49
13
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6693 |
TAME
N-[(4-甲基苯基)磺酰基]-L-精氨酸甲酯,Tosylarginine methyl ester,N-4-Tosyl-L-arginine methyl ester |
APC | Cell Cycle/Checkpoint |
TAME (N-4-Tosyl-L-arginine methyl ester) 是后期促进复合体(APC/C 或 APC)的抑制剂,可与 APC/C 结合并阻止其通过 Cdc20 和 Cdh1 活化,产生有丝分裂阻滞。 | |||
T1731 |
TAME hydrochloride
NA-P-甲苯磺酰-L-精氨酸甲酯盐酸盐,Tos-Arg-OMe HCl,TOS-ARG-OME hydrochloride |
Amino Acids and Derivatives; APC | Cell Cycle/Checkpoint; Metabolism |
TAME hydrochloride (Tos-Arg-OMe HCl) 是后期促进复合体(APC/C 或 APC)的抑制剂,可与 APC/C 结合并阻止其通过 Cdc20 和 Cdh1 活化,产生有丝分裂阻滞。它是一种 od 氨基酸衍生物。 | |||
T1163 |
Betamethasone valerate
Betnovate,倍他米松戊酸酯,Betaderm,Betamethasone 17-valerate,Luxiq |
Glucocorticoid Receptor | Endocrinology/Hormones |
Betamethasone valerate (Luxiq) 的 17 戊酸酯,是一种具有抗炎活性的局部皮质类固醇。它能够抑制放射标记的糖皮质激素地塞米松与人表皮(IC50:5 nM)及小鼠皮肤(IC50:6 nM)的结合。它可用于研究复发性口疮。 | |||
T3597 |
Cutamesine dihydrochloride
AGY94806 dihydrochloride,库他美新二盐酸盐,SA4503 (dihydrochloride),SA4503 dihydrochloride |
Sigma receptor | GPCR/G Protein |
Cutamesine dihydrochloride (SA4503 dihydrochloride) 是一种选择性 σ1 受体激动剂,IC50值为 17.4 nM。 | |||
T0697 |
Aspartame
阿斯巴甜,SC-18862 |
Others; Taste receptor | Metabolism; Others |
Aspartame (SC-18862) 是一种二肽的甲酯,由苯丙氨酸 (50%),天门冬氨酸 (40%) 和甲醇 (10%) 组成。它可用作合成的非营养性甜味剂。 | |||
T50096 |
1,3,3,5,5-pentamethylcyclohexan-1-amine hydrochloride
|
Others | Others |
1,3,3,5,5-pentamethylcyclohexan-1-amine hydrochloride,又称PAC,是一种环胺,通常用作不对称合成中的手性助剂,包括Diels-Alder 反应、羟醛反应和Michael 加成。 | |||
T1559 |
Betamethasone dipropionate
Diprolene AF,SCH 11460,二丙酸倍他米松,Betamethasone 17,21-dipropionate,Diprolene,倍他米松二丙酸酯,Diprosone |
Glucocorticoid Receptor | Endocrinology/Hormones |
Betamethasone dipropionate (SCH 11460) 是糖皮质激素类固醇,具有免疫抑制、抗炎作用。 | |||
T7120 |
Cefetamet pivoxil hydrochloride
盐酸头孢他美酯,Ro 15-8075 |
Antibacterial; Antibiotic | Microbiology/Virology |
Cefetamet pivoxil hydrochloride (Ro 15-8075) 是一种可口服的头孢类抗生素。 | |||
T20763 |
Betamethasone disodium phosphate
Vista-Methasone,NSC90616,Betamethasone 21-phosphate disodium salt,NSC-90616 |
Others | Others |
Betamethasone disodium phosphate (Betamethasone 21-phosphate disodium salt) 是一种具有抗炎活性的皮质类固醇,通过减少促炎细胞因子的分泌促进 M1 至 M2 巨噬细胞极化,可用于研究瘢痕疙瘩和类风湿性关节炎。 | |||
T5837 |
Tamerit
|
Others | Others |
Tamerit 是一种化学发光物质,pKa 值为 6.74 和 15.1,荧光波长为 425 nm。它是法医检测血迹的诊断工具,可用于刑事侦查、生物工程、化学示踪等领域。 | |||
T33639 |
Neotame
NC 00723,HSDB 7965,NC-00723,NC00723,纽甜 |
Others | Others |
Neotame (HSDB 7965) 是阿斯巴甜的衍生物,是低热量、高效的人造甜味剂,非营养性甜味剂和增味剂,其甜度是糖的 7000-13,000 倍,可用于多种食品。 | |||
T30787 |
Cefetamet sodium
Ro 15-8074/001,Ro15-8074/001,Ro-15-8074/001 |
||
Cefetamet sodium is a third-generation cephalosporin. | |||
T30062 | Aniline, 4,4'-pentamethylenedioxybis(3-chloro-, dihydrochloride | ||
Aniline, 4,4'-pentamethylenedioxybis(3-chloro-, dihydrochloride is a bioactive chemical. | |||
T13579 |
Betamethasone acibutate
|
Others | Others |
Betamethasone acibutate, a glucocorticoid, is derived from Betamethasone. | |||
T25932 |
Pentamethonium bromide
NSC148343,NSC 148343,NSC-148343 |
||
Pentamethonium bromide is a vasodilator agent. | |||
T125893 |
1,2,3,4,7-Pentamethoxy-9H-xanthen-9-one
