4
2
Cat. No. | Product Name | Target | Signaling Pathways |
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T69057 |
Elliptinium acetate
NSC 264137,Celiptium,NSC 264137 ; Celiptium |
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Elliptinium acetate (NSC 264137)为DNA插层剂,对L1210细胞显示出明显细胞毒性,并能与其核酸进行共价结合。该化合物主要用于癌症研究,特别是转移性乳腺癌。 | |||
T13462 |
(+)-DHMEQ
(1R,2R,6R)-Dehydroxymethylepoxyquinomicin,(1R,2R,6R)-DHMEQ |
Others | Others |
(+)-DHMEQ is an antioxidant transcription factor Nrf2 activator. (+)-DHMEQ is the enantiomer of (-)-DHMEQ. | |||
T11018 |
DHMEQ racemate
rel-DHMEQ |
NF-κB | NF-κB |
DHMEQ racemate is an NF-κB inhibitor. The activity of DHMEQ racemate is lower than (-)-DHMEQ. | |||
T82222 |
H-D-MeAla-EtVaI-VaI-MeLeu-AIa-D-AIa-MeLeu-MeLeu-MeVaI-MeBmt(OAc)-Abu-O-CH2-CH2-NHMe
|
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H-D-MeAla-EtVal-Val-MeLeu-AIa-D-AIa-MeLeu-MeLeu-MeVal-MeBmt(OAc)-Abu-O-CH2-CH2-NHMe 是一种非免疫抑制性的环孢菌素A衍生物,具备研究先天性肌营养不良症潜力[1]。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN3525 |
Boehmenan
|
ERK; Phosphatase; EGFR; PARP; MEK; Wnt/beta-catenin; Akt; Caspase; STAT; p53 | Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; JAK/STAT signaling; MAPK; Metabolism; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells; Tyrosine Kinase/Adaptors |
(±)-Boehmenan shows potent protein-tyrosine phosphatase 1B (PTP1B) inhibitory activity in vitro with the IC(50) values of 43.5 uM, it inhibits PTP1B activity in a competitive manner. Boehmenan exhibits the potent cytotoxic effects against many cancer cell | |||
TN5423 |
Bisdemethoxyboehmenan
|
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Bisdemethoxyboehmenan 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5423,CAS号为 146918-26-5。 |