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Cat. No.	Product Name	Target	Signaling Pathways
T6972	RS-1	DNA/RNA Synthesis	Cell Cycle/Checkpoint; DNA Damage/DNA Repair
	RS-1 是一种 RAD51 的激活剂，同时可增强 CRISPR/Cas9 的活性。
T24741	RS1-PDK1 inhibitor RS-1,RS1,RS 1	PDK	PI3K/Akt/mTOR signaling
	RS1-PDK1 inhibitor (RS 1) 是一种选择性的蛋白激酶PDK1抑制剂，可用来治疗和预防疾病或失调。
T7519	RS-127445 hydrochloride 4-(4-氟-1-萘基)-6-(1-甲基乙基)-2-嘧啶胺盐酸盐,RS 127445,MT 500	5-HT Receptor	GPCR/G Protein; Neuroscience
	RS-127445 hydrochloride (MT 500) 是一种可口服的，高亲和力选择性5-HT2B 受体拮抗剂，pKi 为 9.5，比作用于其他受体和离子通道的选择性高 1000 倍。
T21468	CVT-2738 UNII-NYS3I6283H,CVT 2738,EC 610-916-8,CVT2738,RS-94287,N-(2,6-二甲基苯基)-1-哌嗪乙酰胺	Others	Others
	CVT-2738 (RS-94287) 是雷诺嗪的代谢物。 Ranolazine 是一种部分脂肪酸氧化 (pFOX) 抑制剂和抗心绞痛药物。
T6018	Zosuquidar trihydrochloride 唑喹达三盐酸盐,Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride	P-gp	Membrane transporter/Ion channel; Neuroscience
	Zosuquidar trihydrochloride (LY-335979 trihydrochloride) 是一种P-糖蛋白抑制剂，Ki 值为 59 nM。
T68051	Delequamine RS 15385-197	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Delequamine (RS 15385-197) 是一种有效的选择性 α2-肾上腺素受体拮抗剂。
T11032	DHPG (RS)-3,5-DHPG,DL-Α-(3,5-二羟基苯基)甘氨酸	GluR	Neuroscience
	DHPG ((RS)-3,5-DHPG) 是一种氨基酸，是选择性代谢型谷氨酸受体 mGluR 的激动剂，也是与磷脂酶 D 耦合的 mGluR 的有效拮抗剂。
T16799	RS-246204	Others	Others
	RS-246204 is an R-spondin-1 substitute compound. RS-246204 is able to initiate small intestinal organoids without the use of the R-spondin-1 protein.
T24740	RS-104966
	RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.
T60242	(RS)-AMPA monohydrate
	(RS)-AMPA ((±)-AMPA) monohydrate 是谷氨酸的一种类似物，对兴奋性神经递质 L-谷氨酸 (L-glutamic acid) 有激动作用。(RS)-AMPA monohydrate 不会干扰海藻酸或 NMDA 受体的结合位点。
T13439	(RS)-Butyryltimolol	Cysteine Protease	Proteases/Proteasome
	(RS)-Butyryltimolol 是 Butyryltimolol 的消旋体。Butyryltimolol 是 Timolol 的有效前药。Timolol 用于青光眼研究，但是难以透过角膜，经化学结构修饰后得到 Butyryltimolol，透过眼角膜的能力增强。Butyryltimolol 进入眼球后，经酶水解再生成 Timolol 而起作用。Butyryltimolol 是一种 β-肾上腺素能 (β-adrenergic) 阻滞剂。
T70661	Azalanstat mesylate
	Azalanstat mesylate is an anti-obesity drug acting as a lanosterol 14α-demethylase inhibitor. Azalanstat mesylate has been shown to inhibit cholesterol synthesis in HepG2 cells, human fibroblasts, hamster hepatocytes and hamster liver, by inhibiting the cytochrome P450 enzyme lanosterol 14 alpha-demethylase. When administered orally to hamsters fed regular chow, RS-21607 (50 mg/kg/day) lowered serum cholesterol in a dose-dependent manner (ED50 = 62 mg/kg) in a period of 1 week. It preferentially...
T70660	Azalanstat HCl
	Azalanstat HCl is an anti-obesity drug acting as a lanosterol 14α-demethylase inhibitor. Azalanstat HCl has been shown to inhibit cholesterol synthesis in HepG2 cells, human fibroblasts, hamster hepatocytes and hamster liver, by inhibiting the cytochrome P450 enzyme lanosterol 14 alpha-demethylase. When administered orally to hamsters fed regular chow, RS-21607 (50 mg/kg/day) lowered serum cholesterol in a dose-dependent manner (ED50 = 62 mg/kg) in a period of 1 week. It preferentially lowered l...
T10462L	Bavisant dihydrochloride hydrate JNJ31001074AAC	Others	Others
	Bavisant dihydrochloride hydrate (JNJ31001074AAC) is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatment for ADHD. in vivo: Mean change

化合物

Cat.No: T6972

Target: DNA/RNA Synthesis

RS1-PDK1 inhibitor

Cat.No: T24741

Synonym: RS-1,RS1,RS 1

Target: PDK

RS-127445 hydrochloride

Cat.No: T7519

Synonym: 4-(4-氟-1-萘基)-6-(1-甲基乙基)-2-嘧啶胺盐酸盐,RS 127445,MT 500

Target: 5-HT Receptor

Cat.No: T21468

Synonym: UNII-NYS3I6283H,CVT 2738,EC 610-916-8,CVT2738,RS-94287,N-(2,6-二甲基苯基)-1-哌嗪乙酰胺

Target: Others

Zosuquidar trihydrochloride

Cat.No: T6018

Synonym: 唑喹达三盐酸盐,Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride

Target: P-gp

Cat.No: T68051

Synonym: RS 15385-197

Target: Adrenergic Receptor

Cat.No: T11032

Synonym: (RS)-3,5-DHPG,DL-Α-(3,5-二羟基苯基)甘氨酸

Target: GluR

Cat.No: T16799

Target: Others

Cat.No: T24740

(RS)-AMPA monohydrate

Cat.No: T60242

(RS)-Butyryltimolol

Cat.No: T13439

Target: Cysteine Protease

Azalanstat mesylate

Cat.No: T70661

Cat.No: T70660

Bavisant dihydrochloride hydrate

Cat.No: T10462L

Synonym: JNJ31001074AAC

Target: Others

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