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1

抑制剂 & 化合物

18

天然产物

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Cat. No. Product Name Target Signaling Pathways
T29887 Aloe emodin anthrone

Aloe emodin anthrone is a stimulant-laxative which has been shown to enhance colonic membrane permeability of water-soluble and poorly permeable compounds.

化合物

Aloe emodin anthrone
Cat.No: T29887
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2869 Emodin

Frangula emodin,大黄素

SARS-CoV; Casein Kinase; Autophagy Autophagy; Metabolism; Microbiology/Virology; Stem Cells
Emodin (Frangula emodin) 是蒽醌衍生物,有抗SARS-CoV 作用。它阻断 SARS 冠状病毒刺突蛋白和血管紧张素转化酶 2 的相互作用。它抑制酪蛋白激酶 2 ,具有抗炎和抗癌作用。它可改善饮食诱导的肥胖小鼠的代谢紊乱。
T2843 Aloe emodin

芦荟大黄素,NSC 38628,3-Hydroxymethylchrysazine,Rhabarberone,Aloe-emodin

Autophagy; HSV Autophagy; Microbiology/Virology
Aloe emodin (Rhabarberone) 是从芦荟叶中提取出的一种羟基蒽醌,在体内外有抗肿瘤活性。
T3900 Emodin-8-glucoside

大黄素-8-β-D-吡喃葡萄糖苷,Emodin glucoside B,Anthraglycoside B

Others Others
Emodin-8-glucoside (Anthraglycoside B) 是从芦荟中分离出的蒽醌衍生物,与 DNA 的小沟结合。它具有保护缺血和再灌注引起的局灶性脑损伤的作用。它直接刺激成骨细胞的细胞增殖和分化。
T2S0389 Emodin-1-O-β-D-glucopyranoside

大黄素-1-O-Β-D-吡喃葡萄糖苷,大黄素-1-O-β-D-葡萄糖苷,Emodin-1-O-glucoside

Others Others
Emodin-1-O-β-D-glucopyranoside (Emodin-1-O-glucoside) 是一种非竞争性细菌神经氨酸酶抑制剂,IC50为 0.85 μM,提取自药用植物虎杖中。
TN1053 Aloe-emodin-8-O-β-D-glucopyranoside

Aloe-emodin-8-O-beta-D-glucopyranoside,芦荟大黄素-8-O-β-D-葡萄糖苷

Phosphatase Metabolism
Aloe-emodin-8-O-β-D-glucopyranoside (Aloe-emodin-8-O-beta-D-glucopyranoside) 是一种分离自Saussrurea lappa 中的化合物,是一种温和的人类蛋白酪氨酸磷酸酶 1B 抑制剂,其IC50=26.6 μM。
TN6774 Emodin 6-O-β-D-glucoside

大黄素-6-O-β-D-葡萄糖苷,Glucoemodin

Others Others
Emodin 6-O-β-D-glucoside (Glucoemodin) 是一种从 Reynoutria japonica 中提取的活性化合物。它具有显著的抗炎和屏障保护活性,可用于研究动脉粥样硬化及糖尿病并发症。
TN6740 Emodinanthrone

大黄素蒽酮,Emodin anthranol,Emodin anthrone,emodinol

Others; Antibiotic Microbiology/Virology; Others
Emodinanthrone 是一种蒽醌类化合物,是大黄素的前体,具有抗生素活性。它抑制大肠杆菌膜囊泡中呼吸驱动的溶质转运。
TN1604 Emodin-1-O-β-gentiobioside

Emodin-1-O-beta-gentiobioside,大黄素-1-O-Β-龙胆二糖苷

Others Others
Emodin-1-O-beta-gentiobioside is a natural product
T29888 Aloe-emodin-glucoside

Aloe-emodin-glucoside is a stimulant-laxative which has been shown to enhance colonic membrane permeability of water-soluble and poorly permeable compounds.
TN1371 Aloe-emodin-3-(hydroxymethyl)-O-β-D-glucopyranoside

芦荟大黄素-3-(羟甲基)-O-Β-D-葡萄糖苷,ALOE-EMODIN-GLUCOSIDE,Aloe-emodin-3-(hydroxymethyl)-O-beta-D-glucopyranoside

Others Others
Aloe-emodin-3-(hydroxymethyl)-O-beta-D-glucopyranoside is a natural product
TN2559 1-O-Methylnataloe-emodin

Others Others
1-O-Methylnataloe-emodin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2559,CAS号为 103392-51-4。
TN6482 Emodin-8-O-beta-gentiobioside

