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9

抑制剂 & 化合物

9

天然产物

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Cat. No. Product Name Target Signaling Pathways
T10328 Anti-parasitic agent 3

Others Others
Anti-parasitic agent 3 是一种抗寄生虫剂,对耐药寄生虫具有活性。
T11013L1 Dextrorotation nimorazole phosphate ester TFA

Others Others
Dextrorotation nimorazole phosphate ester TFA 是一种抗厌氧菌和抗原虫感染的试剂。
T0356 Nitromide

硝米特,3, 5-Dinitrobenzamide,3,5-Dinitrobenzamide

Parasite Microbiology/Virology
Nitromide (3,5-Dinitrobenzamide) 是一种抗寄生虫药。
T11013L2 Levorotation nimorazole phosphate ester TFA

Others Others
Levorotation nimorazole phosphate ester TFA 是一种抗厌氧菌和抗原虫感染的试剂。
T12022 Metronidazole Benzoate

Benzoyl metronidazole

Antibacterial Microbiology/Virology
Metronidazole Benzoate (Benzoyl metronidazole) 是甲硝唑和苯甲酸衍生物,具有抗菌,抗寄生虫,抗滴虫等作用,常用于治疗由厌氧菌引起的感染。
T39425 Umifoxolaner

Umifoxolaner is an anti-parasitic agent (veterinary).
T61538 Antiparasitic agent-10

Antiparasitic agent-10 (Compound 94) is a potent anti-parasitic agent specifically designed to target and combat parasitic infections. It demonstrates notable anti-schistosomal activity, particularly against adults of Schistosoma mansoni. As a result, this compound holds significant potential for utilization in Schistosomiasis research as a viable treatment option [1].
T11013 Dextrorotation nimorazole phosphate ester

Others Others
Dextrorotation nimorazole phosphate ester is an anti-anaerobic and anti-parasitic agent. D-morpholine ornidazole organic phosphate is a newly developed, highly efficient, well-tolerated fourth-generation nitroimidazole derivative. Objective: Antibacterial
T69469 Panepoxydone

Panepoxydone 是一种 NF-κB 活化抑制剂。Panepoxydone 通过抑制 IκB 的磷酸化来干扰 NF-κB 介导的信号转导。Panepoxydone 具有抗肿瘤、抗炎、抗疟疾和抗寄生虫活性。

化合物

Anti-parasitic agent 3
Cat.No: T10328
Synonym:
Target: Others
Dextrorotation nimorazole phosphate ester TFA
Cat.No: T11013L1
Synonym:
Target: Others
Nitromide
Cat.No: T0356
Synonym: 硝米特,3, 5-Dinitrobenzamide,3,5-Dinitrobenzamide
Target: Parasite
Levorotation nimorazole phosphate ester TFA
Cat.No: T11013L2
Synonym:
Target: Others
Metronidazole Benzoate
Cat.No: T12022
Synonym: Benzoyl metronidazole
Target: Antibacterial
Umifoxolaner
Cat.No: T39425
Synonym:
Target:
Antiparasitic agent-10
Cat.No: T61538
Synonym:
Target:
Dextrorotation nimorazole phosphate ester
Cat.No: T11013
Synonym:
Target: Others
Panepoxydone
Cat.No: T69469
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5807 Stylopine hydrochloride

NOS; COX Immunology/Inflammation; Neuroscience
Stylopine hydrochloride 是一种生物碱类化合物,从紫堇属之植物块茎中分离得到,具有抗炎症和抗寄生虫作用。
T2S0961 Chalcone

benzylideneacetophenone,phenyl styryl ketone,Cinnamophenone,benzalacetophenone,β-phenylacrylophenone,查耳酮

EGFR; Antibacterial Angiogenesis; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Chalcone (Cinnamophenone) 是从甘草中分离得到的一种芳香酮,可合成查耳酮衍生物。它具有多种生物和药理的活性,如抗炎、抗菌、抗癌、抗氧化、抗寄生虫等活性。
T1082 Benzyl isothiocyanate

Benzoylthiocarbimide,苄基异硫氰酸酯,异硫氰酸苯甲酯,Isothiocyanic Acid Benzoyl Ester

Apoptosis; Antibacterial; Antibiotic Apoptosis; Microbiology/Virology
Benzyl isothiocyanate (Benzoylthiocarbimide) 是一种具有杀菌活性的天然异硫氰酸酯,最初存在于十字花科蔬菜中。 它显示出免疫调节、抗寄生虫、抗生素、抗氧化、抗动脉粥样硬化、抗血管生成、抗转移、抗癌化疗和化学预防活性。
T68953 Arecoline

