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抑制剂 & 化合物

11

天然产物

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Cat. No. Product Name Target Signaling Pathways
T3647 HTHQ

HX 1171,HTHQ(1-O-Hexyl-2,3,5-trimethylhydroquinone),1-O-hexyl-2,3,5-trimethylhydroquinone

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
HTHQ (HTHQ(1-O-Hexyl-2,3,5-trimethylhydroquinone)) 是一种强力的亲脂性酚类抗氧化剂。它通过与活性氧直接反应,清除 ROS,从而形成更稳定的自由基,具有很强的抗氧化活性。

化合物

HTHQ
Cat.No: T3647
Synonym: HX 1171,HTHQ(1-O-Hexyl-2,3,5-trimethylhydroquinone),1-O-hexyl-2,3,5-trimethylhydroquinone
Target: Reactive Oxygen Species
Cat. No. Product Name Target Signaling Pathways
TN1772 Isoastilbin

Anti-infection; Tyrosinase; Antibacterial Microbiology/Virology; Proteases/Proteasome
Isoastilbin 是Rhizoma Smilacis glabrae 和Astragalus membranaceus 中的二氢黄酮醇糖苷。它抑制酪氨酸酶活性,还抑制葡萄糖基转移酶,IC50值为 54.3 μg/mL。它具有神经保护、抗氧化、抗微生物和抗凋亡活性,可研究阿尔茨海默氏病。
T11589 Hydroxycitric acid tripotassium hydrate

柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate

ATP Citrate Lyase; HIF/HIF Prolyl-Hydroxylase; HIF Angiogenesis; Chromatin/Epigenetic; Metabolism
Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) 是一种藤黄果的主要活性成分,也是一种柠檬酸的衍生物。它可竞争性抑制柠檬酸裂解酶 (ATP citrate lyase) ,并具有减肥作用。它有效抑制结石形成,并抑制HIF,具有抗氧化,抗炎和抗肿瘤活性。
T0256 Citric acid trilithium salt tetrahydrate

Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate

Dehydrogenase; GSK-3; HIF/HIF Prolyl-Hydroxylase; Antibacterial; GluR Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling; Stem Cells
Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) 是一种用于治疗精神疾病的药物。它也是一种医药和建筑材料, 可用于氨基酸定量分析时的梯度洗脱。
TN5031 Sitostenone

豆甾-4-烯-3-酮

Others Others
Sitostenone 具有抗氧化活性。 Stigmasta-4-en-3-one(Sitostenone)可用于治疗雄激素依赖性疾病,尤其是治疗良性前列腺增生。
TN4220 Homobutein

3-O-Methylbutein,2',4,4'-Trihydroxy-3-methoxychalcone

Antioxidant; NF-κB; HDAC; Parasite; Immunology/Inflammation related Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology; NF-κB; oxidation-reduction
Homobutein (3-O-Methylbutein) 是 HDAC 和 NF-κB 的双重抑制剂,IC50 分别为 190 和 38 μM。 Homobutein 是一种铁螯合剂,具有抗癌、抗炎、抗寄生虫和抗氧化活性。
T6S2038 Ziyuglycoside II

Apoptosis; Antioxidant; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Ziyuglycoside II 是从地榆中提取的一种三萜皂苷,可诱导活性氧 产生和凋亡,具有抗炎和抗癌作用。
TMS2180 Zeaxanthin

Anchovyxanthin,All-Trans-Zeaxanthin,玉米

Antioxidant; Endogenous Metabolite Metabolism; oxidation-reduction
Zeaxanthin (All-Trans-Zeaxanthin) 是食物获得类胡萝卜素,存在于眼睛的黄斑部,具有抗氧化活性。
TN4358 Junipediol A

Others Others
Junipediol A shows antioxidation activity.
TN4360 Junipediol B

Others Others
Junipediol B shows antioxidation activity.
TN2958 3'-Methoxydaidzin

Others Others
3'-Methoxydaidzin has antioxidation activity, it may be a potential neuroprotective substance in Gegen Qinlian decoction.
TN5227 (+/-)-Vestitol

NOS; CXCR; Antifection Autophagy; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology
Vestitol has antioxidation, anti-inflammatory and antimicrobial activities, it can strongly act in a low dose and concentration and have a promising potential to be applied in the pharmaceutical and food industries. Vestitol inhibits neutrophils migration

天然产物

Isoastilbin
Cat.No: TN1772
Synonym:
Target: Anti-infection, Tyrosinase, Antibacterial
Hydroxycitric acid tripotassium hydrate
Cat.No: T11589
Synonym: 柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate
Target: ATP Citrate Lyase, HIF/HIF Prolyl-Hydroxylase, HIF
Citric acid trilithium salt tetrahydrate
Cat.No: T0256
Synonym: Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate
Target: Dehydrogenase, GSK-3, HIF/HIF Prolyl-Hydroxylase, Antibacterial, GluR
Sitostenone
Cat.No: TN5031
Synonym: 豆甾-4-烯-3-酮
Target: Others
Homobutein
Cat.No: TN4220
Synonym: 3-O-Methylbutein,2',4,4'-Trihydroxy-3-methoxychalcone
Target: Antioxidant, NF-κB, HDAC, Parasite, Immunology/Inflammation related
Ziyuglycoside II
Cat.No: T6S2038
Synonym:
Target: Apoptosis, Antioxidant, Reactive Oxygen Species
Zeaxanthin
Cat.No: TMS2180
Synonym: Anchovyxanthin,All-Trans-Zeaxanthin,玉米
Target: Antioxidant, Endogenous Metabolite
Junipediol A
Cat.No: TN4358
Synonym:
Target: Others
Junipediol B
Cat.No: TN4360
Synonym:
Target: Others
3'-Methoxydaidzin
Cat.No: TN2958
Synonym:
Target: Others
(+/-)-Vestitol
Cat.No: TN5227
Synonym:
Target: NOS, CXCR, Antifection
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