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26

抑制剂 & 化合物

20

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
TP1493L1	PSA1 141-150 acetate PSA1 141-150 acetate(160215-60-1 free base)	Others	Others
	PSA1 141-150 acetate 用于癌症实验的免疫治疗，它是一种前列腺特异性抗原 1 肽。
TP1493	PSA1 (141-150) PSA1 141-150
	This Prostate Specific Antigen 1 peptide was used in the immunotherapy of cancer experiments.
T5092	AIM-100 AIM100	ACK	Tyrosine Kinase/Adaptors
	AIM-100 是选择性的 Ack1 抑制剂 (IC50:21.58 nM)。它还抑制 Tyr267磷酸化，但不抑制其他激酶，包括 PI3K 和 AKT 亚家族成员。它具有抗癌活性。
T19379	Ipsalazide	Autophagy	Autophagy
	Ipsalazide 是一种新型柳氮磺吡啶类似物，可用于治疗炎症性肠病。
T22871	Ipsapirone	5-HT Receptor	GPCR/G Protein; Neuroscience
	Ipsapirone 是 5-HT1A 受体的部分激动剂，在高剂量时对 5-HT2 和 α1-肾上腺素能功能产生抑制作用。
T13237L	Ropsacitinib Tyk2-IN-8,PF-06826647	Tyrosine Kinases	Tyrosine Kinase/Adaptors
	Ropsacitinib (PF-06826647) 是一种选择性TYK2抑制剂。Ropsacitinib 与Tyk2催化活性JH1结构域结合(IC50:17nM)。
T39349	Vocacapsaicin hydrochloride CA-008 hydrochloride	TRP/TRPV Channel	Membrane transporter/Ion channel
	Vocacapsaicin hydrochloride (CA-008 hydrochloride) 是非阿片类 TRPV1 激动剂，是辣椒素的原料，可用于缓解疼痛。
T1109	(Z)-Capsaicin Zucapsaicin,Civamide,cis-Capsaicin,珠卡赛辛,(Z)-辣椒素	TRP/TRPV Channel; HSV	Membrane transporter/Ion channel; Microbiology/Virology
	(Z)-Capsaicin (Zucapsaicin) 是天然辣椒素的合成顺式异构体，用于治疗膝骨关节炎。它是一种可口服的 TRPV1激动剂，可研究神经性疼痛。
T80966	Topsalysin PRX-302
	Topsalysin为PSA激活的前体蛋白质，同时是与人前列腺特异性抗原融合的孔隙形成蛋白（合成原气溶素）。研究显示Topsalysin能够抑制小鼠模型中的肿瘤生长。
TP1063	Psalmotoxin 1 PcTx1,Psalmopoeus cambridgei toxin-1
	Psalmotoxin 1 is a potent and selective acid-sensing ion channel 1a (ASIC1a) blocker.
T28459	Psammaplysene A
	Psammaplysene A is a FOXO1a nuclear export inhibitor.
T124402	7-O-Acetyllycopsamine N-oxide
	7-O-Acetyllycopsamine N-oxide 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T124402。
T39348	Vocacapsaicin CA-008,Vocacapsaicin
	Vocacapsaicin (CA-008), a prodrug of Capsaicin and a first-in-class non-opioid TRPV1 agonist, offers significant and enduring pain relief.
T28460	Psammaplysene B
	Psammaplysene B is a FOXO1a nuclear export inhibitor.
T16273	Napsagatran hydrate Ro 46-6240/010 hydrate,Ro 46-6240 hydrate	Others	Others
	Napsagatran hydrate is a novel and specific inhibitor of thrombin.
T23912	CPSA
	CPSA is an effective and selective AKR1C1 inhibitor.
T123864	Lycopsamine N-oxide
	Lycopsamine N-oxide 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T123864。
T8683	Mipsagargin G-202	Others	Others
	Mipsagargin (G-202) 是一种抑制 DNA 生物合成的新型抗生素。
T82645	Cyclic PSAP peptide
	Cyclic PSAP peptide（DWLPK）是一种环五肽，具有活性分子特性，在体内能够抑制肿瘤转移扩散和发展。
T27623	Ipsapirone hydrochloride BAY q 7821,BAY q-7821,BAY q7821,Ipsapirone HCl
	Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.
T125760	Dipsacussaponin C
	Dipsacussaponin C 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T125760。
T29110	VPC-13163 2,3-dihydro-2,3'-Bi-1H-indole,VPC13163,NSC52361,NSC 52361,VPC 13163	Others	Others
	VPC-13163 (NSC-52361) 对 LNCaP 和耐恩杂鲁胺的前列腺癌细胞系 (MR49F) 具有很强的抗增殖活性，而它不影响 AR 独立 PC3 细胞系的生长。它还抑制 LNCaP 和 MR49F 中的前列腺特异性抗原 (PSA) 并降低 AR 靶基因 PSA 和 TMPRSS2 的表达。这些发现表明 VPC-13566 表现出 AR BF3 特定的作用机制。
T77574	ROS inducer 1	ROS; Antibiotic	Immunology/Inflammation; Microbiology/Virology
	ROS inducer 1 是一种具有杀菌作用的小分子化合物，对 Xanthomonas axonopodis pv. citri (Xac)、Xanthomonas oryzae pv. oryzae (Xoo)和 Pseudomonas syringae pv. actinidiae (Psa) 具有抑制作用。ROS inducer 1 诱 Xanthomonas 细胞内 ROS 的产生可用于研究农作物细菌感染。
T80552	Prostate Specific Antigen Substrate
	Prostate Specific Antigen Substrate为前列腺特异性抗原（PSA）的荧光底物，专用于检测PSA的酶活性。
T78976	Antibacterial agent 141
	Antibacterialagent 141（Compound B14）针对四种植物病原体Xoo、Xac、Psa与Cmm展现出了抗菌效果，其EC50值为1.28 μM。该化合物能够抑制细胞膜形成并改变细胞透性。
T76675	Clazakizumab
	Clazakizumab是一种具有高亲和力和特异性的单克隆抗体，针对IL-6(白细胞介素-6)细胞因子。它可能对抑制COVID-19中因SARS-CoV-2引起的细胞因子反应有帮助。此外，Clazakizumab也被用于研究银屑病关节炎(PsA)和肾抗体介导的排斥反应。

