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抑制剂 & 化合物

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天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T0482	Sertraline hydrochloride Sertraline HCl,CP-51974-1 HCl,盐酸舍曲林	5-HT Receptor; Serotonin Transporter	GPCR/G Protein; Neuroscience
	Sertraline hydrochloride (Sertraline HCl) 是选择性 5- 羟色胺再吸收抑制剂类的抗抑郁剂，可用于多种疾病的研究，如重度抑郁症和强迫症。
T1483	Citalopram hydrobromide Lu 10-171,Nitalapram HBr,Bonitrile HBr,XU-62-320,Lu 10-171 HBr,氢溴酸西酞普兰,Citalopram HBr	5-HT Receptor; Serotonin Transporter; Autophagy	Autophagy; GPCR/G Protein; Neuroscience
	Citalopram hydrobromide (XU-62-320) 是一种选择性 5-羟色胺再摄取抑制剂，可选择性地抑制 CNS 神经元对 5-羟色胺的再摄取，从而增强中枢神经系统中的 5-羟色胺能活性，也具有抗抑郁活性。它抑制兔血小板中 5-HT 的摄取，IC50为 14 nM。
T6232	Vilazodone Hydrochloride 盐酸维拉佐酮,SB659746A,EMD 68843,Vilazodone HCl	Others; 5-HT Receptor; Serotonin Transporter	GPCR/G Protein; Neuroscience; Others
	Vilazodone Hydrochloride (EMD 68843) 是 5-HT1A 受体和特异性 5-羟色胺再摄取抑制剂(SSRI) 的部分激动剂，用于治疗重度抑郁症。
T1636L	Paroxetine hydrochloride hemihydrate Paroxetine Hydrochloride,Paxil,Paroxetine HCl,Seroxat	5-HT Receptor	GPCR/G Protein; Neuroscience
	Paroxetine hydrochloride hemihydrate (Paxil) 是一种抗抑郁药，为高效的五羟色胺再摄取抑制剂，能抑制 GRK2 活性，IC50 为 14 μM。
T6493	Escitalopram Oxalate 草酸右旋西酞普兰,依他普仑草酸盐,Cipralex,(S)-(+)Citalopram oxalate	Others; 5-HT Receptor; Serotonin Transporter	GPCR/G Protein; Neuroscience; Others
	Escitalopram Oxalate ((S)-(+)Citalopram oxalate) 是一种外消旋 Citalopram 的 S-对映体，是一种选择性 5-羟色胺再摄取抑制剂，Ki=0.89 nM，比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性，是一种研究抑郁症的抗抑郁药。
T20828	Citalopram Cipram,Lu 10-171,Lu-10-171 Lu10-171	5-HT Receptor	GPCR/G Protein; Neuroscience
	Citalopram (Lu 10-171) 是一种具有口服活性的、选择性的血清素再摄取抑制剂 (SSRI)，是一种选择性5-羟色胺再摄取抑制剂，是一种 S(+)-对映体 (Escitalopram) 和 R(-)-对映体的外消旋混合物。Citalopram 具有抗抑郁活性，可增强血清素能神经传递，可用于研究老年痴呆。
T1279	Vilazodone 维拉佐酮,SB659746A,EMD 68843	5-HT Receptor; Serotonin Transporter	GPCR/G Protein; Neuroscience
	Vilazodone (SB659746A) 是一种可口服的选择性 5 -羟色胺再摄取抑制剂 (SSRI) 和部分5-HT1A 受体激动剂。它有抗抑郁作用，可用于抑郁症和情绪性疾病的研究。
T6461	Dapoxetine hydrochloride LY-210448,LY-210448 hydrochloride,Dapoxetine HCl,盐酸达泊西汀,Priligy	5-HT Receptor; Serotonin Transporter	GPCR/G Protein; Neuroscience
	Dapoxetine hydrochloride (LY-210448 hydrochloride) 是一种具有口服活性的、选择性的血清素再摄取 (serotonin reuptake) 抑制剂 (SSRI)，可用于研究早泄 (PE) 。
T67956L	Litoxetine HCl litoxetine HCL(86811-09-8 Free base)	5-HT Receptor	GPCR/G Protein; Neuroscience
	Litoxetine HCl 是一种选择性5-羟色胺（5-HT）再摄取抑制剂（SSRI）和混合5-羟色胺拮抗剂，可用于治疗尿失禁。Litoxetine HCl 在没有抗毒蕈碱特性的浓度下（10 nM-1 microM）引起大鼠离体食道肌肉粘膜的浓度依赖性松弛，使卡巴胆碱张力降低达37%,更高浓度的Litoxetine HCl（3微摩-300微摩）与明显的松弛有关，直至取消卡巴胆碱张力。以前在离体豚鼠肠道中证明的利托西汀的抗心律失常活性，在浓度大于1 microM 时在大鼠离体食道肌肉粘膜中发挥了作用。 Litoxetine HCl 的5-HT 释放作用可以解释利托西汀对未处理的大鼠组织中的5-HT 诱导的松弛的效力，这种效力被pCPA 处理所逆转。
T68683	Sertraline Free Base
	Sertraline Free Base is a Selective Serotonin Reuptake Inhibitor (SSRI). It can treat depression, obsessive-compulsive disorder (OCD), posttraumatic stress disorder (PTSD), premenstrual dysphoric disorder (PMDD), social anxiety disorder, and panic disorder.
T68579	Fluvoxamine acid
	Fluvoxamine acid is a medication which functions as a selective serotonin reuptake inhibitor (SSRI) and σ1 receptor agonist. Fluvoxamine is used primarily for the treatment of obsessive-compulsive disorder (OCD), and is also used to treat major depressive disorder (MDD), and anxiety disorders such as panic disorder and post-traumatic stress disorder (PTSD).
T28042	MIN-117 Wf516,Wf 516,Wf-516
	MIN-117, a SSRI/5-HT receptor antagonist, is potentially used for the treatment of depression.
T35920	N-methyl Paroxetine
	N-methyl Paroxetine is a derivative of the selective serotonin reuptake inhibitor (SSRI) antidepressant paroxetine that inhibits [3H]paroxetine binding to rat cortical membranes (Ki = 4.3 nM). It inhibits serotonin uptake in rat brain synaptosomes with an IC50 value of 22 nM. N-methyl Paroxetine has been used as a precursor in the synthesis of paroxetine and is a potential impurity in commercial preparations of paroxetine.
T68670	Panuramine
	Panuramine is an antidepressant which was synthesized in 1981 by Wyeth. It acts as a potent and selective serotonin reuptake inhibitor (SSRI).
T68680	CP-53631
	CP-53631 is a selective serotonin reuptake inhibitor (SSRI)
T13300	Vilazodone-d8 维拉佐酮D8	Others	Others
	Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.
T22395	Paroxetine mesylate	Others	Others
	Paroxetine Mesylate, the mesylate salt form of paroxetine, is a phenylpiperidine derivative and a selective serotonin reuptake inhibitor (SSRI) with anxiolytic and antidepressant properties.
T71389	Fluoxetine oxalate
	Fluoxetine oxalate is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class. It is used for the treatment of major depressive disorder, obsessive–compulsive disorder, bulimia nervosa, panic disorder, and premenstrual dysphoric disorder.
T71587	Fluoxetine succinate ester
	Fluoxetine succinate ester is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class. It is used for the treatment of major depressive disorder, obsessive–compulsive disorder, bulimia nervosa, panic disorder, and premenstrual dysphoric disorder.
T36521	Alaproclate (hydrochloride)
	Alaproclate is a selective serotonin reuptake inhibitor (SSRI).1,2 It inhibits depletion of serotonin (5-HT) induced by 4-methyl-α-ethyl-m-tyramine in rat cerebral cortex, hippocampus, hypothalamus, and striatum (EC50s = 18, 4, 8, and 12 mg/kg, respectively).1 Alaproclate inhibits NMDA-evoked currents and depolarization-induced voltage-dependent potassium currents in rat hippocampal neurons (IC50s = 1.1 and 6.9 μM, respectively) and does not inhibit GABA-evoked currents when used at concentratio...