Reactive Oxygen Species; AChR Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Arecoline 是一种来自棕榈科植物槟榔的天然生物碱,是有效的烟碱和毒蕈碱乙酰胆碱受体的部分激动剂。Arecoline 具有抗焦虑和抗寄生虫活性,可诱导氧化应激,可用于研究阿尔茨海默病和老年性痴呆。
T3897 Isoschaftoside

Anti-infection; Antifungal Microbiology/Virology
Isoschaftosid 是从 Desmodium uncinatum 根部分泌物中提取的 c- 糖基黄酮类天然产物,有抗肿瘤、抗氧化和抗菌活性,它还对 M. incognita 具有很强的杀线虫活性。
T0461 Berberine chloride

Berberine hydrochloride,盐酸小檗碱,Benzodioxide,Natural Yellow 18,盐酸黄连素

Reactive Oxygen Species; Topoisomerase; Antibacterial; Antibiotic; Autophagy Autophagy; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Berberine chloride (Natural Yellow 18) 是一种来自小檗科 Hydrastis canadensis L. 的生物碱,也存在于许多其他植物中,常用作抗生素。它对肠胃外的毒性相对较大,但已用于口服用于各种真菌和寄生虫感染以及止泻。
T3794 Pentagalloylglucose

Penta-O-galloyl-β-D-glucose,1,2,3,4,6-O-Pentagalloylglucose,1,2,3,4,6-Penta-O-galloyl-beta-D-glucopyranose,1,2,3,4,6-五没食子酰葡萄糖

Influenza Virus Microbiology/Virology
1,2,3,4,6-O-Pentagalloylglucose (Penta-O-galloyl-β-D-glucose) 存在于多种植物中,具有重要的药理作用。Pentagalloylglucose 表现出显著的抗狂犬病病毒 (RABV) 活性。
T14114 Acivicin

阿西维辛,AT-125,U-42126

Others Others
Acivicin (AT-125) is a γ-glutamyl transpeptidase (GGT) inhibitor derived from the Streptomyces sviceus natural product. It possesses anti-cancer and anti-parasitic properties and can effectively cross the blood-brain barrier[1][2].
T77207 Acivicin hydrochloride

Acivicin hydrochloride (AT-125 hydrochloride),一种猪链霉菌的天然产物,兼具透过血脑屏障的能力,是γ-谷氨酰转肽酶 (GGT) 的抑制剂,具有抗癌和抗寄生虫的特性。

天然产物

Stylopine hydrochloride
Cat.No: T5807
Synonym:
Target: NOS, COX
Chalcone
Cat.No: T2S0961
Synonym: benzylideneacetophenone,phenyl styryl ketone,Cinnamophenone,benzalacetophenone,β-phenylacrylophenone,查耳酮
Target: EGFR, Antibacterial
Benzyl isothiocyanate
Cat.No: T1082
Synonym: Benzoylthiocarbimide,苄基异硫氰酸酯,异硫氰酸苯甲酯,Isothiocyanic Acid Benzoyl Ester
Target: Apoptosis, Antibacterial, Antibiotic
Arecoline
Cat.No: T68953
Synonym:
Target: Reactive Oxygen Species, AChR
Isoschaftoside
Cat.No: T3897
Synonym:
Target: Anti-infection, Antifungal
Berberine chloride
Cat.No: T0461
Synonym: Berberine hydrochloride,盐酸小檗碱,Benzodioxide,Natural Yellow 18,盐酸黄连素
Target: Reactive Oxygen Species, Topoisomerase, Antibacterial, Antibiotic, Autophagy
Pentagalloylglucose
Cat.No: T3794
Synonym: Penta-O-galloyl-β-D-glucose,1,2,3,4,6-O-Pentagalloylglucose,1,2,3,4,6-Penta-O-galloyl-beta-D-glucopyranose,1,2,3,4,6-五没食子酰葡萄糖
Target: Influenza Virus
Acivicin
Cat.No: T14114
Synonym: 阿西维辛,AT-125,U-42126
Target: Others
Acivicin hydrochloride
Cat.No: T77207
Synonym:
Target:
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