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抑制剂 & 化合物

19

天然产物

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Cat. No. Product Name Target Signaling Pathways
T32558 Lanosteryl acetate

Lanosterol acetate

Lanosteryl acetate is a bioactive chemical.

化合物

Lanosteryl acetate
Cat.No: T32558
Synonym: Lanosterol acetate
Target:
Cat. No. Product Name Target Signaling Pathways
T3227 Danshensu

Salvianic acid A,Dan shen suan A,丹参素

Apoptosis; Nrf2; Autophagy Apoptosis; Autophagy; Immunology/Inflammation
Danshensu (Dan shen suan A) 是丹参的有效成分,能够激活 Nrf2信号通路,具有保护心血管作用。
T2944 Danshensu sodium salt

Sodium Danshensu,(±)-DanShenSu sodium salt,丹参素钠,(±)-DanShenSu sodium sal

P450; Autophagy Autophagy; Metabolism
Danshensu sodium salt (Sodium Danshensu) 是从中国草本丹参中提取的一种天然产物,可以抑制去氧肾上腺素和CaCl2 在无Ca2+ 培养基中引起的血管收缩。
T39825 (Rac)-Salvianic acid A

(Rac)-丹参素,(Rac)-Danshensu

(Rac)-Salvianic acid A, also known as (Rac)-Danshensu, is a phenolic acid compound that possesses exceptional radical scavenging and antioxidant properties.
TN2113 Przewaquinone A

丹参素 A

Others Others
Przewaquinone A has antitumor activity.
T3890 Verbenalin

Verbenalol β-D-glucopyranoside,马鞭草苷,Verbenaloside,Verbenalol glucoside,Cornin

Others Others
Verbenalin (Verbenaloside) 是马鞭草苷,具有抗炎、抗真菌、抗病毒等活性。它能减轻脑缺血再灌注损伤。它可用于前列腺炎的研究。
T7914 Acenaphthylene

Others Others
Acenaphthylene 是多环芳烃。其中多环芳烃是自然衍生于煤和焦油沉积物中,并由有机质的不完全燃烧得到。
T3414 Morroniside

莫诺苷,奎宁树

Apoptosis; MMP; Pyroptosis Apoptosis; Immunology/Inflammation; Proteases/Proteasome
Morroniside 通过抑制神经元凋亡和 MMP9/2 的表达从而发挥神经保护作用,可作为 db/db 小鼠肝脏炎症反应和脂质代谢的调节剂。它通过抑制高血糖和氧化应激表现出对糖尿病肾损伤和人脐静脉内皮细胞的保护作用。
T3746 Dimethyl phthalate

邻苯二甲酸二甲酯,Solvanom,Avolin,Fermine,避蚊酯

Others Others
Dimethyl phthalate (Fermine) 是一种邻苯二甲酸酯 (PAEs),是一种已知的内分泌干扰物,也是一种普遍存在的污染物。它常作为增塑剂,赋予硬质聚氯乙烯 (PVC) 树脂以柔韧性。
TN1160 1,2,3,6-Tetragalloylglucose

1,2,3,6-Tetra-O-galloyl-β-D-glucose,1,2,3,6-四-O-没食子酰-Β-D-葡萄糖,TeGG

LDL; UGT Metabolism
1,2,3,6-Tetragalloylglucose (TeGG) 是 UDP-葡萄糖醛酸转移酶 1 家族成员,是多肽A1 的抑制剂(Ki:1.68 μM)。
TN4368 Kaempferol-3,7-di-O-β-glucoside

Kaempferol 3,7-di-O-glucoside

Glucosidase; Amylase Metabolism
Kaempferol-3,7-di-O-β-glucoside (Kaempferol 3,7-diglucoside) 是一种来自 Morettia philaena 的黄酮醇,对 α-淀粉酶 (α-amylase)、α-葡萄糖苷酶 (α-glucosidase) 和乙酰胆碱酯酶 (Acetylcholinesterase) 具有抑制作用。Kaempferol-3,7-di-O-β-glucoside 具有神经保护活性,可减缓分化神经元细胞 SH-SY5Y 免受 Amyloid β 肽诱导的损伤。Kaempferol-3,7-di-O-β-glucoside 可用于研究阿尔茨海默氏症类的神经系统疾病。
T6S1294 Nicotiflorin

Nictoflorin,Kaempferol-3-O-Rutinoside,山奈酚-3-O-芸香糖苷,Nicotifloroside

Others Others
Nicotiflorin (Kaempferol-3-O-Rutinoside) 是一种黄酮苷,从传统中药Flos Carthami 中提取得到。它有抗糖化活性和神经保护作用。
T3863 Chikusetsusaponin IVa

竹节参皂苷IVa,Calenduloside F,竹节人参皂苷 IVA

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
Chikusetsusaponin IVa (Calenduloside F) 是一种三萜皂苷中主要的活性成分,是一种蛋白激酶的激活剂,对血栓及一些代谢性疾病具有抵抗作用。
TQ0188 Miquelianin

槲皮素-3-O-葡萄糖醛酸苷,Quercetin 3-glucuronide,Quercetin 3-O-glucuronide

stilbene oxidase; Endogenous Metabolite Metabolism
Miquelianin (Quercetin 3-glucuronide) 是槲皮素的代谢产物,属于类黄酮化合物。
T6000 Delta-Tocopherol

