM。它被用于杀虫剂和各种漱口水以及其他个人护理产品中。
T0401 Benzethonium chloride

Hyamine,Phemeride,苄索氯铵,Quatrachlor

AChR Neuroscience
Benzethonium chloride (Quatrachlor) 是合成季铵盐,具有表面活性剂、防腐剂和广谱抗菌特性。它作用于在爪蟾卵母细胞,抑制人重组α7和α4β2神经元烟碱性乙酰胆碱受体。
T14951 Chlorhexidine digluconate

Apoptosis; Antibiotic Apoptosis; Microbiology/Virology
Chlorhexidine digluconate 是一种广谱防腐剂和消毒剂,具有广谱抗菌活性,抑制革兰氏阳性菌和革兰氏阴性菌,可诱导细胞坏死和凋亡,可用于研究细菌感染。
T0289 9-Aminoacridine

Aminacrine,9-氨基吖啶

Others; HIV Protease; Antibacterial Microbiology/Virology; Others; Proteases/Proteasome
9-Aminoacridine 是一种具有龋齿传播特性的抗菌剂,可用作局部消毒剂。它也是一种高度荧光染料,实验用作一种诱变剂,是细胞内 pH 的指示剂。
T0339 Resorcinol monoacetate

乙醯間二酚(1,3-苯二醇单乙酸酯 ),Resorcin monoacetate

Others Others
Resorcinol monoacetate (Resorcin monoacetate) 是一种防腐剂,及消毒剂,是用于合成其他药品的化学中间体。有用于痤疮,脂溢性皮炎,湿疹,银屑病和其它皮肤病的研究潜力。
T1000 Chlorhexidine

氯己定,Chlorhexidinum,Nolvasan,Rotersept

CAT; Antibacterial; Antibiotic; Antifection Microbiology/Virology; oxidation-reduction
Chlorhexidine (Rotersept) 是一种抗菌剂和防腐剂。它可用于注射前、手术前或外伤后清洁皮肤。
T0900 Cetylpyridinium chloride monohydrate

Hexadecylpyridinium chloride monohydrate,十六烷基氯化吡啶

Antibacterial; Antibiotic Microbiology/Virology
Cetylpyridinium chloride monohydrate (Hexadecylpyridinium chloride monohydrate) 是阳离子季铵, 是一种能杀死细菌和其他微生物的防腐剂, 用于某些类型的漱口水, 牙膏, 咽喉和鼻腔喷雾剂中, 可有效预防牙斑和减少牙龈炎。
T13152 Thymol iodide

Others Others
Thymol iodide is a compound of Iodide and Thymol. It is mostly used as mild antiseptic and fungicide.
T20020 Auramine hydrochloride

NSC4045,NSC 47707,NSC-47707,NSC 4045,NSC-4045,NSC47707

Auramine hydrochloride is an aniline dye. Auramine hydrochloride is used as a disinfectant and an antiseptic agent.
T19754 Cetrimide

Cetrimide is an antiseptic. It is used to irrigate root canals to ensure the disinfection and removal of microbial residues.
T0438L Proflavine dihydrochloride

Proflavine HCl

Proflavine dihydrochloride is a topical antiseptic.
T28230 Olanexidine Gluconate

OPB2045G,OPB 2045,OPB-2045G,OPB2045,OPB-2045,OPB 2045G

Olanexidine gluconate is an antiseptic/disinfectant compound with potent bactericidal activity against Gram-negative and Gram-positive bacteria.
T25151 Bibrocathol

Bibrocathin,Bibrocatholum

Bibrocathol is a well-established antiseptic drug used for the treatment of acute eyelid diseases like blepharitis.
T20188 Polynoxylin

Formaldehyde, urea polymer,Gabrite,Hygromull,HSDB 7203

Polynoxylin is an antiseptic. It is used for local treatment of the skin and the mouth.
T21280 Aminacrine hydrochloride monohydrate