|
||
1,2,3,4,7-Pentamethoxy-9H-xanthen-9-one 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125893。 | |||
T25004 |
Advantame anhydrous
Advantame |
||
Advantame anhydrous is a non-caloric sweetener, synthesized from isovanillin and aspartame. The U.S. Food and Drug Administration has approved Advantame for general use in foods and beverages except for meat and poultry as a food additive. | |||
T34781 |
Tameridone
R 51 163,R 51163 |
||
Tameridone is a sedative used for cattle. | |||
T83161 | Advantame | ||
Advantame为阿斯巴甜衍生物,属于无热量合成甜味剂,广泛应用于食品添加剂领域。 | |||
T66637 |
(S)-3-((((9H-Fluoren-9-yl)methoxy)carbonyl)amino)-6-(3-((2,2,4,6,7-pentamethyl-2,3-dihydrobenzofuran-5-yl)sulfonyl)guanidino)hexanoic acid
|
||
(S)-3-((((9H-Fluoren-9-yl)methoxy)carbonyl)amino)-6-(3-((2,2,4,6,7-pentamethyl-2,3-dihydrobenzofuran-5-yl)sulfonyl)guanidino)hexanoic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66637,CAS号为 401915-53-5。 | |||
T38100 |
Betamethasone 21-phosphate (sodium salt hydrate)
|
||
Betamethasone 21-phosphate is a synthetic glucocorticoid.1It prevents increases in macrophage and eosinophil numbers in bronchoalveolar lavage fluid (BALF) and decreases in blood leukocyte numbers in a guinea pig model of parainfluenza-3 viral infection when administered at a dose of 8 mg/kg but does not prevent airway hyperresponsiveness after infection.2Betamethasone 21-phosphate inhibits cell infiltration into the aqueous humor in a rat model of endotoxin-induced uveitis when administered top... | |||
T28455 |
ProTAME
pro-Tosyl-L-Arginine Methyl Ester |
||
ProTAME is an inhibitor of APC/CFzr and APC/CCdc20. Combinations of proTAME with topoisomerase inhibitors, doxorubicin and etoposide, significantly increase cell death in primary cells and Multiple Myeloma (MM) cell lines, particularly if TOPIIα levels ar | |||
T16152 |
Betamethasone 17-benzoate
|
Kinesin | Cytoskeletal Signaling |
Betamethasone 17-benzoate is a representative steroid. It also can be used in the treatment of recurrent aphothous ulcers (RAU). | |||
T33830 |
o-Toluidine, 4,4'-pentamethylenedioxydi-, dihydrochloride
|
||
o-Toluidine, 4,4'-pentamethylenedioxydi-, dihydrochloride is a bioactive chemical. | |||
T29866 |
Alitame
HSDB 7825,CP-54,802,CP 54802 |
||
Alitame is a non-nutritive sweetener that is 2000 times sweeter than sucrose. It is formed from aspartic acid, alanine & an amide. | |||
T65124 |
Dipentamethylenethiuram Tetrasulfide
|
||
Dipentamethylenethiuram Tetrasulfide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65124,CAS号为 120-54-7。 | |||
T19001 |
Heptamethine cyanine dye-1
ADS 815EI |
Others | Others |
Heptamethine cyanine dye-1, a near-infrared cyanine dye, is used for fluorescence imaging in biological systems. | |||
T79663 |
E07 aptamer
|
SARS-CoV | Microbiology/Virology |
SARS-CoV-2 nsp14-IN-4(Compound 12q)是一种选择性抑制剂,针对SARS-CoV-2 nsp14 methyltransferase,具有IC50为19 ± 2.5 nM。该化合物不带中性离子性质,能够穿透细胞膜。它可用于COVID-19及其病原体SARS-CoV-2的相关研究。 | |||
T125825 |
Pentamethylene bisacetamide
|
||
Pentamethylene bisacetamide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125825,CAS号为 146695-99-0。 | |||
