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Cat. No.	Product Name	Target	Signaling Pathways
T23087	NPY 5RA972	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	NPY 5RA972 是一种神经肽 Y Y5 受体拮抗剂
TP2194L	Neuropeptide Y (scrambled) Acetate Pro-Neuropeptide Y (scrambled) Acetate,NPY (scrambled) Acetate	Others	Others
	Neuropeptide Y (scrambled) Acetate (Pro-Neuropeptide Y (scrambled) Acetate) 是一种 Neuropeptide Y 的杂序肽，Neuropeptide Y 参与阿尔茨海默病 (AD) ，可能具有神经保护作用。
T83677	Neuropeptide Y (porcine, bovine) TFA NPY (porcine, bovine)
	神经肽Y（Neuropeptide Y, NPY）是一种参与调节食欲、血管收缩、心脏收缩力和肠道分泌的神经肽，同时也是NPY受体Y1、Y2和Y5的激动剂。它在全身范围内表达。NPY能够在表达大鼠Y1或Y2以及表达大鼠Y5的HEK293细胞中选择性抑制由forskolin诱导的cAMP积累，而对表达大鼠Y4受体的L-M(TK-)细胞的影响较小（EC50分别为0.15、2.7、0.66和>1,000 nM)。在分离的豚鼠心脏模型中，NPY能够增加灌注压（EC30 = 1.3 nM）。神经内注射NPY（300 pmol/动物）能够在大鼠中增加食物摄取量。
T71749	SF-22	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	SF-22 是一种可透过血脑屏障的神经肽 Y 受体(Y2R) 拮抗剂，具有潜在抗炎活性，可用于研究神经系统紊乱带来的疾病。
T23094	NTNCB hydrochloride	Others; Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience; Others
	NTNCB hydrochloride 是一种神经肽 Y Y5 受体的拮抗剂。
T8963	CYM2503	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	CYM2503 是 GAL2 受体的正变构调节剂 (PAM)，可在体外增强甘丙肽诱导的 IP1 产生。它对受体的正构甘丙肽结合位点没有亲和力（通过其无法置换碘化甘丙肽或自行诱导 IP1 积累来衡量）。
TQ0286	MK-0557	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	MK-0557 是神经肽 Y5 受体的选择性口服拮抗剂，Ki 值为1.6 nM。
TP2206	[Leu31,Pro34]-Neuropeptide Y (porcine) LEU 31, PRO34]-神经肽Y(猪)	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	[Leu31,Pro34]- Neuropeptide Y (porcine) 是神经肽 Y (NPY) 的一种类似物，是对NPY Y1受体有选择性的激动作用。它表现出抗焦虑作用。
TP1380	Galanin (1-16), mouse, porcine, rat	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	Galanin (1-16), mouse, porcine, rat 是一种有效的甘丙肽受体激动剂，Kd 为 3 nM。
T17222	Velneperit 韦利贝特,S2367	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	Velneperit (S2367) 是一种有效且选择性的神经肽 Y (NPY) Y5 受体，有用于治疗肥胖症的研究潜力。
T10539	BIBO3304 TFA	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	BIBO3304 TFA 是一种可口服的、选择性的神经肽 Y(NPY) Y1受体高效拮抗剂，对人和大鼠 Y1 受体均具有高亲和力，IC50分别为 0.38 和 0.72 nM。
T5587	CGP71683 hydrochloride CGP71683A,盐酸CGP71683	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	CGP71683 hydrochloride (CGP71683A) 是竞争性的神经肽受体拮抗剂，Ki 值为 1.3 nM。
T1997	JNJ-31020028 JNJ 31020028	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	JNJ-31020028是神经肽Y2受体选择性可脑渗透抑制剂，对人Y2和鼠源Y2受体pIC50值分别为8.07和8.22，其神经肽 Y2 受体的选择性比人 Y1/Y4/Y5 受体高 100 倍。
TP1059	Peptide YY (PYY) (3-36), human Peptide YY (3-36)	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) 是一种肠胃激素肽，可以激动Y2受体，具有降低食欲的功效。
T5455	HT-2157 SNAP37889,SNAP-37889	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	HT-2157 (SNAP-37889) 是一种高亲和力、选择性和竞争性的甘丙肽 3 受体 (Gal3) 拮抗剂。
T8456	GALNON	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	Galnon 是一种甘丙肽受体激动剂，可改善内在的皮质骨组织特性。
T12895	SHA 68	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	SHA 68 是一种有效且选择性的神经肽 S 受体 (NPSR) 非肽拮抗剂，对 NPSR Asn107和 NPSR Ile107的IC50分别为 22.0 和 23.8 nM，具有有限的血脑屏障渗透能力和用于神经痛的活性。
T75913	[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic polypeptide TFA
