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3

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T1283 Clinafloxacin

克林沙星,PD 127391,CI-960,AM-1091

Antibacterial; Antibiotic Microbiology/Virology
Clinafloxacin (CI-960) 是一种高效广谱氟喹诺酮类抗生素,抑制革兰氏阳性、革兰氏阴性和厌氧病原体。它对金黄色葡萄球菌的 DNA 促旋酶和拓扑异构酶 IV 有抑制作用,IC50值分别为 0.92 µg/ml 和 1.62 µg/ml。
T20510 Novobiocin

U-6391,U 6391,U6391,Cathomycin,Albamycin

Apoptosis; Virus Protease; HSP; DNA gyrase; Antibacterial; Antibiotic Apoptosis; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Novobiocin 是一种具有口服活性和有效性的的抗生素。Novobiocin 是 DNA 促旋酶抑制剂和热休克蛋白 90 (Hsp90) 拮抗剂,对促旋酶和Hsp90 具有抑制作用。 Novobiocin 具有抗正痘活性,可用于研究高度耐药性肺炎球菌感染。
T19678 Cefaloridine

Cephaloridine,Sch 11527

Cefaloridine is a first-generation semisynthetic derivative of cephalosporin C. It is unique among cephalosporins in that it exists as a zwitterion. Cephaloridine was very effective to cure pneumococcal pneumonia. It has a high clinical and bacteriologica

化合物

Clinafloxacin
Cat.No: T1283
Synonym: 克林沙星,PD 127391,CI-960,AM-1091
Target: Antibacterial, Antibiotic
Novobiocin
Cat.No: T20510
Synonym: U-6391,U 6391,U6391,Cathomycin,Albamycin
Target: Apoptosis, Virus Protease, HSP, DNA gyrase, Antibacterial, Antibiotic
Cefaloridine
Cat.No: T19678
Synonym: Cephaloridine,Sch 11527
Target:
Cat. No. Product Name Target Signaling Pathways
T0974 Novobiocin Sodium

Albamycinsodium,新生霉素钠,Cathomycin,Albamycin

Potassium Channel; DNA gyrase; Topoisomerase; Antibacterial; Antibiotic; ABC; Autophagy Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology
Novobiocin Sodium (Albamycinsodium) 是源自 Streptomyces niveus 的抗生素。 它的化学结构类似于香豆素。Novobiocin 与 DNA 促旋酶结合并阻断三磷酸腺苷活性。
T5S2347 Deoxyshikonin

去氧紫草素,Arnebin 7

Others; HIF/HIF Prolyl-Hydroxylase; Antibacterial Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Others
Deoxyshikonin (Arnebin 7) 是从紫草中分离的天然产物,具有抗肿瘤活性,在体外具有促血管生成作用。它和没食子酸十二烷基酯在体内外均与青霉素有显着的协同抗菌活性。
TN2176 Sanggenol A

Influenza Virus; Antifection Microbiology/Virology
Sanggenol A 抑制甲型流感病毒和肺炎球菌神经氨酸酶,因此可作为双重作用的抗感染试剂。

天然产物

Novobiocin Sodium
Cat.No: T0974
Synonym: Albamycinsodium,新生霉素钠,Cathomycin,Albamycin
Target: Potassium Channel, DNA gyrase, Topoisomerase, Antibacterial, Antibiotic, ABC, Autophagy
Deoxyshikonin
Cat.No: T5S2347
Synonym: 去氧紫草素,Arnebin 7
Target: Others, HIF/HIF Prolyl-Hydroxylase, Antibacterial
Sanggenol A
Cat.No: TN2176
Synonym:
Target: Influenza Virus, Antifection
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