23
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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0916 |
Butamben
Butyl 4-aminobenzoate,4-氨基苯甲酸丁酯 |
Potassium Channel; Calcium Channel; Sodium Channel | Membrane transporter/Ion channel; Metabolism |
Butamben (Butyl 4-aminobenzoate) 是一种长效局部麻醉剂,用于治疗慢性疼痛。 | |||
T13963 |
W-2429
NSC294836 |
Others | Others |
W-2429 is a non-narcotic analgesic agent. | |||
T1169 |
Moguisteine
莫吉司坦,BBR-2173 |
Others | Others |
Moguisteine (BBR-2173) 是一种具有止咳作用的化合物。 | |||
T0484 |
Deracoxib
SC 46,SC 046,地拉考昔,SC 59046 |
Apoptosis; COX | Apoptosis; Immunology/Inflammation; Neuroscience |
Deracoxib (SC 46) 是非甾体、非麻醉性抗炎药。 它也是选择性 cyclooxygenase-2 抑制剂,IC50 值:70 至 150 μM,抑制 3 种骨肉瘤细胞系。 | |||
T7160 |
Lofexidine
|
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Lofexidine 是一种选择性α2 受体激动剂,常用于缓解海洛因和其他阿片类戒断的躯体症状。 | |||
T0201 |
Meptazinol hydrochloride
Meptazinol HCl,盐酸美普他酚 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Meptazinol hydrochloride (Meptazinol HCl) 是一种独特的中枢opioid 类镇痛剂,用作具有镇痛特性的麻醉拮抗剂。 | |||
T0055 |
Glafenine
Glafenin,格拉非宁 |
COX | Immunology/Inflammation; Neuroscience |
Glafenine (Glafenin) 是一种可用于缓解疼痛研究的非甾体抗炎药。 | |||
T23580 |
20681-S
20681 S |
||
20681-S has narcotic antagonistic properties and antinociceptive. | |||
T26362 |
Brifentanil hydrochloride
A3331,A-3331,A 3331 |
||
Brifentanil hydrochloride is a potent narcotic analgesic. | |||
T68608 |
Methylnaltrexone
|
||
Methylnaltrexone is a narcotic antagonists. | |||
T26362L |
Brifentanil
|
||
Brifentanil is a narcotic analgesic. | |||
T68358 |
(R)-Methylnaltrexone
|
||
Methylnaltrexone is a narcotic antagonist. | |||
T69086 | MR 2266 | ||
MR 2266 is a narcotic antagonist. | |||
T27925 |
LY 88329
LY-88329,LY88329 |
||
LY 88329 is a narcotic antagonist in the class of phenylpiperidine. | |||
T27928 |
LY 99335
LY99335,LY-99335 |
||
LY 99335 is a narcotic antagonist in the class of phenylpiperidine. | |||
T69370 |
Cyclazocine
|
||
Cyclazocine is an analgesic with mixed narcotic agonist-antagonist properties. | |||
T23944 |
DA 5018
DA-5018,DA5018 |
||
DA 5018 is a capsaicin derivative and is also a new non-narcotic analgesic. It has an antipruritic effect. | |||
T16810 |
Ruzadolane
卢扎朵仑,UP 26-91 |
Others | Others |
Ruzadolane(以前称为UP 26-91)是一种5-羟色胺受体拮抗剂,被开发为一种非麻醉性中枢镇痛剂,用于治疗焦虑症和疼痛。 | |||
T69121 |
Oxpheneridine
|
||
Oxpheneridine is a mu opioid receptor agonist that possesses the spasmolytic activity and acts as a narcotic analgesic. | |||
T60501 | Tipepidine | ||
Tipepidine 是一种非麻醉性镇咳药,具有抗抑郁样作用。 Tipepidine 可逆地抑制多巴胺 (DA) D2 受体介导的 GIRK 电流 (IDA(GIRK) ),IC50值为 7.0 μM,随后激活 VTA 多巴胺神经元。 | |||
T73233 |
Ciramadol
WY 15705 |
||
Ciramadol (WY 15705) 是一种有效的镇痛剂,具有麻醉激动剂和拮抗剂的特点。Ciramadol (WY 15705) 可用于术后疼痛治疗研究。 | |||
T25420 |
FK 33-824
FK-33-824,Sandoz FK 33-824,FK33-824,SAN 33-824,Damme |
||
FK 33-824 ,with similar actions to those of methionine enkephalin(ENKEPHALIN, METHIONINE),is a stable synthetic analog of that. Its effects can be reversed by narcotic antagonists such as naloxone. | |||
T11302 | Flumexadol | 5-HT Receptor | GPCR/G Protein; Neuroscience |
Flumexadol is a selective and affinity 5-HT2C receptor agonist with a Ki of 25 nM for the (+)-enantiomer of Flumexadol, and is 40-fold selective over the 5-HT2A receptor. Flumexadol is an orally active non-narcotic analgesic. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0739 |
Guaifenesin
Glycerol guaiacolate,Guaiacol glyceryl ether,愈创甘油醚,Guaiphenesin |
Others | Others |
Guaifenesin (Guaiphenesin) 是一种祛痰剂,来自于 Guajacum officinale Linné 木材中。它可以增加痰液体积和降低其粘度,缓解咳嗽不适,促进有效的咳嗽。 |