	[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide 为高效且选择性的神经肽 YY5 受体激动剂，其与 hY5 受体的结合 IC50 值为 0.24 nM，已知可促进饮食摄入。
T4445	Tolfenpyrad	Antibacterial	Microbiology/Virology
	Tolfenpyrad 是杀虫剂，用于对抗对现有杀虫剂（如有机磷酸酯和氨基甲酸酯）具有抗药性的害虫。
T0435	Sulfinpyrazone (+/-)-Sulfinpyrazone,G-28315,苯磺保泰松,NSC 75925	COX	Immunology/Inflammation; Neuroscience
	Sulfinpyrazone (NSC-75925) 是一种口服有效的尿酸剂，具有抗血栓和血小板抑制作用。它可作用于慢性和间歇性痛风性关节炎。
T6607	Nitenpyram 烯啶虫胺,Niterndipoine,烯啶蟲胺,Bestguard,Capstar	AChR	Neuroscience
	Nitenpyram (Capstar) 是一种烟碱型乙酰胆碱受体 (AchR) 激动剂，IC50为 14 nM，用作治疗牲畜和宠物寄生虫的兽药。
T8692	(Rac)-Benpyrine	TNF	Apoptosis
	(Rac)-Benpyrine 是一种有效且具有口服活性的 TNF-α 抑制剂，是Benpyrine 的外消旋体。它可研究TNF-α介导的炎症和自身免疫性疾病。
T4446	Tebufenpyrad Pyranica,吡螨胺,MK239,Comanche	Mitochondrial Metabolism	Metabolism
	Tebufenpyrad (Comanche) 是一种重要的农业化学杀螨剂，其作用类似于已知的线粒体毒物 rotenone。
T19714	Fenpyroximate	Others	Others
	Fenpyroximate 是一种有效的杀螨剂。
TP1963	[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide cpp1-7-npy19-23-ala31-aib32-gln34-hpancreatic-polypeptide,[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - hPancreatic Polypeptide
	Potent, selective peptide agonist for the neuropeptide Y Y5 receptor (IC50 values for inhibition of NPY binding to human Y5, Y1, Y2 and Y4 receptors are 0.24, 530, > 500, and 51 nM respectively, Ki at Y5 = 0.1 - 0.15 nM). Stimulates food intake in vivo.
T38763	Mefenpyr-diethyl
	Mefenpyr-diethyl is an herbicide safener, which protects crops against herbicide injury.
T33968	Phenchlobenpyrrone
	Phenchlobenpyrrone has potential as a treatment for Alzheimer's disease.
T76553	TAT (47-57) GGG-Cys(Npys)
	TAT (47-57) GGG-Cys(Npys)为一种细胞穿透肽(CPP)，显示了在细胞内药物递送研究中的应用潜力。
T36486	Benpyrine
	Benpyrine is a highly specific and orally active TNF-α inhibitor with a KD value of 82.1 μM. Benpyrine tightly binds to TNF-α and blocks its interaction with TNFR1, with an IC50 value of 0.109 μM. Benpyrine has the potential for TNF-α mediated inflammatory and autoimmune disease research[1]. Benpyrine (5-20 μM; 14 hours; RAW264.7 cells) pretreatment results in a dose-dependent decrease in the phosphorylation of IκBα in RAW264.7 cells (stimulated with 10 ng/mL TNF-α or 1 μg/mL LPS). Benpyrine abo...
T76545	Cys(Npys)-TAT (47-57)
	Cys(Npys)-TAT(47-57)为TAT多肽中的一个段，可通过静电相互作用与质粒DNA结合。该段对应TAT的转导域，并含有活化的C端半胱氨酸残基。TAT为HIV-1编码的一种核转录激活蛋白。
T21611L	BWX 46 Acetate BWX 46 Acetate(172997-92-1 Free base)	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	BWX 46 Acetate 是一种有效的、高度选择性的神经肽 Y (NPY) 受体激动剂，IC50 为 0.5 nM。
TP1044L	Pancreatic Polypeptide, rat acetate	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	Pancreatic Polypeptide, rat acetate 是 NPY 受体的激动剂，对 NPYR4 具有高亲和力。
TP1984L	[D-Trp34]-Neuropeptide Y Acetate [D-Trp34]-Neuropeptide Y Acetate (153549-84-9 Free base)	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	[D-Trp34]-Neuropeptide Y Acetate 是有效的、选择性的神经肽 Y (NPY) Y5 受体激动剂，在 NPY Y1，Y2，Y4 和 y6 受体上的效力较低。[D-Trp34]-Neuropeptide Y Acetate 可以显著增加大鼠的食物摄入量。
T24121	GW438014A GW 438014 A,GW-438014-A	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	GW438014A 是一种有效且具有选择性的 NPY-Y5 受体拮抗剂。GW438014A 对食物摄入并减少肥胖啮齿动物的体重增加具有抑制作用。
