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Cat. No. | Product Name | Target | Signaling Pathways |
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T37212 |
5-hydroxy-Nω-methyl Tryptamine (oxalate)
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5-hydroxy-Nω-methyl Tryptamine is a metabolite of serotonin in humans that has also been found in plants. It is an agonist of the 5-HT receptor subtype 5-HT7 (IC50 = 23 pM in a radioligand binding assay). 5-hydroxy-Nω-methyl Tryptamine increases intracellular cyclic AMP production in HEK293 cells expressing 5-HT7 (EC50 = 22 nM). It inhibits serotonin uptake in HEK293 cells expressing human serotonin transporters (IC50 = 490 nM). Elevated levels of urinary 5-hydroxy-Nω-methyl tryptamine have been... | |||
T24604 |
PDAT
Propyl Dimethyl Amino Tryptamine |
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PDAT is a noncompetitive Indolethylamine N-methyltransferase inhibitor. | |||
T124997 | Tryptamine hydrochloride | ||
Tryptamine hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124997,CAS号为 343-94-2。 | |||
TNU0617 |
N10-pivaloyl tryptamine
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Heterocyclic compound-indole, intermediate and building block | |||
T50111 |
6-Fluorotryptamine hydrochloride
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Others | Others |
6-Fluorotryptamine hydrochloride 是一种用作分子结构单元的化合物,是天然色胺生物碱血清素的衍生物。它是5-HT2A 和5-HT2C 血清素受体的激动剂,使其成为开发治疗各种精神和神经疾病的新药的潜在候选者。 | |||
T77673 |
7-FluorotryptaMine HCl
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GPR; Arrestin | Endocrinology/Hormones; GPCR/G Protein |
7-FluorotryptaMine HCl 是一种有效的芳香单胺 GPRC5A 激动剂,可诱导 GPRC5A 介导的 β-arrestin 募集。7-FluorotryptaMine HCl 可用于研究与免疫和癌症相关的信号通路。 | |||
T22520 |
5-Carboxamidotryptamine maleate
5-CT maleate |
5-HT Receptor | GPCR/G Protein; Neuroscience |
5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) 是一种 受体激动剂,具有降压和升血糖的作用。 | |||
T8600 |
N-ACETYLTRYPTAMINE
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Melatonin Receptor | GPCR/G Protein |
N-Acetyltryptamine 是视网膜褪黑素受体的部分激动剂,可用于 5-羟色胺 N-乙酰转移酶活性的检测。 | |||
T40631 |
4-Hydroxytryptamine creatinine sulfate
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4-Hydroxytryptamine creatinine sulfate, a derivative of tryptamine, acts as an agonist for neurotransmitters. | |||
T60526 | N-Salicyloyltryptamine | ||
N-Salicyloyltryptamine(STP) 是一种色胺类似物,具有抗惊厥、抗炎、镇痛和血管舒张的作用。N-Salicyloyltryptamine 作为电压依赖性离子通道(包括Na+、Ca2+、K+离子通道)抑制剂,可抑制 K+电流,IC50值为 34.6 μM ( /to)。 | |||
T22561 |
α-Methyl-5-hydroxytryptamine maleate
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Others | Others |
5-HT2B receptor agonist | |||
T22524 |
5-Nonyloxytryptamine oxalate
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Others | Others |
5-HT1B agonist | |||
T67851 |
rac Desmethyl Citalopram Hydrochloride
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5-HT Receptor | GPCR/G Protein; Neuroscience |
rac Desmethyl Citalopram Hydrochloride 是一种5-羟色胺摄取抑制剂,IC50值为0.013μM。 | |||
T0235 |
Modaline sulfate
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MAO; Monoamine Oxidase | Metabolism; Neuroscience |
Modaline sulfate 是一种 MAO 抑制剂,用于研究抑郁症。 | |||
T1442 |
Pizotifen
Pizotyline,BC-105,苯噻啶 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Pizotifen (Pizotyline) 是5-HT2受体的有效拮抗剂,并对5-HT1C 有高亲和力。它是一种强血清素和色胺拮抗剂,具有较弱的抗胆碱能、抗组胺和抗激肽作用,还具有镇静和刺激食欲的特性。 | |||
T34431 |
RU 27849
RU-27849,RU27849 |
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RU 27849 is used to study the binding of tryptamine recognition sites. | |||
T70408 |
Rizatriptan sulfate
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Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine. | |||
T70656 | CP 132484 | ||
CP 132484 is a tryptamine derivative which acts as a potent and selective agonist for the 5-HT₂ family of serotonin receptors. It has reasonable selectivity for 5-HT2A and 5-HT2C subtypes over 5-HT2B, but is only slightly selective for 5-HT2A over 5-HT2C. | |||
T22044 |
BGC 20-761
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BGC20-761 是一种选择性的5-HT6和多巴胺受体 (dopamine receptor) 拮抗剂,对人 5-HT6,5-HT2A,D2 受体的Ki 值分别为 20,69,和 140 nM。BGC20-761 可增强长期记忆。BGC20-761 具有作为抗精神病药物的潜在效用。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T0647 |
Tryptamine
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Dehydrogenase; 5-HT Receptor; Endogenous Metabolite; TRP/TRPV Channel | GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Tryptamine 是一种在动物、植物和真菌中发现的单胺生物碱。它含有吲哚环结构,结构类似于色氨酸。在哺乳动物的大脑中发现了微量这种物质,并被认为是一种神经递质或神经调节剂。 | |||
T4860 |
5-Hydroxytryptamine creatinine sulfate monohydrate
Serotonin creatinine sulfate monohydrate,5-Hydroxytryptamine creatinine sulfate complex,5-五羟色胺肌酸酐 |
Others; Endogenous Metabolite | Metabolism; Others |
5-Hydroxytryptamine creatinine sulfate monohydrate (Serotonin creatinine sulfate monohydrate) 是内源性代谢产物的一种。 | |||
T1354 |
N-Acetyl-5-hydroxytryptamine
Normelatonin,N-乙酰-5-羟色胺,O-Demethylmelatonin,N-Acetylserotonin |
Trk receptor; Endogenous Metabolite | Metabolism; Tyrosine Kinase/Adaptors |
N-Acetyl-5-hydroxytryptamine (O-Demethylmelatonin) 是褪黑激素的直接前体,能够有效激活TrkB 受体。 | |||
TN6571 |
Nb-Feruloyltryptamine
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Nb-Feruloyltryptamine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6571,CAS号为 53905-13-8。 |