15
5
Cat. No. | Product Name | Target | Signaling Pathways |
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T9915 |
Eculizumab
|
Complement System | Immunology/Inflammation |
Eculizumab 是针对补体 C5 的长效人源化单克隆抗体。它对 C5 裂解为 C5a 和 C5b 具有抑制作用,并抑制了末端补体系统的部署,其中包括膜攻击复合物的形成。它可用于溶血的研究。 | |||
T6581 |
Methyclothiazide
Duretic,Enduron,甲氯噻嗪,Aquatensen |
Others; Carbonic Anhydrase | Metabolism; Others |
Methyclothiazide (Aquatensen) 是一种具有口服活性的利尿剂,也是一种降压剂。它能够拮抗体外的电压依赖性钙通道的 (VDCC) 活性,也可以抑制内源性血管收缩刺激导致的血管反应。 | |||
T26781 |
BF-1
BF1 |
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BF-1 is a 5-Hydroxytryptamine receptor 2B antagonist. BF-1 was tested as potential migraine prophylactic drug by blocking BW723C86 (5-((thiophen-2-yl)methoxy)-α-methyltryptamine) or meta-chlorophenylpiperazine (mCPP) induced neurogenic dural plasma protei | |||
T35362 |
NSC622608
|
Others | Others |
NSC622608 是 V 域 Ig 抑制 T 细胞活化 (VISTA) 的小分子配体,VISTA 是影响 T 细胞攻击肿瘤能力的免疫检查点。 | |||
T76831 |
Tesidolumab
LFG316 |
Complement System | Immunology/Inflammation |
Tesidolumab (LFG316) 是一种全人IgG1/λ抗c5单克隆抗体。Tesidolumab (LFG316)对crovalimab和C5有抑制作用, 阻断C5的切割,防止膜攻击复合体的后续形成,可用于研究血管外溶血。 | |||
T21757 |
BRL 52537 hydrochloride
|
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
BRL 52537 hydrochloride 是一种选择性和特异性 KOR 激动剂,与缺血性神经元损伤的神经保护有关。它用于研究中风和心脏病发作的潜在治疗方法以及更一般的大脑研究。 | |||
T1551 |
Tegaserod maleate
HTF-919,马来酸替加色罗,SDZ-HTF-919 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Tegaserod maleate (SDZ-HTF-919) 是选择性5-HT4受体的部分激动剂和5-HT2B 受体的拮抗剂,用于治疗肠易激综合征和便秘。 | |||
T39463 |
Asundexian
BAY 2433334,Asundexian,BAY2433334,BAY-2433334 |
Factor Xa | Metabolism |
Asundexian (BAY-2433334) 是一种高效且具有口服活性凝血因子 FXIa 抑制剂,可直接且可逆地与FXIa 的活性位点结合,从而抑制其活性。Asundexian 对缓冲液中的人 FXIa 的 IC50 为 1 nM。Asundexian 具有抗肿瘤活性,可用于研究急性缺血性卒中、短暂性脑缺血发作和缺血性卒中。 | |||
T23671 |
AH 7725
AH-7725,AH7725 |
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AH 7725 is an inhibitor of the asthma attack. | |||
T37337 |
N-3-oxo-hexadecanoyl-L-Homoserine lactone
|
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N-3-oxo-hexadecanoyl-L-Homoserine lactone is an unusual, substituted, long-chain N-acyl-homoserine lactone (AHL) produced by some bacteria, including strains of Agrobacterium vitis and Pseudomonas. Like other AHLs, this C16-containing form is thought to be involved in quorum sensing. Substituted, long-chain AHLs, including N-3-oxo-tetradecanoyl-L-homoserine lactone , prime for systemic acquired resistance to pathogen attack in plants. | |||
T24901 |
Troponin I (104-115)
Ac-Gly-lys-phe-lys-arg-pro-pro-leu-arg-arg-val-arg-NH2,Tni peptide (104-115) |