Aminacrine HCl monohydrate

Aminacrine hydrochloride monohydrate, a highly fluorescent anti-infective dye, is used as a topical antiseptic and mutagen due to its interaction with DNA. It is also used as an intracellular pH indicator.
T61493 Olanexidine

Olanexidine is a broad-spectrum antibacterial agent and antiseptic, effective against both Gram-positive and Gram-negative bacteria. It is commonly utilized in the research of infection and inflammation [1] [2] [3].
T0265 Merbromin

红汞,Mercury dibromofluorescein disodium salt

Others; Antibacterial Microbiology/Virology; Others
Merbromin (Mercury dibromofluorescein disodium salt) 有效抑制 Zika 病毒 (ZIKV) 复制,通过抑制 ZIKVpro 表现出抗 ZIKV 效力。它用作割伤和擦伤的局部消毒剂,并用作生物染料。
T69995 Chlorhexidine-d8 HCl

Chlorhexidine-d8 is intended for use as an internal standard for the quantification of chlorhexidine by GC- or LC-MS. Chlorhexidine is a bis(biguanide) antimicrobial disinfectant and antiseptic agent. It inhibits growth of clinical methicillin-resistant S. aureus (MRSA) isolates (MIC90 = 4 μg/ml). It is also active against canine isolates of MRSA, methicillin-susceptible S. aureus (MSSA), methicillin-resistant S. pseudintermedius (MRSP), and methicillin-susceptible S. pseudintermedius (MSSP; MIC...