TP1137L	Pancreatic Polypeptide (human) acetate	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	Pancreatic Polypeptide (human) acetate 是一种 C 末端酰胺化的 36 个氨基酸肽，可作为神经肽 Y (NPY) Y4/Y5 受体激动剂。
TP1618L	PACAP-38 (31-38), human, mouse, rat acetate PACAP-38 (31-38), human, mouse, rat acetate(138764-85-9 Free base)	PACAP	GPCR/G Protein
	PACAP-38 (31-38), human, mouse, rat acetate 是 PAC1 受体的激活剂。PACAP-38 (31-38), human, mouse, rat acetate 对交感神经元 NPY 和儿茶酚胺的产生具有强效、有效和持续的刺激作用，可用于神经营养和神经保护研究。
T70952	UR-MK299
	UR-MK299 is a NPY Y1 receptor antagonist.
T35599	Neuropeptide Y (3-36) (human, rat) (trifluoroacetate salt)
	Neuropeptide Y (NPY) (3-36) is a C-terminal fragment of NPY, a neuropeptide involved in controlling appetite, blood pressure, cardiac contractility, and intestinal secretion. NPY (3-36) is an endogenous peptide produced by cleavage of NPY by dipeptidyl peptidase 4 (DPP-4). It binds selectively to the NPY receptor Y2 (Ki = 0.41 nM in CHP 234 cells) over the Y1 receptor, where it does not bind at concentrations up to 1 μM. NPY (3-36) (0.1 nM) increases migration of human umbilical vein endothelial...
T23287	S 25585	Others	Others
	S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.
T29171	Y2 Antagonist 36
	Y2 Antagonist 36 is a highly potent, soluble and selective antagonist of NPY Y2.
T22935	LU AA33810	Others	Others
	LU AA33810 is a neuropeptide Y (NPY) Y5 receptor antagonist.
T10921	CYM 9484	Others	Others
	CYM 9484 is a selective and potent neuropeptide Y (NPY) Y2 receptor antagonist with IC50 value of 19 nM.
T71091	Y2-Antagonist-2
	Y2-Antagonist-2 is a novel, selective, soluble non-peptidic NPY Y2 receptor antagonist with enhanced CNS exposure.
T75911	[D-Trp34]-Neuropeptide Y TFA
	[D-Trp34]-Neuropeptide Y TFA，一种高效且选择性的神经肽Y (NPY) Y5受体激动剂，其在NPY Y1、Y2、Y4及Y6受体上的活性显著低于Y5受体。该化合物能显著提高大鼠的食物摄入量。
TP1618	PACAP-38 (31-38), human, mouse, rat
	PACAP-38 (31-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine production.
T26800	BIBO3304 BIBO-3304,BIBO 3304
	BIBO3304 is a selective NPY Y1 receptor antagonist (IC50 values are 0.38 and 0.72 nM at human and rat receptors respectively). BIBO3304 inhibits NPY- and fasting-induced feeding in vivo following central administration.
T69220	GW438014 free base
	GW438014A is a selective NPY-Y5 receptor antagonist.
TP2194	Neuropeptide Y (scrambled)	Others	Others
	Neuropeptide Y (NPY) is a 36-amino acid neuropeptide that exerts its activity via G-protein-coupled receptors. NPY is widely distributed in the peripheral and central nervous systems. It modulates a variety of physiological processes, e.g. the central reg
T14572	BIIE-0246 AR-H 053591	Others	Others
	BIIE-0246 is a potent and highly selective non-peptide neuropeptide Y (NPY) Y2 receptor antagonist. With an IC50 of 15 nM.
TP2215	Agouti-related Protein (AGRP) (25-82), human	Others	Others
	Agouti-related peptide (AgRP) is a neuropeptide produced in the brain by the AgRP/NPY neuron. It is only synthesized in NPY containing cell bodies located in the ventromedial part of the arcuate nucleus in the hypothalamus. The appetite-stimulating effect