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Troponin I is a cardiac and skeletal muscle protein useful in the laboratory diagnosis of a heart attack. Troponin I is a part of the troponin protein complex, where it binds to actin in thin myofilaments to hold the actin-tropomyosin complex in place. | |||
T73060 |
Pralidoxime
|
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Pralidoxime 是一种有效的乙酰胆碱酯酶 (AChE) 的再激活剂。Pralidoxime 通过肟部分对结合神经毒剂磷中心的亲核攻击,重新激活受神经毒剂抑制的 AChE。Pralidoxime 是一种有机磷中毒的解毒剂。 | |||
T22202 |
iMAC2
|
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iMAC2 是一种有效的MAC 抑制剂,IC50为 28 nM,LD50为15000 nM。iMAC2 显示出抗凋亡作用,并且iMAC2 阻断细胞色素 c 的释放。 | |||
T37394 |
13(S)-HpOTrE
|
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13(S)-HpOTrE is a monohydroperoxy polyunsaturated fatty acid produced in soybeans by the action of soybean LO-2 on esterified α-linolenic acid.[1] Incubation of soybean seedling biomembranes with soybean LO-2 catalyzes the formation of both 9- and 13-HpOTrE in a molar ratio of 10:1.1 In plants, 13(S)-HpOTrE can be metabolized by the hydroperoxide lyase pathway producing aldehyde and oxoacid fragments, or by the hydroperoxide dehydratase pathway producing jasmonic acid.[2],[3],[4] Treatment of to... | |||
T83764 |
Sulfane Sulfur Probe 4
SSP4 |
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Sulfane sulfur probe 4 (SSP4) 是用于检测含硫化氢衍生的多硫化物、过硫化物和硫化物的荧光探针。在含硫磺物种存在下,SSP4 经核苷酸攻击反应生成荧光素,其激发/发射峰值分别为494/515 nm,以及两分子的1,2-苯并二硫杂环-3-酮。SSP4 已应用于确定H2S3在原代小鼠神经元中的定位,并检测L. japonicus 幼苗根部的多硫化物。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T19458 |
N-Hydroxypipecolic acid
1-Hydroxy-2-piperidinecarboxylic acid,NHP |
Others | Others |
N-Hydroxypipecolic acid (NHP) 是植物代谢产物和系统性获得性抗性调节剂,可与免疫信号水杨酸协调建立系统性获得性抗性,诱导系统获得性耐药对细菌和卵菌感染。它在植物叶片中系统地积累,以应对病原菌的侵袭。 | |||
T2793 |
Tetrahydropalmatine
DL-Tetrahydropalmatine,四氢帕马丁,延胡索乙素,Rotundine |
Apoptosis; Others; Dopamine Receptor | Apoptosis; GPCR/G Protein; Neuroscience; Others |
Tetrahydropalmatine (DL-Tetrahydropalmatine) 通过抑制大鼠杏仁核的多巴胺释放来抑制癫痫发作,用于缓解疼痛的研究。 | |||
T3093 |
Spermine tetrahydrochloride
精胺盐酸盐,Spermine Tetrahydrochloride,Neuridine tetrahydrochloride,Musculamine tetrahydrochloride,Gerontine tetrahydrochloride |
Others; Endogenous Metabolite | Metabolism; Others |
Spermine tetrahydrochloride (Musculamine tetrahydrochloride) 是内源性代谢产物的一种。 | |||
TN7105 |
Phenazine-1-carboxylic acid
|
Antifungal | Microbiology/Virology |
Phenazine-1-carboxy acid 对所有植物病原真菌均显示出很强的抗真菌活性,抑制真菌生长约 90-100%。 | |||
T4715 |
2'-Deoxyguanosine monohydrate
2'-脱氧鸟苷一水合物,Guanine-2'-deoxyriboside |
Others; Endogenous Metabolite | Metabolism; Others |
2'-Deoxyguanosine monohydrate (Guanine-2'-deoxyriboside) 是内源性代谢产物的一种。 |