化合物

PSA1 141-150 acetate

Cat.No: TP1493L1

Synonym: PSA1 141-150 acetate(160215-60-1 free base)

Target: Others

PSA1 (141-150)

Cat.No: TP1493

Synonym: PSA1 141-150

Cat.No: T5092

Synonym: AIM100

Target: ACK

Cat.No: T19379

Target: Autophagy

Cat.No: T22871

Target: 5-HT Receptor

Cat.No: T13237L

Synonym: Tyk2-IN-8,PF-06826647

Target: Tyrosine Kinases

Vocacapsaicin hydrochloride

Cat.No: T39349

Synonym: CA-008 hydrochloride

Target: TRP/TRPV Channel

Cat.No: T1109

Synonym: Zucapsaicin,Civamide,cis-Capsaicin,珠卡赛辛,(Z)-辣椒素

Target: TRP/TRPV Channel, HSV

Cat.No: T80966

Synonym: PRX-302

Psalmotoxin 1

Cat.No: TP1063

Synonym: PcTx1,Psalmopoeus cambridgei toxin-1

Psammaplysene A

Cat.No: T28459

7-O-Acetyllycopsamine N-oxide

Cat.No: T124402

Cat.No: T39348

Synonym: CA-008,Vocacapsaicin

Psammaplysene B

Cat.No: T28460

Napsagatran hydrate

Cat.No: T16273

Synonym: Ro 46-6240/010 hydrate,Ro 46-6240 hydrate

Target: Others

Cat.No: T23912

Lycopsamine N-oxide

Cat.No: T123864

Cat.No: T8683

Synonym: G-202

Target: Others

Cyclic PSAP peptide

Cat.No: T82645

Ipsapirone hydrochloride

Cat.No: T27623

Synonym: BAY q 7821,BAY q-7821,BAY q7821,Ipsapirone HCl

Dipsacussaponin C

Cat.No: T125760

Cat.No: T29110

Synonym: 2,3-dihydro-2,3'-Bi-1H-indole,VPC13163,NSC52361,NSC 52361,VPC 13163

Target: Others

Cat.No: T77574

Target: ROS, Antibiotic

Prostate Specific Antigen Substrate

Cat.No: T80552

Antibacterial agent 141

Cat.No: T78976

Cat.No: T76675

Cat. No.	Product Name	Target	Signaling Pathways
T7177	Capsazepine	Apoptosis; TRP/TRPV Channel	Apoptosis; Membrane transporter/Ion channel
	Capsazepine 是一种 TRPV1 受体的拮抗剂， IC50值为 562 nM。它可阻断由激活 TRPV1 离子通道的辣椒素引起的热痛感，是辣椒素拮抗剂。
T2163	Dihydrocapsaicin CCRIS1589,二氢辣椒素,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide	Others; TRP/TRPV Channel	Membrane transporter/Ion channel; Others
	Dihydrocapsaicin (CCRIS1589) 是一种天然来源的辣椒素，是TRPV1的选择性激动剂，同时可以增加 p-Akt 水平。它可以增强低温诱导的神经保护。
TN1739	Homodihydrocapsaicin I 高二氢辣椒素,高二氢辣椒素I	Others	Others
	Homodihydrocapsaicin I 是一种辣椒素，分离自辣椒果实中。
T3372	Dipsacoside B	Others	Others
	Dipsacoside B 是主要的具有生物活性的皂素，可用作标志物。
T1062	Capsaicin Qutenza,8-Methyl-N-vanillyl-trans-6-nonenamide,天然辣椒素,Vanilloid,辣椒素,(E)-Capsaicin,Zostrix	Apoptosis; TRP/TRPV Channel; Autophagy	Apoptosis; Autophagy; Membrane transporter/Ion channel
	Capsaicin ((E)-Capsaicin) 属于天然产物，提取自辣椒，是一种 TRPV1 激动剂 (EC50=0.29 μM)。Capsaicin 具有抗肿瘤、抗炎、抗氧化、神经保护等活性。
T3421	Nordihydrocapsaicin	Others	Others
	Nordihydrocapsaicin(诺地氢辣椒碱)是Capsaicin(辣椒素)的模拟物和同源物，属于在Capsicum(辣椒)中发现的Capsaicinoid(辣椒素类)化合物。
T39018	Capsaicin β-D-glucopyranoside
	Capsaicin β-D-glucopyranoside, a glucoside converted by Capsaicin, is the bioactive compound found in chili peppers responsible for their characteristic pungent flavor.
T36303	Psammaplin A