T33810 |
o-Phenylenediamine, 4,4'-pentamethylenedioxybis-
|
||
o-Phenylenediamine, 4,4'-pentamethylenedioxybis- is a bioactive chemical. | |||
T30056 |
Aniline, 4,4'-(octamethylenedioxy)bis(N-methyl-, dihydrochloride
|
||
Aniline, 4,4'-(octamethylenedioxy)bis(N-methyl-, dihydrochloride is a bioactive chemical. | |||
T24453 |
Metamelfalan
NSC-67781,Metamelfalanum,NSC67781,NSC 67781,m-L-Sarcolysin |
||
Metamelfalan is an alkylating nitrogen mustard with potential antineoplastic activity. It causes crosslinking of DNA, thereby preventing DNA replication and eventually cellular proliferation. | |||
T30172 |
Aspartame acesulfame
乙酰舒泛-阿司帕坦盐,Aspartame acesulfame salt,Acesulfame mixture with aspartame |
||
Aspartame acesulfame, as an artificial sweetener, is 350 times sweeter than sucrose. | |||
T20165 |
Alitame anhydrous
CP54802,CP-54802,CP 54802 |
||
Alitame anhydrous is a non-nutritive sweetener. It is 2000 times sweeter than sucrose. | |||
T30052 |
Aniline, 4,4'-(heptamethylenedioxy)di-, dihydrochloride
|
||
Aniline, 4,4'-(heptamethylenedioxy)di-, dihydrochloride is a bioactive chemical. | |||
T75274 |
Cefetamet
|
||
Cefetamet 是一种头孢类抗生素。Cefetamet 具有研究上、下社区获得性呼吸道感染的潜力。 | |||
T126486 |
5,6,7,3',4'-Pentamethoxyflavanone
|
||
5,6,7,3',4'-Pentamethoxyflavanone 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126486。 | |||
T65094 |
3,3-Pentamethylene glutarimide
|
||
3,3-Pentamethylene glutarimide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65094,CAS号为 1130-32-1。 | |||
T30429 |
beta-Alitame
|
||
beta-Alitame is a non-nutritive sweetener that is 2000 times sweeter than sucrose. It is formed from aspartic acid, alanine & an amide. | |||
T26974 |
Cefetamet Hydrochloride
Cefetamet HCl,Cefetamet |
||
Cefetamet is a potent antibiotic to treat respiratory and urinary tract infections. | |||
T21103 |
Betamethasone acetate
Betamethasone 21-acetate |
||
Betamethasone acetate, the 21-acetate ester of betamethasone, is a synthetic glucocorticoid corticosteroid and a corticosteroid ester. | |||
T30057 | Aniline, 4,4'-(pentamethylenedioxy)bis(N-methyl-, dihydrochloride | ||
Aniline, 4,4'-(pentamethylenedioxy)bis(N-methyl-, dihydrochloride is a bioactive chemical. | |||
T65844 |
(S)-2-((tert-Butoxycarbonyl)amino)-5-(3-((2,2,4,6,7-pentamethyl-2,3-dihydrobenzofuran-5-yl)sulfonyl)guanidino)pentanoic acid
|
||
(S)-2-((tert-Butoxycarbonyl)amino)-5-(3-((2,2,4,6,7-pentamethyl-2,3-dihydrobenzofuran-5-yl)sulfonyl)guanidino)pentanoic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65844,CAS号为 200124-22-7。 | |||
T1729 |
3',4',5',5,7-Pentamethoxyflavanone
|
Others | Others |
3',4',5',5,7-Pentamethoxyflavanone 是一种天然黄酮化合物,在 Neoraptua magnifica var. magnifica 中发现。 | |||
T78537 |
Cefetamet pivoxyl
Ro 15-8075 free base |
Antibiotic | Microbiology/Virology |
Cefetamet pivoxyl为头孢类抗生素,能抑制355种肠道病原体Keime、革兰氏阴性菌(ausgenommenPseudomonas aeruginosa)及嗜肺军团菌。 | |||
T68775 |
Etamestrol
|
||
Etamestrol is a synthetic, steroidal estrogen described as an ovulation inhibitor or hormonal contraceptive | |||
T32017 |
m-Heptamethyleniminomethylbenzylguanidine sulfate
