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1

抑制剂 & 化合物

15

天然产物

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Cat. No. Product Name Target Signaling Pathways
T2806L Lappaconitine HCl

Lappaconitine hydrochloride

Lappaconitine HCl is a centrally acting non-opioid analgesic and class-I antiarrhythmic. It acts by binding to the site-2 receptor and irreversibly blocking hH1 sodium channels.

化合物

Lappaconitine HCl
Cat.No: T2806L
Synonym: Lappaconitine hydrochloride
Target:
Cat. No. Product Name Target Signaling Pathways
T3827 Rhein-8-glucoside calcium

大黄酸-8-O-β-D-葡萄糖苷,Rhein-8-O-β-D-glucopyranoside,Rhein-8-glucoside calcium salt

Phosphatase; Antibacterial Metabolism; Microbiology/Virology
Rhein-8-glucoside calcium (Rhein-8-glucoside calcium salt) salt 是一种从 Saussurea lappa 根的 EtOH 提取物中,分离得到的蒽醌类 hPTP1B 抑制剂,IC50值为11.5 μM,具有抗菌作用。
T32570 Lappaconine

20-ethyl-1,14,16-trimethoxyaconitane-4,6,8-triol,O(sup 1)-Methyllappaconidine

Others Others
Lappaconine (20-ethyl-1,14,16-trimethoxyaconitane-4,6,8-triol) 衍生自去甲二萜生物碱。
T6560 Lappaconitine hydrobromide

氢溴酸高乌甲素,Lappaconite HBr,Allapinine

Others Others
Lappaconitine hydrobromide (Allapinine) 是天然生物碱类化合物,具有抗心律失常作用。
T2806 Lappaconitine

高乌甲素,(+)-Lappaconitine

P2X Receptor; Sodium Channel Membrane transporter/Ion channel; Neuroscience
Lappaconitine ((+)-Lappaconitine) 是从高乌头中分离得到的一种天然产物,可用于缓解疼痛的研究。
TN4410 Lappaol C

P-gp; JNK MAPK; Membrane transporter/Ion channel; Neuroscience
Lappaol C has antioxidant and antiaging properties, it may promote the C. elegans longevity and stress resistance through a JNK-1-DAF-16 cascade. Lappaol C also has potential chemosensitizing activity, it may be candidates for developing novel adjuvant an
TN6463 Lappaol B

Lappaol B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6463,CAS号为 62359-60-8。
TN6462 Isolappaol C

Isolappaol C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6462,CAS号为 929905-15-7。
TN4411 Lappaol F

CDK; P-gp; JNK Cell Cycle/Checkpoint; MAPK; Membrane transporter/Ion channel; Neuroscience
1. Lappaol F has antioxidant and antiaging properties, it may promote the C. elegans longevity and stress resistance through a JNK-1-DAF-16 cascade. <br/> 2. Lappaol F has potential chemosensitizing activity, it may be candidates for developing novel adju
TN1072 Lappaol A

P-gp; JNK MAPK; Membrane transporter/Ion channel; Neuroscience
Lappaol A has antioxidant and antiaging properties, it may promote the C. elegans longevity and stress resistance through a JNK-1-DAF-16 cascade. Lappaol A also has potential chemosensitizing activity, it may be candidates for developing novel adjuvant an
TN6461 Isolappaol A

Isolappaol A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6461,CAS号为 131400-96-9。
T2957 Arctigenin

牛蒡苷元,牛蒡子苷元,(-)-Arctigenin

Apoptosis; MMP; Influenza Virus; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Arctigenin ((-)-Arctigenin) 是一种存在于牛蒡中的木脂素,具有抗氧化、抗肿瘤、抗炎和抗病毒活性。它可研究代谢紊乱和中枢神经系统功能障碍。
T7456 4-Ethyloctanoic acid

Others Others
4-Ethyloctanoic acid 是天然产物,可从云木香中分离得到,广泛用作安全调味料和食品添加剂。
TN1053 Aloe-emodin-8-O-β-D-glucopyranoside

Aloe-emodin-8-O-beta-D-glucopyranoside,芦荟大黄素-8-O-β-D-葡萄糖苷

Phosphatase Metabolism
Aloe-emodin-8-O-β-D-glucopyranoside (Aloe-emodin-8-O-beta-D-glucopyranoside) 是一种分离自Saussrurea lappa 中的化合物,是一种温和的人类蛋白酪氨酸磷酸酶 1B 抑制剂,其IC50=26.6 μM。
TN2383 Arctinol B

Others Others
Arctinol B is a natural product from Arctium lappa L
T80778 weak Hepatoprotective agent-1

Weak Hepatoprotective agent-1 (Compound 11),一种从Arctium lappa L. 分离得到的天然产物,在10 μM浓度下具有弱肝保护活性。

天然产物

Rhein-8-glucoside calcium
Cat.No: T3827
Synonym: 大黄酸-8-O-β-D-葡萄糖苷,Rhein-8-O-β-D-glucopyranoside,Rhein-8-glucoside calcium salt
Target: Phosphatase, Antibacterial
Lappaconine
Cat.No: T32570
Synonym: 20-ethyl-1,14,16-trimethoxyaconitane-4,6,8-triol,O(sup 1)-Methyllappaconidine
Target: Others
Lappaconitine hydrobromide
Cat.No: T6560
Synonym: 氢溴酸高乌甲素,Lappaconite HBr,Allapinine
Target: Others
Lappaconitine
Cat.No: T2806
Synonym: 高乌甲素,(+)-Lappaconitine
Target: P2X Receptor, Sodium Channel
Lappaol C
Cat.No: TN4410
Synonym:
Target: P-gp, JNK
Lappaol B
Cat.No: TN6463
Synonym:
Target:
Isolappaol C
Cat.No: TN6462
Synonym:
Target:
Lappaol F
Cat.No: TN4411
Synonym:
Target: CDK, P-gp, JNK
Lappaol A
Cat.No: TN1072
Synonym:
Target: P-gp, JNK
Isolappaol A
Cat.No: TN6461
Synonym:
Target:
Arctigenin
Cat.No: T2957
Synonym: 牛蒡苷元,牛蒡子苷元,(-)-Arctigenin
Target: Apoptosis, MMP, Influenza Virus, Autophagy
4-Ethyloctanoic acid
Cat.No: T7456
Synonym:
Target: Others
Aloe-emodin-8-O-β-D-glucopyranoside
Cat.No: TN1053
Synonym: Aloe-emodin-8-O-beta-D-glucopyranoside,芦荟大黄素-8-O-β-D-葡萄糖苷
Target: Phosphatase
Arctinol B
Cat.No: TN2383
Synonym:
Target: Others
weak Hepatoprotective agent-1
Cat.No: T80778
Synonym:
Target:
TargetMol Loading
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