(+)-DELTA-生育酚,D-DELTA-TOCOPHEROL

Endogenous Metabolite Metabolism
Delta-Tocopherol 是维生素 E 的异构体,具有抗氧化活性。
TN1331 7-O-Methyl morroniside

金银花,7-O-甲基莫诺甙

Others Others
7-O-Methyl morroniside is a natural product from Lonicera morrowii.
TN1330 7-O-Ethylmorroniside

7-乙氧基莫诺苷,7-O-ethyl-morroniside,7-氧乙基莫诺苷,金银花

Others Others
7-O-ethyl-morroniside is a natural product from Lonicera morrowii.
TN4613 (-)-N-methylcoclaurine

N-Methylcoclaurine

Others Others
N-Methylcoclaurine shows binding affinities for the ĸ opioid receptor with the equilibrium dissociation constant (Ki) value of 0.9 ± 0.1 uM. N-methylcoclaurine also shows promising butyrylcholinesterase inhibition activities, with the IC50 value of 1
TN1919 (+)-Medioresinol

梣皮树脂醇,皮树脂醇,Medioresinol

Beta Amyloid; ROS; Antifection Immunology/Inflammation; Microbiology/Virology; Neuroscience
Medioresinol possesses antioxidative, a lesishmanicidal activity and cardiovascular disease risk reduction, it has antiamyloidogenic activity via reduction in the amount of α²-secretase, it is a potentially valuable antiamyloidogenic agent for the prevent
TN2928 Pygenic acid A

3-Epicorosolic acid,脓毒酸A

3-Epicorosolic acid has a potent inhibitory effect on Epstein-Barr virus early antigen (EBV-EA) induction, it has potential anti-inflammatory activities as well as cancer chemopreventive activity.3-Epicorosolic acid shows both potent α-glucosidase and pro

天然产物

Danshensu
Cat.No: T3227
Synonym: Salvianic acid A,Dan shen suan A,丹参素
Target: Apoptosis, Nrf2, Autophagy
Danshensu sodium salt
Cat.No: T2944
Synonym: Sodium Danshensu,(±)-DanShenSu sodium salt,丹参素钠,(±)-DanShenSu sodium sal
Target: P450, Autophagy
(Rac)-Salvianic acid A
Cat.No: T39825
Synonym: (Rac)-丹参素,(Rac)-Danshensu
Target:
Przewaquinone A
Cat.No: TN2113
Synonym: 丹参素 A
Target: Others
Verbenalin
Cat.No: T3890
Synonym: Verbenalol β-D-glucopyranoside,马鞭草苷,Verbenaloside,Verbenalol glucoside,Cornin
Target: Others
Acenaphthylene
Cat.No: T7914
Synonym:
Target: Others
Morroniside
Cat.No: T3414
Synonym: 莫诺苷,奎宁树
Target: Apoptosis, MMP, Pyroptosis
Dimethyl phthalate
Cat.No: T3746
Synonym: 邻苯二甲酸二甲酯,Solvanom,Avolin,Fermine,避蚊酯
Target: Others
1,2,3,6-Tetragalloylglucose
Cat.No: TN1160
Synonym: 1,2,3,6-Tetra-O-galloyl-β-D-glucose,1,2,3,6-四-O-没食子酰-Β-D-葡萄糖,TeGG
Target: LDL, UGT
Kaempferol-3,7-di-O-β-glucoside
Cat.No: TN4368
Synonym: Kaempferol 3,7-di-O-glucoside
Target: Glucosidase, Amylase
Nicotiflorin
Cat.No: T6S1294
Synonym: Nictoflorin,Kaempferol-3-O-Rutinoside,山奈酚-3-O-芸香糖苷,Nicotifloroside
Target: Others
Chikusetsusaponin IVa
Cat.No: T3863
Synonym: 竹节参皂苷IVa,Calenduloside F,竹节人参皂苷 IVA
Target: AMPK
Miquelianin
Cat.No: TQ0188
Synonym: 槲皮素-3-O-葡萄糖醛酸苷,Quercetin 3-glucuronide,Quercetin 3-O-glucuronide
Target: stilbene oxidase, Endogenous Metabolite
Delta-Tocopherol
Cat.No: T6000
Synonym: (+)-DELTA-生育酚,D-DELTA-TOCOPHEROL
Target: Endogenous Metabolite
7-O-Methyl morroniside
Cat.No: TN1331
Synonym: 金银花,7-O-甲基莫诺甙
Target: Others
7-O-Ethylmorroniside
Cat.No: TN1330
Synonym: 7-乙氧基莫诺苷,7-O-ethyl-morroniside,7-氧乙基莫诺苷,金银花
Target: Others
(-)-N-methylcoclaurine
Cat.No: TN4613
Synonym: N-Methylcoclaurine
Target: Others
(+)-Medioresinol
Cat.No: TN1919
Synonym: 梣皮树脂醇,皮树脂醇,Medioresinol
Target: Beta Amyloid, ROS, Antifection
Pygenic acid A
Cat.No: TN2928
Synonym: 3-Epicorosolic acid,脓毒酸A
Target:
TargetMol Loading
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