	Psammaplin A, a marine metabolite, functions as a robust inhibitor of HDAC and DNA methyltransferases, displaying notable potency and selectivity as a DAC1 inhibitor, with an IC50 value of 0.9 nM. It exhibits antimicrobial effects against Gram-positive bacteria and inhibits both DNA synthesis and DNA gyrase activity, also demonstrating antitumor activity[1][2].
T33029	7-Acetyllycopsamine Lycopsamine `1-acetate,7-乙酰基环磷酰胺
	Lycopsamine `1-acetate is a bioactive chemical.
TN1122	Dipsanoside A	Others	Others
	Dipsanoside A is a natural product
T82187	Homocapsaicin II
	Homocapsaicin II, 提取自Capsicum annuum L果实，为一种辣椒素类化合物。
TN1123	Dipsanoside B 续断苷 B,续断苷B	Others	Others
	Dipsanoside B is a natural product
TN3588	Capsanthin	Others	Others
	Capsanthin 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN3588，CAS号为 465-42-9。
T22729	Dipsacobioside	Others	Others
	Dipsacobioside is extracted from Anemone hupehensis.
T33028	Lycopsamine
	Lycopsamine is a bioactive chemical.
T83309	5,22-Dioxokopsane
	5,22-Dioxokopsane为源自Kopsia officinalis的单萜类吲哚生物碱。
TN5878	7,2',4'-Trihydroxy-5-methoxy-3-phenylcoumarin
	7,2',4'-Trihydroxy-5-methoxy-3-arylcoumarin shows activity in inhibiting prostate specific antigen (PSA) secreted from androgen dependent prostate cancer cell line, LNCaP cells.
TN3416	Angelol M	Others	Others
	Angelol M shows activity in inhibiting prostate specific antigen (PSA) secreted from androgen dependent prostate cancer cell line, LNCaP cells.
T75467	Asperglaucin A
	Asperglaucin A 代表一种不寻常的类苯酞衍生物。Asperglaucin A 对两种植物病原体Pseudomonas syringae pv actinidae(Psa) 和Bacillus cereus 具有有效的抗菌活性，MIC 值为 6.25 μM。
T75468	Asperglaucin B
	Asperglaucin B 是一种来自真菌Aspergillus chevalieriSQ-8 的烷基化水杨醛衍生物，具有抗菌活性。Asperglaucin B 对两种植物病原体Pseudomonas syringae pv actinidae(Psa)和Bacillus cereus 显示出有效的抗菌活性，MIC 值为 6.25 μM。

天然产物

Cat.No: T7177

Target: Apoptosis, TRP/TRPV Channel

Dihydrocapsaicin

Cat.No: T2163

Synonym: CCRIS1589,二氢辣椒素,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide

Target: Others, TRP/TRPV Channel

Homodihydrocapsaicin I

Cat.No: TN1739

Synonym: 高二氢辣椒素,高二氢辣椒素I

Target: Others

Cat.No: T3372

Target: Others

Cat.No: T1062

Synonym: Qutenza,8-Methyl-N-vanillyl-trans-6-nonenamide,天然辣椒素,Vanilloid,辣椒素,(E)-Capsaicin,Zostrix

Target: Apoptosis, TRP/TRPV Channel, Autophagy

Nordihydrocapsaicin

Cat.No: T3421

Target: Others

Capsaicin β-D-glucopyranoside

Cat.No: T39018

Cat.No: T36303

7-Acetyllycopsamine

Cat.No: T33029

Synonym: Lycopsamine `1-acetate,7-乙酰基环磷酰胺

Cat.No: TN1122

Target: Others

Homocapsaicin II

Cat.No: T82187

Cat.No: TN1123

Synonym: 续断苷 B,续断苷B

Target: Others

Cat.No: TN3588

Target: Others

Cat.No: T22729

Target: Others

Cat.No: T33028

5,22-Dioxokopsane

Cat.No: T83309

7,2',4'-Trihydroxy-5-methoxy-3-phenylcoumarin

Cat.No: TN5878

Cat.No: TN3416

Target: Others

Cat.No: T75467

Cat.No: T75468

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