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10

抑制剂 & 化合物

2

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Cat. No. Product Name Target Signaling Pathways
T0891 Dapsone

DDS,4,4‘-Sulfonyldianiline,氨苯砜,Bis(4-aminophenyl) sulfone,Sulphadione,4,4'-Diaminodiphenylsulfone,4-Aminophenyl sulfone

Reactive Oxygen Species; Antibacterial; Antibiotic; Parasite Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Dapsone (Sulphadione) 是具有口服活性和血脑渗透通透性的磺酰类抗生素,具有抑菌、抗细菌和抗原虫活性。它有抗麻风活性,抑制麻风杆菌细胞提取物中叶酸的合成。它可研究皮肤病。
T0441 Pasiniazid

Pasiniazide,帕司烟肼,Paraniazide,Isonicotinic acid hydrazide p-aminosalicylate

COX; NADPH Immunology/Inflammation; Metabolism; Neuroscience
Pasiniazid (Paraniazide) 是抗麻风及抗结核药。
T0748 Sulfameter

5-Methoxysulfadiazine,Sulfametoxydiazine,磺胺对甲氧嘧啶

DHFR; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Sulfameter (Sulfametoxydiazine) 是一种长效磺胺类抗生素,具有抗菌活性。它可研究尿路感染和麻风病。
T12644L (S)-Thalidomide

(S)-(-)-Thalidomide

Apoptosis Apoptosis
(S)-Thalidomide ((S)-(-)-Thalidomide) 是 Thalidomide 的 S 型异构体,具有免疫调节,抗炎,抗癌,抗血管生成活性和促凋亡活性,可用于研究麻风结节性红斑和骨髓瘤。
T35903 N-acetyl Dapsone

Antibacterial; Parasite Microbiology/Virology
N-acetyl Dapsone 是一种抗炎和抗菌化合物,广泛用于治疗麻风病、疟疾、痤疮和各种免疫疾病。
T27018 CID21480113

CID21480113, an antibacterial agent, is effective in treating dapsone resistant leprosy.
T34747 Sulfoxone sodium

Sulfoxone,Aldesulfone,Adesulfone Sodium,NSC 27222,Diasone

Sulfoxone sodium ( Adesulfone Sodium) is an anti-leprosy drug.
T19868 Thiambutosine

SC 682,SC-682,SU-1906,SU 1906,SC682,SU1906

Thiambutosine was a candidate that is used for treatment of lepromatous leprosy.
T26733 B 746

B-746,B746

B 746 is an antibacterial agent primarily. B 746 is used in therapy for leprosy and Mycobacterium avium infections as well as against Mycobacterium tuberculosis, including those with multi-drug resistance.
T61592 Thalidomide-piperazine hydrochloride

Thalidomide-piperazine hydrochloride is a chemical compound with potential applications in the research of leprosy and multiple myeloma. It serves as a valuable tool in developmental biology, facilitating significant discoveries in the biochemical pathways of limb development [1].

化合物

Dapsone
Cat.No: T0891
Synonym: DDS,4,4‘-Sulfonyldianiline,氨苯砜,Bis(4-aminophenyl) sulfone,Sulphadione,4,4'-Diaminodiphenylsulfone,4-Aminophenyl sulfone
Target: Reactive Oxygen Species, Antibacterial, Antibiotic, Parasite
Pasiniazid
Cat.No: T0441
Synonym: Pasiniazide,帕司烟肼,Paraniazide,Isonicotinic acid hydrazide p-aminosalicylate
Target: COX, NADPH
Sulfameter
Cat.No: T0748
Synonym: 5-Methoxysulfadiazine,Sulfametoxydiazine,磺胺对甲氧嘧啶
Target: DHFR, Antibacterial, Antibiotic
(S)-Thalidomide
Cat.No: T12644L
Synonym: (S)-(-)-Thalidomide
Target: Apoptosis
N-acetyl Dapsone
Cat.No: T35903
Synonym:
Target: Antibacterial, Parasite
CID21480113
Cat.No: T27018
Synonym:
Target:
Sulfoxone sodium
Cat.No: T34747
Synonym: Sulfoxone,Aldesulfone,Adesulfone Sodium,NSC 27222,Diasone
Target:
Thiambutosine
Cat.No: T19868
Synonym: SC 682,SC-682,SU-1906,SU 1906,SC682,SU1906
Target:
B 746
Cat.No: T26733
Synonym: B-746,B746
Target:
Thalidomide-piperazine hydrochloride
Cat.No: T61592
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T8347 Rifamycin S

Reactive Oxygen Species; ROS; Antibacterial; Antibiotic Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Rifamycin S 是一种 DNA 依赖性 RNA 聚合酶抑制剂,是一种醌和一种针对革兰氏阳性细菌的抗生素试剂。它是涉及两个电子的可逆氧化还原系统的氧化形式。它能产生活性氧并抑制微粒体脂质过氧化,可研究肺结核和麻风病。
T0070 Pentoxifylline

Oxpentifylline,PTX,己酮可可碱,BL-191

HIV Protease; PDE; Adenosine Receptor; Autophagy Autophagy; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Pentoxifylline (PTX) 是一种具有口服活性的磷酸二酯酶非选择性抑制剂,具有免疫调节、抗炎、抗纤溶、抗增殖和血液流变学改善作用。它可研究周围血管疾病、脑血管疾病和其他一些涉及局部微循环缺陷的疾病。

天然产物

Rifamycin S
Cat.No: T8347
Synonym:
Target: Reactive Oxygen Species, ROS, Antibacterial, Antibiotic
Pentoxifylline
Cat.No: T0070
Synonym: Oxpentifylline,PTX,己酮可可碱,BL-191
Target: HIV Protease, PDE, Adenosine Receptor, Autophagy
TargetMol Loading
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