化合物

Methenamine Hippurate
Cat.No: T8365
Synonym:
Target: Antibacterial
Taurolidine
Cat.No: T7533
Synonym:
Target: Apoptosis, Others, Antibacterial, Antibiotic
Ethacridine lactate monohydrate
Cat.No: T1440
Synonym: 乳酸依沙吖啶一水物,利凡诺
Target: Antibacterial, Antibiotic
Hexylresorcinol
Cat.No: T0314
Synonym: 己雷锁辛,4-己基间苯二酚,4-Hexylresorcinol
Target: Apoptosis, Tyrosinase, Antibacterial, Parasite
8-Hydroxyquinoline hemisulfate
Cat.No: T7887
Synonym: 8-羟基喹啉硫酸盐,Oxyquinoline sulfate
Target: Others, Antibacterial, Antibiotic
Ethacridine lactate
Cat.No: T5967
Synonym: 乳酸依沙吖啶,Acrinol,6,9-DIAMINO-2-ETHOXYACRIDINE LACTATE
Target: Others, Antibacterial
Chlorindanol
Cat.No: T1253
Synonym: 7-Chloro-4-indanol,Lanesta,Clorindanol,4-氯-7-羟基氢化茚,7-氯-4-羟基氢化茚
Target: Others
Hexetidine
Cat.No: T0328
Synonym: NSC-17764,海克替啶
Target: Antibacterial, Antifungal
Methyl Blue
Cat.No: T19027
Synonym:
Target: Others
Amantanium bromide
Cat.No: T10295
Synonym: 金刚溴铵,Amantanil bromidum
Target: Others
Cetrimonium bromide
Cat.No: T0497
Synonym: Lauroseptol,Cetyltrimethylammonium Bromide,西曲溴铵,CTAB
Target: Antibiotic
BISMUTH SUBGALLATE
Cat.No: T4502
Synonym: 次没食子酸铋,Dermatol Puder,Bismuth Gallate
Target: Others
Proflavine
Cat.No: T22408
Synonym: 吡啶-3,6-二胺,3,6-Diaminoacridine
Target: Antibacterial
8-Hydroxyquinoline
Cat.No: T0404
Synonym: Hydroxyquinoline,8-Quinolinol,羟基喹啉,Oxine,8-羟基喹啉,8-Oxychinolin
Target: Others, Antibacterial, Antibiotic
Proflavine Hemisulfate
Cat.No: T0438
Synonym: 3,6-Diaminoacridine hemisulfate,Proflavin hemisulfate,硫酸原黄素
Target: Others, Potassium Channel, DNA, Thrombin, Antibacterial, Autophagy
Cetylpyridinium Chloride
Cat.No: T6439
Synonym: 西吡氯铵,Cetamium,Pristacin,Hexadecylpyridinium Chloride
Target: Others, HBV, Antibacterial
Benzethonium chloride
Cat.No: T0401
Synonym: Hyamine,Phemeride,苄索氯铵,Quatrachlor
Target: AChR
Chlorhexidine digluconate
Cat.No: T14951
Synonym:
Target: Apoptosis, Antibiotic
9-Aminoacridine
Cat.No: T0289
Synonym: Aminacrine,9-氨基吖啶
Target: Others, HIV Protease, Antibacterial
Resorcinol monoacetate
Cat.No: T0339
Synonym: 乙醯間二酚(1,3-苯二醇单乙酸酯 ),Resorcin monoacetate
Target: Others
Chlorhexidine
Cat.No: T1000
Synonym: 氯己定,Chlorhexidinum,Nolvasan,Rotersept
Target: CAT, Antibacterial, Antibiotic, Antifection
Cetylpyridinium chloride monohydrate
Cat.No: T0900
Synonym: Hexadecylpyridinium chloride monohydrate,十六烷基氯化吡啶
Target: Antibacterial, Antibiotic
Thymol iodide
Cat.No: T13152
Synonym:
Target: Others
Auramine hydrochloride
Cat.No: T20020
Synonym: NSC4045,NSC 47707,NSC-47707,NSC 4045,NSC-4045,NSC47707
Target:
Cetrimide
Cat.No: T19754
Synonym:
Target:
Proflavine dihydrochloride
Cat.No: T0438L
Synonym: Proflavine HCl
Target:
Olanexidine Gluconate
Cat.No: T28230
Synonym: OPB2045G,OPB 2045,OPB-2045G,OPB2045,OPB-2045,OPB 2045G
Target:
Bibrocathol
Cat.No: T25151
Synonym: Bibrocathin,Bibrocatholum
Target:
Polynoxylin
Cat.No: T20188
Synonym: Formaldehyde, urea polymer,Gabrite,Hygromull,HSDB 7203
Target:
Aminacrine hydrochloride monohydrate
Cat.No: T21280
Synonym: Aminacrine HCl monohydrate
Target:
Olanexidine
Cat.No: T61493
Synonym:
Target:
Merbromin
Cat.No: T0265
Synonym: 红汞,Mercury dibromofluorescein disodium salt
Target: Others, Antibacterial
Chlorhexidine-d8 HCl
Cat.No: T69995
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN3690 Comanthoside B

Comanthosid B

Antibacterial Microbiology/Virology
Comanthoside B (Comanthosid B) 是一种黄酮类苷,分离自芦花属植物,具有抗菌、抗炎活性。
TN2730 2,5-Dihydroxybenzaldehyde

Gentisaldehyde,2,5-二羟基苯甲醛

Anti-infection; Antibacterial Microbiology/Virology
2,5-Dihydroxybenzaldehyde (Gentisaldehyde) 是一种天然抗微生物剂,可抑制Mycobacterium avium subsp. paratuberculosis 的生长。它还抑制金黄色葡萄球菌菌株,MIC50为 500 mg/L。
T0144 Ftaxilide

Histanorm,安息香酸,伏保克西里

Antibacterial Microbiology/Virology
Ftaxilide (Histanorm) 是新型抗结核剂。
T0011 2-Phenylethanol

苯乙醇,Phenethyl alcohol,2-Phenylethyl alcohol,Benzyl carbinol,Phenylethanol,Benzeneethanol