Guanidine, (3-(hexahydro-1(2H)-azocinylmethyl)benzyl)-, sulfate |
||
Guanidine, (3-(hexahydro-1(2H)-azocinylmethyl)benzyl)-, sulfate is a bioactive chemical. | |||
T66180 |
4,4-Pentamethylenepiperidine HCl
|
||
4,4-Pentamethylenepiperidine HCl 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66180,CAS号为 1125-01-5。 | |||
T13578 |
Betamethasone-17-butyrate-21-propionate
|
Others | Others |
Betamethasone-17-butyrate-21-propionate is a topical corticosteroid and may be used in the treatment of inflammatory skin diseases. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2A2486 |
3',4',5',5,7-Pentamethoxyflavone
5,7,3',4',5'-Pentamethoxyflavone |
Nrf2 | Immunology/Inflammation |
3',4',5',5,7-Pentamethoxyflavone 是从 Rutaceae 中发现的的一种天然黄铜类化合物,通过抑制Nrf2 通路克服化疗活性分子从而对癌细胞展现出耐药性。 | |||
T14008 |
2,2,5,7,8-Pentamethyl-6-Chromanol
PMC |
Androgen Receptor | Endocrinology/Hormones |
2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) 是维生素 E (α-tocopherol) 的抗氧化部分,能够有效的调节雄激素受体 (androgen receptor) 信号,及抗前列腺癌细胞系的抗癌活性。 | |||
T20754 |
Deltamethrin
Butoss,RU-22974,Esbecythrin,溴氰菊酯,K-Othrin,Decamethrin,RU 22974 |
Others | Others |
Deltamethrin (RU 22974) 是一种具有神经毒性的拟除虫菊酯杀虫剂,在大鼠中能够产生一系列可逆的运动症状(如包括后肢僵硬、舞蹈性关节炎)。 | |||
TN2121 |
3,5,7,3′,4′-Pentamethoxyflavone
栎精-3,5,7,3',4'-五甲醚,槲皮素3,5,7,3',4'-五甲基醚,Quercetin 3,5,7,3,4-pentamethyl ether |
Others | Others |
3,5,7,3′,4′-Pentamethoxyflavone (Quercetin 3,5,7,3,4-pentamethyl ether) 是一种分离自小花山奈中的多甲氧基黄酮。在分化早期,它可以调控转录因子,促进 3T3-L1 前脂肪细胞形成脂肪。 | |||
TN6195 | 5-Hydroxy-3,6,7,8,3'-pentamethoxy-4',5'-methylenedioxyflavone | ||
5-Hydroxy-3,6,7,8,3'-pentamethoxy-4',5'-methylenedioxyflavone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6195,CAS号为 82669-01-0。 | |||
T83412 | 2,3,4,6,7-Pentamethoxy-9,10-dihydrophenanthrene | ||
2,3,4,6,7-Pentamethoxy-9,10-dihydrophenanthrene为活性化合物,可自Bulbophyllum vaginatum分离得到。 | |||
TN6256 |
pentamethoxy-6,7-methylenedioxyflavone
3'-Hydroxy-3,5,8,4',5'-pentamethoxy-6,7-methylenedioxyflavone |
||
pentamethoxy-6,7-methylenedioxyflavone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6256,CAS号为 82668-94-8。 | |||
TN6355 | 6-Hydroxy-5,7,3',4',5'-pentamethoxyflavone | ||
6-Hydroxy-5,7,3',4',5'-pentamethoxyflavone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6355,CAS号为 29043-06-9。 | |||
TN7116 |
6'-Hydroxy-3,4,2',3',4'-pentamethoxychalcone
|
Others | Others |
6'-Hydroxy-3,4,2',3',4'-pentamethoxychalcone 是一种来自 Piper obliquum 的烯基酚,具有抗炎和抗菌活性。 | |||
TN6248 | 3'-Hydroxy-3,5,6,7,8,4',5'-heptamethoxyflavone | ||
3'-Hydroxy-3,5,6,7,8,4',5'-heptamethoxyflavone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6248,CAS号为 5244-28-0。 | |||
TN2864 |
3',4',5',3,5,6,7-Heptamethoxyflavone
|
Antifection | Microbiology/Virology |
3',4',5',3,5,6,7-Heptamethoxyflavone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2864,CAS号为 17245-30-6。 | |||
TN2481 |
1,2,3,6,7-Pentamethoxyxanthone
|
Others | Others |
1,2,3,6,7-Pentamethoxyxanthone is a natural product from Polygala tenuifolia. | |||
TN2382 |
3,5,7,8,3',4',5'-Heptamethoxyflavone
|
Others | Others |
3,5,7,8,3',4',5'-Heptamethoxyflavone is a natural product from Murraya exotica L |