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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T28960 Thaspine HCl

Thaspine,Thaspine HCl, NSC 135784,NSC-135784,NSC135784

Thaspine is a potent topoisomerase IB inhibitor. Taspine downregulates VEGF expression and inhibits proliferation of vascular endothelial cells through PI3 kinase and MAP kinase signaling pathways.
T20656 Verapamil

NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil

P450; Calcium Channel; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Verapamil (CP-16533-1) 是一种钙通道阻滞剂,是一种口服有效的 P-gp 抑制剂。Verapamil 抑制 CYP3A4,可用于治疗高血压、心律失常和心绞痛的研究。

化合物

Thaspine HCl
Cat.No: T28960
Synonym: Thaspine,Thaspine HCl, NSC 135784,NSC-135784,NSC135784
Target:
Verapamil
Cat.No: T20656
Synonym: NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil
Target: P450, Calcium Channel, P-gp
Cat. No. Product Name Target Signaling Pathways
TN5100 Taspine

ERK; EGFR; BCL; VEGFR; MAPK; Akt Angiogenesis; Apoptosis; Cytoskeletal Signaling; JAK/STAT signaling; MAPK; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Taspine shows antitumor activity by modulating the EGFR signaling pathway of Erk1/2 and Akt in vitro and in vivo, it can inhibit growth and induce apoptosis of HUVEC in a dose-dependent manner, it has shown meaningful angiogenesis activity. Taspine exhibi

天然产物

Taspine
Cat.No: TN5100
Synonym:
Target: ERK, EGFR, BCL, VEGFR, MAPK, Akt
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