Emodin-8-O-beta-gentiobioside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6482,CAS号为 66466-22-6。
T79997 (±)-Emodin bianthrone

Parasite Microbiology/Virology
(±)-Emodin bianthrone (compound 10) 是具抗疟、抗结核及抗真菌作用的天然化合物。
T82718 cis-Emodin bianthrone

Cis-Emodin bianthrone为大黄素蒽酮的高聚氧化产物,其丙酮溶液在空气中表现出稳定性。
T83382 2-Hydroxyl emodin-1-methyl ether

2-Hydroxyl emodin-1-methyl ether (Compound 5) 是源自Cassia obtusifolia种子的天然蒽醌类化合物。
T80023 1-O-Methylemodin

1-O-Mmethylemodin为自Zopfiella longicaudata分离得到的天然产物,具备抗真菌活性。
T2S1181 Aloenin

Aloenin A,Aloearbonaside,芦荟宁

Beta-Secretase; AChR Neuroscience
Aloenin (Aloenin A) A 是一种具有清除过氧自由基作用的天然产物,对 β-分泌酶 (BACE) 具有中等抑制活性。
TN2278 Torachrysone

决明柯酮

Antifection Microbiology/Virology
Torachrysone shows promising antioxidant activity. Torachrysone, toralactone , aloe-emodin, rhein and emodin show noticeable antibacterial effects on four strains of methicillin-resistant Staphylococcus aureus with a minimum inhibitory concentration of 2-

天然产物

Emodin
Cat.No: T2869
Synonym: Frangula emodin,大黄素
Target: SARS-CoV, Casein Kinase, Autophagy
Aloe emodin
Cat.No: T2843
Synonym: 芦荟大黄素,NSC 38628,3-Hydroxymethylchrysazine,Rhabarberone,Aloe-emodin
Target: Autophagy, HSV
Emodin-8-glucoside
Cat.No: T3900
Synonym: 大黄素-8-β-D-吡喃葡萄糖苷,Emodin glucoside B,Anthraglycoside B
Target: Others
Emodin-1-O-β-D-glucopyranoside
Cat.No: T2S0389
Synonym: 大黄素-1-O-Β-D-吡喃葡萄糖苷,大黄素-1-O-β-D-葡萄糖苷,Emodin-1-O-glucoside
Target: Others
Aloe-emodin-8-O-β-D-glucopyranoside
Cat.No: TN1053
Synonym: Aloe-emodin-8-O-beta-D-glucopyranoside,芦荟大黄素-8-O-β-D-葡萄糖苷
Target: Phosphatase
Emodin 6-O-β-D-glucoside
Cat.No: TN6774
Synonym: 大黄素-6-O-β-D-葡萄糖苷,Glucoemodin
Target: Others
Emodinanthrone
Cat.No: TN6740
Synonym: 大黄素蒽酮,Emodin anthranol,Emodin anthrone,emodinol
Target: Others, Antibiotic
Emodin-1-O-β-gentiobioside
Cat.No: TN1604
Synonym: Emodin-1-O-beta-gentiobioside,大黄素-1-O-Β-龙胆二糖苷
Target: Others
Aloe-emodin-glucoside
Cat.No: T29888
Synonym:
Target:
Aloe-emodin-3-(hydroxymethyl)-O-β-D-glucopyranoside
Cat.No: TN1371
Synonym: 芦荟大黄素-3-(羟甲基)-O-Β-D-葡萄糖苷,ALOE-EMODIN-GLUCOSIDE,Aloe-emodin-3-(hydroxymethyl)-O-beta-D-glucopyranoside
Target: Others
1-O-Methylnataloe-emodin
Cat.No: TN2559
Synonym:
Target: Others
Emodin-8-O-beta-gentiobioside
Cat.No: TN6482
Synonym:
Target:
(±)-Emodin bianthrone
Cat.No: T79997
Synonym:
Target: Parasite
cis-Emodin bianthrone
Cat.No: T82718
Synonym:
Target:
2-Hydroxyl emodin-1-methyl ether
Cat.No: T83382
Synonym:
Target:
1-O-Methylemodin
Cat.No: T80023
Synonym:
Target:
Aloenin
Cat.No: T2S1181
Synonym: Aloenin A,Aloearbonaside,芦荟宁
Target: Beta-Secretase, AChR
Torachrysone
Cat.No: TN2278
Synonym: 决明柯酮
Target: Antifection
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