化合物

Sertraline hydrochloride

Cat.No: T0482

Synonym: Sertraline HCl,CP-51974-1 HCl,盐酸舍曲林

Target: 5-HT Receptor, Serotonin Transporter

Citalopram hydrobromide

Cat.No: T1483

Synonym: Lu 10-171,Nitalapram HBr,Bonitrile HBr,XU-62-320,Lu 10-171 HBr,氢溴酸西酞普兰,Citalopram HBr

Target: 5-HT Receptor, Serotonin Transporter, Autophagy

Vilazodone Hydrochloride

Cat.No: T6232

Synonym: 盐酸维拉佐酮,SB659746A,EMD 68843,Vilazodone HCl

Target: Others, 5-HT Receptor, Serotonin Transporter

Paroxetine hydrochloride hemihydrate

Cat.No: T1636L

Synonym: Paroxetine Hydrochloride,Paxil,Paroxetine HCl,Seroxat

Target: 5-HT Receptor

Escitalopram Oxalate

Cat.No: T6493

Synonym: 草酸右旋西酞普兰,依他普仑草酸盐,Cipralex,(S)-(+)Citalopram oxalate

Target: Others, 5-HT Receptor, Serotonin Transporter

Cat.No: T20828

Synonym: Cipram,Lu 10-171,Lu-10-171 Lu10-171

Target: 5-HT Receptor

Cat.No: T1279

Synonym: 维拉佐酮,SB659746A,EMD 68843

Target: 5-HT Receptor, Serotonin Transporter

Dapoxetine hydrochloride

Cat.No: T6461

Synonym: LY-210448,LY-210448 hydrochloride,Dapoxetine HCl,盐酸达泊西汀,Priligy

Target: 5-HT Receptor, Serotonin Transporter

Cat.No: T67956L

Synonym: litoxetine HCL(86811-09-8 Free base)

Target: 5-HT Receptor

Sertraline Free Base

Cat.No: T68683

Fluvoxamine acid

Cat.No: T68579

Cat.No: T28042

Synonym: Wf516,Wf 516,Wf-516

N-methyl Paroxetine

Cat.No: T35920

Cat.No: T68670

Cat.No: T68680

Cat.No: T13300

Synonym: 维拉佐酮D8

Target: Others

Paroxetine mesylate

Cat.No: T22395

Target: Others

Fluoxetine oxalate

Cat.No: T71389

Fluoxetine succinate ester

Cat.No: T71587

Alaproclate (hydrochloride)

Cat.No: T36521

Cat. No.	Product Name	Target	Signaling Pathways
T0185	Escitalopram Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram	Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Escitalopram (Seroplex) 是一种外消旋 Citalopram 的 S-对映体，是一种选择性 5-羟色胺再摄取抑制剂，Ki=0.89 nM，比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性，是一种研究抑郁症的抗抑郁药。

天然产物

Cat.No: T0185

Synonym: Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram

Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor

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