化合物

Cat.No: T23087

Target: Neuropeptide Y Receptor

Neuropeptide Y (scrambled) Acetate

Cat.No: TP2194L

Synonym: Pro-Neuropeptide Y (scrambled) Acetate,NPY (scrambled) Acetate

Target: Others

Neuropeptide Y (porcine, bovine) TFA

Cat.No: T83677

Synonym: NPY (porcine, bovine)

Cat.No: T71749

Target: Neuropeptide Y Receptor

NTNCB hydrochloride

Cat.No: T23094

Target: Others, Neuropeptide Y Receptor

Cat.No: T8963

Target: Neuropeptide Y Receptor

Cat.No: TQ0286

Target: Neuropeptide Y Receptor

[Leu31,Pro34]-Neuropeptide Y (porcine)

Cat.No: TP2206

Synonym: LEU 31, PRO34]-神经肽Y(猪)

Target: Neuropeptide Y Receptor

Galanin (1-16), mouse, porcine, rat

Cat.No: TP1380

Target: Neuropeptide Y Receptor

Cat.No: T17222

Synonym: 韦利贝特,S2367

Target: Neuropeptide Y Receptor

Cat.No: T10539

Target: Neuropeptide Y Receptor

CGP71683 hydrochloride

Cat.No: T5587

Synonym: CGP71683A,盐酸CGP71683

Target: Neuropeptide Y Receptor

Cat.No: T1997

Synonym: JNJ 31020028

Target: Neuropeptide Y Receptor

Peptide YY (PYY) (3-36), human

Cat.No: TP1059

Synonym: Peptide YY (3-36)

Target: Neuropeptide Y Receptor

Cat.No: T5455

Synonym: SNAP37889,SNAP-37889

Target: Neuropeptide Y Receptor

Cat.No: T8456

Target: Neuropeptide Y Receptor

Cat.No: T12895

Target: Neuropeptide Y Receptor

[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic polypeptide TFA

Cat.No: T75913

Cat.No: T4445

Target: Antibacterial

Cat.No: T0435

Synonym: (+/-)-Sulfinpyrazone,G-28315,苯磺保泰松,NSC 75925

Target: COX

Cat.No: T6607

Synonym: 烯啶虫胺,Niterndipoine,烯啶蟲胺,Bestguard,Capstar

Target: AChR

(Rac)-Benpyrine

Cat.No: T8692

Target: TNF

Cat.No: T4446

Synonym: Pyranica,吡螨胺,MK239,Comanche

Target: Mitochondrial Metabolism

Cat.No: T19714

Target: Others

[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide

Cat.No: TP1963

Synonym: cpp1-7-npy19-23-ala31-aib32-gln34-hpancreatic-polypeptide,[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - hPancreatic Polypeptide

Mefenpyr-diethyl

Cat.No: T38763

Phenchlobenpyrrone

Cat.No: T33968

TAT (47-57) GGG-Cys(Npys)

Cat.No: T76553

Cat.No: T36486

Cys(Npys)-TAT (47-57)

Cat.No: T76545

Cat.No: T21611L

Synonym: BWX 46 Acetate(172997-92-1 Free base)

Target: Neuropeptide Y Receptor

Pancreatic Polypeptide, rat acetate

Cat.No: TP1044L

Target: Neuropeptide Y Receptor

[D-Trp34]-Neuropeptide Y Acetate

Cat.No: TP1984L

Synonym: [D-Trp34]-Neuropeptide Y Acetate (153549-84-9 Free base)

Target: Neuropeptide Y Receptor

Cat.No: T24121

Synonym: GW 438014 A,GW-438014-A

Target: Neuropeptide Y Receptor

Pancreatic Polypeptide (human) acetate

Cat.No: TP1137L

Target: Neuropeptide Y Receptor

PACAP-38 (31-38), human, mouse, rat acetate

Cat.No: TP1618L

Synonym: PACAP-38 (31-38), human, mouse, rat acetate(138764-85-9 Free base)

Target: PACAP

Cat.No: T70952

Neuropeptide Y (3-36) (human, rat) (trifluoroacetate salt)

Cat.No: T35599

Cat.No: T23287

Target: Others

Y2 Antagonist 36

Cat.No: T29171

Cat.No: T22935

Target: Others

Cat.No: T10921

Target: Others

Y2-Antagonist-2

Cat.No: T71091

[D-Trp34]-Neuropeptide Y TFA

Cat.No: T75911

PACAP-38 (31-38), human, mouse, rat

Cat.No: TP1618

Cat.No: T26800

Synonym: BIBO-3304,BIBO 3304

GW438014 free base

Cat.No: T69220

Neuropeptide Y (scrambled)

Cat.No: TP2194

Target: Others

Cat.No: T14572

Synonym: AR-H 053591

Target: Others

Agouti-related Protein (AGRP) (25-82), human

Cat.No: TP2215

Target: Others

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