Others; Virus Protease; Antibacterial; Antibiotic Microbiology/Virology; Others
2-Phenylethanol (Phenylethanol) 是从玫瑰、风笛、阿勒颇松、桔子花等多种物种中提取得到的一种无色液体。它有一种使人感到愉悦的气味,也是一种从真菌Candida albicans 产生的自体抗生素。它可用作香皂中的防腐剂,也用作香烟添加剂。
T1301 Guaiacol

O-methylcatechol,2-hydroxyanisole,o-methoxyphenol,2-Methoxyphenol,愈创木酚

NF-κB; COX; Endogenous Metabolite Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Guaiacol (2-Methoxyphenol) 是从小叶栲中提取的一种酚类,可抑制 LPS 刺激的COX-2表达和NF-κB 激活,具有抗炎活性。
T2S0490 Eugenol acetate

Acetyleugenol,乙酰丁香酚,Aceteugenol,乙酸丁香酚酯,Eugenyl acetate,1,3,4-Eugenol acetate

Others; Antibacterial; Antifungal Microbiology/Virology; Others
Eugenol acetate (Aceteugenol) 是来自丁香植物 Syzygiumaromaticum 的一种化学成分,具有抗菌、抗毒和抗氧化活性。
T10934 D-Gluconic acid

Dextronic acid,Glycogenic acid,Pentahydroxycaproic acid,Gluconic acid,D-Gluco-hexonic acid,D-Gluconsaeure,Maltonic acid,葡萄糖酸

Endogenous Metabolite Metabolism
D-Gluconic acid (D-Gluco-hexonic acid) 是一种具有杀菌作用和螯合性质的氧化型羧酸。
T8199 (±)-α-Bisabolol

Bisabolol

Apoptosis; Antioxidant Apoptosis; oxidation-reduction
(±)-α-Bisabolol (Bisabolol) 是一种从洋甘菊、念珠菌树等植物精油中提取的倍半萜烯醇,是一种天然防腐剂,具有舒缓、抗刺激、抗炎、抗氧化和抗癌活性。(±)-α-Bisabolol 通过诱导细胞周期停滞、线粒体死亡和抑制 PI3K/Akt 信号通路来发挥作用,对 A549 NSC-LC 细胞产生抗癌作用 (IC50 = 15 μM)。(±)-α-Bisabolol 能强效诱导胶质瘤细胞凋亡。

天然产物

Comanthoside B
Cat.No: TN3690
Synonym: Comanthosid B
Target: Antibacterial
2,5-Dihydroxybenzaldehyde
Cat.No: TN2730
Synonym: Gentisaldehyde,2,5-二羟基苯甲醛
Target: Anti-infection, Antibacterial
Ftaxilide
Cat.No: T0144
Synonym: Histanorm,安息香酸,伏保克西里
Target: Antibacterial
2-Phenylethanol
Cat.No: T0011
Synonym: 苯乙醇,Phenethyl alcohol,2-Phenylethyl alcohol,Benzyl carbinol,Phenylethanol,Benzeneethanol
Target: Others, Virus Protease, Antibacterial, Antibiotic
Guaiacol
Cat.No: T1301
Synonym: O-methylcatechol,2-hydroxyanisole,o-methoxyphenol,2-Methoxyphenol,愈创木酚
Target: NF-κB, COX, Endogenous Metabolite
Eugenol acetate
Cat.No: T2S0490
Synonym: Acetyleugenol,乙酰丁香酚,Aceteugenol,乙酸丁香酚酯,Eugenyl acetate,1,3,4-Eugenol acetate
Target: Others, Antibacterial, Antifungal
D-Gluconic acid
Cat.No: T10934
Synonym: Dextronic acid,Glycogenic acid,Pentahydroxycaproic acid,Gluconic acid,D-Gluco-hexonic acid,D-Gluconsaeure,Maltonic acid,葡萄糖酸
Target: Endogenous Metabolite
(±)-α-Bisabolol
Cat.No: T8199
Synonym: Bisabolol
Target: Apoptosis, Antioxidant
TargetMol Loading
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